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CellMiner Address: https://discover.nci.nih.gov/cellminer/
CellMiner Database Version: 2.16
Human Genome Version: HG-19
Date: 10-28-2026
Table 3: Drugs and compounds with almanac combo scores
NSC #1Drug nameClinical statusMechanism of actionNSC #2Drug nameClinical statusMechanism of action
740MethotrexateFDA approvedDf|DHFR752ThioguanineFDA approvedDs|IMPDH2|IMPDH
740MethotrexateFDA approvedDf|DHFR3053DactinomycinFDA approvedDb|RNA polymerase I
740MethotrexateFDA approvedDf|DHFR3088ChlorambucilFDA approvedA7|AlkAg
740MethotrexateFDA approvedDf|DHFR8806MelphalanFDA approvedA7|AlkAg
740MethotrexateFDA approvedDf|DHFR9706Triethylenemelamine-A7|AlkAg
740MethotrexateFDA approvedDf|DHFR13875HexamethylmelamineFDA approvedDb|AlkAg
740MethotrexateFDA approvedDf|DHFR19893FluorouracilFDA approvedDs|Rs|TYMS
740MethotrexateFDA approvedDf|DHFR24559MithramycinFDA approvedDb|Rs
740MethotrexateFDA approvedDf|DHFR32065HydroxyureaFDA approvedAM|Dr
740MethotrexateFDA approvedDf|DHFR34462Uracil mustardFDA approvedA7|AlkAg
740MethotrexateFDA approvedDf|DHFR38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
740MethotrexateFDA approvedDf|DHFR45388DacarbazineFDA approvedA7|AlkAg
740MethotrexateFDA approvedDf|DHFR49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
740MethotrexateFDA approvedDf|DHFR71423Megestrol acetateFDA approvedHo|PGR
740MethotrexateFDA approvedDf|DHFR79037LomustineFDA approvedA6|AlkAg
740MethotrexateFDA approvedDf|DHFR82151Daunorubicin hydrochlorideFDA approvedTOP2
740MethotrexateFDA approvedDf|DHFR102816AzacitidineFDA approvedDNMT
740MethotrexateFDA approvedDf|DHFR122819TeniposideFDA approvedTOP2
740MethotrexateFDA approvedDf|DHFR123127Doxorubicin hydrochlorideFDA approvedTOP2
740MethotrexateFDA approvedDf|DHFR125066BleomycinFDA approvedDb
740MethotrexateFDA approvedDf|DHFR125973PaclitaxelFDA approvedTUBB|Tu-stab
740MethotrexateFDA approvedDf|DHFR138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
740MethotrexateFDA approvedDf|DHFR141540EtoposideFDA approvedTOP2
740MethotrexateFDA approvedDf|DHFR169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
740MethotrexateFDA approvedDf|DHFR226080RapamycinFDA approvedPK:STK,MTOR
740MethotrexateFDA approvedDf|DHFR246131ValrubicinFDA approvedTOP2
740MethotrexateFDA approvedDf|DHFR279836MitoxantroneFDA approvedTOP2
740MethotrexateFDA approvedDf|DHFR608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
740MethotrexateFDA approvedDf|DHFR628503DocetaxelFDA approvedTUBB|Tu-stab
740MethotrexateFDA approvedDf|DHFR673596SN 38Clinical trialTOP1
740MethotrexateFDA approvedDf|DHFR698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
740MethotrexateFDA approvedDf|DHFR701852VorinostatFDA approvedHDAC
740MethotrexateFDA approvedDf|DHFR713563ExemestaneFDA approvedHo|CYP19A1
740MethotrexateFDA approvedDf|DHFR715055GefitinibFDA approvedPK:YK,EGFR
740MethotrexateFDA approvedDf|DHFR719276FulvestrantFDA approvedAM|Ho|ESR|SERM
740MethotrexateFDA approvedDf|DHFR719344AnastrozoleFDA approvedHo|CYP19A1
740MethotrexateFDA approvedDf|DHFR719345LetrozoleFDA approvedHo|CYP19A1
740MethotrexateFDA approvedDf|DHFR721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
740MethotrexateFDA approvedDf|DHFR732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
740MethotrexateFDA approvedDf|DHFR733504EverolimusFDA approvedPK:STK,MTOR
740MethotrexateFDA approvedDf|DHFR737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
740MethotrexateFDA approvedDf|DHFR745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
740MethotrexateFDA approvedDf|DHFR747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
740MethotrexateFDA approvedDf|DHFR747972LenalidomideFDA approvedFT|Immunomodulatory
740MethotrexateFDA approvedDf|DHFR747974RaloxifeneFDA approvedHo|SERM
740MethotrexateFDA approvedDf|DHFR749226AbirateroneFDA approvedHo|CYP17A1
740MethotrexateFDA approvedDf|DHFR750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
740MethotrexateFDA approvedDf|DHFR753082VemurafenibFDA approvedPK:YK,BRAF
740MethotrexateFDA approvedDf|DHFR754143RomidepsinFDA approvedHDAC
740MethotrexateFDA approvedDf|DHFR754230PralatrexateFDA approvedDf|CTNNB1|DHFR
740MethotrexateFDA approvedDf|DHFR755986VismodegibFDA approvedSMO|PK:YK
740MethotrexateFDA approvedDf|DHFR756645CrizotinibFDA approvedPK:YK,MET,ALK
740MethotrexateFDA approvedDf|DHFR757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
740MethotrexateFDA approvedDf|DHFR760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
740MethotrexateFDA approvedDf|DHFR761432CabazitaxelFDA approvedTUBB|Tu-stab
740MethotrexateFDA approvedDf|DHFR763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
750BusulfanFDA approvedA7|AlkAg740MethotrexateFDA approvedDf|DHFR
750BusulfanFDA approvedA7|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
750BusulfanFDA approvedA7|AlkAg7556-MercaptopurineFDA approvedDs|PPAT
750BusulfanFDA approvedA7|AlkAg762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
750BusulfanFDA approvedA7|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
750BusulfanFDA approvedA7|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
750BusulfanFDA approvedA7|AlkAg6396ThiotepaFDA approvedA7|AlkAg
750BusulfanFDA approvedA7|AlkAg8806MelphalanFDA approvedA7|AlkAg
750BusulfanFDA approvedA7|AlkAg9706Triethylenemelamine-A7|AlkAg
750BusulfanFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
750BusulfanFDA approvedA7|AlkAg18509Aminolevulinic Acid HydrochlorideFDA approvedAM
750BusulfanFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
750BusulfanFDA approvedA7|AlkAg24559MithramycinFDA approvedDb|Rs
750BusulfanFDA approvedA7|AlkAg25154PipobromanFDA approvedA7|AlkAg
750BusulfanFDA approvedA7|AlkAg27640FloxuridineFDA approvedDs|TYMS
750BusulfanFDA approvedA7|AlkAg32065HydroxyureaFDA approvedAM|Dr
750BusulfanFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
750BusulfanFDA approvedA7|AlkAg38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
750BusulfanFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
750BusulfanFDA approvedA7|AlkAg49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
750BusulfanFDA approvedA7|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
750BusulfanFDA approvedA7|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
750BusulfanFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
750BusulfanFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
750BusulfanFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
750BusulfanFDA approvedA7|AlkAg102816AzacitidineFDA approvedDNMT
750BusulfanFDA approvedA7|AlkAg105014CladribineFDA approvedDs|ADA
750BusulfanFDA approvedA7|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
750BusulfanFDA approvedA7|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
750BusulfanFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
750BusulfanFDA approvedA7|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
750BusulfanFDA approvedA7|AlkAg125066BleomycinFDA approvedDb
750BusulfanFDA approvedA7|AlkAg125973PaclitaxelFDA approvedTUBB|Tu-stab
750BusulfanFDA approvedA7|AlkAg138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
750BusulfanFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
750BusulfanFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
750BusulfanFDA approvedA7|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
750BusulfanFDA approvedA7|AlkAg226080RapamycinFDA approvedPK:STK,MTOR
750BusulfanFDA approvedA7|AlkAg241240CarboplatinFDA approvedA7|AlkAg
750BusulfanFDA approvedA7|AlkAg246131ValrubicinFDA approvedTOP2
750BusulfanFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
750BusulfanFDA approvedA7|AlkAg362856TemozolomideFDA approvedA7|AlkAg
750BusulfanFDA approvedA7|AlkAg606869ClofarabineFDA approvedDs
750BusulfanFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
750BusulfanFDA approvedA7|AlkAg613327Gemcitabine HCLFDA approvedDs
750BusulfanFDA approvedA7|AlkAg628503DocetaxelFDA approvedTUBB|Tu-stab
750BusulfanFDA approvedA7|AlkAg673596SN 38Clinical trialTOP1
750BusulfanFDA approvedA7|AlkAg686673NelarabineFDA approvedDs
750BusulfanFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
750BusulfanFDA approvedA7|AlkAg701852VorinostatFDA approvedHDAC
750BusulfanFDA approvedA7|AlkAg712807CapecitabineFDA approvedDs|TYMS
750BusulfanFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
750BusulfanFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
750BusulfanFDA approvedA7|AlkAg719276FulvestrantFDA approvedAM|Ho|ESR|SERM
750BusulfanFDA approvedA7|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
750BusulfanFDA approvedA7|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
750BusulfanFDA approvedA7|AlkAg721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
750BusulfanFDA approvedA7|AlkAg732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
750BusulfanFDA approvedA7|AlkAg733504EverolimusFDA approvedPK:STK,MTOR
750BusulfanFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
750BusulfanFDA approvedA7|AlkAg743414ImatinibFDA approvedBCR-ABL|PK:YK
750BusulfanFDA approvedA7|AlkAg745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
750BusulfanFDA approvedA7|AlkAg747599NilotinibFDA approvedBCR-ABL|PK:YK
750BusulfanFDA approvedA7|AlkAg747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
750BusulfanFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
750BusulfanFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
750BusulfanFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
750BusulfanFDA approvedA7|AlkAg750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
750BusulfanFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
750BusulfanFDA approvedA7|AlkAg754143RomidepsinFDA approvedHDAC
750BusulfanFDA approvedA7|AlkAg754230PralatrexateFDA approvedDf|CTNNB1|DHFR
750BusulfanFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
750BusulfanFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
750BusulfanFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
750BusulfanFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
750BusulfanFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
750BusulfanFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
752ThioguanineFDA approvedDs|IMPDH2|IMPDH3088ChlorambucilFDA approvedA7|AlkAg
752ThioguanineFDA approvedDs|IMPDH2|IMPDH8806MelphalanFDA approvedA7|AlkAg
752ThioguanineFDA approvedDs|IMPDH2|IMPDH9706Triethylenemelamine-A7|AlkAg
752ThioguanineFDA approvedDs|IMPDH2|IMPDH13875HexamethylmelamineFDA approvedDb|AlkAg
752ThioguanineFDA approvedDs|IMPDH2|IMPDH19893FluorouracilFDA approvedDs|Rs|TYMS
752ThioguanineFDA approvedDs|IMPDH2|IMPDH34462Uracil mustardFDA approvedA7|AlkAg
752ThioguanineFDA approvedDs|IMPDH2|IMPDH45388DacarbazineFDA approvedA7|AlkAg
752ThioguanineFDA approvedDs|IMPDH2|IMPDH71423Megestrol acetateFDA approvedHo|PGR
752ThioguanineFDA approvedDs|IMPDH2|IMPDH79037LomustineFDA approvedA6|AlkAg
752ThioguanineFDA approvedDs|IMPDH2|IMPDH82151Daunorubicin hydrochlorideFDA approvedTOP2
752ThioguanineFDA approvedDs|IMPDH2|IMPDH122819TeniposideFDA approvedTOP2
752ThioguanineFDA approvedDs|IMPDH2|IMPDH123127Doxorubicin hydrochlorideFDA approvedTOP2
752ThioguanineFDA approvedDs|IMPDH2|IMPDH141540EtoposideFDA approvedTOP2
752ThioguanineFDA approvedDs|IMPDH2|IMPDH169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
752ThioguanineFDA approvedDs|IMPDH2|IMPDH279836MitoxantroneFDA approvedTOP2
752ThioguanineFDA approvedDs|IMPDH2|IMPDH608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
752ThioguanineFDA approvedDs|IMPDH2|IMPDH698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
752ThioguanineFDA approvedDs|IMPDH2|IMPDH713563ExemestaneFDA approvedHo|CYP19A1
752ThioguanineFDA approvedDs|IMPDH2|IMPDH715055GefitinibFDA approvedPK:YK,EGFR
752ThioguanineFDA approvedDs|IMPDH2|IMPDH737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
752ThioguanineFDA approvedDs|IMPDH2|IMPDH747972LenalidomideFDA approvedFT|Immunomodulatory
752ThioguanineFDA approvedDs|IMPDH2|IMPDH747974RaloxifeneFDA approvedHo|SERM
752ThioguanineFDA approvedDs|IMPDH2|IMPDH749226AbirateroneFDA approvedHo|CYP17A1
752ThioguanineFDA approvedDs|IMPDH2|IMPDH753082VemurafenibFDA approvedPK:YK,BRAF
752ThioguanineFDA approvedDs|IMPDH2|IMPDH755986VismodegibFDA approvedSMO|PK:YK
752ThioguanineFDA approvedDs|IMPDH2|IMPDH756645CrizotinibFDA approvedPK:YK,MET,ALK
752ThioguanineFDA approvedDs|IMPDH2|IMPDH757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
752ThioguanineFDA approvedDs|IMPDH2|IMPDH760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
752ThioguanineFDA approvedDs|IMPDH2|IMPDH761432CabazitaxelFDA approvedTUBB|Tu-stab
752ThioguanineFDA approvedDs|IMPDH2|IMPDH763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
7556-MercaptopurineFDA approvedDs|PPAT740MethotrexateFDA approvedDf|DHFR
7556-MercaptopurineFDA approvedDs|PPAT752ThioguanineFDA approvedDs|IMPDH2|IMPDH
7556-MercaptopurineFDA approvedDs|PPAT3053DactinomycinFDA approvedDb|RNA polymerase I
7556-MercaptopurineFDA approvedDs|PPAT3088ChlorambucilFDA approvedA7|AlkAg
7556-MercaptopurineFDA approvedDs|PPAT6396ThiotepaFDA approvedA7|AlkAg
7556-MercaptopurineFDA approvedDs|PPAT8806MelphalanFDA approvedA7|AlkAg
7556-MercaptopurineFDA approvedDs|PPAT9706Triethylenemelamine-A7|AlkAg
7556-MercaptopurineFDA approvedDs|PPAT13875HexamethylmelamineFDA approvedDb|AlkAg
7556-MercaptopurineFDA approvedDs|PPAT19893FluorouracilFDA approvedDs|Rs|TYMS
7556-MercaptopurineFDA approvedDs|PPAT24559MithramycinFDA approvedDb|Rs
7556-MercaptopurineFDA approvedDs|PPAT27640FloxuridineFDA approvedDs|TYMS
7556-MercaptopurineFDA approvedDs|PPAT32065HydroxyureaFDA approvedAM|Dr
7556-MercaptopurineFDA approvedDs|PPAT34462Uracil mustardFDA approvedA7|AlkAg
7556-MercaptopurineFDA approvedDs|PPAT38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
7556-MercaptopurineFDA approvedDs|PPAT45388DacarbazineFDA approvedA7|AlkAg
7556-MercaptopurineFDA approvedDs|PPAT49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
7556-MercaptopurineFDA approvedDs|PPAT63878Cytarabine hydrochlorideFDA approvedDs
7556-MercaptopurineFDA approvedDs|PPAT67574Vincristine sulfateFDA approvedTUBB|Tu-frag
7556-MercaptopurineFDA approvedDs|PPAT71423Megestrol acetateFDA approvedHo|PGR
7556-MercaptopurineFDA approvedDs|PPAT79037LomustineFDA approvedA6|AlkAg
7556-MercaptopurineFDA approvedDs|PPAT82151Daunorubicin hydrochlorideFDA approvedTOP2
7556-MercaptopurineFDA approvedDs|PPAT102816AzacitidineFDA approvedDNMT
7556-MercaptopurineFDA approvedDs|PPAT105014CladribineFDA approvedDs|ADA
7556-MercaptopurineFDA approvedDs|PPAT118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
7556-MercaptopurineFDA approvedDs|PPAT122758TretinoinFDA approvedHo|RXR|Differentiator
7556-MercaptopurineFDA approvedDs|PPAT122819TeniposideFDA approvedTOP2
7556-MercaptopurineFDA approvedDs|PPAT123127Doxorubicin hydrochlorideFDA approvedTOP2
7556-MercaptopurineFDA approvedDs|PPAT125066BleomycinFDA approvedDb
7556-MercaptopurineFDA approvedDs|PPAT125973PaclitaxelFDA approvedTUBB|Tu-stab
7556-MercaptopurineFDA approvedDs|PPAT138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
7556-MercaptopurineFDA approvedDs|PPAT141540EtoposideFDA approvedTOP2
7556-MercaptopurineFDA approvedDs|PPAT169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
7556-MercaptopurineFDA approvedDs|PPAT180973Tamoxifen citrateFDA approvedHo|SERM
7556-MercaptopurineFDA approvedDs|PPAT241240CarboplatinFDA approvedA7|AlkAg
7556-MercaptopurineFDA approvedDs|PPAT246131ValrubicinFDA approvedTOP2
7556-MercaptopurineFDA approvedDs|PPAT279836MitoxantroneFDA approvedTOP2
7556-MercaptopurineFDA approvedDs|PPAT362856TemozolomideFDA approvedA7|AlkAg
7556-MercaptopurineFDA approvedDs|PPAT608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
7556-MercaptopurineFDA approvedDs|PPAT628503DocetaxelFDA approvedTUBB|Tu-stab
7556-MercaptopurineFDA approvedDs|PPAT673596SN 38Clinical trialTOP1
7556-MercaptopurineFDA approvedDs|PPAT698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
7556-MercaptopurineFDA approvedDs|PPAT701852VorinostatFDA approvedHDAC
7556-MercaptopurineFDA approvedDs|PPAT713563ExemestaneFDA approvedHo|CYP19A1
7556-MercaptopurineFDA approvedDs|PPAT715055GefitinibFDA approvedPK:YK,EGFR
7556-MercaptopurineFDA approvedDs|PPAT719276FulvestrantFDA approvedAM|Ho|ESR|SERM
7556-MercaptopurineFDA approvedDs|PPAT719344AnastrozoleFDA approvedHo|CYP19A1
7556-MercaptopurineFDA approvedDs|PPAT719345LetrozoleFDA approvedHo|CYP19A1
7556-MercaptopurineFDA approvedDs|PPAT719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
7556-MercaptopurineFDA approvedDs|PPAT721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
7556-MercaptopurineFDA approvedDs|PPAT732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
7556-MercaptopurineFDA approvedDs|PPAT733504EverolimusFDA approvedPK:STK,MTOR
7556-MercaptopurineFDA approvedDs|PPAT737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
7556-MercaptopurineFDA approvedDs|PPAT743414ImatinibFDA approvedBCR-ABL|PK:YK
7556-MercaptopurineFDA approvedDs|PPAT745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
7556-MercaptopurineFDA approvedDs|PPAT747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
7556-MercaptopurineFDA approvedDs|PPAT747972LenalidomideFDA approvedFT|Immunomodulatory
7556-MercaptopurineFDA approvedDs|PPAT747974RaloxifeneFDA approvedHo|SERM
7556-MercaptopurineFDA approvedDs|PPAT749226AbirateroneFDA approvedHo|CYP17A1
7556-MercaptopurineFDA approvedDs|PPAT750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
7556-MercaptopurineFDA approvedDs|PPAT753082VemurafenibFDA approvedPK:YK,BRAF
7556-MercaptopurineFDA approvedDs|PPAT754143RomidepsinFDA approvedHDAC
7556-MercaptopurineFDA approvedDs|PPAT754230PralatrexateFDA approvedDf|CTNNB1|DHFR
7556-MercaptopurineFDA approvedDs|PPAT755986VismodegibFDA approvedSMO|PK:YK
7556-MercaptopurineFDA approvedDs|PPAT756645CrizotinibFDA approvedPK:YK,MET,ALK
7556-MercaptopurineFDA approvedDs|PPAT757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
7556-MercaptopurineFDA approvedDs|PPAT760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
7556-MercaptopurineFDA approvedDs|PPAT761432CabazitaxelFDA approvedTUBB|Tu-stab
7556-MercaptopurineFDA approvedDs|PPAT763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg740MethotrexateFDA approvedDf|DHFR
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg7556-MercaptopurineFDA approvedDs|PPAT
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg6396ThiotepaFDA approvedA7|AlkAg
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg8806MelphalanFDA approvedA7|AlkAg
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg9706Triethylenemelamine-A7|AlkAg
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg24559MithramycinFDA approvedDb|Rs
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg27640FloxuridineFDA approvedDs|TYMS
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg32065HydroxyureaFDA approvedAM|Dr
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg102816AzacitidineFDA approvedDNMT
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg105014CladribineFDA approvedDs|ADA
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg125066BleomycinFDA approvedDb
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg125973PaclitaxelFDA approvedTUBB|Tu-stab
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg226080RapamycinFDA approvedPK:STK,MTOR
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg241240CarboplatinFDA approvedA7|AlkAg
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg246131ValrubicinFDA approvedTOP2
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg362856TemozolomideFDA approvedA7|AlkAg
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg606869ClofarabineFDA approvedDs
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg613327Gemcitabine HCLFDA approvedDs
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg628503DocetaxelFDA approvedTUBB|Tu-stab
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg673596SN 38Clinical trialTOP1
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg686673NelarabineFDA approvedDs
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg701852VorinostatFDA approvedHDAC
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg712807CapecitabineFDA approvedDs|TYMS
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg719276FulvestrantFDA approvedAM|Ho|ESR|SERM
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg719344AnastrozoleFDA approvedHo|CYP19A1
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg733504EverolimusFDA approvedPK:STK,MTOR
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg743414ImatinibFDA approvedBCR-ABL|PK:YK
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg747599NilotinibFDA approvedBCR-ABL|PK:YK
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg754143RomidepsinFDA approvedHDAC
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg754230PralatrexateFDA approvedDf|CTNNB1|DHFR
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
1390AllopurinolFDA approvedAM|XDH740MethotrexateFDA approvedDf|DHFR
1390AllopurinolFDA approvedAM|XDH750BusulfanFDA approvedA7|AlkAg
1390AllopurinolFDA approvedAM|XDH752ThioguanineFDA approvedDs|IMPDH2|IMPDH
1390AllopurinolFDA approvedAM|XDH7556-MercaptopurineFDA approvedDs|PPAT
1390AllopurinolFDA approvedAM|XDH762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
1390AllopurinolFDA approvedAM|XDH3053DactinomycinFDA approvedDb|RNA polymerase I
1390AllopurinolFDA approvedAM|XDH3088ChlorambucilFDA approvedA7|AlkAg
1390AllopurinolFDA approvedAM|XDH6396ThiotepaFDA approvedA7|AlkAg
1390AllopurinolFDA approvedAM|XDH8806MelphalanFDA approvedA7|AlkAg
1390AllopurinolFDA approvedAM|XDH9706Triethylenemelamine-A7|AlkAg
1390AllopurinolFDA approvedAM|XDH13875HexamethylmelamineFDA approvedDb|AlkAg
1390AllopurinolFDA approvedAM|XDH18509Aminolevulinic Acid HydrochlorideFDA approvedAM
1390AllopurinolFDA approvedAM|XDH19893FluorouracilFDA approvedDs|Rs|TYMS
1390AllopurinolFDA approvedAM|XDH24559MithramycinFDA approvedDb|Rs
1390AllopurinolFDA approvedAM|XDH25154PipobromanFDA approvedA7|AlkAg
1390AllopurinolFDA approvedAM|XDH27640FloxuridineFDA approvedDs|TYMS
1390AllopurinolFDA approvedAM|XDH32065HydroxyureaFDA approvedAM|Dr
1390AllopurinolFDA approvedAM|XDH34462Uracil mustardFDA approvedA7|AlkAg
1390AllopurinolFDA approvedAM|XDH38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
1390AllopurinolFDA approvedAM|XDH45388DacarbazineFDA approvedA7|AlkAg
1390AllopurinolFDA approvedAM|XDH49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
1390AllopurinolFDA approvedAM|XDH63878Cytarabine hydrochlorideFDA approvedDs
1390AllopurinolFDA approvedAM|XDH67574Vincristine sulfateFDA approvedTUBB|Tu-frag
1390AllopurinolFDA approvedAM|XDH71423Megestrol acetateFDA approvedHo|PGR
1390AllopurinolFDA approvedAM|XDH79037LomustineFDA approvedA6|AlkAg
1390AllopurinolFDA approvedAM|XDH82151Daunorubicin hydrochlorideFDA approvedTOP2
1390AllopurinolFDA approvedAM|XDH102816AzacitidineFDA approvedDNMT
1390AllopurinolFDA approvedAM|XDH105014CladribineFDA approvedDs|ADA
1390AllopurinolFDA approvedAM|XDH118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
1390AllopurinolFDA approvedAM|XDH122758TretinoinFDA approvedHo|RXR|Differentiator
1390AllopurinolFDA approvedAM|XDH122819TeniposideFDA approvedTOP2
1390AllopurinolFDA approvedAM|XDH123127Doxorubicin hydrochlorideFDA approvedTOP2
1390AllopurinolFDA approvedAM|XDH125066BleomycinFDA approvedDb
1390AllopurinolFDA approvedAM|XDH125973PaclitaxelFDA approvedTUBB|Tu-stab
1390AllopurinolFDA approvedAM|XDH138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
1390AllopurinolFDA approvedAM|XDH141540EtoposideFDA approvedTOP2
1390AllopurinolFDA approvedAM|XDH169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
1390AllopurinolFDA approvedAM|XDH180973Tamoxifen citrateFDA approvedHo|SERM
1390AllopurinolFDA approvedAM|XDH226080RapamycinFDA approvedPK:STK,MTOR
1390AllopurinolFDA approvedAM|XDH241240CarboplatinFDA approvedA7|AlkAg
1390AllopurinolFDA approvedAM|XDH246131ValrubicinFDA approvedTOP2
1390AllopurinolFDA approvedAM|XDH279836MitoxantroneFDA approvedTOP2
1390AllopurinolFDA approvedAM|XDH362856TemozolomideFDA approvedA7|AlkAg
1390AllopurinolFDA approvedAM|XDH606869ClofarabineFDA approvedDs
1390AllopurinolFDA approvedAM|XDH608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
1390AllopurinolFDA approvedAM|XDH613327Gemcitabine HCLFDA approvedDs
1390AllopurinolFDA approvedAM|XDH628503DocetaxelFDA approvedTUBB|Tu-stab
1390AllopurinolFDA approvedAM|XDH673596SN 38Clinical trialTOP1
1390AllopurinolFDA approvedAM|XDH686673NelarabineFDA approvedDs
1390AllopurinolFDA approvedAM|XDH698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
1390AllopurinolFDA approvedAM|XDH701852VorinostatFDA approvedHDAC
1390AllopurinolFDA approvedAM|XDH712807CapecitabineFDA approvedDs|TYMS
1390AllopurinolFDA approvedAM|XDH713563ExemestaneFDA approvedHo|CYP19A1
1390AllopurinolFDA approvedAM|XDH715055GefitinibFDA approvedPK:YK,EGFR
1390AllopurinolFDA approvedAM|XDH719276FulvestrantFDA approvedAM|Ho|ESR|SERM
1390AllopurinolFDA approvedAM|XDH719344AnastrozoleFDA approvedHo|CYP19A1
1390AllopurinolFDA approvedAM|XDH719345LetrozoleFDA approvedHo|CYP19A1
1390AllopurinolFDA approvedAM|XDH719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
1390AllopurinolFDA approvedAM|XDH721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
1390AllopurinolFDA approvedAM|XDH732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
1390AllopurinolFDA approvedAM|XDH733504EverolimusFDA approvedPK:STK,MTOR
1390AllopurinolFDA approvedAM|XDH737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
1390AllopurinolFDA approvedAM|XDH743414ImatinibFDA approvedBCR-ABL|PK:YK
1390AllopurinolFDA approvedAM|XDH745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
1390AllopurinolFDA approvedAM|XDH747599NilotinibFDA approvedBCR-ABL|PK:YK
1390AllopurinolFDA approvedAM|XDH747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
1390AllopurinolFDA approvedAM|XDH747972LenalidomideFDA approvedFT|Immunomodulatory
1390AllopurinolFDA approvedAM|XDH747974RaloxifeneFDA approvedHo|SERM
1390AllopurinolFDA approvedAM|XDH749226AbirateroneFDA approvedHo|CYP17A1
1390AllopurinolFDA approvedAM|XDH750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
1390AllopurinolFDA approvedAM|XDH753082VemurafenibFDA approvedPK:YK,BRAF
1390AllopurinolFDA approvedAM|XDH754143RomidepsinFDA approvedHDAC
1390AllopurinolFDA approvedAM|XDH754230PralatrexateFDA approvedDf|CTNNB1|DHFR
1390AllopurinolFDA approvedAM|XDH755986VismodegibFDA approvedSMO|PK:YK
1390AllopurinolFDA approvedAM|XDH756645CrizotinibFDA approvedPK:YK,MET,ALK
1390AllopurinolFDA approvedAM|XDH757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
1390AllopurinolFDA approvedAM|XDH760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
1390AllopurinolFDA approvedAM|XDH761432CabazitaxelFDA approvedTUBB|Tu-stab
1390AllopurinolFDA approvedAM|XDH763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
3053DactinomycinFDA approvedDb|RNA polymerase I752ThioguanineFDA approvedDs|IMPDH2|IMPDH
3053DactinomycinFDA approvedDb|RNA polymerase I3088ChlorambucilFDA approvedA7|AlkAg
3053DactinomycinFDA approvedDb|RNA polymerase I8806MelphalanFDA approvedA7|AlkAg
3053DactinomycinFDA approvedDb|RNA polymerase I13875HexamethylmelamineFDA approvedDb|AlkAg
3053DactinomycinFDA approvedDb|RNA polymerase I19893FluorouracilFDA approvedDs|Rs|TYMS
3053DactinomycinFDA approvedDb|RNA polymerase I34462Uracil mustardFDA approvedA7|AlkAg
3053DactinomycinFDA approvedDb|RNA polymerase I45388DacarbazineFDA approvedA7|AlkAg
3053DactinomycinFDA approvedDb|RNA polymerase I71423Megestrol acetateFDA approvedHo|PGR
3053DactinomycinFDA approvedDb|RNA polymerase I79037LomustineFDA approvedA6|AlkAg
3053DactinomycinFDA approvedDb|RNA polymerase I82151Daunorubicin hydrochlorideFDA approvedTOP2
3053DactinomycinFDA approvedDb|RNA polymerase I122819TeniposideFDA approvedTOP2
3053DactinomycinFDA approvedDb|RNA polymerase I141540EtoposideFDA approvedTOP2
3053DactinomycinFDA approvedDb|RNA polymerase I169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
3053DactinomycinFDA approvedDb|RNA polymerase I279836MitoxantroneFDA approvedTOP2
3053DactinomycinFDA approvedDb|RNA polymerase I608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
3053DactinomycinFDA approvedDb|RNA polymerase I698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
3053DactinomycinFDA approvedDb|RNA polymerase I713563ExemestaneFDA approvedHo|CYP19A1
3053DactinomycinFDA approvedDb|RNA polymerase I715055GefitinibFDA approvedPK:YK,EGFR
3053DactinomycinFDA approvedDb|RNA polymerase I719345LetrozoleFDA approvedHo|CYP19A1
3053DactinomycinFDA approvedDb|RNA polymerase I737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
3053DactinomycinFDA approvedDb|RNA polymerase I747972LenalidomideFDA approvedFT|Immunomodulatory
3053DactinomycinFDA approvedDb|RNA polymerase I747974RaloxifeneFDA approvedHo|SERM
3053DactinomycinFDA approvedDb|RNA polymerase I749226AbirateroneFDA approvedHo|CYP17A1
3053DactinomycinFDA approvedDb|RNA polymerase I753082VemurafenibFDA approvedPK:YK,BRAF
3053DactinomycinFDA approvedDb|RNA polymerase I755986VismodegibFDA approvedSMO|PK:YK
3053DactinomycinFDA approvedDb|RNA polymerase I756645CrizotinibFDA approvedPK:YK,MET,ALK
3053DactinomycinFDA approvedDb|RNA polymerase I757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
3053DactinomycinFDA approvedDb|RNA polymerase I760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
3053DactinomycinFDA approvedDb|RNA polymerase I761432CabazitaxelFDA approvedTUBB|Tu-stab
3053DactinomycinFDA approvedDb|RNA polymerase I763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
3088ChlorambucilFDA approvedA7|AlkAg8806MelphalanFDA approvedA7|AlkAg
3088ChlorambucilFDA approvedA7|AlkAg9706Triethylenemelamine-A7|AlkAg
3088ChlorambucilFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
3088ChlorambucilFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
3088ChlorambucilFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
3088ChlorambucilFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
3088ChlorambucilFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
3088ChlorambucilFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
3088ChlorambucilFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
3088ChlorambucilFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
3088ChlorambucilFDA approvedA7|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
3088ChlorambucilFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
3088ChlorambucilFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
3088ChlorambucilFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
3088ChlorambucilFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
3088ChlorambucilFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
3088ChlorambucilFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
3088ChlorambucilFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
3088ChlorambucilFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
3088ChlorambucilFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
3088ChlorambucilFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
3088ChlorambucilFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
3088ChlorambucilFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
3088ChlorambucilFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
3088ChlorambucilFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
3088ChlorambucilFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
3088ChlorambucilFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
3088ChlorambucilFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
3088ChlorambucilFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
6396ThiotepaFDA approvedA7|AlkAg740MethotrexateFDA approvedDf|DHFR
6396ThiotepaFDA approvedA7|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
6396ThiotepaFDA approvedA7|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
6396ThiotepaFDA approvedA7|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
6396ThiotepaFDA approvedA7|AlkAg8806MelphalanFDA approvedA7|AlkAg
6396ThiotepaFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
6396ThiotepaFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
6396ThiotepaFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
6396ThiotepaFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
6396ThiotepaFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
6396ThiotepaFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
6396ThiotepaFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
6396ThiotepaFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
6396ThiotepaFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
6396ThiotepaFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
6396ThiotepaFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
6396ThiotepaFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
6396ThiotepaFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
6396ThiotepaFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
6396ThiotepaFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
6396ThiotepaFDA approvedA7|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
6396ThiotepaFDA approvedA7|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
6396ThiotepaFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
6396ThiotepaFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
6396ThiotepaFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
6396ThiotepaFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
6396ThiotepaFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
6396ThiotepaFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
6396ThiotepaFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
6396ThiotepaFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
6396ThiotepaFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
6396ThiotepaFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
6396ThiotepaFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
8806MelphalanFDA approvedA7|AlkAg9706Triethylenemelamine-A7|AlkAg
8806MelphalanFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
8806MelphalanFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
8806MelphalanFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
8806MelphalanFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
8806MelphalanFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
8806MelphalanFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
8806MelphalanFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
8806MelphalanFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
8806MelphalanFDA approvedA7|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
8806MelphalanFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
8806MelphalanFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
8806MelphalanFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
8806MelphalanFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
8806MelphalanFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
8806MelphalanFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
8806MelphalanFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
8806MelphalanFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
8806MelphalanFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
8806MelphalanFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
8806MelphalanFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
8806MelphalanFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
8806MelphalanFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
8806MelphalanFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
8806MelphalanFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
8806MelphalanFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
8806MelphalanFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
8806MelphalanFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
9706Triethylenemelamine-A7|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
9706Triethylenemelamine-A7|AlkAg6396ThiotepaFDA approvedA7|AlkAg
9706Triethylenemelamine-A7|AlkAg27640FloxuridineFDA approvedDs|TYMS
9706Triethylenemelamine-A7|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
9706Triethylenemelamine-A7|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
9706Triethylenemelamine-A7|AlkAg102816AzacitidineFDA approvedDNMT
9706Triethylenemelamine-A7|AlkAg105014CladribineFDA approvedDs|ADA
9706Triethylenemelamine-A7|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
9706Triethylenemelamine-A7|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
9706Triethylenemelamine-A7|AlkAg125973PaclitaxelFDA approvedTUBB|Tu-stab
9706Triethylenemelamine-A7|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
9706Triethylenemelamine-A7|AlkAg226080RapamycinFDA approvedPK:STK,MTOR
9706Triethylenemelamine-A7|AlkAg241240CarboplatinFDA approvedA7|AlkAg
9706Triethylenemelamine-A7|AlkAg246131ValrubicinFDA approvedTOP2
9706Triethylenemelamine-A7|AlkAg362856TemozolomideFDA approvedA7|AlkAg
9706Triethylenemelamine-A7|AlkAg606869ClofarabineFDA approvedDs
9706Triethylenemelamine-A7|AlkAg613327Gemcitabine HCLFDA approvedDs
9706Triethylenemelamine-A7|AlkAg628503DocetaxelFDA approvedTUBB|Tu-stab
9706Triethylenemelamine-A7|AlkAg673596SN 38Clinical trialTOP1
9706Triethylenemelamine-A7|AlkAg686673NelarabineFDA approvedDs
9706Triethylenemelamine-A7|AlkAg701852VorinostatFDA approvedHDAC
9706Triethylenemelamine-A7|AlkAg712807CapecitabineFDA approvedDs|TYMS
9706Triethylenemelamine-A7|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
9706Triethylenemelamine-A7|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
9706Triethylenemelamine-A7|AlkAg721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
9706Triethylenemelamine-A7|AlkAg732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
9706Triethylenemelamine-A7|AlkAg733504EverolimusFDA approvedPK:STK,MTOR
9706Triethylenemelamine-A7|AlkAg743414ImatinibFDA approvedBCR-ABL|PK:YK
9706Triethylenemelamine-A7|AlkAg745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
9706Triethylenemelamine-A7|AlkAg747599NilotinibFDA approvedBCR-ABL|PK:YK
9706Triethylenemelamine-A7|AlkAg750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
9706Triethylenemelamine-A7|AlkAg754143RomidepsinFDA approvedHDAC
13875HexamethylmelamineFDA approvedDb|AlkAg9706Triethylenemelamine-A7|AlkAg
13875HexamethylmelamineFDA approvedDb|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
13875HexamethylmelamineFDA approvedDb|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
13875HexamethylmelamineFDA approvedDb|AlkAg45388DacarbazineFDA approvedA7|AlkAg
13875HexamethylmelamineFDA approvedDb|AlkAg71423Megestrol acetateFDA approvedHo|PGR
13875HexamethylmelamineFDA approvedDb|AlkAg79037LomustineFDA approvedA6|AlkAg
13875HexamethylmelamineFDA approvedDb|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
13875HexamethylmelamineFDA approvedDb|AlkAg122819TeniposideFDA approvedTOP2
13875HexamethylmelamineFDA approvedDb|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
13875HexamethylmelamineFDA approvedDb|AlkAg141540EtoposideFDA approvedTOP2
13875HexamethylmelamineFDA approvedDb|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
13875HexamethylmelamineFDA approvedDb|AlkAg279836MitoxantroneFDA approvedTOP2
13875HexamethylmelamineFDA approvedDb|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
13875HexamethylmelamineFDA approvedDb|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
13875HexamethylmelamineFDA approvedDb|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
13875HexamethylmelamineFDA approvedDb|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
13875HexamethylmelamineFDA approvedDb|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
13875HexamethylmelamineFDA approvedDb|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
13875HexamethylmelamineFDA approvedDb|AlkAg747974RaloxifeneFDA approvedHo|SERM
13875HexamethylmelamineFDA approvedDb|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
13875HexamethylmelamineFDA approvedDb|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
13875HexamethylmelamineFDA approvedDb|AlkAg755986VismodegibFDA approvedSMO|PK:YK
13875HexamethylmelamineFDA approvedDb|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
13875HexamethylmelamineFDA approvedDb|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
13875HexamethylmelamineFDA approvedDb|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
13875HexamethylmelamineFDA approvedDb|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
13875HexamethylmelamineFDA approvedDb|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
14229QuinacrineClinical trialDb|AP740MethotrexateFDA approvedDf|DHFR
14229QuinacrineClinical trialDb|AP750BusulfanFDA approvedA7|AlkAg
14229QuinacrineClinical trialDb|AP752ThioguanineFDA approvedDs|IMPDH2|IMPDH
14229QuinacrineClinical trialDb|AP7556-MercaptopurineFDA approvedDs|PPAT
14229QuinacrineClinical trialDb|AP762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
14229QuinacrineClinical trialDb|AP1390AllopurinolFDA approvedAM|XDH
14229QuinacrineClinical trialDb|AP3053DactinomycinFDA approvedDb|RNA polymerase I
14229QuinacrineClinical trialDb|AP3088ChlorambucilFDA approvedA7|AlkAg
14229QuinacrineClinical trialDb|AP6396ThiotepaFDA approvedA7|AlkAg
14229QuinacrineClinical trialDb|AP8806MelphalanFDA approvedA7|AlkAg
14229QuinacrineClinical trialDb|AP9706Triethylenemelamine-A7|AlkAg
14229QuinacrineClinical trialDb|AP13875HexamethylmelamineFDA approvedDb|AlkAg
14229QuinacrineClinical trialDb|AP18509Aminolevulinic Acid HydrochlorideFDA approvedAM
14229QuinacrineClinical trialDb|AP19893FluorouracilFDA approvedDs|Rs|TYMS
14229QuinacrineClinical trialDb|AP24559MithramycinFDA approvedDb|Rs
14229QuinacrineClinical trialDb|AP27640FloxuridineFDA approvedDs|TYMS
14229QuinacrineClinical trialDb|AP32065HydroxyureaFDA approvedAM|Dr
14229QuinacrineClinical trialDb|AP34462Uracil mustardFDA approvedA7|AlkAg
14229QuinacrineClinical trialDb|AP38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
14229QuinacrineClinical trialDb|AP45388DacarbazineFDA approvedA7|AlkAg
14229QuinacrineClinical trialDb|AP49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
14229QuinacrineClinical trialDb|AP63878Cytarabine hydrochlorideFDA approvedDs
14229QuinacrineClinical trialDb|AP67574Vincristine sulfateFDA approvedTUBB|Tu-frag
14229QuinacrineClinical trialDb|AP71423Megestrol acetateFDA approvedHo|PGR
14229QuinacrineClinical trialDb|AP79037LomustineFDA approvedA6|AlkAg
14229QuinacrineClinical trialDb|AP82151Daunorubicin hydrochlorideFDA approvedTOP2
14229QuinacrineClinical trialDb|AP102816AzacitidineFDA approvedDNMT
14229QuinacrineClinical trialDb|AP105014CladribineFDA approvedDs|ADA
14229QuinacrineClinical trialDb|AP118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
14229QuinacrineClinical trialDb|AP122758TretinoinFDA approvedHo|RXR|Differentiator
14229QuinacrineClinical trialDb|AP122819TeniposideFDA approvedTOP2
14229QuinacrineClinical trialDb|AP123127Doxorubicin hydrochlorideFDA approvedTOP2
14229QuinacrineClinical trialDb|AP125066BleomycinFDA approvedDb
14229QuinacrineClinical trialDb|AP125973PaclitaxelFDA approvedTUBB|Tu-stab
14229QuinacrineClinical trialDb|AP138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
14229QuinacrineClinical trialDb|AP141540EtoposideFDA approvedTOP2
14229QuinacrineClinical trialDb|AP169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
14229QuinacrineClinical trialDb|AP180973Tamoxifen citrateFDA approvedHo|SERM
14229QuinacrineClinical trialDb|AP226080RapamycinFDA approvedPK:STK,MTOR
14229QuinacrineClinical trialDb|AP241240CarboplatinFDA approvedA7|AlkAg
14229QuinacrineClinical trialDb|AP246131ValrubicinFDA approvedTOP2
14229QuinacrineClinical trialDb|AP279836MitoxantroneFDA approvedTOP2
14229QuinacrineClinical trialDb|AP362856TemozolomideFDA approvedA7|AlkAg
14229QuinacrineClinical trialDb|AP606869ClofarabineFDA approvedDs
14229QuinacrineClinical trialDb|AP608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
14229QuinacrineClinical trialDb|AP613327Gemcitabine HCLFDA approvedDs
14229QuinacrineClinical trialDb|AP628503DocetaxelFDA approvedTUBB|Tu-stab
14229QuinacrineClinical trialDb|AP673596SN 38Clinical trialTOP1
14229QuinacrineClinical trialDb|AP686673NelarabineFDA approvedDs
14229QuinacrineClinical trialDb|AP698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
14229QuinacrineClinical trialDb|AP701852VorinostatFDA approvedHDAC
14229QuinacrineClinical trialDb|AP712807CapecitabineFDA approvedDs|TYMS
14229QuinacrineClinical trialDb|AP713563ExemestaneFDA approvedHo|CYP19A1
14229QuinacrineClinical trialDb|AP715055GefitinibFDA approvedPK:YK,EGFR
14229QuinacrineClinical trialDb|AP719276FulvestrantFDA approvedAM|Ho|ESR|SERM
14229QuinacrineClinical trialDb|AP719344AnastrozoleFDA approvedHo|CYP19A1
14229QuinacrineClinical trialDb|AP719345LetrozoleFDA approvedHo|CYP19A1
14229QuinacrineClinical trialDb|AP719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
14229QuinacrineClinical trialDb|AP721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
14229QuinacrineClinical trialDb|AP732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
14229QuinacrineClinical trialDb|AP733504EverolimusFDA approvedPK:STK,MTOR
14229QuinacrineClinical trialDb|AP737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
14229QuinacrineClinical trialDb|AP743414ImatinibFDA approvedBCR-ABL|PK:YK
14229QuinacrineClinical trialDb|AP745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
14229QuinacrineClinical trialDb|AP747599NilotinibFDA approvedBCR-ABL|PK:YK
14229QuinacrineClinical trialDb|AP747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
14229QuinacrineClinical trialDb|AP747972LenalidomideFDA approvedFT|Immunomodulatory
14229QuinacrineClinical trialDb|AP747974RaloxifeneFDA approvedHo|SERM
14229QuinacrineClinical trialDb|AP749226AbirateroneFDA approvedHo|CYP17A1
14229QuinacrineClinical trialDb|AP750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
14229QuinacrineClinical trialDb|AP753082VemurafenibFDA approvedPK:YK,BRAF
14229QuinacrineClinical trialDb|AP754143RomidepsinFDA approvedHDAC
14229QuinacrineClinical trialDb|AP754230PralatrexateFDA approvedDf|CTNNB1|DHFR
14229QuinacrineClinical trialDb|AP755986VismodegibFDA approvedSMO|PK:YK
14229QuinacrineClinical trialDb|AP756645CrizotinibFDA approvedPK:YK,MET,ALK
14229QuinacrineClinical trialDb|AP757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
14229QuinacrineClinical trialDb|AP760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
14229QuinacrineClinical trialDb|AP761432CabazitaxelFDA approvedTUBB|Tu-stab
14229QuinacrineClinical trialDb|AP763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
18509Aminolevulinic Acid HydrochlorideFDA approvedAM740MethotrexateFDA approvedDf|DHFR
18509Aminolevulinic Acid HydrochlorideFDA approvedAM752ThioguanineFDA approvedDs|IMPDH2|IMPDH
18509Aminolevulinic Acid HydrochlorideFDA approvedAM7556-MercaptopurineFDA approvedDs|PPAT
18509Aminolevulinic Acid HydrochlorideFDA approvedAM762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
18509Aminolevulinic Acid HydrochlorideFDA approvedAM3053DactinomycinFDA approvedDb|RNA polymerase I
18509Aminolevulinic Acid HydrochlorideFDA approvedAM3088ChlorambucilFDA approvedA7|AlkAg
18509Aminolevulinic Acid HydrochlorideFDA approvedAM6396ThiotepaFDA approvedA7|AlkAg
18509Aminolevulinic Acid HydrochlorideFDA approvedAM8806MelphalanFDA approvedA7|AlkAg
18509Aminolevulinic Acid HydrochlorideFDA approvedAM9706Triethylenemelamine-A7|AlkAg
18509Aminolevulinic Acid HydrochlorideFDA approvedAM13875HexamethylmelamineFDA approvedDb|AlkAg
18509Aminolevulinic Acid HydrochlorideFDA approvedAM19893FluorouracilFDA approvedDs|Rs|TYMS
18509Aminolevulinic Acid HydrochlorideFDA approvedAM24559MithramycinFDA approvedDb|Rs
18509Aminolevulinic Acid HydrochlorideFDA approvedAM27640FloxuridineFDA approvedDs|TYMS
18509Aminolevulinic Acid HydrochlorideFDA approvedAM32065HydroxyureaFDA approvedAM|Dr
18509Aminolevulinic Acid HydrochlorideFDA approvedAM34462Uracil mustardFDA approvedA7|AlkAg
18509Aminolevulinic Acid HydrochlorideFDA approvedAM38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
18509Aminolevulinic Acid HydrochlorideFDA approvedAM45388DacarbazineFDA approvedA7|AlkAg
18509Aminolevulinic Acid HydrochlorideFDA approvedAM49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
18509Aminolevulinic Acid HydrochlorideFDA approvedAM63878Cytarabine hydrochlorideFDA approvedDs
18509Aminolevulinic Acid HydrochlorideFDA approvedAM67574Vincristine sulfateFDA approvedTUBB|Tu-frag
18509Aminolevulinic Acid HydrochlorideFDA approvedAM71423Megestrol acetateFDA approvedHo|PGR
18509Aminolevulinic Acid HydrochlorideFDA approvedAM79037LomustineFDA approvedA6|AlkAg
18509Aminolevulinic Acid HydrochlorideFDA approvedAM82151Daunorubicin hydrochlorideFDA approvedTOP2
18509Aminolevulinic Acid HydrochlorideFDA approvedAM102816AzacitidineFDA approvedDNMT
18509Aminolevulinic Acid HydrochlorideFDA approvedAM105014CladribineFDA approvedDs|ADA
18509Aminolevulinic Acid HydrochlorideFDA approvedAM118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
18509Aminolevulinic Acid HydrochlorideFDA approvedAM122758TretinoinFDA approvedHo|RXR|Differentiator
18509Aminolevulinic Acid HydrochlorideFDA approvedAM122819TeniposideFDA approvedTOP2
18509Aminolevulinic Acid HydrochlorideFDA approvedAM123127Doxorubicin hydrochlorideFDA approvedTOP2
18509Aminolevulinic Acid HydrochlorideFDA approvedAM125066BleomycinFDA approvedDb
18509Aminolevulinic Acid HydrochlorideFDA approvedAM125973PaclitaxelFDA approvedTUBB|Tu-stab
18509Aminolevulinic Acid HydrochlorideFDA approvedAM138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
18509Aminolevulinic Acid HydrochlorideFDA approvedAM141540EtoposideFDA approvedTOP2
18509Aminolevulinic Acid HydrochlorideFDA approvedAM169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
18509Aminolevulinic Acid HydrochlorideFDA approvedAM180973Tamoxifen citrateFDA approvedHo|SERM
18509Aminolevulinic Acid HydrochlorideFDA approvedAM226080RapamycinFDA approvedPK:STK,MTOR
18509Aminolevulinic Acid HydrochlorideFDA approvedAM241240CarboplatinFDA approvedA7|AlkAg
18509Aminolevulinic Acid HydrochlorideFDA approvedAM246131ValrubicinFDA approvedTOP2
18509Aminolevulinic Acid HydrochlorideFDA approvedAM279836MitoxantroneFDA approvedTOP2
18509Aminolevulinic Acid HydrochlorideFDA approvedAM362856TemozolomideFDA approvedA7|AlkAg
18509Aminolevulinic Acid HydrochlorideFDA approvedAM606869ClofarabineFDA approvedDs
18509Aminolevulinic Acid HydrochlorideFDA approvedAM608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
18509Aminolevulinic Acid HydrochlorideFDA approvedAM613327Gemcitabine HCLFDA approvedDs
18509Aminolevulinic Acid HydrochlorideFDA approvedAM628503DocetaxelFDA approvedTUBB|Tu-stab
18509Aminolevulinic Acid HydrochlorideFDA approvedAM673596SN 38Clinical trialTOP1
18509Aminolevulinic Acid HydrochlorideFDA approvedAM686673NelarabineFDA approvedDs
18509Aminolevulinic Acid HydrochlorideFDA approvedAM698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
18509Aminolevulinic Acid HydrochlorideFDA approvedAM701852VorinostatFDA approvedHDAC
18509Aminolevulinic Acid HydrochlorideFDA approvedAM712807CapecitabineFDA approvedDs|TYMS
18509Aminolevulinic Acid HydrochlorideFDA approvedAM713563ExemestaneFDA approvedHo|CYP19A1
18509Aminolevulinic Acid HydrochlorideFDA approvedAM715055GefitinibFDA approvedPK:YK,EGFR
18509Aminolevulinic Acid HydrochlorideFDA approvedAM719276FulvestrantFDA approvedAM|Ho|ESR|SERM
18509Aminolevulinic Acid HydrochlorideFDA approvedAM719344AnastrozoleFDA approvedHo|CYP19A1
18509Aminolevulinic Acid HydrochlorideFDA approvedAM719345LetrozoleFDA approvedHo|CYP19A1
18509Aminolevulinic Acid HydrochlorideFDA approvedAM719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
18509Aminolevulinic Acid HydrochlorideFDA approvedAM732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
18509Aminolevulinic Acid HydrochlorideFDA approvedAM733504EverolimusFDA approvedPK:STK,MTOR
18509Aminolevulinic Acid HydrochlorideFDA approvedAM737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
18509Aminolevulinic Acid HydrochlorideFDA approvedAM743414ImatinibFDA approvedBCR-ABL|PK:YK
18509Aminolevulinic Acid HydrochlorideFDA approvedAM745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
18509Aminolevulinic Acid HydrochlorideFDA approvedAM747599NilotinibFDA approvedBCR-ABL|PK:YK
18509Aminolevulinic Acid HydrochlorideFDA approvedAM747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
18509Aminolevulinic Acid HydrochlorideFDA approvedAM747972LenalidomideFDA approvedFT|Immunomodulatory
18509Aminolevulinic Acid HydrochlorideFDA approvedAM747974RaloxifeneFDA approvedHo|SERM
18509Aminolevulinic Acid HydrochlorideFDA approvedAM749226AbirateroneFDA approvedHo|CYP17A1
18509Aminolevulinic Acid HydrochlorideFDA approvedAM750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
18509Aminolevulinic Acid HydrochlorideFDA approvedAM753082VemurafenibFDA approvedPK:YK,BRAF
18509Aminolevulinic Acid HydrochlorideFDA approvedAM754143RomidepsinFDA approvedHDAC
18509Aminolevulinic Acid HydrochlorideFDA approvedAM754230PralatrexateFDA approvedDf|CTNNB1|DHFR
18509Aminolevulinic Acid HydrochlorideFDA approvedAM755986VismodegibFDA approvedSMO|PK:YK
18509Aminolevulinic Acid HydrochlorideFDA approvedAM756645CrizotinibFDA approvedPK:YK,MET,ALK
18509Aminolevulinic Acid HydrochlorideFDA approvedAM757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
18509Aminolevulinic Acid HydrochlorideFDA approvedAM760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
18509Aminolevulinic Acid HydrochlorideFDA approvedAM761432CabazitaxelFDA approvedTUBB|Tu-stab
18509Aminolevulinic Acid HydrochlorideFDA approvedAM763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
19893FluorouracilFDA approvedDs|Rs|TYMS9706Triethylenemelamine-A7|AlkAg
19893FluorouracilFDA approvedDs|Rs|TYMS34462Uracil mustardFDA approvedA7|AlkAg
19893FluorouracilFDA approvedDs|Rs|TYMS45388DacarbazineFDA approvedA7|AlkAg
19893FluorouracilFDA approvedDs|Rs|TYMS71423Megestrol acetateFDA approvedHo|PGR
19893FluorouracilFDA approvedDs|Rs|TYMS79037LomustineFDA approvedA6|AlkAg
19893FluorouracilFDA approvedDs|Rs|TYMS82151Daunorubicin hydrochlorideFDA approvedTOP2
19893FluorouracilFDA approvedDs|Rs|TYMS122819TeniposideFDA approvedTOP2
19893FluorouracilFDA approvedDs|Rs|TYMS123127Doxorubicin hydrochlorideFDA approvedTOP2
19893FluorouracilFDA approvedDs|Rs|TYMS141540EtoposideFDA approvedTOP2
19893FluorouracilFDA approvedDs|Rs|TYMS169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
19893FluorouracilFDA approvedDs|Rs|TYMS279836MitoxantroneFDA approvedTOP2
19893FluorouracilFDA approvedDs|Rs|TYMS608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
19893FluorouracilFDA approvedDs|Rs|TYMS698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
19893FluorouracilFDA approvedDs|Rs|TYMS713563ExemestaneFDA approvedHo|CYP19A1
19893FluorouracilFDA approvedDs|Rs|TYMS715055GefitinibFDA approvedPK:YK,EGFR
19893FluorouracilFDA approvedDs|Rs|TYMS737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
19893FluorouracilFDA approvedDs|Rs|TYMS747972LenalidomideFDA approvedFT|Immunomodulatory
19893FluorouracilFDA approvedDs|Rs|TYMS747974RaloxifeneFDA approvedHo|SERM
19893FluorouracilFDA approvedDs|Rs|TYMS749226AbirateroneFDA approvedHo|CYP17A1
19893FluorouracilFDA approvedDs|Rs|TYMS753082VemurafenibFDA approvedPK:YK,BRAF
19893FluorouracilFDA approvedDs|Rs|TYMS755986VismodegibFDA approvedSMO|PK:YK
19893FluorouracilFDA approvedDs|Rs|TYMS756645CrizotinibFDA approvedPK:YK,MET,ALK
19893FluorouracilFDA approvedDs|Rs|TYMS757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
19893FluorouracilFDA approvedDs|Rs|TYMS760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
19893FluorouracilFDA approvedDs|Rs|TYMS761432CabazitaxelFDA approvedTUBB|Tu-stab
19893FluorouracilFDA approvedDs|Rs|TYMS763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
24559MithramycinFDA approvedDb|Rs752ThioguanineFDA approvedDs|IMPDH2|IMPDH
24559MithramycinFDA approvedDb|Rs3053DactinomycinFDA approvedDb|RNA polymerase I
24559MithramycinFDA approvedDb|Rs3088ChlorambucilFDA approvedA7|AlkAg
24559MithramycinFDA approvedDb|Rs6396ThiotepaFDA approvedA7|AlkAg
24559MithramycinFDA approvedDb|Rs8806MelphalanFDA approvedA7|AlkAg
24559MithramycinFDA approvedDb|Rs9706Triethylenemelamine-A7|AlkAg
24559MithramycinFDA approvedDb|Rs13875HexamethylmelamineFDA approvedDb|AlkAg
24559MithramycinFDA approvedDb|Rs19893FluorouracilFDA approvedDs|Rs|TYMS
24559MithramycinFDA approvedDb|Rs27640FloxuridineFDA approvedDs|TYMS
24559MithramycinFDA approvedDb|Rs34462Uracil mustardFDA approvedA7|AlkAg
24559MithramycinFDA approvedDb|Rs45388DacarbazineFDA approvedA7|AlkAg
24559MithramycinFDA approvedDb|Rs63878Cytarabine hydrochlorideFDA approvedDs
24559MithramycinFDA approvedDb|Rs67574Vincristine sulfateFDA approvedTUBB|Tu-frag
24559MithramycinFDA approvedDb|Rs71423Megestrol acetateFDA approvedHo|PGR
24559MithramycinFDA approvedDb|Rs79037LomustineFDA approvedA6|AlkAg
24559MithramycinFDA approvedDb|Rs82151Daunorubicin hydrochlorideFDA approvedTOP2
24559MithramycinFDA approvedDb|Rs102816AzacitidineFDA approvedDNMT
24559MithramycinFDA approvedDb|Rs105014CladribineFDA approvedDs|ADA
24559MithramycinFDA approvedDb|Rs118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
24559MithramycinFDA approvedDb|Rs122758TretinoinFDA approvedHo|RXR|Differentiator
24559MithramycinFDA approvedDb|Rs122819TeniposideFDA approvedTOP2
24559MithramycinFDA approvedDb|Rs125973PaclitaxelFDA approvedTUBB|Tu-stab
24559MithramycinFDA approvedDb|Rs141540EtoposideFDA approvedTOP2
24559MithramycinFDA approvedDb|Rs169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
24559MithramycinFDA approvedDb|Rs180973Tamoxifen citrateFDA approvedHo|SERM
24559MithramycinFDA approvedDb|Rs241240CarboplatinFDA approvedA7|AlkAg
24559MithramycinFDA approvedDb|Rs279836MitoxantroneFDA approvedTOP2
24559MithramycinFDA approvedDb|Rs362856TemozolomideFDA approvedA7|AlkAg
24559MithramycinFDA approvedDb|Rs608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
24559MithramycinFDA approvedDb|Rs628503DocetaxelFDA approvedTUBB|Tu-stab
24559MithramycinFDA approvedDb|Rs673596SN 38Clinical trialTOP1
24559MithramycinFDA approvedDb|Rs698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
24559MithramycinFDA approvedDb|Rs701852VorinostatFDA approvedHDAC
24559MithramycinFDA approvedDb|Rs713563ExemestaneFDA approvedHo|CYP19A1
24559MithramycinFDA approvedDb|Rs715055GefitinibFDA approvedPK:YK,EGFR
24559MithramycinFDA approvedDb|Rs719345LetrozoleFDA approvedHo|CYP19A1
24559MithramycinFDA approvedDb|Rs719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
24559MithramycinFDA approvedDb|Rs721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
24559MithramycinFDA approvedDb|Rs732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
24559MithramycinFDA approvedDb|Rs733504EverolimusFDA approvedPK:STK,MTOR
24559MithramycinFDA approvedDb|Rs737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
24559MithramycinFDA approvedDb|Rs743414ImatinibFDA approvedBCR-ABL|PK:YK
24559MithramycinFDA approvedDb|Rs745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
24559MithramycinFDA approvedDb|Rs747972LenalidomideFDA approvedFT|Immunomodulatory
24559MithramycinFDA approvedDb|Rs747974RaloxifeneFDA approvedHo|SERM
24559MithramycinFDA approvedDb|Rs749226AbirateroneFDA approvedHo|CYP17A1
24559MithramycinFDA approvedDb|Rs750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
24559MithramycinFDA approvedDb|Rs753082VemurafenibFDA approvedPK:YK,BRAF
24559MithramycinFDA approvedDb|Rs754143RomidepsinFDA approvedHDAC
24559MithramycinFDA approvedDb|Rs755986VismodegibFDA approvedSMO|PK:YK
24559MithramycinFDA approvedDb|Rs756645CrizotinibFDA approvedPK:YK,MET,ALK
24559MithramycinFDA approvedDb|Rs757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
24559MithramycinFDA approvedDb|Rs760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
24559MithramycinFDA approvedDb|Rs761432CabazitaxelFDA approvedTUBB|Tu-stab
24559MithramycinFDA approvedDb|Rs763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
25154PipobromanFDA approvedA7|AlkAg740MethotrexateFDA approvedDf|DHFR
25154PipobromanFDA approvedA7|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
25154PipobromanFDA approvedA7|AlkAg7556-MercaptopurineFDA approvedDs|PPAT
25154PipobromanFDA approvedA7|AlkAg762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
25154PipobromanFDA approvedA7|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
25154PipobromanFDA approvedA7|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
25154PipobromanFDA approvedA7|AlkAg6396ThiotepaFDA approvedA7|AlkAg
25154PipobromanFDA approvedA7|AlkAg8806MelphalanFDA approvedA7|AlkAg
25154PipobromanFDA approvedA7|AlkAg9706Triethylenemelamine-A7|AlkAg
25154PipobromanFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
25154PipobromanFDA approvedA7|AlkAg14229QuinacrineClinical trialDb|AP
25154PipobromanFDA approvedA7|AlkAg18509Aminolevulinic Acid HydrochlorideFDA approvedAM
25154PipobromanFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
25154PipobromanFDA approvedA7|AlkAg24559MithramycinFDA approvedDb|Rs
25154PipobromanFDA approvedA7|AlkAg27640FloxuridineFDA approvedDs|TYMS
25154PipobromanFDA approvedA7|AlkAg32065HydroxyureaFDA approvedAM|Dr
25154PipobromanFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
25154PipobromanFDA approvedA7|AlkAg38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
25154PipobromanFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
25154PipobromanFDA approvedA7|AlkAg49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
25154PipobromanFDA approvedA7|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
25154PipobromanFDA approvedA7|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
25154PipobromanFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
25154PipobromanFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
25154PipobromanFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
25154PipobromanFDA approvedA7|AlkAg102816AzacitidineFDA approvedDNMT
25154PipobromanFDA approvedA7|AlkAg105014CladribineFDA approvedDs|ADA
25154PipobromanFDA approvedA7|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
25154PipobromanFDA approvedA7|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
25154PipobromanFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
25154PipobromanFDA approvedA7|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
25154PipobromanFDA approvedA7|AlkAg125066BleomycinFDA approvedDb
25154PipobromanFDA approvedA7|AlkAg125973PaclitaxelFDA approvedTUBB|Tu-stab
25154PipobromanFDA approvedA7|AlkAg138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
25154PipobromanFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
25154PipobromanFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
25154PipobromanFDA approvedA7|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
25154PipobromanFDA approvedA7|AlkAg226080RapamycinFDA approvedPK:STK,MTOR
25154PipobromanFDA approvedA7|AlkAg241240CarboplatinFDA approvedA7|AlkAg
25154PipobromanFDA approvedA7|AlkAg246131ValrubicinFDA approvedTOP2
25154PipobromanFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
25154PipobromanFDA approvedA7|AlkAg362856TemozolomideFDA approvedA7|AlkAg
25154PipobromanFDA approvedA7|AlkAg606869ClofarabineFDA approvedDs
25154PipobromanFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
25154PipobromanFDA approvedA7|AlkAg613327Gemcitabine HCLFDA approvedDs
25154PipobromanFDA approvedA7|AlkAg628503DocetaxelFDA approvedTUBB|Tu-stab
25154PipobromanFDA approvedA7|AlkAg673596SN 38Clinical trialTOP1
25154PipobromanFDA approvedA7|AlkAg686673NelarabineFDA approvedDs
25154PipobromanFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
25154PipobromanFDA approvedA7|AlkAg701852VorinostatFDA approvedHDAC
25154PipobromanFDA approvedA7|AlkAg712807CapecitabineFDA approvedDs|TYMS
25154PipobromanFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
25154PipobromanFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
25154PipobromanFDA approvedA7|AlkAg719276FulvestrantFDA approvedAM|Ho|ESR|SERM
25154PipobromanFDA approvedA7|AlkAg719344AnastrozoleFDA approvedHo|CYP19A1
25154PipobromanFDA approvedA7|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
25154PipobromanFDA approvedA7|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
25154PipobromanFDA approvedA7|AlkAg721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
25154PipobromanFDA approvedA7|AlkAg732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
25154PipobromanFDA approvedA7|AlkAg733504EverolimusFDA approvedPK:STK,MTOR
25154PipobromanFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
25154PipobromanFDA approvedA7|AlkAg743414ImatinibFDA approvedBCR-ABL|PK:YK
25154PipobromanFDA approvedA7|AlkAg745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
25154PipobromanFDA approvedA7|AlkAg747599NilotinibFDA approvedBCR-ABL|PK:YK
25154PipobromanFDA approvedA7|AlkAg747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
25154PipobromanFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
25154PipobromanFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
25154PipobromanFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
25154PipobromanFDA approvedA7|AlkAg750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
25154PipobromanFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
25154PipobromanFDA approvedA7|AlkAg754143RomidepsinFDA approvedHDAC
25154PipobromanFDA approvedA7|AlkAg754230PralatrexateFDA approvedDf|CTNNB1|DHFR
25154PipobromanFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
25154PipobromanFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
25154PipobromanFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
25154PipobromanFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
25154PipobromanFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
25154PipobromanFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
26271CyclophosphamideFDA approvedA7|AlkAg740MethotrexateFDA approvedDf|DHFR
26271CyclophosphamideFDA approvedA7|AlkAg750BusulfanFDA approvedA7|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
26271CyclophosphamideFDA approvedA7|AlkAg7556-MercaptopurineFDA approvedDs|PPAT
26271CyclophosphamideFDA approvedA7|AlkAg762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg1390AllopurinolFDA approvedAM|XDH
26271CyclophosphamideFDA approvedA7|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
26271CyclophosphamideFDA approvedA7|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg6396ThiotepaFDA approvedA7|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg8806MelphalanFDA approvedA7|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg9706Triethylenemelamine-A7|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg14229QuinacrineClinical trialDb|AP
26271CyclophosphamideFDA approvedA7|AlkAg18509Aminolevulinic Acid HydrochlorideFDA approvedAM
26271CyclophosphamideFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
26271CyclophosphamideFDA approvedA7|AlkAg24559MithramycinFDA approvedDb|Rs
26271CyclophosphamideFDA approvedA7|AlkAg25154PipobromanFDA approvedA7|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg26980MitomycinFDA approvedA2|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg27640FloxuridineFDA approvedDs|TYMS
26271CyclophosphamideFDA approvedA7|AlkAg32065HydroxyureaFDA approvedAM|Dr
26271CyclophosphamideFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
26271CyclophosphamideFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg459238-MethoxypsoralenFDA approvedDb
26271CyclophosphamideFDA approvedA7|AlkAg49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
26271CyclophosphamideFDA approvedA7|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
26271CyclophosphamideFDA approvedA7|AlkAg66847ThalidomideFDA approvedAng|Immunomodulatory
26271CyclophosphamideFDA approvedA7|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
26271CyclophosphamideFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
26271CyclophosphamideFDA approvedA7|AlkAg77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
26271CyclophosphamideFDA approvedA7|AlkAg85998StreptozocinFDA approvedA7|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg102816AzacitidineFDA approvedDNMT
26271CyclophosphamideFDA approvedA7|AlkAg105014CladribineFDA approvedDs|ADA
26271CyclophosphamideFDA approvedA7|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
26271CyclophosphamideFDA approvedA7|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
26271CyclophosphamideFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
26271CyclophosphamideFDA approvedA7|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
26271CyclophosphamideFDA approvedA7|AlkAg125066BleomycinFDA approvedDb
26271CyclophosphamideFDA approvedA7|AlkAg125973PaclitaxelFDA approvedTUBB|Tu-stab
26271CyclophosphamideFDA approvedA7|AlkAg138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
26271CyclophosphamideFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
26271CyclophosphamideFDA approvedA7|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
26271CyclophosphamideFDA approvedA7|AlkAg226080RapamycinFDA approvedPK:STK,MTOR
26271CyclophosphamideFDA approvedA7|AlkAg241240CarboplatinFDA approvedA7|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg246131ValrubicinFDA approvedTOP2
26271CyclophosphamideFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
26271CyclophosphamideFDA approvedA7|AlkAg362856TemozolomideFDA approvedA7|AlkAg
26271CyclophosphamideFDA approvedA7|AlkAg606869ClofarabineFDA approvedDs
26271CyclophosphamideFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
26271CyclophosphamideFDA approvedA7|AlkAg613327Gemcitabine HCLFDA approvedDs
26271CyclophosphamideFDA approvedA7|AlkAg628503DocetaxelFDA approvedTUBB|Tu-stab
26271CyclophosphamideFDA approvedA7|AlkAg673596SN 38Clinical trialTOP1
26271CyclophosphamideFDA approvedA7|AlkAg686673NelarabineFDA approvedDs
26271CyclophosphamideFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
26271CyclophosphamideFDA approvedA7|AlkAg701852VorinostatFDA approvedHDAC
26271CyclophosphamideFDA approvedA7|AlkAg712807CapecitabineFDA approvedDs|TYMS
26271CyclophosphamideFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
26271CyclophosphamideFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
26271CyclophosphamideFDA approvedA7|AlkAg719276FulvestrantFDA approvedAM|Ho|ESR|SERM
26271CyclophosphamideFDA approvedA7|AlkAg719344AnastrozoleFDA approvedHo|CYP19A1
26271CyclophosphamideFDA approvedA7|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
26271CyclophosphamideFDA approvedA7|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
26271CyclophosphamideFDA approvedA7|AlkAg721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
26271CyclophosphamideFDA approvedA7|AlkAg732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
26271CyclophosphamideFDA approvedA7|AlkAg733504EverolimusFDA approvedPK:STK,MTOR
26271CyclophosphamideFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
26271CyclophosphamideFDA approvedA7|AlkAg743414ImatinibFDA approvedBCR-ABL|PK:YK
26271CyclophosphamideFDA approvedA7|AlkAg745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
26271CyclophosphamideFDA approvedA7|AlkAg747599NilotinibFDA approvedBCR-ABL|PK:YK
26271CyclophosphamideFDA approvedA7|AlkAg747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
26271CyclophosphamideFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
26271CyclophosphamideFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
26271CyclophosphamideFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
26271CyclophosphamideFDA approvedA7|AlkAg750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
26271CyclophosphamideFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
26271CyclophosphamideFDA approvedA7|AlkAg754143RomidepsinFDA approvedHDAC
26271CyclophosphamideFDA approvedA7|AlkAg754230PralatrexateFDA approvedDf|CTNNB1|DHFR
26271CyclophosphamideFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
26271CyclophosphamideFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
26271CyclophosphamideFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
26271CyclophosphamideFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
26271CyclophosphamideFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
26271CyclophosphamideFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
26980MitomycinFDA approvedA2|AlkAg740MethotrexateFDA approvedDf|DHFR
26980MitomycinFDA approvedA2|AlkAg750BusulfanFDA approvedA7|AlkAg
26980MitomycinFDA approvedA2|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
26980MitomycinFDA approvedA2|AlkAg7556-MercaptopurineFDA approvedDs|PPAT
26980MitomycinFDA approvedA2|AlkAg762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
26980MitomycinFDA approvedA2|AlkAg1390AllopurinolFDA approvedAM|XDH
26980MitomycinFDA approvedA2|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
26980MitomycinFDA approvedA2|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
26980MitomycinFDA approvedA2|AlkAg6396ThiotepaFDA approvedA7|AlkAg
26980MitomycinFDA approvedA2|AlkAg8806MelphalanFDA approvedA7|AlkAg
26980MitomycinFDA approvedA2|AlkAg9706Triethylenemelamine-A7|AlkAg
26980MitomycinFDA approvedA2|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
26980MitomycinFDA approvedA2|AlkAg14229QuinacrineClinical trialDb|AP
26980MitomycinFDA approvedA2|AlkAg18509Aminolevulinic Acid HydrochlorideFDA approvedAM
26980MitomycinFDA approvedA2|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
26980MitomycinFDA approvedA2|AlkAg24559MithramycinFDA approvedDb|Rs
26980MitomycinFDA approvedA2|AlkAg25154PipobromanFDA approvedA7|AlkAg
26980MitomycinFDA approvedA2|AlkAg27640FloxuridineFDA approvedDs|TYMS
26980MitomycinFDA approvedA2|AlkAg32065HydroxyureaFDA approvedAM|Dr
26980MitomycinFDA approvedA2|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
26980MitomycinFDA approvedA2|AlkAg38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
26980MitomycinFDA approvedA2|AlkAg45388DacarbazineFDA approvedA7|AlkAg
26980MitomycinFDA approvedA2|AlkAg49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
26980MitomycinFDA approvedA2|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
26980MitomycinFDA approvedA2|AlkAg66847ThalidomideFDA approvedAng|Immunomodulatory
26980MitomycinFDA approvedA2|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
26980MitomycinFDA approvedA2|AlkAg71423Megestrol acetateFDA approvedHo|PGR
26980MitomycinFDA approvedA2|AlkAg77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
26980MitomycinFDA approvedA2|AlkAg79037LomustineFDA approvedA6|AlkAg
26980MitomycinFDA approvedA2|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
26980MitomycinFDA approvedA2|AlkAg85998StreptozocinFDA approvedA7|AlkAg
26980MitomycinFDA approvedA2|AlkAg102816AzacitidineFDA approvedDNMT
26980MitomycinFDA approvedA2|AlkAg105014CladribineFDA approvedDs|ADA
26980MitomycinFDA approvedA2|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
26980MitomycinFDA approvedA2|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
26980MitomycinFDA approvedA2|AlkAg122819TeniposideFDA approvedTOP2
26980MitomycinFDA approvedA2|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
26980MitomycinFDA approvedA2|AlkAg125066BleomycinFDA approvedDb
26980MitomycinFDA approvedA2|AlkAg125973PaclitaxelFDA approvedTUBB|Tu-stab
26980MitomycinFDA approvedA2|AlkAg138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
26980MitomycinFDA approvedA2|AlkAg141540EtoposideFDA approvedTOP2
26980MitomycinFDA approvedA2|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
26980MitomycinFDA approvedA2|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
26980MitomycinFDA approvedA2|AlkAg226080RapamycinFDA approvedPK:STK,MTOR
26980MitomycinFDA approvedA2|AlkAg241240CarboplatinFDA approvedA7|AlkAg
26980MitomycinFDA approvedA2|AlkAg246131ValrubicinFDA approvedTOP2
26980MitomycinFDA approvedA2|AlkAg279836MitoxantroneFDA approvedTOP2
26980MitomycinFDA approvedA2|AlkAg362856TemozolomideFDA approvedA7|AlkAg
26980MitomycinFDA approvedA2|AlkAg606869ClofarabineFDA approvedDs
26980MitomycinFDA approvedA2|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
26980MitomycinFDA approvedA2|AlkAg613327Gemcitabine HCLFDA approvedDs
26980MitomycinFDA approvedA2|AlkAg628503DocetaxelFDA approvedTUBB|Tu-stab
26980MitomycinFDA approvedA2|AlkAg673596SN 38Clinical trialTOP1
26980MitomycinFDA approvedA2|AlkAg686673NelarabineFDA approvedDs
26980MitomycinFDA approvedA2|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
26980MitomycinFDA approvedA2|AlkAg701852VorinostatFDA approvedHDAC
26980MitomycinFDA approvedA2|AlkAg712807CapecitabineFDA approvedDs|TYMS
26980MitomycinFDA approvedA2|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
26980MitomycinFDA approvedA2|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
26980MitomycinFDA approvedA2|AlkAg719276FulvestrantFDA approvedAM|Ho|ESR|SERM
26980MitomycinFDA approvedA2|AlkAg719344AnastrozoleFDA approvedHo|CYP19A1
26980MitomycinFDA approvedA2|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
26980MitomycinFDA approvedA2|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
26980MitomycinFDA approvedA2|AlkAg721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
26980MitomycinFDA approvedA2|AlkAg732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
26980MitomycinFDA approvedA2|AlkAg733504EverolimusFDA approvedPK:STK,MTOR
26980MitomycinFDA approvedA2|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
26980MitomycinFDA approvedA2|AlkAg743414ImatinibFDA approvedBCR-ABL|PK:YK
26980MitomycinFDA approvedA2|AlkAg745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
26980MitomycinFDA approvedA2|AlkAg747599NilotinibFDA approvedBCR-ABL|PK:YK
26980MitomycinFDA approvedA2|AlkAg747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
26980MitomycinFDA approvedA2|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
26980MitomycinFDA approvedA2|AlkAg747974RaloxifeneFDA approvedHo|SERM
26980MitomycinFDA approvedA2|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
26980MitomycinFDA approvedA2|AlkAg750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
26980MitomycinFDA approvedA2|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
26980MitomycinFDA approvedA2|AlkAg754143RomidepsinFDA approvedHDAC
26980MitomycinFDA approvedA2|AlkAg754230PralatrexateFDA approvedDf|CTNNB1|DHFR
26980MitomycinFDA approvedA2|AlkAg755986VismodegibFDA approvedSMO|PK:YK
26980MitomycinFDA approvedA2|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
26980MitomycinFDA approvedA2|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
26980MitomycinFDA approvedA2|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
26980MitomycinFDA approvedA2|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
26980MitomycinFDA approvedA2|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
27640FloxuridineFDA approvedDs|TYMS740MethotrexateFDA approvedDf|DHFR
27640FloxuridineFDA approvedDs|TYMS752ThioguanineFDA approvedDs|IMPDH2|IMPDH
27640FloxuridineFDA approvedDs|TYMS3053DactinomycinFDA approvedDb|RNA polymerase I
27640FloxuridineFDA approvedDs|TYMS3088ChlorambucilFDA approvedA7|AlkAg
27640FloxuridineFDA approvedDs|TYMS6396ThiotepaFDA approvedA7|AlkAg
27640FloxuridineFDA approvedDs|TYMS8806MelphalanFDA approvedA7|AlkAg
27640FloxuridineFDA approvedDs|TYMS13875HexamethylmelamineFDA approvedDb|AlkAg
27640FloxuridineFDA approvedDs|TYMS19893FluorouracilFDA approvedDs|Rs|TYMS
27640FloxuridineFDA approvedDs|TYMS34462Uracil mustardFDA approvedA7|AlkAg
27640FloxuridineFDA approvedDs|TYMS45388DacarbazineFDA approvedA7|AlkAg
27640FloxuridineFDA approvedDs|TYMS71423Megestrol acetateFDA approvedHo|PGR
27640FloxuridineFDA approvedDs|TYMS79037LomustineFDA approvedA6|AlkAg
27640FloxuridineFDA approvedDs|TYMS82151Daunorubicin hydrochlorideFDA approvedTOP2
27640FloxuridineFDA approvedDs|TYMS122819TeniposideFDA approvedTOP2
27640FloxuridineFDA approvedDs|TYMS141540EtoposideFDA approvedTOP2
27640FloxuridineFDA approvedDs|TYMS169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
27640FloxuridineFDA approvedDs|TYMS279836MitoxantroneFDA approvedTOP2
27640FloxuridineFDA approvedDs|TYMS608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
27640FloxuridineFDA approvedDs|TYMS698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
27640FloxuridineFDA approvedDs|TYMS713563ExemestaneFDA approvedHo|CYP19A1
27640FloxuridineFDA approvedDs|TYMS715055GefitinibFDA approvedPK:YK,EGFR
27640FloxuridineFDA approvedDs|TYMS719345LetrozoleFDA approvedHo|CYP19A1
27640FloxuridineFDA approvedDs|TYMS719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
27640FloxuridineFDA approvedDs|TYMS737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
27640FloxuridineFDA approvedDs|TYMS747972LenalidomideFDA approvedFT|Immunomodulatory
27640FloxuridineFDA approvedDs|TYMS747974RaloxifeneFDA approvedHo|SERM
27640FloxuridineFDA approvedDs|TYMS749226AbirateroneFDA approvedHo|CYP17A1
27640FloxuridineFDA approvedDs|TYMS753082VemurafenibFDA approvedPK:YK,BRAF
27640FloxuridineFDA approvedDs|TYMS755986VismodegibFDA approvedSMO|PK:YK
27640FloxuridineFDA approvedDs|TYMS756645CrizotinibFDA approvedPK:YK,MET,ALK
27640FloxuridineFDA approvedDs|TYMS757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
27640FloxuridineFDA approvedDs|TYMS760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
27640FloxuridineFDA approvedDs|TYMS761432CabazitaxelFDA approvedTUBB|Tu-stab
27640FloxuridineFDA approvedDs|TYMS763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
32065HydroxyureaFDA approvedAM|Dr752ThioguanineFDA approvedDs|IMPDH2|IMPDH
32065HydroxyureaFDA approvedAM|Dr3053DactinomycinFDA approvedDb|RNA polymerase I
32065HydroxyureaFDA approvedAM|Dr3088ChlorambucilFDA approvedA7|AlkAg
32065HydroxyureaFDA approvedAM|Dr6396ThiotepaFDA approvedA7|AlkAg
32065HydroxyureaFDA approvedAM|Dr8806MelphalanFDA approvedA7|AlkAg
32065HydroxyureaFDA approvedAM|Dr9706Triethylenemelamine-A7|AlkAg
32065HydroxyureaFDA approvedAM|Dr13875HexamethylmelamineFDA approvedDb|AlkAg
32065HydroxyureaFDA approvedAM|Dr19893FluorouracilFDA approvedDs|Rs|TYMS
32065HydroxyureaFDA approvedAM|Dr24559MithramycinFDA approvedDb|Rs
32065HydroxyureaFDA approvedAM|Dr27640FloxuridineFDA approvedDs|TYMS
32065HydroxyureaFDA approvedAM|Dr34462Uracil mustardFDA approvedA7|AlkAg
32065HydroxyureaFDA approvedAM|Dr45388DacarbazineFDA approvedA7|AlkAg
32065HydroxyureaFDA approvedAM|Dr63878Cytarabine hydrochlorideFDA approvedDs
32065HydroxyureaFDA approvedAM|Dr67574Vincristine sulfateFDA approvedTUBB|Tu-frag
32065HydroxyureaFDA approvedAM|Dr71423Megestrol acetateFDA approvedHo|PGR
32065HydroxyureaFDA approvedAM|Dr79037LomustineFDA approvedA6|AlkAg
32065HydroxyureaFDA approvedAM|Dr82151Daunorubicin hydrochlorideFDA approvedTOP2
32065HydroxyureaFDA approvedAM|Dr102816AzacitidineFDA approvedDNMT
32065HydroxyureaFDA approvedAM|Dr105014CladribineFDA approvedDs|ADA
32065HydroxyureaFDA approvedAM|Dr118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
32065HydroxyureaFDA approvedAM|Dr122758TretinoinFDA approvedHo|RXR|Differentiator
32065HydroxyureaFDA approvedAM|Dr122819TeniposideFDA approvedTOP2
32065HydroxyureaFDA approvedAM|Dr125973PaclitaxelFDA approvedTUBB|Tu-stab
32065HydroxyureaFDA approvedAM|Dr141540EtoposideFDA approvedTOP2
32065HydroxyureaFDA approvedAM|Dr169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
32065HydroxyureaFDA approvedAM|Dr180973Tamoxifen citrateFDA approvedHo|SERM
32065HydroxyureaFDA approvedAM|Dr241240CarboplatinFDA approvedA7|AlkAg
32065HydroxyureaFDA approvedAM|Dr279836MitoxantroneFDA approvedTOP2
32065HydroxyureaFDA approvedAM|Dr362856TemozolomideFDA approvedA7|AlkAg
32065HydroxyureaFDA approvedAM|Dr608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
32065HydroxyureaFDA approvedAM|Dr628503DocetaxelFDA approvedTUBB|Tu-stab
32065HydroxyureaFDA approvedAM|Dr673596SN 38Clinical trialTOP1
32065HydroxyureaFDA approvedAM|Dr698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
32065HydroxyureaFDA approvedAM|Dr701852VorinostatFDA approvedHDAC
32065HydroxyureaFDA approvedAM|Dr713563ExemestaneFDA approvedHo|CYP19A1
32065HydroxyureaFDA approvedAM|Dr715055GefitinibFDA approvedPK:YK,EGFR
32065HydroxyureaFDA approvedAM|Dr719345LetrozoleFDA approvedHo|CYP19A1
32065HydroxyureaFDA approvedAM|Dr719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
32065HydroxyureaFDA approvedAM|Dr721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
32065HydroxyureaFDA approvedAM|Dr732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
32065HydroxyureaFDA approvedAM|Dr733504EverolimusFDA approvedPK:STK,MTOR
32065HydroxyureaFDA approvedAM|Dr737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
32065HydroxyureaFDA approvedAM|Dr743414ImatinibFDA approvedBCR-ABL|PK:YK
32065HydroxyureaFDA approvedAM|Dr745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
32065HydroxyureaFDA approvedAM|Dr747972LenalidomideFDA approvedFT|Immunomodulatory
32065HydroxyureaFDA approvedAM|Dr747974RaloxifeneFDA approvedHo|SERM
32065HydroxyureaFDA approvedAM|Dr749226AbirateroneFDA approvedHo|CYP17A1
32065HydroxyureaFDA approvedAM|Dr750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
32065HydroxyureaFDA approvedAM|Dr753082VemurafenibFDA approvedPK:YK,BRAF
32065HydroxyureaFDA approvedAM|Dr754143RomidepsinFDA approvedHDAC
32065HydroxyureaFDA approvedAM|Dr755986VismodegibFDA approvedSMO|PK:YK
32065HydroxyureaFDA approvedAM|Dr756645CrizotinibFDA approvedPK:YK,MET,ALK
32065HydroxyureaFDA approvedAM|Dr757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
32065HydroxyureaFDA approvedAM|Dr760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
32065HydroxyureaFDA approvedAM|Dr761432CabazitaxelFDA approvedTUBB|Tu-stab
32065HydroxyureaFDA approvedAM|Dr763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
34462Uracil mustardFDA approvedA7|AlkAg9706Triethylenemelamine-A7|AlkAg
34462Uracil mustardFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
34462Uracil mustardFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
34462Uracil mustardFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
34462Uracil mustardFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
34462Uracil mustardFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
34462Uracil mustardFDA approvedA7|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
34462Uracil mustardFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
34462Uracil mustardFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
34462Uracil mustardFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
34462Uracil mustardFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
34462Uracil mustardFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
34462Uracil mustardFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
34462Uracil mustardFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
34462Uracil mustardFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
34462Uracil mustardFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
34462Uracil mustardFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
34462Uracil mustardFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
34462Uracil mustardFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
34462Uracil mustardFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
34462Uracil mustardFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
34462Uracil mustardFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
34462Uracil mustardFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
34462Uracil mustardFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
34462Uracil mustardFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1752ThioguanineFDA approvedDs|IMPDH2|IMPDH
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A13053DactinomycinFDA approvedDb|RNA polymerase I
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A13088ChlorambucilFDA approvedA7|AlkAg
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A16396ThiotepaFDA approvedA7|AlkAg
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A18806MelphalanFDA approvedA7|AlkAg
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A19706Triethylenemelamine-A7|AlkAg
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A113875HexamethylmelamineFDA approvedDb|AlkAg
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A119893FluorouracilFDA approvedDs|Rs|TYMS
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A124559MithramycinFDA approvedDb|Rs
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A127640FloxuridineFDA approvedDs|TYMS
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A132065HydroxyureaFDA approvedAM|Dr
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A134462Uracil mustardFDA approvedA7|AlkAg
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A145388DacarbazineFDA approvedA7|AlkAg
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A149842Vinblastine sulfateFDA approvedTUBB|Tu-frag
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A163878Cytarabine hydrochlorideFDA approvedDs
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A167574Vincristine sulfateFDA approvedTUBB|Tu-frag
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A171423Megestrol acetateFDA approvedHo|PGR
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A179037LomustineFDA approvedA6|AlkAg
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A182151Daunorubicin hydrochlorideFDA approvedTOP2
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1102816AzacitidineFDA approvedDNMT
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1105014CladribineFDA approvedDs|ADA
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1122758TretinoinFDA approvedHo|RXR|Differentiator
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1122819TeniposideFDA approvedTOP2
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1123127Doxorubicin hydrochlorideFDA approvedTOP2
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1125066BleomycinFDA approvedDb
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1125973PaclitaxelFDA approvedTUBB|Tu-stab
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1141540EtoposideFDA approvedTOP2
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1180973Tamoxifen citrateFDA approvedHo|SERM
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1226080RapamycinFDA approvedPK:STK,MTOR
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1241240CarboplatinFDA approvedA7|AlkAg
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1246131ValrubicinFDA approvedTOP2
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1279836MitoxantroneFDA approvedTOP2
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1362856TemozolomideFDA approvedA7|AlkAg
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1606869ClofarabineFDA approvedDs
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1628503DocetaxelFDA approvedTUBB|Tu-stab
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1673596SN 38Clinical trialTOP1
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1686673NelarabineFDA approvedDs
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1701852VorinostatFDA approvedHDAC
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1712807CapecitabineFDA approvedDs|TYMS
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1713563ExemestaneFDA approvedHo|CYP19A1
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1715055GefitinibFDA approvedPK:YK,EGFR
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1719345LetrozoleFDA approvedHo|CYP19A1
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1733504EverolimusFDA approvedPK:STK,MTOR
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1743414ImatinibFDA approvedBCR-ABL|PK:YK
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1747599NilotinibFDA approvedBCR-ABL|PK:YK
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1747972LenalidomideFDA approvedFT|Immunomodulatory
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1747974RaloxifeneFDA approvedHo|SERM
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1749226AbirateroneFDA approvedHo|CYP17A1
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1753082VemurafenibFDA approvedPK:YK,BRAF
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1754143RomidepsinFDA approvedHDAC
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1755986VismodegibFDA approvedSMO|PK:YK
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1756645CrizotinibFDA approvedPK:YK,MET,ALK
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1761432CabazitaxelFDA approvedTUBB|Tu-stab
38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
45388DacarbazineFDA approvedA7|AlkAg9706Triethylenemelamine-A7|AlkAg
45388DacarbazineFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
45388DacarbazineFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
45388DacarbazineFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
45388DacarbazineFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
45388DacarbazineFDA approvedA7|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
45388DacarbazineFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
45388DacarbazineFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
45388DacarbazineFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
45388DacarbazineFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
45388DacarbazineFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
45388DacarbazineFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
45388DacarbazineFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
45388DacarbazineFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
45388DacarbazineFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
45388DacarbazineFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
45388DacarbazineFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
45388DacarbazineFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
45388DacarbazineFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
45388DacarbazineFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
45388DacarbazineFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
45388DacarbazineFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
45388DacarbazineFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
45388DacarbazineFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
459238-MethoxypsoralenFDA approvedDb740MethotrexateFDA approvedDf|DHFR
459238-MethoxypsoralenFDA approvedDb750BusulfanFDA approvedA7|AlkAg
459238-MethoxypsoralenFDA approvedDb752ThioguanineFDA approvedDs|IMPDH2|IMPDH
459238-MethoxypsoralenFDA approvedDb7556-MercaptopurineFDA approvedDs|PPAT
459238-MethoxypsoralenFDA approvedDb762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
459238-MethoxypsoralenFDA approvedDb1390AllopurinolFDA approvedAM|XDH
459238-MethoxypsoralenFDA approvedDb3053DactinomycinFDA approvedDb|RNA polymerase I
459238-MethoxypsoralenFDA approvedDb3088ChlorambucilFDA approvedA7|AlkAg
459238-MethoxypsoralenFDA approvedDb6396ThiotepaFDA approvedA7|AlkAg
459238-MethoxypsoralenFDA approvedDb8806MelphalanFDA approvedA7|AlkAg
459238-MethoxypsoralenFDA approvedDb9706Triethylenemelamine-A7|AlkAg
459238-MethoxypsoralenFDA approvedDb13875HexamethylmelamineFDA approvedDb|AlkAg
459238-MethoxypsoralenFDA approvedDb14229QuinacrineClinical trialDb|AP
459238-MethoxypsoralenFDA approvedDb18509Aminolevulinic Acid HydrochlorideFDA approvedAM
459238-MethoxypsoralenFDA approvedDb19893FluorouracilFDA approvedDs|Rs|TYMS
459238-MethoxypsoralenFDA approvedDb24559MithramycinFDA approvedDb|Rs
459238-MethoxypsoralenFDA approvedDb25154PipobromanFDA approvedA7|AlkAg
459238-MethoxypsoralenFDA approvedDb26980MitomycinFDA approvedA2|AlkAg
459238-MethoxypsoralenFDA approvedDb27640FloxuridineFDA approvedDs|TYMS
459238-MethoxypsoralenFDA approvedDb32065HydroxyureaFDA approvedAM|Dr
459238-MethoxypsoralenFDA approvedDb34462Uracil mustardFDA approvedA7|AlkAg
459238-MethoxypsoralenFDA approvedDb38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
459238-MethoxypsoralenFDA approvedDb45388DacarbazineFDA approvedA7|AlkAg
459238-MethoxypsoralenFDA approvedDb49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
459238-MethoxypsoralenFDA approvedDb63878Cytarabine hydrochlorideFDA approvedDs
459238-MethoxypsoralenFDA approvedDb66847ThalidomideFDA approvedAng|Immunomodulatory
459238-MethoxypsoralenFDA approvedDb67574Vincristine sulfateFDA approvedTUBB|Tu-frag
459238-MethoxypsoralenFDA approvedDb71423Megestrol acetateFDA approvedHo|PGR
459238-MethoxypsoralenFDA approvedDb77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
459238-MethoxypsoralenFDA approvedDb79037LomustineFDA approvedA6|AlkAg
459238-MethoxypsoralenFDA approvedDb82151Daunorubicin hydrochlorideFDA approvedTOP2
459238-MethoxypsoralenFDA approvedDb85998StreptozocinFDA approvedA7|AlkAg
459238-MethoxypsoralenFDA approvedDb102816AzacitidineFDA approvedDNMT
459238-MethoxypsoralenFDA approvedDb105014CladribineFDA approvedDs|ADA
459238-MethoxypsoralenFDA approvedDb118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
459238-MethoxypsoralenFDA approvedDb122758TretinoinFDA approvedHo|RXR|Differentiator
459238-MethoxypsoralenFDA approvedDb122819TeniposideFDA approvedTOP2
459238-MethoxypsoralenFDA approvedDb123127Doxorubicin hydrochlorideFDA approvedTOP2
459238-MethoxypsoralenFDA approvedDb125066BleomycinFDA approvedDb
459238-MethoxypsoralenFDA approvedDb125973PaclitaxelFDA approvedTUBB|Tu-stab
459238-MethoxypsoralenFDA approvedDb138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
459238-MethoxypsoralenFDA approvedDb141540EtoposideFDA approvedTOP2
459238-MethoxypsoralenFDA approvedDb169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
459238-MethoxypsoralenFDA approvedDb180973Tamoxifen citrateFDA approvedHo|SERM
459238-MethoxypsoralenFDA approvedDb226080RapamycinFDA approvedPK:STK,MTOR
459238-MethoxypsoralenFDA approvedDb241240CarboplatinFDA approvedA7|AlkAg
459238-MethoxypsoralenFDA approvedDb246131ValrubicinFDA approvedTOP2
459238-MethoxypsoralenFDA approvedDb279836MitoxantroneFDA approvedTOP2
459238-MethoxypsoralenFDA approvedDb362856TemozolomideFDA approvedA7|AlkAg
459238-MethoxypsoralenFDA approvedDb606869ClofarabineFDA approvedDs
459238-MethoxypsoralenFDA approvedDb608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
459238-MethoxypsoralenFDA approvedDb613327Gemcitabine HCLFDA approvedDs
459238-MethoxypsoralenFDA approvedDb628503DocetaxelFDA approvedTUBB|Tu-stab
459238-MethoxypsoralenFDA approvedDb673596SN 38Clinical trialTOP1
459238-MethoxypsoralenFDA approvedDb686673NelarabineFDA approvedDs
459238-MethoxypsoralenFDA approvedDb698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
459238-MethoxypsoralenFDA approvedDb701852VorinostatFDA approvedHDAC
459238-MethoxypsoralenFDA approvedDb712807CapecitabineFDA approvedDs|TYMS
459238-MethoxypsoralenFDA approvedDb713563ExemestaneFDA approvedHo|CYP19A1
459238-MethoxypsoralenFDA approvedDb715055GefitinibFDA approvedPK:YK,EGFR
459238-MethoxypsoralenFDA approvedDb719276FulvestrantFDA approvedAM|Ho|ESR|SERM
459238-MethoxypsoralenFDA approvedDb719344AnastrozoleFDA approvedHo|CYP19A1
459238-MethoxypsoralenFDA approvedDb719345LetrozoleFDA approvedHo|CYP19A1
459238-MethoxypsoralenFDA approvedDb719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
459238-MethoxypsoralenFDA approvedDb721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
459238-MethoxypsoralenFDA approvedDb732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
459238-MethoxypsoralenFDA approvedDb733504EverolimusFDA approvedPK:STK,MTOR
459238-MethoxypsoralenFDA approvedDb737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
459238-MethoxypsoralenFDA approvedDb743414ImatinibFDA approvedBCR-ABL|PK:YK
459238-MethoxypsoralenFDA approvedDb745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
459238-MethoxypsoralenFDA approvedDb747599NilotinibFDA approvedBCR-ABL|PK:YK
459238-MethoxypsoralenFDA approvedDb747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
459238-MethoxypsoralenFDA approvedDb747972LenalidomideFDA approvedFT|Immunomodulatory
459238-MethoxypsoralenFDA approvedDb747974RaloxifeneFDA approvedHo|SERM
459238-MethoxypsoralenFDA approvedDb749226AbirateroneFDA approvedHo|CYP17A1
459238-MethoxypsoralenFDA approvedDb750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
459238-MethoxypsoralenFDA approvedDb753082VemurafenibFDA approvedPK:YK,BRAF
459238-MethoxypsoralenFDA approvedDb754143RomidepsinFDA approvedHDAC
459238-MethoxypsoralenFDA approvedDb754230PralatrexateFDA approvedDf|CTNNB1|DHFR
459238-MethoxypsoralenFDA approvedDb755986VismodegibFDA approvedSMO|PK:YK
459238-MethoxypsoralenFDA approvedDb756645CrizotinibFDA approvedPK:YK,MET,ALK
459238-MethoxypsoralenFDA approvedDb757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
459238-MethoxypsoralenFDA approvedDb760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
459238-MethoxypsoralenFDA approvedDb761432CabazitaxelFDA approvedTUBB|Tu-stab
459238-MethoxypsoralenFDA approvedDb763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag752ThioguanineFDA approvedDs|IMPDH2|IMPDH
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag3053DactinomycinFDA approvedDb|RNA polymerase I
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag3088ChlorambucilFDA approvedA7|AlkAg
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag6396ThiotepaFDA approvedA7|AlkAg
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag8806MelphalanFDA approvedA7|AlkAg
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag9706Triethylenemelamine-A7|AlkAg
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag13875HexamethylmelamineFDA approvedDb|AlkAg
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag19893FluorouracilFDA approvedDs|Rs|TYMS
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag24559MithramycinFDA approvedDb|Rs
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag27640FloxuridineFDA approvedDs|TYMS
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag32065HydroxyureaFDA approvedAM|Dr
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag34462Uracil mustardFDA approvedA7|AlkAg
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag45388DacarbazineFDA approvedA7|AlkAg
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag63878Cytarabine hydrochlorideFDA approvedDs
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag67574Vincristine sulfateFDA approvedTUBB|Tu-frag
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag71423Megestrol acetateFDA approvedHo|PGR
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag79037LomustineFDA approvedA6|AlkAg
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag82151Daunorubicin hydrochlorideFDA approvedTOP2
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag102816AzacitidineFDA approvedDNMT
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag105014CladribineFDA approvedDs|ADA
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag122758TretinoinFDA approvedHo|RXR|Differentiator
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag122819TeniposideFDA approvedTOP2
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag123127Doxorubicin hydrochlorideFDA approvedTOP2
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag125066BleomycinFDA approvedDb
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag125973PaclitaxelFDA approvedTUBB|Tu-stab
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag141540EtoposideFDA approvedTOP2
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag180973Tamoxifen citrateFDA approvedHo|SERM
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag226080RapamycinFDA approvedPK:STK,MTOR
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag241240CarboplatinFDA approvedA7|AlkAg
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag279836MitoxantroneFDA approvedTOP2
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag362856TemozolomideFDA approvedA7|AlkAg
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag606869ClofarabineFDA approvedDs
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag613327Gemcitabine HCLFDA approvedDs
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag673596SN 38Clinical trialTOP1
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag686673NelarabineFDA approvedDs
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag701852VorinostatFDA approvedHDAC
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag713563ExemestaneFDA approvedHo|CYP19A1
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag715055GefitinibFDA approvedPK:YK,EGFR
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag719345LetrozoleFDA approvedHo|CYP19A1
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag733504EverolimusFDA approvedPK:STK,MTOR
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag743414ImatinibFDA approvedBCR-ABL|PK:YK
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag747599NilotinibFDA approvedBCR-ABL|PK:YK
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag747972LenalidomideFDA approvedFT|Immunomodulatory
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag747974RaloxifeneFDA approvedHo|SERM
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag749226AbirateroneFDA approvedHo|CYP17A1
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag753082VemurafenibFDA approvedPK:YK,BRAF
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag754143RomidepsinFDA approvedHDAC
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag755986VismodegibFDA approvedSMO|PK:YK
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag756645CrizotinibFDA approvedPK:YK,MET,ALK
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag761432CabazitaxelFDA approvedTUBB|Tu-stab
49842Vinblastine sulfateFDA approvedTUBB|Tu-frag763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
63878Cytarabine hydrochlorideFDA approvedDs740MethotrexateFDA approvedDf|DHFR
63878Cytarabine hydrochlorideFDA approvedDs752ThioguanineFDA approvedDs|IMPDH2|IMPDH
63878Cytarabine hydrochlorideFDA approvedDs3053DactinomycinFDA approvedDb|RNA polymerase I
63878Cytarabine hydrochlorideFDA approvedDs3088ChlorambucilFDA approvedA7|AlkAg
63878Cytarabine hydrochlorideFDA approvedDs6396ThiotepaFDA approvedA7|AlkAg
63878Cytarabine hydrochlorideFDA approvedDs8806MelphalanFDA approvedA7|AlkAg
63878Cytarabine hydrochlorideFDA approvedDs13875HexamethylmelamineFDA approvedDb|AlkAg
63878Cytarabine hydrochlorideFDA approvedDs19893FluorouracilFDA approvedDs|Rs|TYMS
63878Cytarabine hydrochlorideFDA approvedDs27640FloxuridineFDA approvedDs|TYMS
63878Cytarabine hydrochlorideFDA approvedDs34462Uracil mustardFDA approvedA7|AlkAg
63878Cytarabine hydrochlorideFDA approvedDs45388DacarbazineFDA approvedA7|AlkAg
63878Cytarabine hydrochlorideFDA approvedDs71423Megestrol acetateFDA approvedHo|PGR
63878Cytarabine hydrochlorideFDA approvedDs79037LomustineFDA approvedA6|AlkAg
63878Cytarabine hydrochlorideFDA approvedDs82151Daunorubicin hydrochlorideFDA approvedTOP2
63878Cytarabine hydrochlorideFDA approvedDs122819TeniposideFDA approvedTOP2
63878Cytarabine hydrochlorideFDA approvedDs141540EtoposideFDA approvedTOP2
63878Cytarabine hydrochlorideFDA approvedDs169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
63878Cytarabine hydrochlorideFDA approvedDs279836MitoxantroneFDA approvedTOP2
63878Cytarabine hydrochlorideFDA approvedDs608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
63878Cytarabine hydrochlorideFDA approvedDs698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
63878Cytarabine hydrochlorideFDA approvedDs713563ExemestaneFDA approvedHo|CYP19A1
63878Cytarabine hydrochlorideFDA approvedDs715055GefitinibFDA approvedPK:YK,EGFR
63878Cytarabine hydrochlorideFDA approvedDs719345LetrozoleFDA approvedHo|CYP19A1
63878Cytarabine hydrochlorideFDA approvedDs719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
63878Cytarabine hydrochlorideFDA approvedDs737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
63878Cytarabine hydrochlorideFDA approvedDs747972LenalidomideFDA approvedFT|Immunomodulatory
63878Cytarabine hydrochlorideFDA approvedDs747974RaloxifeneFDA approvedHo|SERM
63878Cytarabine hydrochlorideFDA approvedDs749226AbirateroneFDA approvedHo|CYP17A1
63878Cytarabine hydrochlorideFDA approvedDs753082VemurafenibFDA approvedPK:YK,BRAF
63878Cytarabine hydrochlorideFDA approvedDs755986VismodegibFDA approvedSMO|PK:YK
63878Cytarabine hydrochlorideFDA approvedDs756645CrizotinibFDA approvedPK:YK,MET,ALK
63878Cytarabine hydrochlorideFDA approvedDs757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
63878Cytarabine hydrochlorideFDA approvedDs760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
63878Cytarabine hydrochlorideFDA approvedDs761432CabazitaxelFDA approvedTUBB|Tu-stab
63878Cytarabine hydrochlorideFDA approvedDs763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
66847ThalidomideFDA approvedAng|Immunomodulatory740MethotrexateFDA approvedDf|DHFR
66847ThalidomideFDA approvedAng|Immunomodulatory750BusulfanFDA approvedA7|AlkAg
66847ThalidomideFDA approvedAng|Immunomodulatory752ThioguanineFDA approvedDs|IMPDH2|IMPDH
66847ThalidomideFDA approvedAng|Immunomodulatory7556-MercaptopurineFDA approvedDs|PPAT
66847ThalidomideFDA approvedAng|Immunomodulatory762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
66847ThalidomideFDA approvedAng|Immunomodulatory1390AllopurinolFDA approvedAM|XDH
66847ThalidomideFDA approvedAng|Immunomodulatory3053DactinomycinFDA approvedDb|RNA polymerase I
66847ThalidomideFDA approvedAng|Immunomodulatory3088ChlorambucilFDA approvedA7|AlkAg
66847ThalidomideFDA approvedAng|Immunomodulatory6396ThiotepaFDA approvedA7|AlkAg
66847ThalidomideFDA approvedAng|Immunomodulatory8806MelphalanFDA approvedA7|AlkAg
66847ThalidomideFDA approvedAng|Immunomodulatory9706Triethylenemelamine-A7|AlkAg
66847ThalidomideFDA approvedAng|Immunomodulatory13875HexamethylmelamineFDA approvedDb|AlkAg
66847ThalidomideFDA approvedAng|Immunomodulatory14229QuinacrineClinical trialDb|AP
66847ThalidomideFDA approvedAng|Immunomodulatory18509Aminolevulinic Acid HydrochlorideFDA approvedAM
66847ThalidomideFDA approvedAng|Immunomodulatory19893FluorouracilFDA approvedDs|Rs|TYMS
66847ThalidomideFDA approvedAng|Immunomodulatory24559MithramycinFDA approvedDb|Rs
66847ThalidomideFDA approvedAng|Immunomodulatory25154PipobromanFDA approvedA7|AlkAg
66847ThalidomideFDA approvedAng|Immunomodulatory27640FloxuridineFDA approvedDs|TYMS
66847ThalidomideFDA approvedAng|Immunomodulatory32065HydroxyureaFDA approvedAM|Dr
66847ThalidomideFDA approvedAng|Immunomodulatory34462Uracil mustardFDA approvedA7|AlkAg
66847ThalidomideFDA approvedAng|Immunomodulatory38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
66847ThalidomideFDA approvedAng|Immunomodulatory45388DacarbazineFDA approvedA7|AlkAg
66847ThalidomideFDA approvedAng|Immunomodulatory49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
66847ThalidomideFDA approvedAng|Immunomodulatory63878Cytarabine hydrochlorideFDA approvedDs
66847ThalidomideFDA approvedAng|Immunomodulatory67574Vincristine sulfateFDA approvedTUBB|Tu-frag
66847ThalidomideFDA approvedAng|Immunomodulatory71423Megestrol acetateFDA approvedHo|PGR
66847ThalidomideFDA approvedAng|Immunomodulatory79037LomustineFDA approvedA6|AlkAg
66847ThalidomideFDA approvedAng|Immunomodulatory82151Daunorubicin hydrochlorideFDA approvedTOP2
66847ThalidomideFDA approvedAng|Immunomodulatory102816AzacitidineFDA approvedDNMT
66847ThalidomideFDA approvedAng|Immunomodulatory105014CladribineFDA approvedDs|ADA
66847ThalidomideFDA approvedAng|Immunomodulatory118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
66847ThalidomideFDA approvedAng|Immunomodulatory122758TretinoinFDA approvedHo|RXR|Differentiator
66847ThalidomideFDA approvedAng|Immunomodulatory122819TeniposideFDA approvedTOP2
66847ThalidomideFDA approvedAng|Immunomodulatory123127Doxorubicin hydrochlorideFDA approvedTOP2
66847ThalidomideFDA approvedAng|Immunomodulatory125066BleomycinFDA approvedDb
66847ThalidomideFDA approvedAng|Immunomodulatory125973PaclitaxelFDA approvedTUBB|Tu-stab
66847ThalidomideFDA approvedAng|Immunomodulatory138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
66847ThalidomideFDA approvedAng|Immunomodulatory141540EtoposideFDA approvedTOP2
66847ThalidomideFDA approvedAng|Immunomodulatory169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
66847ThalidomideFDA approvedAng|Immunomodulatory180973Tamoxifen citrateFDA approvedHo|SERM
66847ThalidomideFDA approvedAng|Immunomodulatory226080RapamycinFDA approvedPK:STK,MTOR
66847ThalidomideFDA approvedAng|Immunomodulatory241240CarboplatinFDA approvedA7|AlkAg
66847ThalidomideFDA approvedAng|Immunomodulatory246131ValrubicinFDA approvedTOP2
66847ThalidomideFDA approvedAng|Immunomodulatory279836MitoxantroneFDA approvedTOP2
66847ThalidomideFDA approvedAng|Immunomodulatory362856TemozolomideFDA approvedA7|AlkAg
66847ThalidomideFDA approvedAng|Immunomodulatory606869ClofarabineFDA approvedDs
66847ThalidomideFDA approvedAng|Immunomodulatory608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
66847ThalidomideFDA approvedAng|Immunomodulatory613327Gemcitabine HCLFDA approvedDs
66847ThalidomideFDA approvedAng|Immunomodulatory628503DocetaxelFDA approvedTUBB|Tu-stab
66847ThalidomideFDA approvedAng|Immunomodulatory673596SN 38Clinical trialTOP1
66847ThalidomideFDA approvedAng|Immunomodulatory686673NelarabineFDA approvedDs
66847ThalidomideFDA approvedAng|Immunomodulatory698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
66847ThalidomideFDA approvedAng|Immunomodulatory701852VorinostatFDA approvedHDAC
66847ThalidomideFDA approvedAng|Immunomodulatory712807CapecitabineFDA approvedDs|TYMS
66847ThalidomideFDA approvedAng|Immunomodulatory713563ExemestaneFDA approvedHo|CYP19A1
66847ThalidomideFDA approvedAng|Immunomodulatory715055GefitinibFDA approvedPK:YK,EGFR
66847ThalidomideFDA approvedAng|Immunomodulatory719276FulvestrantFDA approvedAM|Ho|ESR|SERM
66847ThalidomideFDA approvedAng|Immunomodulatory719344AnastrozoleFDA approvedHo|CYP19A1
66847ThalidomideFDA approvedAng|Immunomodulatory719345LetrozoleFDA approvedHo|CYP19A1
66847ThalidomideFDA approvedAng|Immunomodulatory719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
66847ThalidomideFDA approvedAng|Immunomodulatory721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
66847ThalidomideFDA approvedAng|Immunomodulatory732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
66847ThalidomideFDA approvedAng|Immunomodulatory733504EverolimusFDA approvedPK:STK,MTOR
66847ThalidomideFDA approvedAng|Immunomodulatory737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
66847ThalidomideFDA approvedAng|Immunomodulatory743414ImatinibFDA approvedBCR-ABL|PK:YK
66847ThalidomideFDA approvedAng|Immunomodulatory745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
66847ThalidomideFDA approvedAng|Immunomodulatory747599NilotinibFDA approvedBCR-ABL|PK:YK
66847ThalidomideFDA approvedAng|Immunomodulatory747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
66847ThalidomideFDA approvedAng|Immunomodulatory747972LenalidomideFDA approvedFT|Immunomodulatory
66847ThalidomideFDA approvedAng|Immunomodulatory747974RaloxifeneFDA approvedHo|SERM
66847ThalidomideFDA approvedAng|Immunomodulatory749226AbirateroneFDA approvedHo|CYP17A1
66847ThalidomideFDA approvedAng|Immunomodulatory750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
66847ThalidomideFDA approvedAng|Immunomodulatory753082VemurafenibFDA approvedPK:YK,BRAF
66847ThalidomideFDA approvedAng|Immunomodulatory754143RomidepsinFDA approvedHDAC
66847ThalidomideFDA approvedAng|Immunomodulatory754230PralatrexateFDA approvedDf|CTNNB1|DHFR
66847ThalidomideFDA approvedAng|Immunomodulatory755986VismodegibFDA approvedSMO|PK:YK
66847ThalidomideFDA approvedAng|Immunomodulatory756645CrizotinibFDA approvedPK:YK,MET,ALK
66847ThalidomideFDA approvedAng|Immunomodulatory757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
66847ThalidomideFDA approvedAng|Immunomodulatory760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
66847ThalidomideFDA approvedAng|Immunomodulatory761432CabazitaxelFDA approvedTUBB|Tu-stab
66847ThalidomideFDA approvedAng|Immunomodulatory763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
67574Vincristine sulfateFDA approvedTUBB|Tu-frag740MethotrexateFDA approvedDf|DHFR
67574Vincristine sulfateFDA approvedTUBB|Tu-frag752ThioguanineFDA approvedDs|IMPDH2|IMPDH
67574Vincristine sulfateFDA approvedTUBB|Tu-frag3053DactinomycinFDA approvedDb|RNA polymerase I
67574Vincristine sulfateFDA approvedTUBB|Tu-frag3088ChlorambucilFDA approvedA7|AlkAg
67574Vincristine sulfateFDA approvedTUBB|Tu-frag6396ThiotepaFDA approvedA7|AlkAg
67574Vincristine sulfateFDA approvedTUBB|Tu-frag8806MelphalanFDA approvedA7|AlkAg
67574Vincristine sulfateFDA approvedTUBB|Tu-frag13875HexamethylmelamineFDA approvedDb|AlkAg
67574Vincristine sulfateFDA approvedTUBB|Tu-frag19893FluorouracilFDA approvedDs|Rs|TYMS
67574Vincristine sulfateFDA approvedTUBB|Tu-frag27640FloxuridineFDA approvedDs|TYMS
67574Vincristine sulfateFDA approvedTUBB|Tu-frag34462Uracil mustardFDA approvedA7|AlkAg
67574Vincristine sulfateFDA approvedTUBB|Tu-frag45388DacarbazineFDA approvedA7|AlkAg
67574Vincristine sulfateFDA approvedTUBB|Tu-frag63878Cytarabine hydrochlorideFDA approvedDs
67574Vincristine sulfateFDA approvedTUBB|Tu-frag71423Megestrol acetateFDA approvedHo|PGR
67574Vincristine sulfateFDA approvedTUBB|Tu-frag79037LomustineFDA approvedA6|AlkAg
67574Vincristine sulfateFDA approvedTUBB|Tu-frag82151Daunorubicin hydrochlorideFDA approvedTOP2
67574Vincristine sulfateFDA approvedTUBB|Tu-frag122819TeniposideFDA approvedTOP2
67574Vincristine sulfateFDA approvedTUBB|Tu-frag141540EtoposideFDA approvedTOP2
67574Vincristine sulfateFDA approvedTUBB|Tu-frag169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
67574Vincristine sulfateFDA approvedTUBB|Tu-frag279836MitoxantroneFDA approvedTOP2
67574Vincristine sulfateFDA approvedTUBB|Tu-frag608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
67574Vincristine sulfateFDA approvedTUBB|Tu-frag698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
67574Vincristine sulfateFDA approvedTUBB|Tu-frag713563ExemestaneFDA approvedHo|CYP19A1
67574Vincristine sulfateFDA approvedTUBB|Tu-frag715055GefitinibFDA approvedPK:YK,EGFR
67574Vincristine sulfateFDA approvedTUBB|Tu-frag719345LetrozoleFDA approvedHo|CYP19A1
67574Vincristine sulfateFDA approvedTUBB|Tu-frag719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
67574Vincristine sulfateFDA approvedTUBB|Tu-frag737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
67574Vincristine sulfateFDA approvedTUBB|Tu-frag747972LenalidomideFDA approvedFT|Immunomodulatory
67574Vincristine sulfateFDA approvedTUBB|Tu-frag747974RaloxifeneFDA approvedHo|SERM
67574Vincristine sulfateFDA approvedTUBB|Tu-frag749226AbirateroneFDA approvedHo|CYP17A1
67574Vincristine sulfateFDA approvedTUBB|Tu-frag753082VemurafenibFDA approvedPK:YK,BRAF
67574Vincristine sulfateFDA approvedTUBB|Tu-frag755986VismodegibFDA approvedSMO|PK:YK
67574Vincristine sulfateFDA approvedTUBB|Tu-frag756645CrizotinibFDA approvedPK:YK,MET,ALK
67574Vincristine sulfateFDA approvedTUBB|Tu-frag757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
67574Vincristine sulfateFDA approvedTUBB|Tu-frag760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
67574Vincristine sulfateFDA approvedTUBB|Tu-frag761432CabazitaxelFDA approvedTUBB|Tu-stab
67574Vincristine sulfateFDA approvedTUBB|Tu-frag763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
71423Megestrol acetateFDA approvedHo|PGR9706Triethylenemelamine-A7|AlkAg
71423Megestrol acetateFDA approvedHo|PGR79037LomustineFDA approvedA6|AlkAg
71423Megestrol acetateFDA approvedHo|PGR82151Daunorubicin hydrochlorideFDA approvedTOP2
71423Megestrol acetateFDA approvedHo|PGR122819TeniposideFDA approvedTOP2
71423Megestrol acetateFDA approvedHo|PGR123127Doxorubicin hydrochlorideFDA approvedTOP2
71423Megestrol acetateFDA approvedHo|PGR141540EtoposideFDA approvedTOP2
71423Megestrol acetateFDA approvedHo|PGR169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
71423Megestrol acetateFDA approvedHo|PGR279836MitoxantroneFDA approvedTOP2
71423Megestrol acetateFDA approvedHo|PGR608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
71423Megestrol acetateFDA approvedHo|PGR698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
71423Megestrol acetateFDA approvedHo|PGR713563ExemestaneFDA approvedHo|CYP19A1
71423Megestrol acetateFDA approvedHo|PGR715055GefitinibFDA approvedPK:YK,EGFR
71423Megestrol acetateFDA approvedHo|PGR737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
71423Megestrol acetateFDA approvedHo|PGR747972LenalidomideFDA approvedFT|Immunomodulatory
71423Megestrol acetateFDA approvedHo|PGR747974RaloxifeneFDA approvedHo|SERM
71423Megestrol acetateFDA approvedHo|PGR749226AbirateroneFDA approvedHo|CYP17A1
71423Megestrol acetateFDA approvedHo|PGR753082VemurafenibFDA approvedPK:YK,BRAF
71423Megestrol acetateFDA approvedHo|PGR755986VismodegibFDA approvedSMO|PK:YK
71423Megestrol acetateFDA approvedHo|PGR756645CrizotinibFDA approvedPK:YK,MET,ALK
71423Megestrol acetateFDA approvedHo|PGR757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
71423Megestrol acetateFDA approvedHo|PGR760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
71423Megestrol acetateFDA approvedHo|PGR761432CabazitaxelFDA approvedTUBB|Tu-stab
71423Megestrol acetateFDA approvedHo|PGR763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg740MethotrexateFDA approvedDf|DHFR
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg750BusulfanFDA approvedA7|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg7556-MercaptopurineFDA approvedDs|PPAT
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg1390AllopurinolFDA approvedAM|XDH
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg6396ThiotepaFDA approvedA7|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg8806MelphalanFDA approvedA7|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg9706Triethylenemelamine-A7|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg14229QuinacrineClinical trialDb|AP
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg18509Aminolevulinic Acid HydrochlorideFDA approvedAM
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg24559MithramycinFDA approvedDb|Rs
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg25154PipobromanFDA approvedA7|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg27640FloxuridineFDA approvedDs|TYMS
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg32065HydroxyureaFDA approvedAM|Dr
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg66847ThalidomideFDA approvedAng|Immunomodulatory
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg85998StreptozocinFDA approvedA7|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg102816AzacitidineFDA approvedDNMT
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg105014CladribineFDA approvedDs|ADA
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg125066BleomycinFDA approvedDb
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg125973PaclitaxelFDA approvedTUBB|Tu-stab
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg226080RapamycinFDA approvedPK:STK,MTOR
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg241240CarboplatinFDA approvedA7|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg246131ValrubicinFDA approvedTOP2
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg362856TemozolomideFDA approvedA7|AlkAg
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg606869ClofarabineFDA approvedDs
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg613327Gemcitabine HCLFDA approvedDs
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg628503DocetaxelFDA approvedTUBB|Tu-stab
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg673596SN 38Clinical trialTOP1
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg686673NelarabineFDA approvedDs
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg701852VorinostatFDA approvedHDAC
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg712807CapecitabineFDA approvedDs|TYMS
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg719276FulvestrantFDA approvedAM|Ho|ESR|SERM
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg719344AnastrozoleFDA approvedHo|CYP19A1
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg733504EverolimusFDA approvedPK:STK,MTOR
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg743414ImatinibFDA approvedBCR-ABL|PK:YK
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg747599NilotinibFDA approvedBCR-ABL|PK:YK
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg754143RomidepsinFDA approvedHDAC
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg754230PralatrexateFDA approvedDf|CTNNB1|DHFR
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
77213Procarbazine hydrochlorideFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
79037LomustineFDA approvedA6|AlkAg9706Triethylenemelamine-A7|AlkAg
79037LomustineFDA approvedA6|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
79037LomustineFDA approvedA6|AlkAg122819TeniposideFDA approvedTOP2
79037LomustineFDA approvedA6|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
79037LomustineFDA approvedA6|AlkAg141540EtoposideFDA approvedTOP2
79037LomustineFDA approvedA6|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
79037LomustineFDA approvedA6|AlkAg279836MitoxantroneFDA approvedTOP2
79037LomustineFDA approvedA6|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
79037LomustineFDA approvedA6|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
79037LomustineFDA approvedA6|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
79037LomustineFDA approvedA6|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
79037LomustineFDA approvedA6|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
79037LomustineFDA approvedA6|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
79037LomustineFDA approvedA6|AlkAg747974RaloxifeneFDA approvedHo|SERM
79037LomustineFDA approvedA6|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
79037LomustineFDA approvedA6|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
79037LomustineFDA approvedA6|AlkAg755986VismodegibFDA approvedSMO|PK:YK
79037LomustineFDA approvedA6|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
79037LomustineFDA approvedA6|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
79037LomustineFDA approvedA6|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
79037LomustineFDA approvedA6|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
79037LomustineFDA approvedA6|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
82151Daunorubicin hydrochlorideFDA approvedTOP29706Triethylenemelamine-A7|AlkAg
82151Daunorubicin hydrochlorideFDA approvedTOP2122819TeniposideFDA approvedTOP2
82151Daunorubicin hydrochlorideFDA approvedTOP2123127Doxorubicin hydrochlorideFDA approvedTOP2
82151Daunorubicin hydrochlorideFDA approvedTOP2141540EtoposideFDA approvedTOP2
82151Daunorubicin hydrochlorideFDA approvedTOP2169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
82151Daunorubicin hydrochlorideFDA approvedTOP2279836MitoxantroneFDA approvedTOP2
82151Daunorubicin hydrochlorideFDA approvedTOP2608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
82151Daunorubicin hydrochlorideFDA approvedTOP2698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
82151Daunorubicin hydrochlorideFDA approvedTOP2713563ExemestaneFDA approvedHo|CYP19A1
82151Daunorubicin hydrochlorideFDA approvedTOP2715055GefitinibFDA approvedPK:YK,EGFR
82151Daunorubicin hydrochlorideFDA approvedTOP2737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
82151Daunorubicin hydrochlorideFDA approvedTOP2747972LenalidomideFDA approvedFT|Immunomodulatory
82151Daunorubicin hydrochlorideFDA approvedTOP2747974RaloxifeneFDA approvedHo|SERM
82151Daunorubicin hydrochlorideFDA approvedTOP2749226AbirateroneFDA approvedHo|CYP17A1
82151Daunorubicin hydrochlorideFDA approvedTOP2753082VemurafenibFDA approvedPK:YK,BRAF
82151Daunorubicin hydrochlorideFDA approvedTOP2755986VismodegibFDA approvedSMO|PK:YK
82151Daunorubicin hydrochlorideFDA approvedTOP2756645CrizotinibFDA approvedPK:YK,MET,ALK
82151Daunorubicin hydrochlorideFDA approvedTOP2757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
82151Daunorubicin hydrochlorideFDA approvedTOP2760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
82151Daunorubicin hydrochlorideFDA approvedTOP2761432CabazitaxelFDA approvedTUBB|Tu-stab
82151Daunorubicin hydrochlorideFDA approvedTOP2763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
85998StreptozocinFDA approvedA7|AlkAg740MethotrexateFDA approvedDf|DHFR
85998StreptozocinFDA approvedA7|AlkAg750BusulfanFDA approvedA7|AlkAg
85998StreptozocinFDA approvedA7|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
85998StreptozocinFDA approvedA7|AlkAg7556-MercaptopurineFDA approvedDs|PPAT
85998StreptozocinFDA approvedA7|AlkAg762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
85998StreptozocinFDA approvedA7|AlkAg1390AllopurinolFDA approvedAM|XDH
85998StreptozocinFDA approvedA7|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
85998StreptozocinFDA approvedA7|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
85998StreptozocinFDA approvedA7|AlkAg6396ThiotepaFDA approvedA7|AlkAg
85998StreptozocinFDA approvedA7|AlkAg8806MelphalanFDA approvedA7|AlkAg
85998StreptozocinFDA approvedA7|AlkAg9706Triethylenemelamine-A7|AlkAg
85998StreptozocinFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
85998StreptozocinFDA approvedA7|AlkAg14229QuinacrineClinical trialDb|AP
85998StreptozocinFDA approvedA7|AlkAg18509Aminolevulinic Acid HydrochlorideFDA approvedAM
85998StreptozocinFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
85998StreptozocinFDA approvedA7|AlkAg24559MithramycinFDA approvedDb|Rs
85998StreptozocinFDA approvedA7|AlkAg25154PipobromanFDA approvedA7|AlkAg
85998StreptozocinFDA approvedA7|AlkAg27640FloxuridineFDA approvedDs|TYMS
85998StreptozocinFDA approvedA7|AlkAg32065HydroxyureaFDA approvedAM|Dr
85998StreptozocinFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
85998StreptozocinFDA approvedA7|AlkAg38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
85998StreptozocinFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
85998StreptozocinFDA approvedA7|AlkAg49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
85998StreptozocinFDA approvedA7|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
85998StreptozocinFDA approvedA7|AlkAg66847ThalidomideFDA approvedAng|Immunomodulatory
85998StreptozocinFDA approvedA7|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
85998StreptozocinFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
85998StreptozocinFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
85998StreptozocinFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
85998StreptozocinFDA approvedA7|AlkAg102816AzacitidineFDA approvedDNMT
85998StreptozocinFDA approvedA7|AlkAg105014CladribineFDA approvedDs|ADA
85998StreptozocinFDA approvedA7|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
85998StreptozocinFDA approvedA7|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
85998StreptozocinFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
85998StreptozocinFDA approvedA7|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
85998StreptozocinFDA approvedA7|AlkAg125066BleomycinFDA approvedDb
85998StreptozocinFDA approvedA7|AlkAg125973PaclitaxelFDA approvedTUBB|Tu-stab
85998StreptozocinFDA approvedA7|AlkAg138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
85998StreptozocinFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
85998StreptozocinFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
85998StreptozocinFDA approvedA7|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
85998StreptozocinFDA approvedA7|AlkAg226080RapamycinFDA approvedPK:STK,MTOR
85998StreptozocinFDA approvedA7|AlkAg241240CarboplatinFDA approvedA7|AlkAg
85998StreptozocinFDA approvedA7|AlkAg246131ValrubicinFDA approvedTOP2
85998StreptozocinFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
85998StreptozocinFDA approvedA7|AlkAg362856TemozolomideFDA approvedA7|AlkAg
85998StreptozocinFDA approvedA7|AlkAg606869ClofarabineFDA approvedDs
85998StreptozocinFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
85998StreptozocinFDA approvedA7|AlkAg613327Gemcitabine HCLFDA approvedDs
85998StreptozocinFDA approvedA7|AlkAg628503DocetaxelFDA approvedTUBB|Tu-stab
85998StreptozocinFDA approvedA7|AlkAg673596SN 38Clinical trialTOP1
85998StreptozocinFDA approvedA7|AlkAg686673NelarabineFDA approvedDs
85998StreptozocinFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
85998StreptozocinFDA approvedA7|AlkAg701852VorinostatFDA approvedHDAC
85998StreptozocinFDA approvedA7|AlkAg712807CapecitabineFDA approvedDs|TYMS
85998StreptozocinFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
85998StreptozocinFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
85998StreptozocinFDA approvedA7|AlkAg719276FulvestrantFDA approvedAM|Ho|ESR|SERM
85998StreptozocinFDA approvedA7|AlkAg719344AnastrozoleFDA approvedHo|CYP19A1
85998StreptozocinFDA approvedA7|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
85998StreptozocinFDA approvedA7|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
85998StreptozocinFDA approvedA7|AlkAg721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
85998StreptozocinFDA approvedA7|AlkAg732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
85998StreptozocinFDA approvedA7|AlkAg733504EverolimusFDA approvedPK:STK,MTOR
85998StreptozocinFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
85998StreptozocinFDA approvedA7|AlkAg743414ImatinibFDA approvedBCR-ABL|PK:YK
85998StreptozocinFDA approvedA7|AlkAg745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
85998StreptozocinFDA approvedA7|AlkAg747599NilotinibFDA approvedBCR-ABL|PK:YK
85998StreptozocinFDA approvedA7|AlkAg747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
85998StreptozocinFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
85998StreptozocinFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
85998StreptozocinFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
85998StreptozocinFDA approvedA7|AlkAg750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
85998StreptozocinFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
85998StreptozocinFDA approvedA7|AlkAg754143RomidepsinFDA approvedHDAC
85998StreptozocinFDA approvedA7|AlkAg754230PralatrexateFDA approvedDf|CTNNB1|DHFR
85998StreptozocinFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
85998StreptozocinFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
85998StreptozocinFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
85998StreptozocinFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
85998StreptozocinFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
85998StreptozocinFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
92859Trisenox 3FDA approvedApo740MethotrexateFDA approvedDf|DHFR
92859Trisenox 3FDA approvedApo750BusulfanFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo752ThioguanineFDA approvedDs|IMPDH2|IMPDH
92859Trisenox 3FDA approvedApo7556-MercaptopurineFDA approvedDs|PPAT
92859Trisenox 3FDA approvedApo762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo1390AllopurinolFDA approvedAM|XDH
92859Trisenox 3FDA approvedApo3053DactinomycinFDA approvedDb|RNA polymerase I
92859Trisenox 3FDA approvedApo3088ChlorambucilFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo6396ThiotepaFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo8806MelphalanFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo9706Triethylenemelamine-A7|AlkAg
92859Trisenox 3FDA approvedApo13875HexamethylmelamineFDA approvedDb|AlkAg
92859Trisenox 3FDA approvedApo14229QuinacrineClinical trialDb|AP
92859Trisenox 3FDA approvedApo18509Aminolevulinic Acid HydrochlorideFDA approvedAM
92859Trisenox 3FDA approvedApo19893FluorouracilFDA approvedDs|Rs|TYMS
92859Trisenox 3FDA approvedApo24559MithramycinFDA approvedDb|Rs
92859Trisenox 3FDA approvedApo25154PipobromanFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo26271CyclophosphamideFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo26980MitomycinFDA approvedA2|AlkAg
92859Trisenox 3FDA approvedApo27640FloxuridineFDA approvedDs|TYMS
92859Trisenox 3FDA approvedApo32065HydroxyureaFDA approvedAM|Dr
92859Trisenox 3FDA approvedApo34462Uracil mustardFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
92859Trisenox 3FDA approvedApo45388DacarbazineFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo459238-MethoxypsoralenFDA approvedDb
92859Trisenox 3FDA approvedApo49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
92859Trisenox 3FDA approvedApo63878Cytarabine hydrochlorideFDA approvedDs
92859Trisenox 3FDA approvedApo66847ThalidomideFDA approvedAng|Immunomodulatory
92859Trisenox 3FDA approvedApo67574Vincristine sulfateFDA approvedTUBB|Tu-frag
92859Trisenox 3FDA approvedApo71423Megestrol acetateFDA approvedHo|PGR
92859Trisenox 3FDA approvedApo77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo79037LomustineFDA approvedA6|AlkAg
92859Trisenox 3FDA approvedApo82151Daunorubicin hydrochlorideFDA approvedTOP2
92859Trisenox 3FDA approvedApo85998StreptozocinFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo102816AzacitidineFDA approvedDNMT
92859Trisenox 3FDA approvedApo105014CladribineFDA approvedDs|ADA
92859Trisenox 3FDA approvedApo109724IfosfamideFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
92859Trisenox 3FDA approvedApo119875CisplatinFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo122758TretinoinFDA approvedHo|RXR|Differentiator
92859Trisenox 3FDA approvedApo122819TeniposideFDA approvedTOP2
92859Trisenox 3FDA approvedApo123127Doxorubicin hydrochlorideFDA approvedTOP2
92859Trisenox 3FDA approvedApo125066BleomycinFDA approvedDb
92859Trisenox 3FDA approvedApo125973PaclitaxelFDA approvedTUBB|Tu-stab
92859Trisenox 3FDA approvedApo127716DecitabineFDA approvedAM|DNMT
92859Trisenox 3FDA approvedApo138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
92859Trisenox 3FDA approvedApo141540EtoposideFDA approvedTOP2
92859Trisenox 3FDA approvedApo169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
92859Trisenox 3FDA approvedApo180973Tamoxifen citrateFDA approvedHo|SERM
92859Trisenox 3FDA approvedApo218321PentostatinFDA approvedDs|AM|ADA
92859Trisenox 3FDA approvedApo226080RapamycinFDA approvedPK:STK,MTOR
92859Trisenox 3FDA approvedApo241240CarboplatinFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo246131ValrubicinFDA approvedTOP2
92859Trisenox 3FDA approvedApo266046OxaliplatinFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo279836MitoxantroneFDA approvedTOP2
92859Trisenox 3FDA approvedApo296961EthiofosFDA approvedRP
92859Trisenox 3FDA approvedApo362856TemozolomideFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod
92859Trisenox 3FDA approvedApo409962CarmustineFDA approvedA7|AlkAg
92859Trisenox 3FDA approvedApo606869ClofarabineFDA approvedDs
92859Trisenox 3FDA approvedApo608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
92859Trisenox 3FDA approvedApo609699Topotecan hydrochlorideFDA approvedTOP1
92859Trisenox 3FDA approvedApo613327Gemcitabine HCLFDA approvedDs
92859Trisenox 3FDA approvedApo628503DocetaxelFDA approvedTUBB|Tu-stab
92859Trisenox 3FDA approvedApo673596SN 38Clinical trialTOP1
92859Trisenox 3FDA approvedApo681239Proscript boronic acidFDA approvedPSM
92859Trisenox 3FDA approvedApo686673NelarabineFDA approvedDs
92859Trisenox 3FDA approvedApo698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
92859Trisenox 3FDA approvedApo701852VorinostatFDA approvedHDAC
92859Trisenox 3FDA approvedApo702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg
92859Trisenox 3FDA approvedApo712807CapecitabineFDA approvedDs|TYMS
92859Trisenox 3FDA approvedApo713563ExemestaneFDA approvedHo|CYP19A1
92859Trisenox 3FDA approvedApo715055GefitinibFDA approvedPK:YK,EGFR
92859Trisenox 3FDA approvedApo718781Erlotinib HCLFDA approvedPK:YK,EGFR
92859Trisenox 3FDA approvedApo719276FulvestrantFDA approvedAM|Ho|ESR|SERM
92859Trisenox 3FDA approvedApo719344AnastrozoleFDA approvedHo|CYP19A1
92859Trisenox 3FDA approvedApo719345LetrozoleFDA approvedHo|CYP19A1
92859Trisenox 3FDA approvedApo719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
92859Trisenox 3FDA approvedApo721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
92859Trisenox 3FDA approvedApo732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
92859Trisenox 3FDA approvedApo733504EverolimusFDA approvedPK:STK,MTOR
92859Trisenox 3FDA approvedApo737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
92859Trisenox 3FDA approvedApo743414ImatinibFDA approvedBCR-ABL|PK:YK
92859Trisenox 3FDA approvedApo745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
92859Trisenox 3FDA approvedApo747599NilotinibFDA approvedBCR-ABL|PK:YK
92859Trisenox 3FDA approvedApo747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
92859Trisenox 3FDA approvedApo747972LenalidomideFDA approvedFT|Immunomodulatory
92859Trisenox 3FDA approvedApo747973IxabepiloneFDA approvedTUBB|Tu-stab
92859Trisenox 3FDA approvedApo747974RaloxifeneFDA approvedHo|SERM
92859Trisenox 3FDA approvedApo749226AbirateroneFDA approvedHo|CYP17A1
92859Trisenox 3FDA approvedApo750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
92859Trisenox 3FDA approvedApo753082VemurafenibFDA approvedPK:YK,BRAF
92859Trisenox 3FDA approvedApo754143RomidepsinFDA approvedHDAC
92859Trisenox 3FDA approvedApo754230PralatrexateFDA approvedDf|CTNNB1|DHFR
92859Trisenox 3FDA approvedApo755986VismodegibFDA approvedSMO|PK:YK
92859Trisenox 3FDA approvedApo756645CrizotinibFDA approvedPK:YK,MET,ALK
92859Trisenox 3FDA approvedApo757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
92859Trisenox 3FDA approvedApo760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
92859Trisenox 3FDA approvedApo761432CabazitaxelFDA approvedTUBB|Tu-stab
92859Trisenox 3FDA approvedApo763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
102816AzacitidineFDA approvedDNMT752ThioguanineFDA approvedDs|IMPDH2|IMPDH
102816AzacitidineFDA approvedDNMT3053DactinomycinFDA approvedDb|RNA polymerase I
102816AzacitidineFDA approvedDNMT3088ChlorambucilFDA approvedA7|AlkAg
102816AzacitidineFDA approvedDNMT6396ThiotepaFDA approvedA7|AlkAg
102816AzacitidineFDA approvedDNMT8806MelphalanFDA approvedA7|AlkAg
102816AzacitidineFDA approvedDNMT13875HexamethylmelamineFDA approvedDb|AlkAg
102816AzacitidineFDA approvedDNMT19893FluorouracilFDA approvedDs|Rs|TYMS
102816AzacitidineFDA approvedDNMT27640FloxuridineFDA approvedDs|TYMS
102816AzacitidineFDA approvedDNMT34462Uracil mustardFDA approvedA7|AlkAg
102816AzacitidineFDA approvedDNMT45388DacarbazineFDA approvedA7|AlkAg
102816AzacitidineFDA approvedDNMT49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
102816AzacitidineFDA approvedDNMT63878Cytarabine hydrochlorideFDA approvedDs
102816AzacitidineFDA approvedDNMT67574Vincristine sulfateFDA approvedTUBB|Tu-frag
102816AzacitidineFDA approvedDNMT71423Megestrol acetateFDA approvedHo|PGR
102816AzacitidineFDA approvedDNMT79037LomustineFDA approvedA6|AlkAg
102816AzacitidineFDA approvedDNMT82151Daunorubicin hydrochlorideFDA approvedTOP2
102816AzacitidineFDA approvedDNMT105014CladribineFDA approvedDs|ADA
102816AzacitidineFDA approvedDNMT118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
102816AzacitidineFDA approvedDNMT122758TretinoinFDA approvedHo|RXR|Differentiator
102816AzacitidineFDA approvedDNMT122819TeniposideFDA approvedTOP2
102816AzacitidineFDA approvedDNMT125973PaclitaxelFDA approvedTUBB|Tu-stab
102816AzacitidineFDA approvedDNMT141540EtoposideFDA approvedTOP2
102816AzacitidineFDA approvedDNMT169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
102816AzacitidineFDA approvedDNMT180973Tamoxifen citrateFDA approvedHo|SERM
102816AzacitidineFDA approvedDNMT226080RapamycinFDA approvedPK:STK,MTOR
102816AzacitidineFDA approvedDNMT241240CarboplatinFDA approvedA7|AlkAg
102816AzacitidineFDA approvedDNMT246131ValrubicinFDA approvedTOP2
102816AzacitidineFDA approvedDNMT279836MitoxantroneFDA approvedTOP2
102816AzacitidineFDA approvedDNMT362856TemozolomideFDA approvedA7|AlkAg
102816AzacitidineFDA approvedDNMT606869ClofarabineFDA approvedDs
102816AzacitidineFDA approvedDNMT608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
102816AzacitidineFDA approvedDNMT613327Gemcitabine HCLFDA approvedDs
102816AzacitidineFDA approvedDNMT628503DocetaxelFDA approvedTUBB|Tu-stab
102816AzacitidineFDA approvedDNMT673596SN 38Clinical trialTOP1
102816AzacitidineFDA approvedDNMT686673NelarabineFDA approvedDs
102816AzacitidineFDA approvedDNMT698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
102816AzacitidineFDA approvedDNMT712807CapecitabineFDA approvedDs|TYMS
102816AzacitidineFDA approvedDNMT713563ExemestaneFDA approvedHo|CYP19A1
102816AzacitidineFDA approvedDNMT715055GefitinibFDA approvedPK:YK,EGFR
102816AzacitidineFDA approvedDNMT719276FulvestrantFDA approvedAM|Ho|ESR|SERM
102816AzacitidineFDA approvedDNMT719344AnastrozoleFDA approvedHo|CYP19A1
102816AzacitidineFDA approvedDNMT719345LetrozoleFDA approvedHo|CYP19A1
102816AzacitidineFDA approvedDNMT719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
102816AzacitidineFDA approvedDNMT737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
102816AzacitidineFDA approvedDNMT743414ImatinibFDA approvedBCR-ABL|PK:YK
102816AzacitidineFDA approvedDNMT747599NilotinibFDA approvedBCR-ABL|PK:YK
102816AzacitidineFDA approvedDNMT747972LenalidomideFDA approvedFT|Immunomodulatory
102816AzacitidineFDA approvedDNMT747974RaloxifeneFDA approvedHo|SERM
102816AzacitidineFDA approvedDNMT749226AbirateroneFDA approvedHo|CYP17A1
102816AzacitidineFDA approvedDNMT753082VemurafenibFDA approvedPK:YK,BRAF
102816AzacitidineFDA approvedDNMT754143RomidepsinFDA approvedHDAC
102816AzacitidineFDA approvedDNMT755986VismodegibFDA approvedSMO|PK:YK
102816AzacitidineFDA approvedDNMT756645CrizotinibFDA approvedPK:YK,MET,ALK
102816AzacitidineFDA approvedDNMT757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
102816AzacitidineFDA approvedDNMT760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
102816AzacitidineFDA approvedDNMT761432CabazitaxelFDA approvedTUBB|Tu-stab
102816AzacitidineFDA approvedDNMT763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
105014CladribineFDA approvedDs|ADA740MethotrexateFDA approvedDf|DHFR
105014CladribineFDA approvedDs|ADA752ThioguanineFDA approvedDs|IMPDH2|IMPDH
105014CladribineFDA approvedDs|ADA3053DactinomycinFDA approvedDb|RNA polymerase I
105014CladribineFDA approvedDs|ADA3088ChlorambucilFDA approvedA7|AlkAg
105014CladribineFDA approvedDs|ADA6396ThiotepaFDA approvedA7|AlkAg
105014CladribineFDA approvedDs|ADA8806MelphalanFDA approvedA7|AlkAg
105014CladribineFDA approvedDs|ADA13875HexamethylmelamineFDA approvedDb|AlkAg
105014CladribineFDA approvedDs|ADA19893FluorouracilFDA approvedDs|Rs|TYMS
105014CladribineFDA approvedDs|ADA27640FloxuridineFDA approvedDs|TYMS
105014CladribineFDA approvedDs|ADA34462Uracil mustardFDA approvedA7|AlkAg
105014CladribineFDA approvedDs|ADA45388DacarbazineFDA approvedA7|AlkAg
105014CladribineFDA approvedDs|ADA63878Cytarabine hydrochlorideFDA approvedDs
105014CladribineFDA approvedDs|ADA67574Vincristine sulfateFDA approvedTUBB|Tu-frag
105014CladribineFDA approvedDs|ADA71423Megestrol acetateFDA approvedHo|PGR
105014CladribineFDA approvedDs|ADA79037LomustineFDA approvedA6|AlkAg
105014CladribineFDA approvedDs|ADA82151Daunorubicin hydrochlorideFDA approvedTOP2
105014CladribineFDA approvedDs|ADA122819TeniposideFDA approvedTOP2
105014CladribineFDA approvedDs|ADA141540EtoposideFDA approvedTOP2
105014CladribineFDA approvedDs|ADA169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
105014CladribineFDA approvedDs|ADA279836MitoxantroneFDA approvedTOP2
105014CladribineFDA approvedDs|ADA608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
105014CladribineFDA approvedDs|ADA698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
105014CladribineFDA approvedDs|ADA713563ExemestaneFDA approvedHo|CYP19A1
105014CladribineFDA approvedDs|ADA715055GefitinibFDA approvedPK:YK,EGFR
105014CladribineFDA approvedDs|ADA719345LetrozoleFDA approvedHo|CYP19A1
105014CladribineFDA approvedDs|ADA719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
105014CladribineFDA approvedDs|ADA737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
105014CladribineFDA approvedDs|ADA747972LenalidomideFDA approvedFT|Immunomodulatory
105014CladribineFDA approvedDs|ADA747974RaloxifeneFDA approvedHo|SERM
105014CladribineFDA approvedDs|ADA749226AbirateroneFDA approvedHo|CYP17A1
105014CladribineFDA approvedDs|ADA753082VemurafenibFDA approvedPK:YK,BRAF
105014CladribineFDA approvedDs|ADA755986VismodegibFDA approvedSMO|PK:YK
105014CladribineFDA approvedDs|ADA756645CrizotinibFDA approvedPK:YK,MET,ALK
105014CladribineFDA approvedDs|ADA757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
105014CladribineFDA approvedDs|ADA760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
105014CladribineFDA approvedDs|ADA761432CabazitaxelFDA approvedTUBB|Tu-stab
105014CladribineFDA approvedDs|ADA763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
109724IfosfamideFDA approvedA7|AlkAg740MethotrexateFDA approvedDf|DHFR
109724IfosfamideFDA approvedA7|AlkAg750BusulfanFDA approvedA7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
109724IfosfamideFDA approvedA7|AlkAg7556-MercaptopurineFDA approvedDs|PPAT
109724IfosfamideFDA approvedA7|AlkAg762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg1390AllopurinolFDA approvedAM|XDH
109724IfosfamideFDA approvedA7|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
109724IfosfamideFDA approvedA7|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg6396ThiotepaFDA approvedA7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg8806MelphalanFDA approvedA7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg9706Triethylenemelamine-A7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
109724IfosfamideFDA approvedA7|AlkAg14229QuinacrineClinical trialDb|AP
109724IfosfamideFDA approvedA7|AlkAg18509Aminolevulinic Acid HydrochlorideFDA approvedAM
109724IfosfamideFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
109724IfosfamideFDA approvedA7|AlkAg24559MithramycinFDA approvedDb|Rs
109724IfosfamideFDA approvedA7|AlkAg25154PipobromanFDA approvedA7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg26271CyclophosphamideFDA approvedA7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg26980MitomycinFDA approvedA2|AlkAg
109724IfosfamideFDA approvedA7|AlkAg27640FloxuridineFDA approvedDs|TYMS
109724IfosfamideFDA approvedA7|AlkAg32065HydroxyureaFDA approvedAM|Dr
109724IfosfamideFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
109724IfosfamideFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg459238-MethoxypsoralenFDA approvedDb
109724IfosfamideFDA approvedA7|AlkAg49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
109724IfosfamideFDA approvedA7|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
109724IfosfamideFDA approvedA7|AlkAg66847ThalidomideFDA approvedAng|Immunomodulatory
109724IfosfamideFDA approvedA7|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
109724IfosfamideFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
109724IfosfamideFDA approvedA7|AlkAg77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
109724IfosfamideFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
109724IfosfamideFDA approvedA7|AlkAg85998StreptozocinFDA approvedA7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg102816AzacitidineFDA approvedDNMT
109724IfosfamideFDA approvedA7|AlkAg105014CladribineFDA approvedDs|ADA
109724IfosfamideFDA approvedA7|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
109724IfosfamideFDA approvedA7|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
109724IfosfamideFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
109724IfosfamideFDA approvedA7|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
109724IfosfamideFDA approvedA7|AlkAg125066BleomycinFDA approvedDb
109724IfosfamideFDA approvedA7|AlkAg125973PaclitaxelFDA approvedTUBB|Tu-stab
109724IfosfamideFDA approvedA7|AlkAg138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
109724IfosfamideFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
109724IfosfamideFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
109724IfosfamideFDA approvedA7|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
109724IfosfamideFDA approvedA7|AlkAg226080RapamycinFDA approvedPK:STK,MTOR
109724IfosfamideFDA approvedA7|AlkAg241240CarboplatinFDA approvedA7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg246131ValrubicinFDA approvedTOP2
109724IfosfamideFDA approvedA7|AlkAg266046OxaliplatinFDA approvedA7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
109724IfosfamideFDA approvedA7|AlkAg362856TemozolomideFDA approvedA7|AlkAg
109724IfosfamideFDA approvedA7|AlkAg606869ClofarabineFDA approvedDs
109724IfosfamideFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
109724IfosfamideFDA approvedA7|AlkAg613327Gemcitabine HCLFDA approvedDs
109724IfosfamideFDA approvedA7|AlkAg628503DocetaxelFDA approvedTUBB|Tu-stab
109724IfosfamideFDA approvedA7|AlkAg673596SN 38Clinical trialTOP1
109724IfosfamideFDA approvedA7|AlkAg686673NelarabineFDA approvedDs
109724IfosfamideFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
109724IfosfamideFDA approvedA7|AlkAg701852VorinostatFDA approvedHDAC
109724IfosfamideFDA approvedA7|AlkAg712807CapecitabineFDA approvedDs|TYMS
109724IfosfamideFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
109724IfosfamideFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
109724IfosfamideFDA approvedA7|AlkAg719276FulvestrantFDA approvedAM|Ho|ESR|SERM
109724IfosfamideFDA approvedA7|AlkAg719344AnastrozoleFDA approvedHo|CYP19A1
109724IfosfamideFDA approvedA7|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
109724IfosfamideFDA approvedA7|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
109724IfosfamideFDA approvedA7|AlkAg721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
109724IfosfamideFDA approvedA7|AlkAg732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
109724IfosfamideFDA approvedA7|AlkAg733504EverolimusFDA approvedPK:STK,MTOR
109724IfosfamideFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
109724IfosfamideFDA approvedA7|AlkAg743414ImatinibFDA approvedBCR-ABL|PK:YK
109724IfosfamideFDA approvedA7|AlkAg745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
109724IfosfamideFDA approvedA7|AlkAg747599NilotinibFDA approvedBCR-ABL|PK:YK
109724IfosfamideFDA approvedA7|AlkAg747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
109724IfosfamideFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
109724IfosfamideFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
109724IfosfamideFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
109724IfosfamideFDA approvedA7|AlkAg750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
109724IfosfamideFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
109724IfosfamideFDA approvedA7|AlkAg754143RomidepsinFDA approvedHDAC
109724IfosfamideFDA approvedA7|AlkAg754230PralatrexateFDA approvedDf|CTNNB1|DHFR
109724IfosfamideFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
109724IfosfamideFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
109724IfosfamideFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
109724IfosfamideFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
109724IfosfamideFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
109724IfosfamideFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1740MethotrexateFDA approvedDf|DHFR
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1752ThioguanineFDA approvedDs|IMPDH2|IMPDH
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT13053DactinomycinFDA approvedDb|RNA polymerase I
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT13088ChlorambucilFDA approvedA7|AlkAg
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT16396ThiotepaFDA approvedA7|AlkAg
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT18806MelphalanFDA approvedA7|AlkAg
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT113875HexamethylmelamineFDA approvedDb|AlkAg
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT119893FluorouracilFDA approvedDs|Rs|TYMS
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT127640FloxuridineFDA approvedDs|TYMS
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT134462Uracil mustardFDA approvedA7|AlkAg
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT145388DacarbazineFDA approvedA7|AlkAg
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT163878Cytarabine hydrochlorideFDA approvedDs
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT167574Vincristine sulfateFDA approvedTUBB|Tu-frag
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT171423Megestrol acetateFDA approvedHo|PGR
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT179037LomustineFDA approvedA6|AlkAg
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT182151Daunorubicin hydrochlorideFDA approvedTOP2
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1105014CladribineFDA approvedDs|ADA
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1122819TeniposideFDA approvedTOP2
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1141540EtoposideFDA approvedTOP2
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1279836MitoxantroneFDA approvedTOP2
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1713563ExemestaneFDA approvedHo|CYP19A1
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1715055GefitinibFDA approvedPK:YK,EGFR
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1719345LetrozoleFDA approvedHo|CYP19A1
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1747972LenalidomideFDA approvedFT|Immunomodulatory
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1747974RaloxifeneFDA approvedHo|SERM
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1749226AbirateroneFDA approvedHo|CYP17A1
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1753082VemurafenibFDA approvedPK:YK,BRAF
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1755986VismodegibFDA approvedSMO|PK:YK
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1756645CrizotinibFDA approvedPK:YK,MET,ALK
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1761432CabazitaxelFDA approvedTUBB|Tu-stab
118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
119875CisplatinFDA approvedA7|AlkAg740MethotrexateFDA approvedDf|DHFR
119875CisplatinFDA approvedA7|AlkAg750BusulfanFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
119875CisplatinFDA approvedA7|AlkAg7556-MercaptopurineFDA approvedDs|PPAT
119875CisplatinFDA approvedA7|AlkAg762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg1390AllopurinolFDA approvedAM|XDH
119875CisplatinFDA approvedA7|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
119875CisplatinFDA approvedA7|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg6396ThiotepaFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg8806MelphalanFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg9706Triethylenemelamine-A7|AlkAg
119875CisplatinFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
119875CisplatinFDA approvedA7|AlkAg14229QuinacrineClinical trialDb|AP
119875CisplatinFDA approvedA7|AlkAg18509Aminolevulinic Acid HydrochlorideFDA approvedAM
119875CisplatinFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
119875CisplatinFDA approvedA7|AlkAg24559MithramycinFDA approvedDb|Rs
119875CisplatinFDA approvedA7|AlkAg25154PipobromanFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg26271CyclophosphamideFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg26980MitomycinFDA approvedA2|AlkAg
119875CisplatinFDA approvedA7|AlkAg27640FloxuridineFDA approvedDs|TYMS
119875CisplatinFDA approvedA7|AlkAg32065HydroxyureaFDA approvedAM|Dr
119875CisplatinFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
119875CisplatinFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg459238-MethoxypsoralenFDA approvedDb
119875CisplatinFDA approvedA7|AlkAg49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
119875CisplatinFDA approvedA7|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
119875CisplatinFDA approvedA7|AlkAg66847ThalidomideFDA approvedAng|Immunomodulatory
119875CisplatinFDA approvedA7|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
119875CisplatinFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
119875CisplatinFDA approvedA7|AlkAg77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
119875CisplatinFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
119875CisplatinFDA approvedA7|AlkAg85998StreptozocinFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg102816AzacitidineFDA approvedDNMT
119875CisplatinFDA approvedA7|AlkAg105014CladribineFDA approvedDs|ADA
119875CisplatinFDA approvedA7|AlkAg109724IfosfamideFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
119875CisplatinFDA approvedA7|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
119875CisplatinFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
119875CisplatinFDA approvedA7|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
119875CisplatinFDA approvedA7|AlkAg125066BleomycinFDA approvedDb
119875CisplatinFDA approvedA7|AlkAg125973PaclitaxelFDA approvedTUBB|Tu-stab
119875CisplatinFDA approvedA7|AlkAg127716DecitabineFDA approvedAM|DNMT
119875CisplatinFDA approvedA7|AlkAg138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
119875CisplatinFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
119875CisplatinFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
119875CisplatinFDA approvedA7|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
119875CisplatinFDA approvedA7|AlkAg218321PentostatinFDA approvedDs|AM|ADA
119875CisplatinFDA approvedA7|AlkAg226080RapamycinFDA approvedPK:STK,MTOR
119875CisplatinFDA approvedA7|AlkAg241240CarboplatinFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg246131ValrubicinFDA approvedTOP2
119875CisplatinFDA approvedA7|AlkAg266046OxaliplatinFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
119875CisplatinFDA approvedA7|AlkAg296961EthiofosFDA approvedRP
119875CisplatinFDA approvedA7|AlkAg362856TemozolomideFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod
119875CisplatinFDA approvedA7|AlkAg409962CarmustineFDA approvedA7|AlkAg
119875CisplatinFDA approvedA7|AlkAg606869ClofarabineFDA approvedDs
119875CisplatinFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
119875CisplatinFDA approvedA7|AlkAg609699Topotecan hydrochlorideFDA approvedTOP1
119875CisplatinFDA approvedA7|AlkAg613327Gemcitabine HCLFDA approvedDs
119875CisplatinFDA approvedA7|AlkAg628503DocetaxelFDA approvedTUBB|Tu-stab
119875CisplatinFDA approvedA7|AlkAg673596SN 38Clinical trialTOP1
119875CisplatinFDA approvedA7|AlkAg681239Proscript boronic acidFDA approvedPSM
119875CisplatinFDA approvedA7|AlkAg686673NelarabineFDA approvedDs
119875CisplatinFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
119875CisplatinFDA approvedA7|AlkAg701852VorinostatFDA approvedHDAC
119875CisplatinFDA approvedA7|AlkAg702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg
119875CisplatinFDA approvedA7|AlkAg712807CapecitabineFDA approvedDs|TYMS
119875CisplatinFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
119875CisplatinFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
119875CisplatinFDA approvedA7|AlkAg718781Erlotinib HCLFDA approvedPK:YK,EGFR
119875CisplatinFDA approvedA7|AlkAg719276FulvestrantFDA approvedAM|Ho|ESR|SERM
119875CisplatinFDA approvedA7|AlkAg719344AnastrozoleFDA approvedHo|CYP19A1
119875CisplatinFDA approvedA7|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
119875CisplatinFDA approvedA7|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
119875CisplatinFDA approvedA7|AlkAg721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
119875CisplatinFDA approvedA7|AlkAg732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
119875CisplatinFDA approvedA7|AlkAg733504EverolimusFDA approvedPK:STK,MTOR
119875CisplatinFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
119875CisplatinFDA approvedA7|AlkAg743414ImatinibFDA approvedBCR-ABL|PK:YK
119875CisplatinFDA approvedA7|AlkAg745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
119875CisplatinFDA approvedA7|AlkAg747599NilotinibFDA approvedBCR-ABL|PK:YK
119875CisplatinFDA approvedA7|AlkAg747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
119875CisplatinFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
119875CisplatinFDA approvedA7|AlkAg747973IxabepiloneFDA approvedTUBB|Tu-stab
119875CisplatinFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
119875CisplatinFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
119875CisplatinFDA approvedA7|AlkAg750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
119875CisplatinFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
119875CisplatinFDA approvedA7|AlkAg754143RomidepsinFDA approvedHDAC
119875CisplatinFDA approvedA7|AlkAg754230PralatrexateFDA approvedDf|CTNNB1|DHFR
119875CisplatinFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
119875CisplatinFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
119875CisplatinFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
119875CisplatinFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
119875CisplatinFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
119875CisplatinFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
122758TretinoinFDA approvedHo|RXR|Differentiator740MethotrexateFDA approvedDf|DHFR
122758TretinoinFDA approvedHo|RXR|Differentiator752ThioguanineFDA approvedDs|IMPDH2|IMPDH
122758TretinoinFDA approvedHo|RXR|Differentiator3053DactinomycinFDA approvedDb|RNA polymerase I
122758TretinoinFDA approvedHo|RXR|Differentiator3088ChlorambucilFDA approvedA7|AlkAg
122758TretinoinFDA approvedHo|RXR|Differentiator6396ThiotepaFDA approvedA7|AlkAg
122758TretinoinFDA approvedHo|RXR|Differentiator8806MelphalanFDA approvedA7|AlkAg
122758TretinoinFDA approvedHo|RXR|Differentiator13875HexamethylmelamineFDA approvedDb|AlkAg
122758TretinoinFDA approvedHo|RXR|Differentiator19893FluorouracilFDA approvedDs|Rs|TYMS
122758TretinoinFDA approvedHo|RXR|Differentiator27640FloxuridineFDA approvedDs|TYMS
122758TretinoinFDA approvedHo|RXR|Differentiator34462Uracil mustardFDA approvedA7|AlkAg
122758TretinoinFDA approvedHo|RXR|Differentiator45388DacarbazineFDA approvedA7|AlkAg
122758TretinoinFDA approvedHo|RXR|Differentiator63878Cytarabine hydrochlorideFDA approvedDs
122758TretinoinFDA approvedHo|RXR|Differentiator67574Vincristine sulfateFDA approvedTUBB|Tu-frag
122758TretinoinFDA approvedHo|RXR|Differentiator71423Megestrol acetateFDA approvedHo|PGR
122758TretinoinFDA approvedHo|RXR|Differentiator79037LomustineFDA approvedA6|AlkAg
122758TretinoinFDA approvedHo|RXR|Differentiator82151Daunorubicin hydrochlorideFDA approvedTOP2
122758TretinoinFDA approvedHo|RXR|Differentiator105014CladribineFDA approvedDs|ADA
122758TretinoinFDA approvedHo|RXR|Differentiator118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
122758TretinoinFDA approvedHo|RXR|Differentiator122819TeniposideFDA approvedTOP2
122758TretinoinFDA approvedHo|RXR|Differentiator141540EtoposideFDA approvedTOP2
122758TretinoinFDA approvedHo|RXR|Differentiator169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
122758TretinoinFDA approvedHo|RXR|Differentiator279836MitoxantroneFDA approvedTOP2
122758TretinoinFDA approvedHo|RXR|Differentiator608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
122758TretinoinFDA approvedHo|RXR|Differentiator698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
122758TretinoinFDA approvedHo|RXR|Differentiator713563ExemestaneFDA approvedHo|CYP19A1
122758TretinoinFDA approvedHo|RXR|Differentiator715055GefitinibFDA approvedPK:YK,EGFR
122758TretinoinFDA approvedHo|RXR|Differentiator719345LetrozoleFDA approvedHo|CYP19A1
122758TretinoinFDA approvedHo|RXR|Differentiator719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
122758TretinoinFDA approvedHo|RXR|Differentiator737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
122758TretinoinFDA approvedHo|RXR|Differentiator747972LenalidomideFDA approvedFT|Immunomodulatory
122758TretinoinFDA approvedHo|RXR|Differentiator747974RaloxifeneFDA approvedHo|SERM
122758TretinoinFDA approvedHo|RXR|Differentiator749226AbirateroneFDA approvedHo|CYP17A1
122758TretinoinFDA approvedHo|RXR|Differentiator753082VemurafenibFDA approvedPK:YK,BRAF
122758TretinoinFDA approvedHo|RXR|Differentiator755986VismodegibFDA approvedSMO|PK:YK
122758TretinoinFDA approvedHo|RXR|Differentiator756645CrizotinibFDA approvedPK:YK,MET,ALK
122758TretinoinFDA approvedHo|RXR|Differentiator757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
122758TretinoinFDA approvedHo|RXR|Differentiator760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
122758TretinoinFDA approvedHo|RXR|Differentiator761432CabazitaxelFDA approvedTUBB|Tu-stab
122758TretinoinFDA approvedHo|RXR|Differentiator763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
122819TeniposideFDA approvedTOP29706Triethylenemelamine-A7|AlkAg
122819TeniposideFDA approvedTOP2123127Doxorubicin hydrochlorideFDA approvedTOP2
122819TeniposideFDA approvedTOP2141540EtoposideFDA approvedTOP2
122819TeniposideFDA approvedTOP2169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
122819TeniposideFDA approvedTOP2279836MitoxantroneFDA approvedTOP2
122819TeniposideFDA approvedTOP2608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
122819TeniposideFDA approvedTOP2698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
122819TeniposideFDA approvedTOP2713563ExemestaneFDA approvedHo|CYP19A1
122819TeniposideFDA approvedTOP2715055GefitinibFDA approvedPK:YK,EGFR
122819TeniposideFDA approvedTOP2737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
122819TeniposideFDA approvedTOP2747972LenalidomideFDA approvedFT|Immunomodulatory
122819TeniposideFDA approvedTOP2747974RaloxifeneFDA approvedHo|SERM
122819TeniposideFDA approvedTOP2749226AbirateroneFDA approvedHo|CYP17A1
122819TeniposideFDA approvedTOP2753082VemurafenibFDA approvedPK:YK,BRAF
122819TeniposideFDA approvedTOP2755986VismodegibFDA approvedSMO|PK:YK
122819TeniposideFDA approvedTOP2756645CrizotinibFDA approvedPK:YK,MET,ALK
122819TeniposideFDA approvedTOP2757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
122819TeniposideFDA approvedTOP2760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
122819TeniposideFDA approvedTOP2761432CabazitaxelFDA approvedTUBB|Tu-stab
122819TeniposideFDA approvedTOP2763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
123127Doxorubicin hydrochlorideFDA approvedTOP23053DactinomycinFDA approvedDb|RNA polymerase I
123127Doxorubicin hydrochlorideFDA approvedTOP26396ThiotepaFDA approvedA7|AlkAg
123127Doxorubicin hydrochlorideFDA approvedTOP29706Triethylenemelamine-A7|AlkAg
123127Doxorubicin hydrochlorideFDA approvedTOP224559MithramycinFDA approvedDb|Rs
123127Doxorubicin hydrochlorideFDA approvedTOP227640FloxuridineFDA approvedDs|TYMS
123127Doxorubicin hydrochlorideFDA approvedTOP232065HydroxyureaFDA approvedAM|Dr
123127Doxorubicin hydrochlorideFDA approvedTOP263878Cytarabine hydrochlorideFDA approvedDs
123127Doxorubicin hydrochlorideFDA approvedTOP267574Vincristine sulfateFDA approvedTUBB|Tu-frag
123127Doxorubicin hydrochlorideFDA approvedTOP2102816AzacitidineFDA approvedDNMT
123127Doxorubicin hydrochlorideFDA approvedTOP2105014CladribineFDA approvedDs|ADA
123127Doxorubicin hydrochlorideFDA approvedTOP2118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
123127Doxorubicin hydrochlorideFDA approvedTOP2122758TretinoinFDA approvedHo|RXR|Differentiator
123127Doxorubicin hydrochlorideFDA approvedTOP2125973PaclitaxelFDA approvedTUBB|Tu-stab
123127Doxorubicin hydrochlorideFDA approvedTOP2138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
123127Doxorubicin hydrochlorideFDA approvedTOP2180973Tamoxifen citrateFDA approvedHo|SERM
123127Doxorubicin hydrochlorideFDA approvedTOP2226080RapamycinFDA approvedPK:STK,MTOR
123127Doxorubicin hydrochlorideFDA approvedTOP2241240CarboplatinFDA approvedA7|AlkAg
123127Doxorubicin hydrochlorideFDA approvedTOP2362856TemozolomideFDA approvedA7|AlkAg
123127Doxorubicin hydrochlorideFDA approvedTOP2606869ClofarabineFDA approvedDs
123127Doxorubicin hydrochlorideFDA approvedTOP2613327Gemcitabine HCLFDA approvedDs
123127Doxorubicin hydrochlorideFDA approvedTOP2628503DocetaxelFDA approvedTUBB|Tu-stab
123127Doxorubicin hydrochlorideFDA approvedTOP2673596SN 38Clinical trialTOP1
123127Doxorubicin hydrochlorideFDA approvedTOP2686673NelarabineFDA approvedDs
123127Doxorubicin hydrochlorideFDA approvedTOP2701852VorinostatFDA approvedHDAC
123127Doxorubicin hydrochlorideFDA approvedTOP2712807CapecitabineFDA approvedDs|TYMS
123127Doxorubicin hydrochlorideFDA approvedTOP2719345LetrozoleFDA approvedHo|CYP19A1
123127Doxorubicin hydrochlorideFDA approvedTOP2719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
123127Doxorubicin hydrochlorideFDA approvedTOP2721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
123127Doxorubicin hydrochlorideFDA approvedTOP2732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
123127Doxorubicin hydrochlorideFDA approvedTOP2733504EverolimusFDA approvedPK:STK,MTOR
123127Doxorubicin hydrochlorideFDA approvedTOP2743414ImatinibFDA approvedBCR-ABL|PK:YK
123127Doxorubicin hydrochlorideFDA approvedTOP2745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
123127Doxorubicin hydrochlorideFDA approvedTOP2747599NilotinibFDA approvedBCR-ABL|PK:YK
123127Doxorubicin hydrochlorideFDA approvedTOP2747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
123127Doxorubicin hydrochlorideFDA approvedTOP2750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
123127Doxorubicin hydrochlorideFDA approvedTOP2754143RomidepsinFDA approvedHDAC
123127Doxorubicin hydrochlorideFDA approvedTOP2754230PralatrexateFDA approvedDf|CTNNB1|DHFR
125066BleomycinFDA approvedDb752ThioguanineFDA approvedDs|IMPDH2|IMPDH
125066BleomycinFDA approvedDb3053DactinomycinFDA approvedDb|RNA polymerase I
125066BleomycinFDA approvedDb3088ChlorambucilFDA approvedA7|AlkAg
125066BleomycinFDA approvedDb6396ThiotepaFDA approvedA7|AlkAg
125066BleomycinFDA approvedDb8806MelphalanFDA approvedA7|AlkAg
125066BleomycinFDA approvedDb9706Triethylenemelamine-A7|AlkAg
125066BleomycinFDA approvedDb13875HexamethylmelamineFDA approvedDb|AlkAg
125066BleomycinFDA approvedDb19893FluorouracilFDA approvedDs|Rs|TYMS
125066BleomycinFDA approvedDb24559MithramycinFDA approvedDb|Rs
125066BleomycinFDA approvedDb27640FloxuridineFDA approvedDs|TYMS
125066BleomycinFDA approvedDb32065HydroxyureaFDA approvedAM|Dr
125066BleomycinFDA approvedDb34462Uracil mustardFDA approvedA7|AlkAg
125066BleomycinFDA approvedDb45388DacarbazineFDA approvedA7|AlkAg
125066BleomycinFDA approvedDb63878Cytarabine hydrochlorideFDA approvedDs
125066BleomycinFDA approvedDb67574Vincristine sulfateFDA approvedTUBB|Tu-frag
125066BleomycinFDA approvedDb71423Megestrol acetateFDA approvedHo|PGR
125066BleomycinFDA approvedDb79037LomustineFDA approvedA6|AlkAg
125066BleomycinFDA approvedDb82151Daunorubicin hydrochlorideFDA approvedTOP2
125066BleomycinFDA approvedDb102816AzacitidineFDA approvedDNMT
125066BleomycinFDA approvedDb105014CladribineFDA approvedDs|ADA
125066BleomycinFDA approvedDb118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
125066BleomycinFDA approvedDb122758TretinoinFDA approvedHo|RXR|Differentiator
125066BleomycinFDA approvedDb122819TeniposideFDA approvedTOP2
125066BleomycinFDA approvedDb123127Doxorubicin hydrochlorideFDA approvedTOP2
125066BleomycinFDA approvedDb125973PaclitaxelFDA approvedTUBB|Tu-stab
125066BleomycinFDA approvedDb141540EtoposideFDA approvedTOP2
125066BleomycinFDA approvedDb169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
125066BleomycinFDA approvedDb180973Tamoxifen citrateFDA approvedHo|SERM
125066BleomycinFDA approvedDb226080RapamycinFDA approvedPK:STK,MTOR
125066BleomycinFDA approvedDb241240CarboplatinFDA approvedA7|AlkAg
125066BleomycinFDA approvedDb279836MitoxantroneFDA approvedTOP2
125066BleomycinFDA approvedDb362856TemozolomideFDA approvedA7|AlkAg
125066BleomycinFDA approvedDb606869ClofarabineFDA approvedDs
125066BleomycinFDA approvedDb608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
125066BleomycinFDA approvedDb613327Gemcitabine HCLFDA approvedDs
125066BleomycinFDA approvedDb628503DocetaxelFDA approvedTUBB|Tu-stab
125066BleomycinFDA approvedDb673596SN 38Clinical trialTOP1
125066BleomycinFDA approvedDb686673NelarabineFDA approvedDs
125066BleomycinFDA approvedDb698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
125066BleomycinFDA approvedDb701852VorinostatFDA approvedHDAC
125066BleomycinFDA approvedDb712807CapecitabineFDA approvedDs|TYMS
125066BleomycinFDA approvedDb713563ExemestaneFDA approvedHo|CYP19A1
125066BleomycinFDA approvedDb715055GefitinibFDA approvedPK:YK,EGFR
125066BleomycinFDA approvedDb719345LetrozoleFDA approvedHo|CYP19A1
125066BleomycinFDA approvedDb719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
125066BleomycinFDA approvedDb721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
125066BleomycinFDA approvedDb732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
125066BleomycinFDA approvedDb733504EverolimusFDA approvedPK:STK,MTOR
125066BleomycinFDA approvedDb737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
125066BleomycinFDA approvedDb743414ImatinibFDA approvedBCR-ABL|PK:YK
125066BleomycinFDA approvedDb745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
125066BleomycinFDA approvedDb747599NilotinibFDA approvedBCR-ABL|PK:YK
125066BleomycinFDA approvedDb747972LenalidomideFDA approvedFT|Immunomodulatory
125066BleomycinFDA approvedDb747974RaloxifeneFDA approvedHo|SERM
125066BleomycinFDA approvedDb749226AbirateroneFDA approvedHo|CYP17A1
125066BleomycinFDA approvedDb750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
125066BleomycinFDA approvedDb753082VemurafenibFDA approvedPK:YK,BRAF
125066BleomycinFDA approvedDb754143RomidepsinFDA approvedHDAC
125066BleomycinFDA approvedDb755986VismodegibFDA approvedSMO|PK:YK
125066BleomycinFDA approvedDb756645CrizotinibFDA approvedPK:YK,MET,ALK
125066BleomycinFDA approvedDb757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
125066BleomycinFDA approvedDb760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
125066BleomycinFDA approvedDb761432CabazitaxelFDA approvedTUBB|Tu-stab
125066BleomycinFDA approvedDb763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
125973PaclitaxelFDA approvedTUBB|Tu-stab752ThioguanineFDA approvedDs|IMPDH2|IMPDH
125973PaclitaxelFDA approvedTUBB|Tu-stab3053DactinomycinFDA approvedDb|RNA polymerase I
125973PaclitaxelFDA approvedTUBB|Tu-stab3088ChlorambucilFDA approvedA7|AlkAg
125973PaclitaxelFDA approvedTUBB|Tu-stab6396ThiotepaFDA approvedA7|AlkAg
125973PaclitaxelFDA approvedTUBB|Tu-stab8806MelphalanFDA approvedA7|AlkAg
125973PaclitaxelFDA approvedTUBB|Tu-stab13875HexamethylmelamineFDA approvedDb|AlkAg
125973PaclitaxelFDA approvedTUBB|Tu-stab19893FluorouracilFDA approvedDs|Rs|TYMS
125973PaclitaxelFDA approvedTUBB|Tu-stab27640FloxuridineFDA approvedDs|TYMS
125973PaclitaxelFDA approvedTUBB|Tu-stab34462Uracil mustardFDA approvedA7|AlkAg
125973PaclitaxelFDA approvedTUBB|Tu-stab45388DacarbazineFDA approvedA7|AlkAg
125973PaclitaxelFDA approvedTUBB|Tu-stab63878Cytarabine hydrochlorideFDA approvedDs
125973PaclitaxelFDA approvedTUBB|Tu-stab67574Vincristine sulfateFDA approvedTUBB|Tu-frag
125973PaclitaxelFDA approvedTUBB|Tu-stab71423Megestrol acetateFDA approvedHo|PGR
125973PaclitaxelFDA approvedTUBB|Tu-stab79037LomustineFDA approvedA6|AlkAg
125973PaclitaxelFDA approvedTUBB|Tu-stab82151Daunorubicin hydrochlorideFDA approvedTOP2
125973PaclitaxelFDA approvedTUBB|Tu-stab105014CladribineFDA approvedDs|ADA
125973PaclitaxelFDA approvedTUBB|Tu-stab118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
125973PaclitaxelFDA approvedTUBB|Tu-stab122758TretinoinFDA approvedHo|RXR|Differentiator
125973PaclitaxelFDA approvedTUBB|Tu-stab122819TeniposideFDA approvedTOP2
125973PaclitaxelFDA approvedTUBB|Tu-stab141540EtoposideFDA approvedTOP2
125973PaclitaxelFDA approvedTUBB|Tu-stab169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
125973PaclitaxelFDA approvedTUBB|Tu-stab180973Tamoxifen citrateFDA approvedHo|SERM
125973PaclitaxelFDA approvedTUBB|Tu-stab226080RapamycinFDA approvedPK:STK,MTOR
125973PaclitaxelFDA approvedTUBB|Tu-stab241240CarboplatinFDA approvedA7|AlkAg
125973PaclitaxelFDA approvedTUBB|Tu-stab279836MitoxantroneFDA approvedTOP2
125973PaclitaxelFDA approvedTUBB|Tu-stab362856TemozolomideFDA approvedA7|AlkAg
125973PaclitaxelFDA approvedTUBB|Tu-stab606869ClofarabineFDA approvedDs
125973PaclitaxelFDA approvedTUBB|Tu-stab608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
125973PaclitaxelFDA approvedTUBB|Tu-stab613327Gemcitabine HCLFDA approvedDs
125973PaclitaxelFDA approvedTUBB|Tu-stab686673NelarabineFDA approvedDs
125973PaclitaxelFDA approvedTUBB|Tu-stab698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
125973PaclitaxelFDA approvedTUBB|Tu-stab712807CapecitabineFDA approvedDs|TYMS
125973PaclitaxelFDA approvedTUBB|Tu-stab713563ExemestaneFDA approvedHo|CYP19A1
125973PaclitaxelFDA approvedTUBB|Tu-stab715055GefitinibFDA approvedPK:YK,EGFR
125973PaclitaxelFDA approvedTUBB|Tu-stab719345LetrozoleFDA approvedHo|CYP19A1
125973PaclitaxelFDA approvedTUBB|Tu-stab719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
125973PaclitaxelFDA approvedTUBB|Tu-stab737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
125973PaclitaxelFDA approvedTUBB|Tu-stab743414ImatinibFDA approvedBCR-ABL|PK:YK
125973PaclitaxelFDA approvedTUBB|Tu-stab747599NilotinibFDA approvedBCR-ABL|PK:YK
125973PaclitaxelFDA approvedTUBB|Tu-stab747972LenalidomideFDA approvedFT|Immunomodulatory
125973PaclitaxelFDA approvedTUBB|Tu-stab747974RaloxifeneFDA approvedHo|SERM
125973PaclitaxelFDA approvedTUBB|Tu-stab749226AbirateroneFDA approvedHo|CYP17A1
125973PaclitaxelFDA approvedTUBB|Tu-stab753082VemurafenibFDA approvedPK:YK,BRAF
125973PaclitaxelFDA approvedTUBB|Tu-stab755986VismodegibFDA approvedSMO|PK:YK
125973PaclitaxelFDA approvedTUBB|Tu-stab756645CrizotinibFDA approvedPK:YK,MET,ALK
125973PaclitaxelFDA approvedTUBB|Tu-stab757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
125973PaclitaxelFDA approvedTUBB|Tu-stab760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
125973PaclitaxelFDA approvedTUBB|Tu-stab761432CabazitaxelFDA approvedTUBB|Tu-stab
125973PaclitaxelFDA approvedTUBB|Tu-stab763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
127716DecitabineFDA approvedAM|DNMT740MethotrexateFDA approvedDf|DHFR
127716DecitabineFDA approvedAM|DNMT750BusulfanFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT752ThioguanineFDA approvedDs|IMPDH2|IMPDH
127716DecitabineFDA approvedAM|DNMT7556-MercaptopurineFDA approvedDs|PPAT
127716DecitabineFDA approvedAM|DNMT762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT1390AllopurinolFDA approvedAM|XDH
127716DecitabineFDA approvedAM|DNMT3053DactinomycinFDA approvedDb|RNA polymerase I
127716DecitabineFDA approvedAM|DNMT3088ChlorambucilFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT6396ThiotepaFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT8806MelphalanFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT9706Triethylenemelamine-A7|AlkAg
127716DecitabineFDA approvedAM|DNMT13875HexamethylmelamineFDA approvedDb|AlkAg
127716DecitabineFDA approvedAM|DNMT14229QuinacrineClinical trialDb|AP
127716DecitabineFDA approvedAM|DNMT18509Aminolevulinic Acid HydrochlorideFDA approvedAM
127716DecitabineFDA approvedAM|DNMT19893FluorouracilFDA approvedDs|Rs|TYMS
127716DecitabineFDA approvedAM|DNMT24559MithramycinFDA approvedDb|Rs
127716DecitabineFDA approvedAM|DNMT25154PipobromanFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT26271CyclophosphamideFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT26980MitomycinFDA approvedA2|AlkAg
127716DecitabineFDA approvedAM|DNMT27640FloxuridineFDA approvedDs|TYMS
127716DecitabineFDA approvedAM|DNMT32065HydroxyureaFDA approvedAM|Dr
127716DecitabineFDA approvedAM|DNMT34462Uracil mustardFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
127716DecitabineFDA approvedAM|DNMT45388DacarbazineFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT459238-MethoxypsoralenFDA approvedDb
127716DecitabineFDA approvedAM|DNMT49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
127716DecitabineFDA approvedAM|DNMT63878Cytarabine hydrochlorideFDA approvedDs
127716DecitabineFDA approvedAM|DNMT66847ThalidomideFDA approvedAng|Immunomodulatory
127716DecitabineFDA approvedAM|DNMT67574Vincristine sulfateFDA approvedTUBB|Tu-frag
127716DecitabineFDA approvedAM|DNMT71423Megestrol acetateFDA approvedHo|PGR
127716DecitabineFDA approvedAM|DNMT77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT79037LomustineFDA approvedA6|AlkAg
127716DecitabineFDA approvedAM|DNMT82151Daunorubicin hydrochlorideFDA approvedTOP2
127716DecitabineFDA approvedAM|DNMT85998StreptozocinFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT102816AzacitidineFDA approvedDNMT
127716DecitabineFDA approvedAM|DNMT105014CladribineFDA approvedDs|ADA
127716DecitabineFDA approvedAM|DNMT109724IfosfamideFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
127716DecitabineFDA approvedAM|DNMT122758TretinoinFDA approvedHo|RXR|Differentiator
127716DecitabineFDA approvedAM|DNMT122819TeniposideFDA approvedTOP2
127716DecitabineFDA approvedAM|DNMT123127Doxorubicin hydrochlorideFDA approvedTOP2
127716DecitabineFDA approvedAM|DNMT125066BleomycinFDA approvedDb
127716DecitabineFDA approvedAM|DNMT125973PaclitaxelFDA approvedTUBB|Tu-stab
127716DecitabineFDA approvedAM|DNMT138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
127716DecitabineFDA approvedAM|DNMT141540EtoposideFDA approvedTOP2
127716DecitabineFDA approvedAM|DNMT169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
127716DecitabineFDA approvedAM|DNMT180973Tamoxifen citrateFDA approvedHo|SERM
127716DecitabineFDA approvedAM|DNMT218321PentostatinFDA approvedDs|AM|ADA
127716DecitabineFDA approvedAM|DNMT226080RapamycinFDA approvedPK:STK,MTOR
127716DecitabineFDA approvedAM|DNMT241240CarboplatinFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT246131ValrubicinFDA approvedTOP2
127716DecitabineFDA approvedAM|DNMT266046OxaliplatinFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT279836MitoxantroneFDA approvedTOP2
127716DecitabineFDA approvedAM|DNMT362856TemozolomideFDA approvedA7|AlkAg
127716DecitabineFDA approvedAM|DNMT369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod
127716DecitabineFDA approvedAM|DNMT606869ClofarabineFDA approvedDs
127716DecitabineFDA approvedAM|DNMT608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
127716DecitabineFDA approvedAM|DNMT609699Topotecan hydrochlorideFDA approvedTOP1
127716DecitabineFDA approvedAM|DNMT613327Gemcitabine HCLFDA approvedDs
127716DecitabineFDA approvedAM|DNMT628503DocetaxelFDA approvedTUBB|Tu-stab
127716DecitabineFDA approvedAM|DNMT673596SN 38Clinical trialTOP1
127716DecitabineFDA approvedAM|DNMT686673NelarabineFDA approvedDs
127716DecitabineFDA approvedAM|DNMT698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
127716DecitabineFDA approvedAM|DNMT701852VorinostatFDA approvedHDAC
127716DecitabineFDA approvedAM|DNMT712807CapecitabineFDA approvedDs|TYMS
127716DecitabineFDA approvedAM|DNMT713563ExemestaneFDA approvedHo|CYP19A1
127716DecitabineFDA approvedAM|DNMT715055GefitinibFDA approvedPK:YK,EGFR
127716DecitabineFDA approvedAM|DNMT719276FulvestrantFDA approvedAM|Ho|ESR|SERM
127716DecitabineFDA approvedAM|DNMT719344AnastrozoleFDA approvedHo|CYP19A1
127716DecitabineFDA approvedAM|DNMT719345LetrozoleFDA approvedHo|CYP19A1
127716DecitabineFDA approvedAM|DNMT719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
127716DecitabineFDA approvedAM|DNMT721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
127716DecitabineFDA approvedAM|DNMT732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
127716DecitabineFDA approvedAM|DNMT733504EverolimusFDA approvedPK:STK,MTOR
127716DecitabineFDA approvedAM|DNMT737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
127716DecitabineFDA approvedAM|DNMT743414ImatinibFDA approvedBCR-ABL|PK:YK
127716DecitabineFDA approvedAM|DNMT745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
127716DecitabineFDA approvedAM|DNMT747599NilotinibFDA approvedBCR-ABL|PK:YK
127716DecitabineFDA approvedAM|DNMT747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
127716DecitabineFDA approvedAM|DNMT747972LenalidomideFDA approvedFT|Immunomodulatory
127716DecitabineFDA approvedAM|DNMT747974RaloxifeneFDA approvedHo|SERM
127716DecitabineFDA approvedAM|DNMT749226AbirateroneFDA approvedHo|CYP17A1
127716DecitabineFDA approvedAM|DNMT750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
127716DecitabineFDA approvedAM|DNMT753082VemurafenibFDA approvedPK:YK,BRAF
127716DecitabineFDA approvedAM|DNMT754143RomidepsinFDA approvedHDAC
127716DecitabineFDA approvedAM|DNMT754230PralatrexateFDA approvedDf|CTNNB1|DHFR
127716DecitabineFDA approvedAM|DNMT755986VismodegibFDA approvedSMO|PK:YK
127716DecitabineFDA approvedAM|DNMT756645CrizotinibFDA approvedPK:YK,MET,ALK
127716DecitabineFDA approvedAM|DNMT757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
127716DecitabineFDA approvedAM|DNMT760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
127716DecitabineFDA approvedAM|DNMT761432CabazitaxelFDA approvedTUBB|Tu-stab
127716DecitabineFDA approvedAM|DNMT763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg6396ThiotepaFDA approvedA7|AlkAg
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg8806MelphalanFDA approvedA7|AlkAg
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg9706Triethylenemelamine-A7|AlkAg
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg24559MithramycinFDA approvedDb|Rs
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg27640FloxuridineFDA approvedDs|TYMS
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg32065HydroxyureaFDA approvedAM|Dr
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg45388DacarbazineFDA approvedA7|AlkAg
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg71423Megestrol acetateFDA approvedHo|PGR
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg79037LomustineFDA approvedA6|AlkAg
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg102816AzacitidineFDA approvedDNMT
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg105014CladribineFDA approvedDs|ADA
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg122819TeniposideFDA approvedTOP2
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg125066BleomycinFDA approvedDb
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg125973PaclitaxelFDA approvedTUBB|Tu-stab
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg141540EtoposideFDA approvedTOP2
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg241240CarboplatinFDA approvedA7|AlkAg
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg246131ValrubicinFDA approvedTOP2
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg279836MitoxantroneFDA approvedTOP2
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg362856TemozolomideFDA approvedA7|AlkAg
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg628503DocetaxelFDA approvedTUBB|Tu-stab
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg673596SN 38Clinical trialTOP1
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg701852VorinostatFDA approvedHDAC
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg733504EverolimusFDA approvedPK:STK,MTOR
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg743414ImatinibFDA approvedBCR-ABL|PK:YK
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg747974RaloxifeneFDA approvedHo|SERM
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg754143RomidepsinFDA approvedHDAC
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg755986VismodegibFDA approvedSMO|PK:YK
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
141540EtoposideFDA approvedTOP29706Triethylenemelamine-A7|AlkAg
141540EtoposideFDA approvedTOP2123127Doxorubicin hydrochlorideFDA approvedTOP2
141540EtoposideFDA approvedTOP2169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
141540EtoposideFDA approvedTOP2279836MitoxantroneFDA approvedTOP2
141540EtoposideFDA approvedTOP2608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
141540EtoposideFDA approvedTOP2698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
141540EtoposideFDA approvedTOP2713563ExemestaneFDA approvedHo|CYP19A1
141540EtoposideFDA approvedTOP2715055GefitinibFDA approvedPK:YK,EGFR
141540EtoposideFDA approvedTOP2737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
141540EtoposideFDA approvedTOP2747972LenalidomideFDA approvedFT|Immunomodulatory
141540EtoposideFDA approvedTOP2747974RaloxifeneFDA approvedHo|SERM
141540EtoposideFDA approvedTOP2749226AbirateroneFDA approvedHo|CYP17A1
141540EtoposideFDA approvedTOP2753082VemurafenibFDA approvedPK:YK,BRAF
141540EtoposideFDA approvedTOP2755986VismodegibFDA approvedSMO|PK:YK
141540EtoposideFDA approvedTOP2756645CrizotinibFDA approvedPK:YK,MET,ALK
141540EtoposideFDA approvedTOP2757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
141540EtoposideFDA approvedTOP2760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
141540EtoposideFDA approvedTOP2761432CabazitaxelFDA approvedTUBB|Tu-stab
141540EtoposideFDA approvedTOP2763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective9706Triethylenemelamine-A7|AlkAg
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective123127Doxorubicin hydrochlorideFDA approvedTOP2
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective279836MitoxantroneFDA approvedTOP2
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective713563ExemestaneFDA approvedHo|CYP19A1
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective715055GefitinibFDA approvedPK:YK,EGFR
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective747972LenalidomideFDA approvedFT|Immunomodulatory
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective747974RaloxifeneFDA approvedHo|SERM
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective749226AbirateroneFDA approvedHo|CYP17A1
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective753082VemurafenibFDA approvedPK:YK,BRAF
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective755986VismodegibFDA approvedSMO|PK:YK
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective756645CrizotinibFDA approvedPK:YK,MET,ALK
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective761432CabazitaxelFDA approvedTUBB|Tu-stab
169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
180973Tamoxifen citrateFDA approvedHo|SERM740MethotrexateFDA approvedDf|DHFR
180973Tamoxifen citrateFDA approvedHo|SERM752ThioguanineFDA approvedDs|IMPDH2|IMPDH
180973Tamoxifen citrateFDA approvedHo|SERM3053DactinomycinFDA approvedDb|RNA polymerase I
180973Tamoxifen citrateFDA approvedHo|SERM3088ChlorambucilFDA approvedA7|AlkAg
180973Tamoxifen citrateFDA approvedHo|SERM6396ThiotepaFDA approvedA7|AlkAg
180973Tamoxifen citrateFDA approvedHo|SERM8806MelphalanFDA approvedA7|AlkAg
180973Tamoxifen citrateFDA approvedHo|SERM13875HexamethylmelamineFDA approvedDb|AlkAg
180973Tamoxifen citrateFDA approvedHo|SERM19893FluorouracilFDA approvedDs|Rs|TYMS
180973Tamoxifen citrateFDA approvedHo|SERM27640FloxuridineFDA approvedDs|TYMS
180973Tamoxifen citrateFDA approvedHo|SERM34462Uracil mustardFDA approvedA7|AlkAg
180973Tamoxifen citrateFDA approvedHo|SERM45388DacarbazineFDA approvedA7|AlkAg
180973Tamoxifen citrateFDA approvedHo|SERM63878Cytarabine hydrochlorideFDA approvedDs
180973Tamoxifen citrateFDA approvedHo|SERM67574Vincristine sulfateFDA approvedTUBB|Tu-frag
180973Tamoxifen citrateFDA approvedHo|SERM71423Megestrol acetateFDA approvedHo|PGR
180973Tamoxifen citrateFDA approvedHo|SERM79037LomustineFDA approvedA6|AlkAg
180973Tamoxifen citrateFDA approvedHo|SERM82151Daunorubicin hydrochlorideFDA approvedTOP2
180973Tamoxifen citrateFDA approvedHo|SERM105014CladribineFDA approvedDs|ADA
180973Tamoxifen citrateFDA approvedHo|SERM118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
180973Tamoxifen citrateFDA approvedHo|SERM122758TretinoinFDA approvedHo|RXR|Differentiator
180973Tamoxifen citrateFDA approvedHo|SERM122819TeniposideFDA approvedTOP2
180973Tamoxifen citrateFDA approvedHo|SERM141540EtoposideFDA approvedTOP2
180973Tamoxifen citrateFDA approvedHo|SERM169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
180973Tamoxifen citrateFDA approvedHo|SERM279836MitoxantroneFDA approvedTOP2
180973Tamoxifen citrateFDA approvedHo|SERM608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
180973Tamoxifen citrateFDA approvedHo|SERM698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
180973Tamoxifen citrateFDA approvedHo|SERM713563ExemestaneFDA approvedHo|CYP19A1
180973Tamoxifen citrateFDA approvedHo|SERM715055GefitinibFDA approvedPK:YK,EGFR
180973Tamoxifen citrateFDA approvedHo|SERM719345LetrozoleFDA approvedHo|CYP19A1
180973Tamoxifen citrateFDA approvedHo|SERM719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
180973Tamoxifen citrateFDA approvedHo|SERM737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
180973Tamoxifen citrateFDA approvedHo|SERM747972LenalidomideFDA approvedFT|Immunomodulatory
180973Tamoxifen citrateFDA approvedHo|SERM747974RaloxifeneFDA approvedHo|SERM
180973Tamoxifen citrateFDA approvedHo|SERM749226AbirateroneFDA approvedHo|CYP17A1
180973Tamoxifen citrateFDA approvedHo|SERM753082VemurafenibFDA approvedPK:YK,BRAF
180973Tamoxifen citrateFDA approvedHo|SERM755986VismodegibFDA approvedSMO|PK:YK
180973Tamoxifen citrateFDA approvedHo|SERM756645CrizotinibFDA approvedPK:YK,MET,ALK
180973Tamoxifen citrateFDA approvedHo|SERM757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
180973Tamoxifen citrateFDA approvedHo|SERM760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
180973Tamoxifen citrateFDA approvedHo|SERM761432CabazitaxelFDA approvedTUBB|Tu-stab
180973Tamoxifen citrateFDA approvedHo|SERM763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
218321PentostatinFDA approvedDs|AM|ADA740MethotrexateFDA approvedDf|DHFR
218321PentostatinFDA approvedDs|AM|ADA750BusulfanFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA752ThioguanineFDA approvedDs|IMPDH2|IMPDH
218321PentostatinFDA approvedDs|AM|ADA7556-MercaptopurineFDA approvedDs|PPAT
218321PentostatinFDA approvedDs|AM|ADA762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA1390AllopurinolFDA approvedAM|XDH
218321PentostatinFDA approvedDs|AM|ADA3053DactinomycinFDA approvedDb|RNA polymerase I
218321PentostatinFDA approvedDs|AM|ADA3088ChlorambucilFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA6396ThiotepaFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA8806MelphalanFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA9706Triethylenemelamine-A7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA13875HexamethylmelamineFDA approvedDb|AlkAg
218321PentostatinFDA approvedDs|AM|ADA14229QuinacrineClinical trialDb|AP
218321PentostatinFDA approvedDs|AM|ADA18509Aminolevulinic Acid HydrochlorideFDA approvedAM
218321PentostatinFDA approvedDs|AM|ADA19893FluorouracilFDA approvedDs|Rs|TYMS
218321PentostatinFDA approvedDs|AM|ADA24559MithramycinFDA approvedDb|Rs
218321PentostatinFDA approvedDs|AM|ADA25154PipobromanFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA26271CyclophosphamideFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA26980MitomycinFDA approvedA2|AlkAg
218321PentostatinFDA approvedDs|AM|ADA27640FloxuridineFDA approvedDs|TYMS
218321PentostatinFDA approvedDs|AM|ADA32065HydroxyureaFDA approvedAM|Dr
218321PentostatinFDA approvedDs|AM|ADA34462Uracil mustardFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
218321PentostatinFDA approvedDs|AM|ADA45388DacarbazineFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA459238-MethoxypsoralenFDA approvedDb
218321PentostatinFDA approvedDs|AM|ADA49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
218321PentostatinFDA approvedDs|AM|ADA63878Cytarabine hydrochlorideFDA approvedDs
218321PentostatinFDA approvedDs|AM|ADA66847ThalidomideFDA approvedAng|Immunomodulatory
218321PentostatinFDA approvedDs|AM|ADA67574Vincristine sulfateFDA approvedTUBB|Tu-frag
218321PentostatinFDA approvedDs|AM|ADA71423Megestrol acetateFDA approvedHo|PGR
218321PentostatinFDA approvedDs|AM|ADA77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA79037LomustineFDA approvedA6|AlkAg
218321PentostatinFDA approvedDs|AM|ADA82151Daunorubicin hydrochlorideFDA approvedTOP2
218321PentostatinFDA approvedDs|AM|ADA85998StreptozocinFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA102816AzacitidineFDA approvedDNMT
218321PentostatinFDA approvedDs|AM|ADA105014CladribineFDA approvedDs|ADA
218321PentostatinFDA approvedDs|AM|ADA109724IfosfamideFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
218321PentostatinFDA approvedDs|AM|ADA122758TretinoinFDA approvedHo|RXR|Differentiator
218321PentostatinFDA approvedDs|AM|ADA122819TeniposideFDA approvedTOP2
218321PentostatinFDA approvedDs|AM|ADA123127Doxorubicin hydrochlorideFDA approvedTOP2
218321PentostatinFDA approvedDs|AM|ADA125066BleomycinFDA approvedDb
218321PentostatinFDA approvedDs|AM|ADA125973PaclitaxelFDA approvedTUBB|Tu-stab
218321PentostatinFDA approvedDs|AM|ADA138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
218321PentostatinFDA approvedDs|AM|ADA141540EtoposideFDA approvedTOP2
218321PentostatinFDA approvedDs|AM|ADA169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
218321PentostatinFDA approvedDs|AM|ADA180973Tamoxifen citrateFDA approvedHo|SERM
218321PentostatinFDA approvedDs|AM|ADA226080RapamycinFDA approvedPK:STK,MTOR
218321PentostatinFDA approvedDs|AM|ADA241240CarboplatinFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA246131ValrubicinFDA approvedTOP2
218321PentostatinFDA approvedDs|AM|ADA266046OxaliplatinFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA279836MitoxantroneFDA approvedTOP2
218321PentostatinFDA approvedDs|AM|ADA296961EthiofosFDA approvedRP
218321PentostatinFDA approvedDs|AM|ADA362856TemozolomideFDA approvedA7|AlkAg
218321PentostatinFDA approvedDs|AM|ADA369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod
218321PentostatinFDA approvedDs|AM|ADA606869ClofarabineFDA approvedDs
218321PentostatinFDA approvedDs|AM|ADA608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
218321PentostatinFDA approvedDs|AM|ADA613327Gemcitabine HCLFDA approvedDs
218321PentostatinFDA approvedDs|AM|ADA628503DocetaxelFDA approvedTUBB|Tu-stab
218321PentostatinFDA approvedDs|AM|ADA673596SN 38Clinical trialTOP1
218321PentostatinFDA approvedDs|AM|ADA686673NelarabineFDA approvedDs
218321PentostatinFDA approvedDs|AM|ADA698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
218321PentostatinFDA approvedDs|AM|ADA701852VorinostatFDA approvedHDAC
218321PentostatinFDA approvedDs|AM|ADA712807CapecitabineFDA approvedDs|TYMS
218321PentostatinFDA approvedDs|AM|ADA713563ExemestaneFDA approvedHo|CYP19A1
218321PentostatinFDA approvedDs|AM|ADA715055GefitinibFDA approvedPK:YK,EGFR
218321PentostatinFDA approvedDs|AM|ADA719276FulvestrantFDA approvedAM|Ho|ESR|SERM
218321PentostatinFDA approvedDs|AM|ADA719344AnastrozoleFDA approvedHo|CYP19A1
218321PentostatinFDA approvedDs|AM|ADA719345LetrozoleFDA approvedHo|CYP19A1
218321PentostatinFDA approvedDs|AM|ADA719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
218321PentostatinFDA approvedDs|AM|ADA721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
218321PentostatinFDA approvedDs|AM|ADA732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
218321PentostatinFDA approvedDs|AM|ADA733504EverolimusFDA approvedPK:STK,MTOR
218321PentostatinFDA approvedDs|AM|ADA737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
218321PentostatinFDA approvedDs|AM|ADA743414ImatinibFDA approvedBCR-ABL|PK:YK
218321PentostatinFDA approvedDs|AM|ADA745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
218321PentostatinFDA approvedDs|AM|ADA747599NilotinibFDA approvedBCR-ABL|PK:YK
218321PentostatinFDA approvedDs|AM|ADA747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
218321PentostatinFDA approvedDs|AM|ADA747972LenalidomideFDA approvedFT|Immunomodulatory
218321PentostatinFDA approvedDs|AM|ADA747974RaloxifeneFDA approvedHo|SERM
218321PentostatinFDA approvedDs|AM|ADA749226AbirateroneFDA approvedHo|CYP17A1
218321PentostatinFDA approvedDs|AM|ADA750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
218321PentostatinFDA approvedDs|AM|ADA753082VemurafenibFDA approvedPK:YK,BRAF
218321PentostatinFDA approvedDs|AM|ADA754143RomidepsinFDA approvedHDAC
218321PentostatinFDA approvedDs|AM|ADA754230PralatrexateFDA approvedDf|CTNNB1|DHFR
218321PentostatinFDA approvedDs|AM|ADA755986VismodegibFDA approvedSMO|PK:YK
218321PentostatinFDA approvedDs|AM|ADA756645CrizotinibFDA approvedPK:YK,MET,ALK
218321PentostatinFDA approvedDs|AM|ADA757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
218321PentostatinFDA approvedDs|AM|ADA760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
218321PentostatinFDA approvedDs|AM|ADA761432CabazitaxelFDA approvedTUBB|Tu-stab
218321PentostatinFDA approvedDs|AM|ADA763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
226080RapamycinFDA approvedPK:STK,MTOR740MethotrexateFDA approvedDf|DHFR
226080RapamycinFDA approvedPK:STK,MTOR752ThioguanineFDA approvedDs|IMPDH2|IMPDH
226080RapamycinFDA approvedPK:STK,MTOR7556-MercaptopurineFDA approvedDs|PPAT
226080RapamycinFDA approvedPK:STK,MTOR3053DactinomycinFDA approvedDb|RNA polymerase I
226080RapamycinFDA approvedPK:STK,MTOR3088ChlorambucilFDA approvedA7|AlkAg
226080RapamycinFDA approvedPK:STK,MTOR6396ThiotepaFDA approvedA7|AlkAg
226080RapamycinFDA approvedPK:STK,MTOR8806MelphalanFDA approvedA7|AlkAg
226080RapamycinFDA approvedPK:STK,MTOR13875HexamethylmelamineFDA approvedDb|AlkAg
226080RapamycinFDA approvedPK:STK,MTOR19893FluorouracilFDA approvedDs|Rs|TYMS
226080RapamycinFDA approvedPK:STK,MTOR24559MithramycinFDA approvedDb|Rs
226080RapamycinFDA approvedPK:STK,MTOR27640FloxuridineFDA approvedDs|TYMS
226080RapamycinFDA approvedPK:STK,MTOR32065HydroxyureaFDA approvedAM|Dr
226080RapamycinFDA approvedPK:STK,MTOR34462Uracil mustardFDA approvedA7|AlkAg
226080RapamycinFDA approvedPK:STK,MTOR38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
226080RapamycinFDA approvedPK:STK,MTOR45388DacarbazineFDA approvedA7|AlkAg
226080RapamycinFDA approvedPK:STK,MTOR49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
226080RapamycinFDA approvedPK:STK,MTOR63878Cytarabine hydrochlorideFDA approvedDs
226080RapamycinFDA approvedPK:STK,MTOR67574Vincristine sulfateFDA approvedTUBB|Tu-frag
226080RapamycinFDA approvedPK:STK,MTOR71423Megestrol acetateFDA approvedHo|PGR
226080RapamycinFDA approvedPK:STK,MTOR79037LomustineFDA approvedA6|AlkAg
226080RapamycinFDA approvedPK:STK,MTOR82151Daunorubicin hydrochlorideFDA approvedTOP2
226080RapamycinFDA approvedPK:STK,MTOR105014CladribineFDA approvedDs|ADA
226080RapamycinFDA approvedPK:STK,MTOR118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
226080RapamycinFDA approvedPK:STK,MTOR122758TretinoinFDA approvedHo|RXR|Differentiator
226080RapamycinFDA approvedPK:STK,MTOR122819TeniposideFDA approvedTOP2
226080RapamycinFDA approvedPK:STK,MTOR138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
226080RapamycinFDA approvedPK:STK,MTOR141540EtoposideFDA approvedTOP2
226080RapamycinFDA approvedPK:STK,MTOR169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
226080RapamycinFDA approvedPK:STK,MTOR180973Tamoxifen citrateFDA approvedHo|SERM
226080RapamycinFDA approvedPK:STK,MTOR241240CarboplatinFDA approvedA7|AlkAg
226080RapamycinFDA approvedPK:STK,MTOR246131ValrubicinFDA approvedTOP2
226080RapamycinFDA approvedPK:STK,MTOR279836MitoxantroneFDA approvedTOP2
226080RapamycinFDA approvedPK:STK,MTOR362856TemozolomideFDA approvedA7|AlkAg
226080RapamycinFDA approvedPK:STK,MTOR606869ClofarabineFDA approvedDs
226080RapamycinFDA approvedPK:STK,MTOR608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
226080RapamycinFDA approvedPK:STK,MTOR613327Gemcitabine HCLFDA approvedDs
226080RapamycinFDA approvedPK:STK,MTOR686673NelarabineFDA approvedDs
226080RapamycinFDA approvedPK:STK,MTOR698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
226080RapamycinFDA approvedPK:STK,MTOR712807CapecitabineFDA approvedDs|TYMS
226080RapamycinFDA approvedPK:STK,MTOR713563ExemestaneFDA approvedHo|CYP19A1
226080RapamycinFDA approvedPK:STK,MTOR715055GefitinibFDA approvedPK:YK,EGFR
226080RapamycinFDA approvedPK:STK,MTOR719344AnastrozoleFDA approvedHo|CYP19A1
226080RapamycinFDA approvedPK:STK,MTOR719345LetrozoleFDA approvedHo|CYP19A1
226080RapamycinFDA approvedPK:STK,MTOR719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
226080RapamycinFDA approvedPK:STK,MTOR737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
226080RapamycinFDA approvedPK:STK,MTOR743414ImatinibFDA approvedBCR-ABL|PK:YK
226080RapamycinFDA approvedPK:STK,MTOR747599NilotinibFDA approvedBCR-ABL|PK:YK
226080RapamycinFDA approvedPK:STK,MTOR747972LenalidomideFDA approvedFT|Immunomodulatory
226080RapamycinFDA approvedPK:STK,MTOR747974RaloxifeneFDA approvedHo|SERM
226080RapamycinFDA approvedPK:STK,MTOR749226AbirateroneFDA approvedHo|CYP17A1
226080RapamycinFDA approvedPK:STK,MTOR753082VemurafenibFDA approvedPK:YK,BRAF
226080RapamycinFDA approvedPK:STK,MTOR755986VismodegibFDA approvedSMO|PK:YK
226080RapamycinFDA approvedPK:STK,MTOR756645CrizotinibFDA approvedPK:YK,MET,ALK
226080RapamycinFDA approvedPK:STK,MTOR757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
226080RapamycinFDA approvedPK:STK,MTOR760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
226080RapamycinFDA approvedPK:STK,MTOR761432CabazitaxelFDA approvedTUBB|Tu-stab
226080RapamycinFDA approvedPK:STK,MTOR763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
241240CarboplatinFDA approvedA7|AlkAg740MethotrexateFDA approvedDf|DHFR
241240CarboplatinFDA approvedA7|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
241240CarboplatinFDA approvedA7|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
241240CarboplatinFDA approvedA7|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
241240CarboplatinFDA approvedA7|AlkAg6396ThiotepaFDA approvedA7|AlkAg
241240CarboplatinFDA approvedA7|AlkAg8806MelphalanFDA approvedA7|AlkAg
241240CarboplatinFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
241240CarboplatinFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
241240CarboplatinFDA approvedA7|AlkAg27640FloxuridineFDA approvedDs|TYMS
241240CarboplatinFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
241240CarboplatinFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
241240CarboplatinFDA approvedA7|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
241240CarboplatinFDA approvedA7|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
241240CarboplatinFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
241240CarboplatinFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
241240CarboplatinFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
241240CarboplatinFDA approvedA7|AlkAg105014CladribineFDA approvedDs|ADA
241240CarboplatinFDA approvedA7|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
241240CarboplatinFDA approvedA7|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
241240CarboplatinFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
241240CarboplatinFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
241240CarboplatinFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
241240CarboplatinFDA approvedA7|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
241240CarboplatinFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
241240CarboplatinFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
241240CarboplatinFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
241240CarboplatinFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
241240CarboplatinFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
241240CarboplatinFDA approvedA7|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
241240CarboplatinFDA approvedA7|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
241240CarboplatinFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
241240CarboplatinFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
241240CarboplatinFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
241240CarboplatinFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
241240CarboplatinFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
241240CarboplatinFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
241240CarboplatinFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
241240CarboplatinFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
241240CarboplatinFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
241240CarboplatinFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
241240CarboplatinFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
246131ValrubicinFDA approvedTOP2752ThioguanineFDA approvedDs|IMPDH2|IMPDH
246131ValrubicinFDA approvedTOP23053DactinomycinFDA approvedDb|RNA polymerase I
246131ValrubicinFDA approvedTOP23088ChlorambucilFDA approvedA7|AlkAg
246131ValrubicinFDA approvedTOP26396ThiotepaFDA approvedA7|AlkAg
246131ValrubicinFDA approvedTOP28806MelphalanFDA approvedA7|AlkAg
246131ValrubicinFDA approvedTOP213875HexamethylmelamineFDA approvedDb|AlkAg
246131ValrubicinFDA approvedTOP219893FluorouracilFDA approvedDs|Rs|TYMS
246131ValrubicinFDA approvedTOP224559MithramycinFDA approvedDb|Rs
246131ValrubicinFDA approvedTOP227640FloxuridineFDA approvedDs|TYMS
246131ValrubicinFDA approvedTOP232065HydroxyureaFDA approvedAM|Dr
246131ValrubicinFDA approvedTOP234462Uracil mustardFDA approvedA7|AlkAg
246131ValrubicinFDA approvedTOP245388DacarbazineFDA approvedA7|AlkAg
246131ValrubicinFDA approvedTOP249842Vinblastine sulfateFDA approvedTUBB|Tu-frag
246131ValrubicinFDA approvedTOP263878Cytarabine hydrochlorideFDA approvedDs
246131ValrubicinFDA approvedTOP267574Vincristine sulfateFDA approvedTUBB|Tu-frag
246131ValrubicinFDA approvedTOP271423Megestrol acetateFDA approvedHo|PGR
246131ValrubicinFDA approvedTOP279037LomustineFDA approvedA6|AlkAg
246131ValrubicinFDA approvedTOP282151Daunorubicin hydrochlorideFDA approvedTOP2
246131ValrubicinFDA approvedTOP2102816AzacitidineFDA approvedDNMT
246131ValrubicinFDA approvedTOP2105014CladribineFDA approvedDs|ADA
246131ValrubicinFDA approvedTOP2118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
246131ValrubicinFDA approvedTOP2122758TretinoinFDA approvedHo|RXR|Differentiator
246131ValrubicinFDA approvedTOP2122819TeniposideFDA approvedTOP2
246131ValrubicinFDA approvedTOP2123127Doxorubicin hydrochlorideFDA approvedTOP2
246131ValrubicinFDA approvedTOP2125066BleomycinFDA approvedDb
246131ValrubicinFDA approvedTOP2125973PaclitaxelFDA approvedTUBB|Tu-stab
246131ValrubicinFDA approvedTOP2141540EtoposideFDA approvedTOP2
246131ValrubicinFDA approvedTOP2169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
246131ValrubicinFDA approvedTOP2180973Tamoxifen citrateFDA approvedHo|SERM
246131ValrubicinFDA approvedTOP2226080RapamycinFDA approvedPK:STK,MTOR
246131ValrubicinFDA approvedTOP2241240CarboplatinFDA approvedA7|AlkAg
246131ValrubicinFDA approvedTOP2279836MitoxantroneFDA approvedTOP2
246131ValrubicinFDA approvedTOP2362856TemozolomideFDA approvedA7|AlkAg
246131ValrubicinFDA approvedTOP2606869ClofarabineFDA approvedDs
246131ValrubicinFDA approvedTOP2608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
246131ValrubicinFDA approvedTOP2613327Gemcitabine HCLFDA approvedDs
246131ValrubicinFDA approvedTOP2673596SN 38Clinical trialTOP1
246131ValrubicinFDA approvedTOP2686673NelarabineFDA approvedDs
246131ValrubicinFDA approvedTOP2698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
246131ValrubicinFDA approvedTOP2713563ExemestaneFDA approvedHo|CYP19A1
246131ValrubicinFDA approvedTOP2715055GefitinibFDA approvedPK:YK,EGFR
246131ValrubicinFDA approvedTOP2719345LetrozoleFDA approvedHo|CYP19A1
246131ValrubicinFDA approvedTOP2719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
246131ValrubicinFDA approvedTOP2732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
246131ValrubicinFDA approvedTOP2733504EverolimusFDA approvedPK:STK,MTOR
246131ValrubicinFDA approvedTOP2737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
246131ValrubicinFDA approvedTOP2743414ImatinibFDA approvedBCR-ABL|PK:YK
246131ValrubicinFDA approvedTOP2745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
246131ValrubicinFDA approvedTOP2747599NilotinibFDA approvedBCR-ABL|PK:YK
246131ValrubicinFDA approvedTOP2747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
246131ValrubicinFDA approvedTOP2747972LenalidomideFDA approvedFT|Immunomodulatory
246131ValrubicinFDA approvedTOP2747974RaloxifeneFDA approvedHo|SERM
246131ValrubicinFDA approvedTOP2749226AbirateroneFDA approvedHo|CYP17A1
246131ValrubicinFDA approvedTOP2750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
246131ValrubicinFDA approvedTOP2753082VemurafenibFDA approvedPK:YK,BRAF
246131ValrubicinFDA approvedTOP2754143RomidepsinFDA approvedHDAC
246131ValrubicinFDA approvedTOP2755986VismodegibFDA approvedSMO|PK:YK
246131ValrubicinFDA approvedTOP2756645CrizotinibFDA approvedPK:YK,MET,ALK
246131ValrubicinFDA approvedTOP2757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
246131ValrubicinFDA approvedTOP2760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
246131ValrubicinFDA approvedTOP2761432CabazitaxelFDA approvedTUBB|Tu-stab
246131ValrubicinFDA approvedTOP2763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
256439Idarubicin hydrochlorideFDA approvedTOP2740MethotrexateFDA approvedDf|DHFR
256439Idarubicin hydrochlorideFDA approvedTOP2750BusulfanFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP2752ThioguanineFDA approvedDs|IMPDH2|IMPDH
256439Idarubicin hydrochlorideFDA approvedTOP27556-MercaptopurineFDA approvedDs|PPAT
256439Idarubicin hydrochlorideFDA approvedTOP2762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP21390AllopurinolFDA approvedAM|XDH
256439Idarubicin hydrochlorideFDA approvedTOP23053DactinomycinFDA approvedDb|RNA polymerase I
256439Idarubicin hydrochlorideFDA approvedTOP23088ChlorambucilFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP26396ThiotepaFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP28806MelphalanFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP29706Triethylenemelamine-A7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP213875HexamethylmelamineFDA approvedDb|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP214229QuinacrineClinical trialDb|AP
256439Idarubicin hydrochlorideFDA approvedTOP218509Aminolevulinic Acid HydrochlorideFDA approvedAM
256439Idarubicin hydrochlorideFDA approvedTOP219893FluorouracilFDA approvedDs|Rs|TYMS
256439Idarubicin hydrochlorideFDA approvedTOP224559MithramycinFDA approvedDb|Rs
256439Idarubicin hydrochlorideFDA approvedTOP225154PipobromanFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP226271CyclophosphamideFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP226980MitomycinFDA approvedA2|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP227640FloxuridineFDA approvedDs|TYMS
256439Idarubicin hydrochlorideFDA approvedTOP232065HydroxyureaFDA approvedAM|Dr
256439Idarubicin hydrochlorideFDA approvedTOP234462Uracil mustardFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP238721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
256439Idarubicin hydrochlorideFDA approvedTOP245388DacarbazineFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP2459238-MethoxypsoralenFDA approvedDb
256439Idarubicin hydrochlorideFDA approvedTOP249842Vinblastine sulfateFDA approvedTUBB|Tu-frag
256439Idarubicin hydrochlorideFDA approvedTOP263878Cytarabine hydrochlorideFDA approvedDs
256439Idarubicin hydrochlorideFDA approvedTOP266847ThalidomideFDA approvedAng|Immunomodulatory
256439Idarubicin hydrochlorideFDA approvedTOP267574Vincristine sulfateFDA approvedTUBB|Tu-frag
256439Idarubicin hydrochlorideFDA approvedTOP271423Megestrol acetateFDA approvedHo|PGR
256439Idarubicin hydrochlorideFDA approvedTOP277213Procarbazine hydrochlorideFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP279037LomustineFDA approvedA6|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP282151Daunorubicin hydrochlorideFDA approvedTOP2
256439Idarubicin hydrochlorideFDA approvedTOP285998StreptozocinFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP292859Trisenox 3FDA approvedApo
256439Idarubicin hydrochlorideFDA approvedTOP2102816AzacitidineFDA approvedDNMT
256439Idarubicin hydrochlorideFDA approvedTOP2105014CladribineFDA approvedDs|ADA
256439Idarubicin hydrochlorideFDA approvedTOP2109724IfosfamideFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP2119875CisplatinFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP2122758TretinoinFDA approvedHo|RXR|Differentiator
256439Idarubicin hydrochlorideFDA approvedTOP2122819TeniposideFDA approvedTOP2
256439Idarubicin hydrochlorideFDA approvedTOP2123127Doxorubicin hydrochlorideFDA approvedTOP2
256439Idarubicin hydrochlorideFDA approvedTOP2125066BleomycinFDA approvedDb
256439Idarubicin hydrochlorideFDA approvedTOP2125973PaclitaxelFDA approvedTUBB|Tu-stab
256439Idarubicin hydrochlorideFDA approvedTOP2127716DecitabineFDA approvedAM|DNMT
256439Idarubicin hydrochlorideFDA approvedTOP2138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP2141540EtoposideFDA approvedTOP2
256439Idarubicin hydrochlorideFDA approvedTOP2169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
256439Idarubicin hydrochlorideFDA approvedTOP2180973Tamoxifen citrateFDA approvedHo|SERM
256439Idarubicin hydrochlorideFDA approvedTOP2218321PentostatinFDA approvedDs|AM|ADA
256439Idarubicin hydrochlorideFDA approvedTOP2226080RapamycinFDA approvedPK:STK,MTOR
256439Idarubicin hydrochlorideFDA approvedTOP2241240CarboplatinFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP2246131ValrubicinFDA approvedTOP2
256439Idarubicin hydrochlorideFDA approvedTOP2256942Epirubicin HCLFDA approvedTOP2
256439Idarubicin hydrochlorideFDA approvedTOP2266046OxaliplatinFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP2279836MitoxantroneFDA approvedTOP2
256439Idarubicin hydrochlorideFDA approvedTOP2296961EthiofosFDA approvedRP
256439Idarubicin hydrochlorideFDA approvedTOP2362856TemozolomideFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP2369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod
256439Idarubicin hydrochlorideFDA approvedTOP2409962CarmustineFDA approvedA7|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP2606869ClofarabineFDA approvedDs
256439Idarubicin hydrochlorideFDA approvedTOP2608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
256439Idarubicin hydrochlorideFDA approvedTOP2609699Topotecan hydrochlorideFDA approvedTOP1
256439Idarubicin hydrochlorideFDA approvedTOP2613327Gemcitabine HCLFDA approvedDs
256439Idarubicin hydrochlorideFDA approvedTOP2628503DocetaxelFDA approvedTUBB|Tu-stab
256439Idarubicin hydrochlorideFDA approvedTOP2673596SN 38Clinical trialTOP1
256439Idarubicin hydrochlorideFDA approvedTOP2681239Proscript boronic acidFDA approvedPSM
256439Idarubicin hydrochlorideFDA approvedTOP2686673NelarabineFDA approvedDs
256439Idarubicin hydrochlorideFDA approvedTOP2698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
256439Idarubicin hydrochlorideFDA approvedTOP2701852VorinostatFDA approvedHDAC
256439Idarubicin hydrochlorideFDA approvedTOP2702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg
256439Idarubicin hydrochlorideFDA approvedTOP2707389Eribulin mesylateFDA approvedTUBB
256439Idarubicin hydrochlorideFDA approvedTOP2712807CapecitabineFDA approvedDs|TYMS
256439Idarubicin hydrochlorideFDA approvedTOP2713563ExemestaneFDA approvedHo|CYP19A1
256439Idarubicin hydrochlorideFDA approvedTOP2715055GefitinibFDA approvedPK:YK,EGFR
256439Idarubicin hydrochlorideFDA approvedTOP2718781Erlotinib HCLFDA approvedPK:YK,EGFR
256439Idarubicin hydrochlorideFDA approvedTOP2719276FulvestrantFDA approvedAM|Ho|ESR|SERM
256439Idarubicin hydrochlorideFDA approvedTOP2719344AnastrozoleFDA approvedHo|CYP19A1
256439Idarubicin hydrochlorideFDA approvedTOP2719345LetrozoleFDA approvedHo|CYP19A1
256439Idarubicin hydrochlorideFDA approvedTOP2719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
256439Idarubicin hydrochlorideFDA approvedTOP2721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
256439Idarubicin hydrochlorideFDA approvedTOP2732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
256439Idarubicin hydrochlorideFDA approvedTOP2733504EverolimusFDA approvedPK:STK,MTOR
256439Idarubicin hydrochlorideFDA approvedTOP2737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
256439Idarubicin hydrochlorideFDA approvedTOP2743414ImatinibFDA approvedBCR-ABL|PK:YK
256439Idarubicin hydrochlorideFDA approvedTOP2745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
256439Idarubicin hydrochlorideFDA approvedTOP2747599NilotinibFDA approvedBCR-ABL|PK:YK
256439Idarubicin hydrochlorideFDA approvedTOP2747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
256439Idarubicin hydrochlorideFDA approvedTOP2747972LenalidomideFDA approvedFT|Immunomodulatory
256439Idarubicin hydrochlorideFDA approvedTOP2747973IxabepiloneFDA approvedTUBB|Tu-stab
256439Idarubicin hydrochlorideFDA approvedTOP2747974RaloxifeneFDA approvedHo|SERM
256439Idarubicin hydrochlorideFDA approvedTOP2749226AbirateroneFDA approvedHo|CYP17A1
256439Idarubicin hydrochlorideFDA approvedTOP2750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
256439Idarubicin hydrochlorideFDA approvedTOP2754143RomidepsinFDA approvedHDAC
256439Idarubicin hydrochlorideFDA approvedTOP2754230PralatrexateFDA approvedDf|CTNNB1|DHFR
256439Idarubicin hydrochlorideFDA approvedTOP2755986VismodegibFDA approvedSMO|PK:YK
256439Idarubicin hydrochlorideFDA approvedTOP2756645CrizotinibFDA approvedPK:YK,MET,ALK
256439Idarubicin hydrochlorideFDA approvedTOP2757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
256439Idarubicin hydrochlorideFDA approvedTOP2760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
256439Idarubicin hydrochlorideFDA approvedTOP2761432CabazitaxelFDA approvedTUBB|Tu-stab
256439Idarubicin hydrochlorideFDA approvedTOP2763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
256942Epirubicin HCLFDA approvedTOP2740MethotrexateFDA approvedDf|DHFR
256942Epirubicin HCLFDA approvedTOP2750BusulfanFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP2752ThioguanineFDA approvedDs|IMPDH2|IMPDH
256942Epirubicin HCLFDA approvedTOP27556-MercaptopurineFDA approvedDs|PPAT
256942Epirubicin HCLFDA approvedTOP2762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP21390AllopurinolFDA approvedAM|XDH
256942Epirubicin HCLFDA approvedTOP23053DactinomycinFDA approvedDb|RNA polymerase I
256942Epirubicin HCLFDA approvedTOP23088ChlorambucilFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP26396ThiotepaFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP28806MelphalanFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP29706Triethylenemelamine-A7|AlkAg
256942Epirubicin HCLFDA approvedTOP213875HexamethylmelamineFDA approvedDb|AlkAg
256942Epirubicin HCLFDA approvedTOP214229QuinacrineClinical trialDb|AP
256942Epirubicin HCLFDA approvedTOP218509Aminolevulinic Acid HydrochlorideFDA approvedAM
256942Epirubicin HCLFDA approvedTOP219893FluorouracilFDA approvedDs|Rs|TYMS
256942Epirubicin HCLFDA approvedTOP224559MithramycinFDA approvedDb|Rs
256942Epirubicin HCLFDA approvedTOP225154PipobromanFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP226271CyclophosphamideFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP226980MitomycinFDA approvedA2|AlkAg
256942Epirubicin HCLFDA approvedTOP227640FloxuridineFDA approvedDs|TYMS
256942Epirubicin HCLFDA approvedTOP232065HydroxyureaFDA approvedAM|Dr
256942Epirubicin HCLFDA approvedTOP234462Uracil mustardFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP238721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
256942Epirubicin HCLFDA approvedTOP245388DacarbazineFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP2459238-MethoxypsoralenFDA approvedDb
256942Epirubicin HCLFDA approvedTOP249842Vinblastine sulfateFDA approvedTUBB|Tu-frag
256942Epirubicin HCLFDA approvedTOP263878Cytarabine hydrochlorideFDA approvedDs
256942Epirubicin HCLFDA approvedTOP266847ThalidomideFDA approvedAng|Immunomodulatory
256942Epirubicin HCLFDA approvedTOP267574Vincristine sulfateFDA approvedTUBB|Tu-frag
256942Epirubicin HCLFDA approvedTOP271423Megestrol acetateFDA approvedHo|PGR
256942Epirubicin HCLFDA approvedTOP277213Procarbazine hydrochlorideFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP279037LomustineFDA approvedA6|AlkAg
256942Epirubicin HCLFDA approvedTOP282151Daunorubicin hydrochlorideFDA approvedTOP2
256942Epirubicin HCLFDA approvedTOP285998StreptozocinFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP292859Trisenox 3FDA approvedApo
256942Epirubicin HCLFDA approvedTOP2102816AzacitidineFDA approvedDNMT
256942Epirubicin HCLFDA approvedTOP2105014CladribineFDA approvedDs|ADA
256942Epirubicin HCLFDA approvedTOP2109724IfosfamideFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP2119875CisplatinFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP2122758TretinoinFDA approvedHo|RXR|Differentiator
256942Epirubicin HCLFDA approvedTOP2122819TeniposideFDA approvedTOP2
256942Epirubicin HCLFDA approvedTOP2123127Doxorubicin hydrochlorideFDA approvedTOP2
256942Epirubicin HCLFDA approvedTOP2125066BleomycinFDA approvedDb
256942Epirubicin HCLFDA approvedTOP2125973PaclitaxelFDA approvedTUBB|Tu-stab
256942Epirubicin HCLFDA approvedTOP2127716DecitabineFDA approvedAM|DNMT
256942Epirubicin HCLFDA approvedTOP2138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
256942Epirubicin HCLFDA approvedTOP2141540EtoposideFDA approvedTOP2
256942Epirubicin HCLFDA approvedTOP2169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
256942Epirubicin HCLFDA approvedTOP2180973Tamoxifen citrateFDA approvedHo|SERM
256942Epirubicin HCLFDA approvedTOP2218321PentostatinFDA approvedDs|AM|ADA
256942Epirubicin HCLFDA approvedTOP2226080RapamycinFDA approvedPK:STK,MTOR
256942Epirubicin HCLFDA approvedTOP2241240CarboplatinFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP2246131ValrubicinFDA approvedTOP2
256942Epirubicin HCLFDA approvedTOP2256439Idarubicin hydrochlorideFDA approvedTOP2
256942Epirubicin HCLFDA approvedTOP2266046OxaliplatinFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP2279836MitoxantroneFDA approvedTOP2
256942Epirubicin HCLFDA approvedTOP2296961EthiofosFDA approvedRP
256942Epirubicin HCLFDA approvedTOP2362856TemozolomideFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP2369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod
256942Epirubicin HCLFDA approvedTOP2409962CarmustineFDA approvedA7|AlkAg
256942Epirubicin HCLFDA approvedTOP2606869ClofarabineFDA approvedDs
256942Epirubicin HCLFDA approvedTOP2608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
256942Epirubicin HCLFDA approvedTOP2609699Topotecan hydrochlorideFDA approvedTOP1
256942Epirubicin HCLFDA approvedTOP2613327Gemcitabine HCLFDA approvedDs
256942Epirubicin HCLFDA approvedTOP2628503DocetaxelFDA approvedTUBB|Tu-stab
256942Epirubicin HCLFDA approvedTOP2673596SN 38Clinical trialTOP1
256942Epirubicin HCLFDA approvedTOP2681239Proscript boronic acidFDA approvedPSM
256942Epirubicin HCLFDA approvedTOP2686673NelarabineFDA approvedDs
256942Epirubicin HCLFDA approvedTOP2698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
256942Epirubicin HCLFDA approvedTOP2701852VorinostatFDA approvedHDAC
256942Epirubicin HCLFDA approvedTOP2702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg
256942Epirubicin HCLFDA approvedTOP2707389Eribulin mesylateFDA approvedTUBB
256942Epirubicin HCLFDA approvedTOP2712807CapecitabineFDA approvedDs|TYMS
256942Epirubicin HCLFDA approvedTOP2713563ExemestaneFDA approvedHo|CYP19A1
256942Epirubicin HCLFDA approvedTOP2715055GefitinibFDA approvedPK:YK,EGFR
256942Epirubicin HCLFDA approvedTOP2718781Erlotinib HCLFDA approvedPK:YK,EGFR
256942Epirubicin HCLFDA approvedTOP2719276FulvestrantFDA approvedAM|Ho|ESR|SERM
256942Epirubicin HCLFDA approvedTOP2719344AnastrozoleFDA approvedHo|CYP19A1
256942Epirubicin HCLFDA approvedTOP2719345LetrozoleFDA approvedHo|CYP19A1
256942Epirubicin HCLFDA approvedTOP2719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
256942Epirubicin HCLFDA approvedTOP2721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
256942Epirubicin HCLFDA approvedTOP2732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
256942Epirubicin HCLFDA approvedTOP2733504EverolimusFDA approvedPK:STK,MTOR
256942Epirubicin HCLFDA approvedTOP2737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
256942Epirubicin HCLFDA approvedTOP2743414ImatinibFDA approvedBCR-ABL|PK:YK
256942Epirubicin HCLFDA approvedTOP2745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
256942Epirubicin HCLFDA approvedTOP2747599NilotinibFDA approvedBCR-ABL|PK:YK
256942Epirubicin HCLFDA approvedTOP2747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
256942Epirubicin HCLFDA approvedTOP2747972LenalidomideFDA approvedFT|Immunomodulatory
256942Epirubicin HCLFDA approvedTOP2747973IxabepiloneFDA approvedTUBB|Tu-stab
256942Epirubicin HCLFDA approvedTOP2747974RaloxifeneFDA approvedHo|SERM
256942Epirubicin HCLFDA approvedTOP2749226AbirateroneFDA approvedHo|CYP17A1
256942Epirubicin HCLFDA approvedTOP2750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
256942Epirubicin HCLFDA approvedTOP2754143RomidepsinFDA approvedHDAC
256942Epirubicin HCLFDA approvedTOP2754230PralatrexateFDA approvedDf|CTNNB1|DHFR
256942Epirubicin HCLFDA approvedTOP2755986VismodegibFDA approvedSMO|PK:YK
256942Epirubicin HCLFDA approvedTOP2756645CrizotinibFDA approvedPK:YK,MET,ALK
256942Epirubicin HCLFDA approvedTOP2757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
256942Epirubicin HCLFDA approvedTOP2760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
256942Epirubicin HCLFDA approvedTOP2761432CabazitaxelFDA approvedTUBB|Tu-stab
256942Epirubicin HCLFDA approvedTOP2763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
266046OxaliplatinFDA approvedA7|AlkAg740MethotrexateFDA approvedDf|DHFR
266046OxaliplatinFDA approvedA7|AlkAg750BusulfanFDA approvedA7|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
266046OxaliplatinFDA approvedA7|AlkAg7556-MercaptopurineFDA approvedDs|PPAT
266046OxaliplatinFDA approvedA7|AlkAg762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg1390AllopurinolFDA approvedAM|XDH
266046OxaliplatinFDA approvedA7|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
266046OxaliplatinFDA approvedA7|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg6396ThiotepaFDA approvedA7|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg8806MelphalanFDA approvedA7|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg9706Triethylenemelamine-A7|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg14229QuinacrineClinical trialDb|AP
266046OxaliplatinFDA approvedA7|AlkAg18509Aminolevulinic Acid HydrochlorideFDA approvedAM
266046OxaliplatinFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
266046OxaliplatinFDA approvedA7|AlkAg24559MithramycinFDA approvedDb|Rs
266046OxaliplatinFDA approvedA7|AlkAg25154PipobromanFDA approvedA7|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg26271CyclophosphamideFDA approvedA7|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg26980MitomycinFDA approvedA2|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg27640FloxuridineFDA approvedDs|TYMS
266046OxaliplatinFDA approvedA7|AlkAg32065HydroxyureaFDA approvedAM|Dr
266046OxaliplatinFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
266046OxaliplatinFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg459238-MethoxypsoralenFDA approvedDb
266046OxaliplatinFDA approvedA7|AlkAg49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
266046OxaliplatinFDA approvedA7|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
266046OxaliplatinFDA approvedA7|AlkAg66847ThalidomideFDA approvedAng|Immunomodulatory
266046OxaliplatinFDA approvedA7|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
266046OxaliplatinFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
266046OxaliplatinFDA approvedA7|AlkAg77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
266046OxaliplatinFDA approvedA7|AlkAg85998StreptozocinFDA approvedA7|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg102816AzacitidineFDA approvedDNMT
266046OxaliplatinFDA approvedA7|AlkAg105014CladribineFDA approvedDs|ADA
266046OxaliplatinFDA approvedA7|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
266046OxaliplatinFDA approvedA7|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
266046OxaliplatinFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
266046OxaliplatinFDA approvedA7|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
266046OxaliplatinFDA approvedA7|AlkAg125066BleomycinFDA approvedDb
266046OxaliplatinFDA approvedA7|AlkAg125973PaclitaxelFDA approvedTUBB|Tu-stab
266046OxaliplatinFDA approvedA7|AlkAg127716DecitabineFDA approvedAM|DNMT
266046OxaliplatinFDA approvedA7|AlkAg138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
266046OxaliplatinFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
266046OxaliplatinFDA approvedA7|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
266046OxaliplatinFDA approvedA7|AlkAg218321PentostatinFDA approvedDs|AM|ADA
266046OxaliplatinFDA approvedA7|AlkAg226080RapamycinFDA approvedPK:STK,MTOR
266046OxaliplatinFDA approvedA7|AlkAg241240CarboplatinFDA approvedA7|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg246131ValrubicinFDA approvedTOP2
266046OxaliplatinFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
266046OxaliplatinFDA approvedA7|AlkAg362856TemozolomideFDA approvedA7|AlkAg
266046OxaliplatinFDA approvedA7|AlkAg606869ClofarabineFDA approvedDs
266046OxaliplatinFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
266046OxaliplatinFDA approvedA7|AlkAg609699Topotecan hydrochlorideFDA approvedTOP1
266046OxaliplatinFDA approvedA7|AlkAg613327Gemcitabine HCLFDA approvedDs
266046OxaliplatinFDA approvedA7|AlkAg628503DocetaxelFDA approvedTUBB|Tu-stab
266046OxaliplatinFDA approvedA7|AlkAg673596SN 38Clinical trialTOP1
266046OxaliplatinFDA approvedA7|AlkAg686673NelarabineFDA approvedDs
266046OxaliplatinFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
266046OxaliplatinFDA approvedA7|AlkAg701852VorinostatFDA approvedHDAC
266046OxaliplatinFDA approvedA7|AlkAg712807CapecitabineFDA approvedDs|TYMS
266046OxaliplatinFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
266046OxaliplatinFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
266046OxaliplatinFDA approvedA7|AlkAg719276FulvestrantFDA approvedAM|Ho|ESR|SERM
266046OxaliplatinFDA approvedA7|AlkAg719344AnastrozoleFDA approvedHo|CYP19A1
266046OxaliplatinFDA approvedA7|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
266046OxaliplatinFDA approvedA7|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
266046OxaliplatinFDA approvedA7|AlkAg721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
266046OxaliplatinFDA approvedA7|AlkAg732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
266046OxaliplatinFDA approvedA7|AlkAg733504EverolimusFDA approvedPK:STK,MTOR
266046OxaliplatinFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
266046OxaliplatinFDA approvedA7|AlkAg743414ImatinibFDA approvedBCR-ABL|PK:YK
266046OxaliplatinFDA approvedA7|AlkAg745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
266046OxaliplatinFDA approvedA7|AlkAg747599NilotinibFDA approvedBCR-ABL|PK:YK
266046OxaliplatinFDA approvedA7|AlkAg747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
266046OxaliplatinFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
266046OxaliplatinFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
266046OxaliplatinFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
266046OxaliplatinFDA approvedA7|AlkAg750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
266046OxaliplatinFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
266046OxaliplatinFDA approvedA7|AlkAg754143RomidepsinFDA approvedHDAC
266046OxaliplatinFDA approvedA7|AlkAg754230PralatrexateFDA approvedDf|CTNNB1|DHFR
266046OxaliplatinFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
266046OxaliplatinFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
266046OxaliplatinFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
266046OxaliplatinFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
266046OxaliplatinFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
266046OxaliplatinFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
279836MitoxantroneFDA approvedTOP29706Triethylenemelamine-A7|AlkAg
279836MitoxantroneFDA approvedTOP2123127Doxorubicin hydrochlorideFDA approvedTOP2
279836MitoxantroneFDA approvedTOP2608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
279836MitoxantroneFDA approvedTOP2698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
279836MitoxantroneFDA approvedTOP2713563ExemestaneFDA approvedHo|CYP19A1
279836MitoxantroneFDA approvedTOP2715055GefitinibFDA approvedPK:YK,EGFR
279836MitoxantroneFDA approvedTOP2737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
279836MitoxantroneFDA approvedTOP2747972LenalidomideFDA approvedFT|Immunomodulatory
279836MitoxantroneFDA approvedTOP2747974RaloxifeneFDA approvedHo|SERM
279836MitoxantroneFDA approvedTOP2749226AbirateroneFDA approvedHo|CYP17A1
279836MitoxantroneFDA approvedTOP2753082VemurafenibFDA approvedPK:YK,BRAF
279836MitoxantroneFDA approvedTOP2755986VismodegibFDA approvedSMO|PK:YK
279836MitoxantroneFDA approvedTOP2756645CrizotinibFDA approvedPK:YK,MET,ALK
279836MitoxantroneFDA approvedTOP2757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
279836MitoxantroneFDA approvedTOP2760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
279836MitoxantroneFDA approvedTOP2761432CabazitaxelFDA approvedTUBB|Tu-stab
279836MitoxantroneFDA approvedTOP2763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
296961EthiofosFDA approvedRP740MethotrexateFDA approvedDf|DHFR
296961EthiofosFDA approvedRP750BusulfanFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP752ThioguanineFDA approvedDs|IMPDH2|IMPDH
296961EthiofosFDA approvedRP7556-MercaptopurineFDA approvedDs|PPAT
296961EthiofosFDA approvedRP762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP1390AllopurinolFDA approvedAM|XDH
296961EthiofosFDA approvedRP3053DactinomycinFDA approvedDb|RNA polymerase I
296961EthiofosFDA approvedRP3088ChlorambucilFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP6396ThiotepaFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP8806MelphalanFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP9706Triethylenemelamine-A7|AlkAg
296961EthiofosFDA approvedRP13875HexamethylmelamineFDA approvedDb|AlkAg
296961EthiofosFDA approvedRP14229QuinacrineClinical trialDb|AP
296961EthiofosFDA approvedRP18509Aminolevulinic Acid HydrochlorideFDA approvedAM
296961EthiofosFDA approvedRP19893FluorouracilFDA approvedDs|Rs|TYMS
296961EthiofosFDA approvedRP24559MithramycinFDA approvedDb|Rs
296961EthiofosFDA approvedRP25154PipobromanFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP26271CyclophosphamideFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP26980MitomycinFDA approvedA2|AlkAg
296961EthiofosFDA approvedRP27640FloxuridineFDA approvedDs|TYMS
296961EthiofosFDA approvedRP32065HydroxyureaFDA approvedAM|Dr
296961EthiofosFDA approvedRP34462Uracil mustardFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
296961EthiofosFDA approvedRP45388DacarbazineFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP459238-MethoxypsoralenFDA approvedDb
296961EthiofosFDA approvedRP49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
296961EthiofosFDA approvedRP63878Cytarabine hydrochlorideFDA approvedDs
296961EthiofosFDA approvedRP66847ThalidomideFDA approvedAng|Immunomodulatory
296961EthiofosFDA approvedRP67574Vincristine sulfateFDA approvedTUBB|Tu-frag
296961EthiofosFDA approvedRP71423Megestrol acetateFDA approvedHo|PGR
296961EthiofosFDA approvedRP77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP79037LomustineFDA approvedA6|AlkAg
296961EthiofosFDA approvedRP82151Daunorubicin hydrochlorideFDA approvedTOP2
296961EthiofosFDA approvedRP85998StreptozocinFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP102816AzacitidineFDA approvedDNMT
296961EthiofosFDA approvedRP105014CladribineFDA approvedDs|ADA
296961EthiofosFDA approvedRP109724IfosfamideFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
296961EthiofosFDA approvedRP122758TretinoinFDA approvedHo|RXR|Differentiator
296961EthiofosFDA approvedRP122819TeniposideFDA approvedTOP2
296961EthiofosFDA approvedRP123127Doxorubicin hydrochlorideFDA approvedTOP2
296961EthiofosFDA approvedRP125066BleomycinFDA approvedDb
296961EthiofosFDA approvedRP125973PaclitaxelFDA approvedTUBB|Tu-stab
296961EthiofosFDA approvedRP127716DecitabineFDA approvedAM|DNMT
296961EthiofosFDA approvedRP138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
296961EthiofosFDA approvedRP141540EtoposideFDA approvedTOP2
296961EthiofosFDA approvedRP169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
296961EthiofosFDA approvedRP180973Tamoxifen citrateFDA approvedHo|SERM
296961EthiofosFDA approvedRP226080RapamycinFDA approvedPK:STK,MTOR
296961EthiofosFDA approvedRP241240CarboplatinFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP246131ValrubicinFDA approvedTOP2
296961EthiofosFDA approvedRP266046OxaliplatinFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP279836MitoxantroneFDA approvedTOP2
296961EthiofosFDA approvedRP362856TemozolomideFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod
296961EthiofosFDA approvedRP409962CarmustineFDA approvedA7|AlkAg
296961EthiofosFDA approvedRP606869ClofarabineFDA approvedDs
296961EthiofosFDA approvedRP608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
296961EthiofosFDA approvedRP613327Gemcitabine HCLFDA approvedDs
296961EthiofosFDA approvedRP628503DocetaxelFDA approvedTUBB|Tu-stab
296961EthiofosFDA approvedRP673596SN 38Clinical trialTOP1
296961EthiofosFDA approvedRP686673NelarabineFDA approvedDs
296961EthiofosFDA approvedRP698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
296961EthiofosFDA approvedRP701852VorinostatFDA approvedHDAC
296961EthiofosFDA approvedRP712807CapecitabineFDA approvedDs|TYMS
296961EthiofosFDA approvedRP713563ExemestaneFDA approvedHo|CYP19A1
296961EthiofosFDA approvedRP715055GefitinibFDA approvedPK:YK,EGFR
296961EthiofosFDA approvedRP719276FulvestrantFDA approvedAM|Ho|ESR|SERM
296961EthiofosFDA approvedRP719344AnastrozoleFDA approvedHo|CYP19A1
296961EthiofosFDA approvedRP719345LetrozoleFDA approvedHo|CYP19A1
296961EthiofosFDA approvedRP719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
296961EthiofosFDA approvedRP721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
296961EthiofosFDA approvedRP732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
296961EthiofosFDA approvedRP733504EverolimusFDA approvedPK:STK,MTOR
296961EthiofosFDA approvedRP737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
296961EthiofosFDA approvedRP743414ImatinibFDA approvedBCR-ABL|PK:YK
296961EthiofosFDA approvedRP745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
296961EthiofosFDA approvedRP747599NilotinibFDA approvedBCR-ABL|PK:YK
296961EthiofosFDA approvedRP747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
296961EthiofosFDA approvedRP747972LenalidomideFDA approvedFT|Immunomodulatory
296961EthiofosFDA approvedRP747974RaloxifeneFDA approvedHo|SERM
296961EthiofosFDA approvedRP749226AbirateroneFDA approvedHo|CYP17A1
296961EthiofosFDA approvedRP750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
296961EthiofosFDA approvedRP753082VemurafenibFDA approvedPK:YK,BRAF
296961EthiofosFDA approvedRP754143RomidepsinFDA approvedHDAC
296961EthiofosFDA approvedRP754230PralatrexateFDA approvedDf|CTNNB1|DHFR
296961EthiofosFDA approvedRP755986VismodegibFDA approvedSMO|PK:YK
296961EthiofosFDA approvedRP756645CrizotinibFDA approvedPK:YK,MET,ALK
296961EthiofosFDA approvedRP757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
296961EthiofosFDA approvedRP760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
296961EthiofosFDA approvedRP761432CabazitaxelFDA approvedTUBB|Tu-stab
296961EthiofosFDA approvedRP763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
362856TemozolomideFDA approvedA7|AlkAg740MethotrexateFDA approvedDf|DHFR
362856TemozolomideFDA approvedA7|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
362856TemozolomideFDA approvedA7|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
362856TemozolomideFDA approvedA7|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
362856TemozolomideFDA approvedA7|AlkAg6396ThiotepaFDA approvedA7|AlkAg
362856TemozolomideFDA approvedA7|AlkAg8806MelphalanFDA approvedA7|AlkAg
362856TemozolomideFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
362856TemozolomideFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
362856TemozolomideFDA approvedA7|AlkAg27640FloxuridineFDA approvedDs|TYMS
362856TemozolomideFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
362856TemozolomideFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
362856TemozolomideFDA approvedA7|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
362856TemozolomideFDA approvedA7|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
362856TemozolomideFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
362856TemozolomideFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
362856TemozolomideFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
362856TemozolomideFDA approvedA7|AlkAg105014CladribineFDA approvedDs|ADA
362856TemozolomideFDA approvedA7|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
362856TemozolomideFDA approvedA7|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
362856TemozolomideFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
362856TemozolomideFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
362856TemozolomideFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
362856TemozolomideFDA approvedA7|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
362856TemozolomideFDA approvedA7|AlkAg241240CarboplatinFDA approvedA7|AlkAg
362856TemozolomideFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
362856TemozolomideFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
362856TemozolomideFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
362856TemozolomideFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
362856TemozolomideFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
362856TemozolomideFDA approvedA7|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
362856TemozolomideFDA approvedA7|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
362856TemozolomideFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
362856TemozolomideFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
362856TemozolomideFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
362856TemozolomideFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
362856TemozolomideFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
362856TemozolomideFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
362856TemozolomideFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
362856TemozolomideFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
362856TemozolomideFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
362856TemozolomideFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
362856TemozolomideFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod740MethotrexateFDA approvedDf|DHFR
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod750BusulfanFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod752ThioguanineFDA approvedDs|IMPDH2|IMPDH
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod7556-MercaptopurineFDA approvedDs|PPAT
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod1390AllopurinolFDA approvedAM|XDH
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod3053DactinomycinFDA approvedDb|RNA polymerase I
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod3088ChlorambucilFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod6396ThiotepaFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod8806MelphalanFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod9706Triethylenemelamine-A7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod13875HexamethylmelamineFDA approvedDb|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod14229QuinacrineClinical trialDb|AP
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod18509Aminolevulinic Acid HydrochlorideFDA approvedAM
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod19893FluorouracilFDA approvedDs|Rs|TYMS
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod24559MithramycinFDA approvedDb|Rs
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod25154PipobromanFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod26271CyclophosphamideFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod26980MitomycinFDA approvedA2|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod27640FloxuridineFDA approvedDs|TYMS
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod32065HydroxyureaFDA approvedAM|Dr
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod34462Uracil mustardFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod45388DacarbazineFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod459238-MethoxypsoralenFDA approvedDb
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod63878Cytarabine hydrochlorideFDA approvedDs
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod66847ThalidomideFDA approvedAng|Immunomodulatory
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod67574Vincristine sulfateFDA approvedTUBB|Tu-frag
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod71423Megestrol acetateFDA approvedHo|PGR
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod79037LomustineFDA approvedA6|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod82151Daunorubicin hydrochlorideFDA approvedTOP2
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod85998StreptozocinFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod102816AzacitidineFDA approvedDNMT
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod105014CladribineFDA approvedDs|ADA
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod109724IfosfamideFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod122758TretinoinFDA approvedHo|RXR|Differentiator
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod122819TeniposideFDA approvedTOP2
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod123127Doxorubicin hydrochlorideFDA approvedTOP2
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod125066BleomycinFDA approvedDb
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod125973PaclitaxelFDA approvedTUBB|Tu-stab
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod141540EtoposideFDA approvedTOP2
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod180973Tamoxifen citrateFDA approvedHo|SERM
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod226080RapamycinFDA approvedPK:STK,MTOR
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod241240CarboplatinFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod246131ValrubicinFDA approvedTOP2
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod266046OxaliplatinFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod279836MitoxantroneFDA approvedTOP2
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod362856TemozolomideFDA approvedA7|AlkAg
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod606869ClofarabineFDA approvedDs
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod613327Gemcitabine HCLFDA approvedDs
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod628503DocetaxelFDA approvedTUBB|Tu-stab
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod673596SN 38Clinical trialTOP1
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod686673NelarabineFDA approvedDs
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod701852VorinostatFDA approvedHDAC
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod712807CapecitabineFDA approvedDs|TYMS
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod713563ExemestaneFDA approvedHo|CYP19A1
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod715055GefitinibFDA approvedPK:YK,EGFR
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod719276FulvestrantFDA approvedAM|Ho|ESR|SERM
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod719344AnastrozoleFDA approvedHo|CYP19A1
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod719345LetrozoleFDA approvedHo|CYP19A1
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod733504EverolimusFDA approvedPK:STK,MTOR
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod743414ImatinibFDA approvedBCR-ABL|PK:YK
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod747599NilotinibFDA approvedBCR-ABL|PK:YK
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod747972LenalidomideFDA approvedFT|Immunomodulatory
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod747974RaloxifeneFDA approvedHo|SERM
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod749226AbirateroneFDA approvedHo|CYP17A1
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod753082VemurafenibFDA approvedPK:YK,BRAF
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod754143RomidepsinFDA approvedHDAC
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod754230PralatrexateFDA approvedDf|CTNNB1|DHFR
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod755986VismodegibFDA approvedSMO|PK:YK
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod756645CrizotinibFDA approvedPK:YK,MET,ALK
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod761432CabazitaxelFDA approvedTUBB|Tu-stab
369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
409962CarmustineFDA approvedA7|AlkAg740MethotrexateFDA approvedDf|DHFR
409962CarmustineFDA approvedA7|AlkAg750BusulfanFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
409962CarmustineFDA approvedA7|AlkAg7556-MercaptopurineFDA approvedDs|PPAT
409962CarmustineFDA approvedA7|AlkAg762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg1390AllopurinolFDA approvedAM|XDH
409962CarmustineFDA approvedA7|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
409962CarmustineFDA approvedA7|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg6396ThiotepaFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg8806MelphalanFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg9706Triethylenemelamine-A7|AlkAg
409962CarmustineFDA approvedA7|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
409962CarmustineFDA approvedA7|AlkAg14229QuinacrineClinical trialDb|AP
409962CarmustineFDA approvedA7|AlkAg18509Aminolevulinic Acid HydrochlorideFDA approvedAM
409962CarmustineFDA approvedA7|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
409962CarmustineFDA approvedA7|AlkAg24559MithramycinFDA approvedDb|Rs
409962CarmustineFDA approvedA7|AlkAg25154PipobromanFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg26271CyclophosphamideFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg26980MitomycinFDA approvedA2|AlkAg
409962CarmustineFDA approvedA7|AlkAg27640FloxuridineFDA approvedDs|TYMS
409962CarmustineFDA approvedA7|AlkAg32065HydroxyureaFDA approvedAM|Dr
409962CarmustineFDA approvedA7|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
409962CarmustineFDA approvedA7|AlkAg45388DacarbazineFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg459238-MethoxypsoralenFDA approvedDb
409962CarmustineFDA approvedA7|AlkAg49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
409962CarmustineFDA approvedA7|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
409962CarmustineFDA approvedA7|AlkAg66847ThalidomideFDA approvedAng|Immunomodulatory
409962CarmustineFDA approvedA7|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
409962CarmustineFDA approvedA7|AlkAg71423Megestrol acetateFDA approvedHo|PGR
409962CarmustineFDA approvedA7|AlkAg77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg79037LomustineFDA approvedA6|AlkAg
409962CarmustineFDA approvedA7|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
409962CarmustineFDA approvedA7|AlkAg85998StreptozocinFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg102816AzacitidineFDA approvedDNMT
409962CarmustineFDA approvedA7|AlkAg105014CladribineFDA approvedDs|ADA
409962CarmustineFDA approvedA7|AlkAg109724IfosfamideFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
409962CarmustineFDA approvedA7|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
409962CarmustineFDA approvedA7|AlkAg122819TeniposideFDA approvedTOP2
409962CarmustineFDA approvedA7|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
409962CarmustineFDA approvedA7|AlkAg125066BleomycinFDA approvedDb
409962CarmustineFDA approvedA7|AlkAg125973PaclitaxelFDA approvedTUBB|Tu-stab
409962CarmustineFDA approvedA7|AlkAg127716DecitabineFDA approvedAM|DNMT
409962CarmustineFDA approvedA7|AlkAg138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
409962CarmustineFDA approvedA7|AlkAg141540EtoposideFDA approvedTOP2
409962CarmustineFDA approvedA7|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
409962CarmustineFDA approvedA7|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
409962CarmustineFDA approvedA7|AlkAg218321PentostatinFDA approvedDs|AM|ADA
409962CarmustineFDA approvedA7|AlkAg226080RapamycinFDA approvedPK:STK,MTOR
409962CarmustineFDA approvedA7|AlkAg241240CarboplatinFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg246131ValrubicinFDA approvedTOP2
409962CarmustineFDA approvedA7|AlkAg266046OxaliplatinFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg279836MitoxantroneFDA approvedTOP2
409962CarmustineFDA approvedA7|AlkAg362856TemozolomideFDA approvedA7|AlkAg
409962CarmustineFDA approvedA7|AlkAg369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod
409962CarmustineFDA approvedA7|AlkAg606869ClofarabineFDA approvedDs
409962CarmustineFDA approvedA7|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
409962CarmustineFDA approvedA7|AlkAg609699Topotecan hydrochlorideFDA approvedTOP1
409962CarmustineFDA approvedA7|AlkAg613327Gemcitabine HCLFDA approvedDs
409962CarmustineFDA approvedA7|AlkAg628503DocetaxelFDA approvedTUBB|Tu-stab
409962CarmustineFDA approvedA7|AlkAg673596SN 38Clinical trialTOP1
409962CarmustineFDA approvedA7|AlkAg686673NelarabineFDA approvedDs
409962CarmustineFDA approvedA7|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
409962CarmustineFDA approvedA7|AlkAg701852VorinostatFDA approvedHDAC
409962CarmustineFDA approvedA7|AlkAg712807CapecitabineFDA approvedDs|TYMS
409962CarmustineFDA approvedA7|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
409962CarmustineFDA approvedA7|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
409962CarmustineFDA approvedA7|AlkAg719276FulvestrantFDA approvedAM|Ho|ESR|SERM
409962CarmustineFDA approvedA7|AlkAg719344AnastrozoleFDA approvedHo|CYP19A1
409962CarmustineFDA approvedA7|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
409962CarmustineFDA approvedA7|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
409962CarmustineFDA approvedA7|AlkAg721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
409962CarmustineFDA approvedA7|AlkAg732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
409962CarmustineFDA approvedA7|AlkAg733504EverolimusFDA approvedPK:STK,MTOR
409962CarmustineFDA approvedA7|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
409962CarmustineFDA approvedA7|AlkAg743414ImatinibFDA approvedBCR-ABL|PK:YK
409962CarmustineFDA approvedA7|AlkAg745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
409962CarmustineFDA approvedA7|AlkAg747599NilotinibFDA approvedBCR-ABL|PK:YK
409962CarmustineFDA approvedA7|AlkAg747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
409962CarmustineFDA approvedA7|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
409962CarmustineFDA approvedA7|AlkAg747974RaloxifeneFDA approvedHo|SERM
409962CarmustineFDA approvedA7|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
409962CarmustineFDA approvedA7|AlkAg750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
409962CarmustineFDA approvedA7|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
409962CarmustineFDA approvedA7|AlkAg754143RomidepsinFDA approvedHDAC
409962CarmustineFDA approvedA7|AlkAg754230PralatrexateFDA approvedDf|CTNNB1|DHFR
409962CarmustineFDA approvedA7|AlkAg755986VismodegibFDA approvedSMO|PK:YK
409962CarmustineFDA approvedA7|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
409962CarmustineFDA approvedA7|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
409962CarmustineFDA approvedA7|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
409962CarmustineFDA approvedA7|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
409962CarmustineFDA approvedA7|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
606869ClofarabineFDA approvedDs740MethotrexateFDA approvedDf|DHFR
606869ClofarabineFDA approvedDs752ThioguanineFDA approvedDs|IMPDH2|IMPDH
606869ClofarabineFDA approvedDs7556-MercaptopurineFDA approvedDs|PPAT
606869ClofarabineFDA approvedDs3053DactinomycinFDA approvedDb|RNA polymerase I
606869ClofarabineFDA approvedDs3088ChlorambucilFDA approvedA7|AlkAg
606869ClofarabineFDA approvedDs6396ThiotepaFDA approvedA7|AlkAg
606869ClofarabineFDA approvedDs8806MelphalanFDA approvedA7|AlkAg
606869ClofarabineFDA approvedDs13875HexamethylmelamineFDA approvedDb|AlkAg
606869ClofarabineFDA approvedDs19893FluorouracilFDA approvedDs|Rs|TYMS
606869ClofarabineFDA approvedDs24559MithramycinFDA approvedDb|Rs
606869ClofarabineFDA approvedDs27640FloxuridineFDA approvedDs|TYMS
606869ClofarabineFDA approvedDs32065HydroxyureaFDA approvedAM|Dr
606869ClofarabineFDA approvedDs34462Uracil mustardFDA approvedA7|AlkAg
606869ClofarabineFDA approvedDs38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
606869ClofarabineFDA approvedDs45388DacarbazineFDA approvedA7|AlkAg
606869ClofarabineFDA approvedDs49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
606869ClofarabineFDA approvedDs63878Cytarabine hydrochlorideFDA approvedDs
606869ClofarabineFDA approvedDs67574Vincristine sulfateFDA approvedTUBB|Tu-frag
606869ClofarabineFDA approvedDs71423Megestrol acetateFDA approvedHo|PGR
606869ClofarabineFDA approvedDs79037LomustineFDA approvedA6|AlkAg
606869ClofarabineFDA approvedDs82151Daunorubicin hydrochlorideFDA approvedTOP2
606869ClofarabineFDA approvedDs105014CladribineFDA approvedDs|ADA
606869ClofarabineFDA approvedDs118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
606869ClofarabineFDA approvedDs122758TretinoinFDA approvedHo|RXR|Differentiator
606869ClofarabineFDA approvedDs122819TeniposideFDA approvedTOP2
606869ClofarabineFDA approvedDs138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
606869ClofarabineFDA approvedDs141540EtoposideFDA approvedTOP2
606869ClofarabineFDA approvedDs169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
606869ClofarabineFDA approvedDs180973Tamoxifen citrateFDA approvedHo|SERM
606869ClofarabineFDA approvedDs241240CarboplatinFDA approvedA7|AlkAg
606869ClofarabineFDA approvedDs246131ValrubicinFDA approvedTOP2
606869ClofarabineFDA approvedDs279836MitoxantroneFDA approvedTOP2
606869ClofarabineFDA approvedDs362856TemozolomideFDA approvedA7|AlkAg
606869ClofarabineFDA approvedDs608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
606869ClofarabineFDA approvedDs686673NelarabineFDA approvedDs
606869ClofarabineFDA approvedDs698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
606869ClofarabineFDA approvedDs712807CapecitabineFDA approvedDs|TYMS
606869ClofarabineFDA approvedDs713563ExemestaneFDA approvedHo|CYP19A1
606869ClofarabineFDA approvedDs715055GefitinibFDA approvedPK:YK,EGFR
606869ClofarabineFDA approvedDs719276FulvestrantFDA approvedAM|Ho|ESR|SERM
606869ClofarabineFDA approvedDs719344AnastrozoleFDA approvedHo|CYP19A1
606869ClofarabineFDA approvedDs719345LetrozoleFDA approvedHo|CYP19A1
606869ClofarabineFDA approvedDs719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
606869ClofarabineFDA approvedDs737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
606869ClofarabineFDA approvedDs743414ImatinibFDA approvedBCR-ABL|PK:YK
606869ClofarabineFDA approvedDs747599NilotinibFDA approvedBCR-ABL|PK:YK
606869ClofarabineFDA approvedDs747972LenalidomideFDA approvedFT|Immunomodulatory
606869ClofarabineFDA approvedDs747974RaloxifeneFDA approvedHo|SERM
606869ClofarabineFDA approvedDs749226AbirateroneFDA approvedHo|CYP17A1
606869ClofarabineFDA approvedDs753082VemurafenibFDA approvedPK:YK,BRAF
606869ClofarabineFDA approvedDs755986VismodegibFDA approvedSMO|PK:YK
606869ClofarabineFDA approvedDs756645CrizotinibFDA approvedPK:YK,MET,ALK
606869ClofarabineFDA approvedDs757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
606869ClofarabineFDA approvedDs760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
606869ClofarabineFDA approvedDs761432CabazitaxelFDA approvedTUBB|Tu-stab
606869ClofarabineFDA approvedDs763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag9706Triethylenemelamine-A7|AlkAg
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag123127Doxorubicin hydrochlorideFDA approvedTOP2
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag713563ExemestaneFDA approvedHo|CYP19A1
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag715055GefitinibFDA approvedPK:YK,EGFR
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag747972LenalidomideFDA approvedFT|Immunomodulatory
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag747974RaloxifeneFDA approvedHo|SERM
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag749226AbirateroneFDA approvedHo|CYP17A1
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag753082VemurafenibFDA approvedPK:YK,BRAF
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag755986VismodegibFDA approvedSMO|PK:YK
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag756645CrizotinibFDA approvedPK:YK,MET,ALK
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag761432CabazitaxelFDA approvedTUBB|Tu-stab
608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
609699Topotecan hydrochlorideFDA approvedTOP1740MethotrexateFDA approvedDf|DHFR
609699Topotecan hydrochlorideFDA approvedTOP1750BusulfanFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP1752ThioguanineFDA approvedDs|IMPDH2|IMPDH
609699Topotecan hydrochlorideFDA approvedTOP17556-MercaptopurineFDA approvedDs|PPAT
609699Topotecan hydrochlorideFDA approvedTOP1762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP11390AllopurinolFDA approvedAM|XDH
609699Topotecan hydrochlorideFDA approvedTOP13053DactinomycinFDA approvedDb|RNA polymerase I
609699Topotecan hydrochlorideFDA approvedTOP13088ChlorambucilFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP16396ThiotepaFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP18806MelphalanFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP19706Triethylenemelamine-A7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP113875HexamethylmelamineFDA approvedDb|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP114229QuinacrineClinical trialDb|AP
609699Topotecan hydrochlorideFDA approvedTOP118509Aminolevulinic Acid HydrochlorideFDA approvedAM
609699Topotecan hydrochlorideFDA approvedTOP119893FluorouracilFDA approvedDs|Rs|TYMS
609699Topotecan hydrochlorideFDA approvedTOP124559MithramycinFDA approvedDb|Rs
609699Topotecan hydrochlorideFDA approvedTOP125154PipobromanFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP126271CyclophosphamideFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP126980MitomycinFDA approvedA2|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP127640FloxuridineFDA approvedDs|TYMS
609699Topotecan hydrochlorideFDA approvedTOP132065HydroxyureaFDA approvedAM|Dr
609699Topotecan hydrochlorideFDA approvedTOP134462Uracil mustardFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP138721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
609699Topotecan hydrochlorideFDA approvedTOP145388DacarbazineFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP1459238-MethoxypsoralenFDA approvedDb
609699Topotecan hydrochlorideFDA approvedTOP149842Vinblastine sulfateFDA approvedTUBB|Tu-frag
609699Topotecan hydrochlorideFDA approvedTOP163878Cytarabine hydrochlorideFDA approvedDs
609699Topotecan hydrochlorideFDA approvedTOP166847ThalidomideFDA approvedAng|Immunomodulatory
609699Topotecan hydrochlorideFDA approvedTOP167574Vincristine sulfateFDA approvedTUBB|Tu-frag
609699Topotecan hydrochlorideFDA approvedTOP171423Megestrol acetateFDA approvedHo|PGR
609699Topotecan hydrochlorideFDA approvedTOP177213Procarbazine hydrochlorideFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP179037LomustineFDA approvedA6|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP182151Daunorubicin hydrochlorideFDA approvedTOP2
609699Topotecan hydrochlorideFDA approvedTOP185998StreptozocinFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP1102816AzacitidineFDA approvedDNMT
609699Topotecan hydrochlorideFDA approvedTOP1105014CladribineFDA approvedDs|ADA
609699Topotecan hydrochlorideFDA approvedTOP1109724IfosfamideFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP1118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
609699Topotecan hydrochlorideFDA approvedTOP1122758TretinoinFDA approvedHo|RXR|Differentiator
609699Topotecan hydrochlorideFDA approvedTOP1122819TeniposideFDA approvedTOP2
609699Topotecan hydrochlorideFDA approvedTOP1123127Doxorubicin hydrochlorideFDA approvedTOP2
609699Topotecan hydrochlorideFDA approvedTOP1125066BleomycinFDA approvedDb
609699Topotecan hydrochlorideFDA approvedTOP1125973PaclitaxelFDA approvedTUBB|Tu-stab
609699Topotecan hydrochlorideFDA approvedTOP1138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP1141540EtoposideFDA approvedTOP2
609699Topotecan hydrochlorideFDA approvedTOP1169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
609699Topotecan hydrochlorideFDA approvedTOP1180973Tamoxifen citrateFDA approvedHo|SERM
609699Topotecan hydrochlorideFDA approvedTOP1218321PentostatinFDA approvedDs|AM|ADA
609699Topotecan hydrochlorideFDA approvedTOP1226080RapamycinFDA approvedPK:STK,MTOR
609699Topotecan hydrochlorideFDA approvedTOP1241240CarboplatinFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP1246131ValrubicinFDA approvedTOP2
609699Topotecan hydrochlorideFDA approvedTOP1266046OxaliplatinFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP1279836MitoxantroneFDA approvedTOP2
609699Topotecan hydrochlorideFDA approvedTOP1296961EthiofosFDA approvedRP
609699Topotecan hydrochlorideFDA approvedTOP1362856TemozolomideFDA approvedA7|AlkAg
609699Topotecan hydrochlorideFDA approvedTOP1369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod
609699Topotecan hydrochlorideFDA approvedTOP1606869ClofarabineFDA approvedDs
609699Topotecan hydrochlorideFDA approvedTOP1608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
609699Topotecan hydrochlorideFDA approvedTOP1613327Gemcitabine HCLFDA approvedDs
609699Topotecan hydrochlorideFDA approvedTOP1628503DocetaxelFDA approvedTUBB|Tu-stab
609699Topotecan hydrochlorideFDA approvedTOP1673596SN 38Clinical trialTOP1
609699Topotecan hydrochlorideFDA approvedTOP1686673NelarabineFDA approvedDs
609699Topotecan hydrochlorideFDA approvedTOP1698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
609699Topotecan hydrochlorideFDA approvedTOP1701852VorinostatFDA approvedHDAC
609699Topotecan hydrochlorideFDA approvedTOP1712807CapecitabineFDA approvedDs|TYMS
609699Topotecan hydrochlorideFDA approvedTOP1713563ExemestaneFDA approvedHo|CYP19A1
609699Topotecan hydrochlorideFDA approvedTOP1715055GefitinibFDA approvedPK:YK,EGFR
609699Topotecan hydrochlorideFDA approvedTOP1719276FulvestrantFDA approvedAM|Ho|ESR|SERM
609699Topotecan hydrochlorideFDA approvedTOP1719344AnastrozoleFDA approvedHo|CYP19A1
609699Topotecan hydrochlorideFDA approvedTOP1719345LetrozoleFDA approvedHo|CYP19A1
609699Topotecan hydrochlorideFDA approvedTOP1719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
609699Topotecan hydrochlorideFDA approvedTOP1721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
609699Topotecan hydrochlorideFDA approvedTOP1732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
609699Topotecan hydrochlorideFDA approvedTOP1733504EverolimusFDA approvedPK:STK,MTOR
609699Topotecan hydrochlorideFDA approvedTOP1737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
609699Topotecan hydrochlorideFDA approvedTOP1743414ImatinibFDA approvedBCR-ABL|PK:YK
609699Topotecan hydrochlorideFDA approvedTOP1745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
609699Topotecan hydrochlorideFDA approvedTOP1747599NilotinibFDA approvedBCR-ABL|PK:YK
609699Topotecan hydrochlorideFDA approvedTOP1747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
609699Topotecan hydrochlorideFDA approvedTOP1747972LenalidomideFDA approvedFT|Immunomodulatory
609699Topotecan hydrochlorideFDA approvedTOP1747974RaloxifeneFDA approvedHo|SERM
609699Topotecan hydrochlorideFDA approvedTOP1749226AbirateroneFDA approvedHo|CYP17A1
609699Topotecan hydrochlorideFDA approvedTOP1750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
609699Topotecan hydrochlorideFDA approvedTOP1753082VemurafenibFDA approvedPK:YK,BRAF
609699Topotecan hydrochlorideFDA approvedTOP1754143RomidepsinFDA approvedHDAC
609699Topotecan hydrochlorideFDA approvedTOP1754230PralatrexateFDA approvedDf|CTNNB1|DHFR
609699Topotecan hydrochlorideFDA approvedTOP1755986VismodegibFDA approvedSMO|PK:YK
609699Topotecan hydrochlorideFDA approvedTOP1756645CrizotinibFDA approvedPK:YK,MET,ALK
609699Topotecan hydrochlorideFDA approvedTOP1757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
609699Topotecan hydrochlorideFDA approvedTOP1760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
609699Topotecan hydrochlorideFDA approvedTOP1761432CabazitaxelFDA approvedTUBB|Tu-stab
609699Topotecan hydrochlorideFDA approvedTOP1763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
613327Gemcitabine HCLFDA approvedDs740MethotrexateFDA approvedDf|DHFR
613327Gemcitabine HCLFDA approvedDs752ThioguanineFDA approvedDs|IMPDH2|IMPDH
613327Gemcitabine HCLFDA approvedDs7556-MercaptopurineFDA approvedDs|PPAT
613327Gemcitabine HCLFDA approvedDs3053DactinomycinFDA approvedDb|RNA polymerase I
613327Gemcitabine HCLFDA approvedDs3088ChlorambucilFDA approvedA7|AlkAg
613327Gemcitabine HCLFDA approvedDs6396ThiotepaFDA approvedA7|AlkAg
613327Gemcitabine HCLFDA approvedDs8806MelphalanFDA approvedA7|AlkAg
613327Gemcitabine HCLFDA approvedDs13875HexamethylmelamineFDA approvedDb|AlkAg
613327Gemcitabine HCLFDA approvedDs19893FluorouracilFDA approvedDs|Rs|TYMS
613327Gemcitabine HCLFDA approvedDs24559MithramycinFDA approvedDb|Rs
613327Gemcitabine HCLFDA approvedDs27640FloxuridineFDA approvedDs|TYMS
613327Gemcitabine HCLFDA approvedDs32065HydroxyureaFDA approvedAM|Dr
613327Gemcitabine HCLFDA approvedDs34462Uracil mustardFDA approvedA7|AlkAg
613327Gemcitabine HCLFDA approvedDs38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
613327Gemcitabine HCLFDA approvedDs45388DacarbazineFDA approvedA7|AlkAg
613327Gemcitabine HCLFDA approvedDs49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
613327Gemcitabine HCLFDA approvedDs63878Cytarabine hydrochlorideFDA approvedDs
613327Gemcitabine HCLFDA approvedDs67574Vincristine sulfateFDA approvedTUBB|Tu-frag
613327Gemcitabine HCLFDA approvedDs71423Megestrol acetateFDA approvedHo|PGR
613327Gemcitabine HCLFDA approvedDs79037LomustineFDA approvedA6|AlkAg
613327Gemcitabine HCLFDA approvedDs82151Daunorubicin hydrochlorideFDA approvedTOP2
613327Gemcitabine HCLFDA approvedDs105014CladribineFDA approvedDs|ADA
613327Gemcitabine HCLFDA approvedDs118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
613327Gemcitabine HCLFDA approvedDs122758TretinoinFDA approvedHo|RXR|Differentiator
613327Gemcitabine HCLFDA approvedDs122819TeniposideFDA approvedTOP2
613327Gemcitabine HCLFDA approvedDs138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
613327Gemcitabine HCLFDA approvedDs141540EtoposideFDA approvedTOP2
613327Gemcitabine HCLFDA approvedDs169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
613327Gemcitabine HCLFDA approvedDs180973Tamoxifen citrateFDA approvedHo|SERM
613327Gemcitabine HCLFDA approvedDs241240CarboplatinFDA approvedA7|AlkAg
613327Gemcitabine HCLFDA approvedDs279836MitoxantroneFDA approvedTOP2
613327Gemcitabine HCLFDA approvedDs362856TemozolomideFDA approvedA7|AlkAg
613327Gemcitabine HCLFDA approvedDs606869ClofarabineFDA approvedDs
613327Gemcitabine HCLFDA approvedDs608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
613327Gemcitabine HCLFDA approvedDs686673NelarabineFDA approvedDs
613327Gemcitabine HCLFDA approvedDs698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
613327Gemcitabine HCLFDA approvedDs712807CapecitabineFDA approvedDs|TYMS
613327Gemcitabine HCLFDA approvedDs713563ExemestaneFDA approvedHo|CYP19A1
613327Gemcitabine HCLFDA approvedDs715055GefitinibFDA approvedPK:YK,EGFR
613327Gemcitabine HCLFDA approvedDs719276FulvestrantFDA approvedAM|Ho|ESR|SERM
613327Gemcitabine HCLFDA approvedDs719344AnastrozoleFDA approvedHo|CYP19A1
613327Gemcitabine HCLFDA approvedDs719345LetrozoleFDA approvedHo|CYP19A1
613327Gemcitabine HCLFDA approvedDs719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
613327Gemcitabine HCLFDA approvedDs737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
613327Gemcitabine HCLFDA approvedDs743414ImatinibFDA approvedBCR-ABL|PK:YK
613327Gemcitabine HCLFDA approvedDs747599NilotinibFDA approvedBCR-ABL|PK:YK
613327Gemcitabine HCLFDA approvedDs747972LenalidomideFDA approvedFT|Immunomodulatory
613327Gemcitabine HCLFDA approvedDs747974RaloxifeneFDA approvedHo|SERM
613327Gemcitabine HCLFDA approvedDs749226AbirateroneFDA approvedHo|CYP17A1
613327Gemcitabine HCLFDA approvedDs753082VemurafenibFDA approvedPK:YK,BRAF
613327Gemcitabine HCLFDA approvedDs755986VismodegibFDA approvedSMO|PK:YK
613327Gemcitabine HCLFDA approvedDs756645CrizotinibFDA approvedPK:YK,MET,ALK
613327Gemcitabine HCLFDA approvedDs757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
613327Gemcitabine HCLFDA approvedDs760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
613327Gemcitabine HCLFDA approvedDs761432CabazitaxelFDA approvedTUBB|Tu-stab
613327Gemcitabine HCLFDA approvedDs763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
628503DocetaxelFDA approvedTUBB|Tu-stab752ThioguanineFDA approvedDs|IMPDH2|IMPDH
628503DocetaxelFDA approvedTUBB|Tu-stab3053DactinomycinFDA approvedDb|RNA polymerase I
628503DocetaxelFDA approvedTUBB|Tu-stab3088ChlorambucilFDA approvedA7|AlkAg
628503DocetaxelFDA approvedTUBB|Tu-stab6396ThiotepaFDA approvedA7|AlkAg
628503DocetaxelFDA approvedTUBB|Tu-stab8806MelphalanFDA approvedA7|AlkAg
628503DocetaxelFDA approvedTUBB|Tu-stab13875HexamethylmelamineFDA approvedDb|AlkAg
628503DocetaxelFDA approvedTUBB|Tu-stab19893FluorouracilFDA approvedDs|Rs|TYMS
628503DocetaxelFDA approvedTUBB|Tu-stab27640FloxuridineFDA approvedDs|TYMS
628503DocetaxelFDA approvedTUBB|Tu-stab34462Uracil mustardFDA approvedA7|AlkAg
628503DocetaxelFDA approvedTUBB|Tu-stab45388DacarbazineFDA approvedA7|AlkAg
628503DocetaxelFDA approvedTUBB|Tu-stab49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
628503DocetaxelFDA approvedTUBB|Tu-stab63878Cytarabine hydrochlorideFDA approvedDs
628503DocetaxelFDA approvedTUBB|Tu-stab67574Vincristine sulfateFDA approvedTUBB|Tu-frag
628503DocetaxelFDA approvedTUBB|Tu-stab71423Megestrol acetateFDA approvedHo|PGR
628503DocetaxelFDA approvedTUBB|Tu-stab79037LomustineFDA approvedA6|AlkAg
628503DocetaxelFDA approvedTUBB|Tu-stab82151Daunorubicin hydrochlorideFDA approvedTOP2
628503DocetaxelFDA approvedTUBB|Tu-stab105014CladribineFDA approvedDs|ADA
628503DocetaxelFDA approvedTUBB|Tu-stab118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
628503DocetaxelFDA approvedTUBB|Tu-stab122758TretinoinFDA approvedHo|RXR|Differentiator
628503DocetaxelFDA approvedTUBB|Tu-stab122819TeniposideFDA approvedTOP2
628503DocetaxelFDA approvedTUBB|Tu-stab125973PaclitaxelFDA approvedTUBB|Tu-stab
628503DocetaxelFDA approvedTUBB|Tu-stab141540EtoposideFDA approvedTOP2
628503DocetaxelFDA approvedTUBB|Tu-stab169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
628503DocetaxelFDA approvedTUBB|Tu-stab180973Tamoxifen citrateFDA approvedHo|SERM
628503DocetaxelFDA approvedTUBB|Tu-stab226080RapamycinFDA approvedPK:STK,MTOR
628503DocetaxelFDA approvedTUBB|Tu-stab241240CarboplatinFDA approvedA7|AlkAg
628503DocetaxelFDA approvedTUBB|Tu-stab246131ValrubicinFDA approvedTOP2
628503DocetaxelFDA approvedTUBB|Tu-stab279836MitoxantroneFDA approvedTOP2
628503DocetaxelFDA approvedTUBB|Tu-stab362856TemozolomideFDA approvedA7|AlkAg
628503DocetaxelFDA approvedTUBB|Tu-stab606869ClofarabineFDA approvedDs
628503DocetaxelFDA approvedTUBB|Tu-stab608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
628503DocetaxelFDA approvedTUBB|Tu-stab613327Gemcitabine HCLFDA approvedDs
628503DocetaxelFDA approvedTUBB|Tu-stab686673NelarabineFDA approvedDs
628503DocetaxelFDA approvedTUBB|Tu-stab698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
628503DocetaxelFDA approvedTUBB|Tu-stab712807CapecitabineFDA approvedDs|TYMS
628503DocetaxelFDA approvedTUBB|Tu-stab713563ExemestaneFDA approvedHo|CYP19A1
628503DocetaxelFDA approvedTUBB|Tu-stab715055GefitinibFDA approvedPK:YK,EGFR
628503DocetaxelFDA approvedTUBB|Tu-stab719276FulvestrantFDA approvedAM|Ho|ESR|SERM
628503DocetaxelFDA approvedTUBB|Tu-stab719344AnastrozoleFDA approvedHo|CYP19A1
628503DocetaxelFDA approvedTUBB|Tu-stab719345LetrozoleFDA approvedHo|CYP19A1
628503DocetaxelFDA approvedTUBB|Tu-stab719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
628503DocetaxelFDA approvedTUBB|Tu-stab737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
628503DocetaxelFDA approvedTUBB|Tu-stab743414ImatinibFDA approvedBCR-ABL|PK:YK
628503DocetaxelFDA approvedTUBB|Tu-stab747599NilotinibFDA approvedBCR-ABL|PK:YK
628503DocetaxelFDA approvedTUBB|Tu-stab747972LenalidomideFDA approvedFT|Immunomodulatory
628503DocetaxelFDA approvedTUBB|Tu-stab747974RaloxifeneFDA approvedHo|SERM
628503DocetaxelFDA approvedTUBB|Tu-stab749226AbirateroneFDA approvedHo|CYP17A1
628503DocetaxelFDA approvedTUBB|Tu-stab753082VemurafenibFDA approvedPK:YK,BRAF
628503DocetaxelFDA approvedTUBB|Tu-stab755986VismodegibFDA approvedSMO|PK:YK
628503DocetaxelFDA approvedTUBB|Tu-stab756645CrizotinibFDA approvedPK:YK,MET,ALK
628503DocetaxelFDA approvedTUBB|Tu-stab757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
628503DocetaxelFDA approvedTUBB|Tu-stab760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
628503DocetaxelFDA approvedTUBB|Tu-stab761432CabazitaxelFDA approvedTUBB|Tu-stab
628503DocetaxelFDA approvedTUBB|Tu-stab763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
673596SN 38Clinical trialTOP1752ThioguanineFDA approvedDs|IMPDH2|IMPDH
673596SN 38Clinical trialTOP13053DactinomycinFDA approvedDb|RNA polymerase I
673596SN 38Clinical trialTOP13088ChlorambucilFDA approvedA7|AlkAg
673596SN 38Clinical trialTOP16396ThiotepaFDA approvedA7|AlkAg
673596SN 38Clinical trialTOP18806MelphalanFDA approvedA7|AlkAg
673596SN 38Clinical trialTOP113875HexamethylmelamineFDA approvedDb|AlkAg
673596SN 38Clinical trialTOP119893FluorouracilFDA approvedDs|Rs|TYMS
673596SN 38Clinical trialTOP127640FloxuridineFDA approvedDs|TYMS
673596SN 38Clinical trialTOP134462Uracil mustardFDA approvedA7|AlkAg
673596SN 38Clinical trialTOP145388DacarbazineFDA approvedA7|AlkAg
673596SN 38Clinical trialTOP149842Vinblastine sulfateFDA approvedTUBB|Tu-frag
673596SN 38Clinical trialTOP163878Cytarabine hydrochlorideFDA approvedDs
673596SN 38Clinical trialTOP167574Vincristine sulfateFDA approvedTUBB|Tu-frag
673596SN 38Clinical trialTOP171423Megestrol acetateFDA approvedHo|PGR
673596SN 38Clinical trialTOP179037LomustineFDA approvedA6|AlkAg
673596SN 38Clinical trialTOP182151Daunorubicin hydrochlorideFDA approvedTOP2
673596SN 38Clinical trialTOP1105014CladribineFDA approvedDs|ADA
673596SN 38Clinical trialTOP1118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
673596SN 38Clinical trialTOP1122758TretinoinFDA approvedHo|RXR|Differentiator
673596SN 38Clinical trialTOP1122819TeniposideFDA approvedTOP2
673596SN 38Clinical trialTOP1125973PaclitaxelFDA approvedTUBB|Tu-stab
673596SN 38Clinical trialTOP1141540EtoposideFDA approvedTOP2
673596SN 38Clinical trialTOP1169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
673596SN 38Clinical trialTOP1180973Tamoxifen citrateFDA approvedHo|SERM
673596SN 38Clinical trialTOP1226080RapamycinFDA approvedPK:STK,MTOR
673596SN 38Clinical trialTOP1241240CarboplatinFDA approvedA7|AlkAg
673596SN 38Clinical trialTOP1279836MitoxantroneFDA approvedTOP2
673596SN 38Clinical trialTOP1362856TemozolomideFDA approvedA7|AlkAg
673596SN 38Clinical trialTOP1606869ClofarabineFDA approvedDs
673596SN 38Clinical trialTOP1608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
673596SN 38Clinical trialTOP1613327Gemcitabine HCLFDA approvedDs
673596SN 38Clinical trialTOP1628503DocetaxelFDA approvedTUBB|Tu-stab
673596SN 38Clinical trialTOP1686673NelarabineFDA approvedDs
673596SN 38Clinical trialTOP1698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
673596SN 38Clinical trialTOP1712807CapecitabineFDA approvedDs|TYMS
673596SN 38Clinical trialTOP1713563ExemestaneFDA approvedHo|CYP19A1
673596SN 38Clinical trialTOP1715055GefitinibFDA approvedPK:YK,EGFR
673596SN 38Clinical trialTOP1719276FulvestrantFDA approvedAM|Ho|ESR|SERM
673596SN 38Clinical trialTOP1719344AnastrozoleFDA approvedHo|CYP19A1
673596SN 38Clinical trialTOP1719345LetrozoleFDA approvedHo|CYP19A1
673596SN 38Clinical trialTOP1719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
673596SN 38Clinical trialTOP1737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
673596SN 38Clinical trialTOP1743414ImatinibFDA approvedBCR-ABL|PK:YK
673596SN 38Clinical trialTOP1747599NilotinibFDA approvedBCR-ABL|PK:YK
673596SN 38Clinical trialTOP1747972LenalidomideFDA approvedFT|Immunomodulatory
673596SN 38Clinical trialTOP1747974RaloxifeneFDA approvedHo|SERM
673596SN 38Clinical trialTOP1749226AbirateroneFDA approvedHo|CYP17A1
673596SN 38Clinical trialTOP1753082VemurafenibFDA approvedPK:YK,BRAF
673596SN 38Clinical trialTOP1754143RomidepsinFDA approvedHDAC
673596SN 38Clinical trialTOP1755986VismodegibFDA approvedSMO|PK:YK
673596SN 38Clinical trialTOP1756645CrizotinibFDA approvedPK:YK,MET,ALK
673596SN 38Clinical trialTOP1757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
673596SN 38Clinical trialTOP1760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
673596SN 38Clinical trialTOP1761432CabazitaxelFDA approvedTUBB|Tu-stab
673596SN 38Clinical trialTOP1763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
681239Proscript boronic acidFDA approvedPSM740MethotrexateFDA approvedDf|DHFR
681239Proscript boronic acidFDA approvedPSM750BusulfanFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM752ThioguanineFDA approvedDs|IMPDH2|IMPDH
681239Proscript boronic acidFDA approvedPSM7556-MercaptopurineFDA approvedDs|PPAT
681239Proscript boronic acidFDA approvedPSM762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM1390AllopurinolFDA approvedAM|XDH
681239Proscript boronic acidFDA approvedPSM3053DactinomycinFDA approvedDb|RNA polymerase I
681239Proscript boronic acidFDA approvedPSM3088ChlorambucilFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM6396ThiotepaFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM8806MelphalanFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM9706Triethylenemelamine-A7|AlkAg
681239Proscript boronic acidFDA approvedPSM13875HexamethylmelamineFDA approvedDb|AlkAg
681239Proscript boronic acidFDA approvedPSM14229QuinacrineClinical trialDb|AP
681239Proscript boronic acidFDA approvedPSM18509Aminolevulinic Acid HydrochlorideFDA approvedAM
681239Proscript boronic acidFDA approvedPSM19893FluorouracilFDA approvedDs|Rs|TYMS
681239Proscript boronic acidFDA approvedPSM24559MithramycinFDA approvedDb|Rs
681239Proscript boronic acidFDA approvedPSM25154PipobromanFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM26271CyclophosphamideFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM26980MitomycinFDA approvedA2|AlkAg
681239Proscript boronic acidFDA approvedPSM27640FloxuridineFDA approvedDs|TYMS
681239Proscript boronic acidFDA approvedPSM32065HydroxyureaFDA approvedAM|Dr
681239Proscript boronic acidFDA approvedPSM34462Uracil mustardFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
681239Proscript boronic acidFDA approvedPSM45388DacarbazineFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM459238-MethoxypsoralenFDA approvedDb
681239Proscript boronic acidFDA approvedPSM49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
681239Proscript boronic acidFDA approvedPSM63878Cytarabine hydrochlorideFDA approvedDs
681239Proscript boronic acidFDA approvedPSM66847ThalidomideFDA approvedAng|Immunomodulatory
681239Proscript boronic acidFDA approvedPSM67574Vincristine sulfateFDA approvedTUBB|Tu-frag
681239Proscript boronic acidFDA approvedPSM71423Megestrol acetateFDA approvedHo|PGR
681239Proscript boronic acidFDA approvedPSM79037LomustineFDA approvedA6|AlkAg
681239Proscript boronic acidFDA approvedPSM82151Daunorubicin hydrochlorideFDA approvedTOP2
681239Proscript boronic acidFDA approvedPSM85998StreptozocinFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM102816AzacitidineFDA approvedDNMT
681239Proscript boronic acidFDA approvedPSM105014CladribineFDA approvedDs|ADA
681239Proscript boronic acidFDA approvedPSM109724IfosfamideFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
681239Proscript boronic acidFDA approvedPSM122758TretinoinFDA approvedHo|RXR|Differentiator
681239Proscript boronic acidFDA approvedPSM122819TeniposideFDA approvedTOP2
681239Proscript boronic acidFDA approvedPSM123127Doxorubicin hydrochlorideFDA approvedTOP2
681239Proscript boronic acidFDA approvedPSM125066BleomycinFDA approvedDb
681239Proscript boronic acidFDA approvedPSM125973PaclitaxelFDA approvedTUBB|Tu-stab
681239Proscript boronic acidFDA approvedPSM127716DecitabineFDA approvedAM|DNMT
681239Proscript boronic acidFDA approvedPSM138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
681239Proscript boronic acidFDA approvedPSM141540EtoposideFDA approvedTOP2
681239Proscript boronic acidFDA approvedPSM169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
681239Proscript boronic acidFDA approvedPSM180973Tamoxifen citrateFDA approvedHo|SERM
681239Proscript boronic acidFDA approvedPSM218321PentostatinFDA approvedDs|AM|ADA
681239Proscript boronic acidFDA approvedPSM226080RapamycinFDA approvedPK:STK,MTOR
681239Proscript boronic acidFDA approvedPSM241240CarboplatinFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM246131ValrubicinFDA approvedTOP2
681239Proscript boronic acidFDA approvedPSM266046OxaliplatinFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM279836MitoxantroneFDA approvedTOP2
681239Proscript boronic acidFDA approvedPSM296961EthiofosFDA approvedRP
681239Proscript boronic acidFDA approvedPSM362856TemozolomideFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod
681239Proscript boronic acidFDA approvedPSM409962CarmustineFDA approvedA7|AlkAg
681239Proscript boronic acidFDA approvedPSM606869ClofarabineFDA approvedDs
681239Proscript boronic acidFDA approvedPSM608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
681239Proscript boronic acidFDA approvedPSM609699Topotecan hydrochlorideFDA approvedTOP1
681239Proscript boronic acidFDA approvedPSM613327Gemcitabine HCLFDA approvedDs
681239Proscript boronic acidFDA approvedPSM628503DocetaxelFDA approvedTUBB|Tu-stab
681239Proscript boronic acidFDA approvedPSM673596SN 38Clinical trialTOP1
681239Proscript boronic acidFDA approvedPSM686673NelarabineFDA approvedDs
681239Proscript boronic acidFDA approvedPSM698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
681239Proscript boronic acidFDA approvedPSM701852VorinostatFDA approvedHDAC
681239Proscript boronic acidFDA approvedPSM702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg
681239Proscript boronic acidFDA approvedPSM712807CapecitabineFDA approvedDs|TYMS
681239Proscript boronic acidFDA approvedPSM713563ExemestaneFDA approvedHo|CYP19A1
681239Proscript boronic acidFDA approvedPSM715055GefitinibFDA approvedPK:YK,EGFR
681239Proscript boronic acidFDA approvedPSM718781Erlotinib HCLFDA approvedPK:YK,EGFR
681239Proscript boronic acidFDA approvedPSM719276FulvestrantFDA approvedAM|Ho|ESR|SERM
681239Proscript boronic acidFDA approvedPSM719344AnastrozoleFDA approvedHo|CYP19A1
681239Proscript boronic acidFDA approvedPSM719345LetrozoleFDA approvedHo|CYP19A1
681239Proscript boronic acidFDA approvedPSM719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
681239Proscript boronic acidFDA approvedPSM721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
681239Proscript boronic acidFDA approvedPSM732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
681239Proscript boronic acidFDA approvedPSM733504EverolimusFDA approvedPK:STK,MTOR
681239Proscript boronic acidFDA approvedPSM737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
681239Proscript boronic acidFDA approvedPSM743414ImatinibFDA approvedBCR-ABL|PK:YK
681239Proscript boronic acidFDA approvedPSM745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
681239Proscript boronic acidFDA approvedPSM747599NilotinibFDA approvedBCR-ABL|PK:YK
681239Proscript boronic acidFDA approvedPSM747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
681239Proscript boronic acidFDA approvedPSM747972LenalidomideFDA approvedFT|Immunomodulatory
681239Proscript boronic acidFDA approvedPSM747973IxabepiloneFDA approvedTUBB|Tu-stab
681239Proscript boronic acidFDA approvedPSM747974RaloxifeneFDA approvedHo|SERM
681239Proscript boronic acidFDA approvedPSM749226AbirateroneFDA approvedHo|CYP17A1
681239Proscript boronic acidFDA approvedPSM750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
681239Proscript boronic acidFDA approvedPSM753082VemurafenibFDA approvedPK:YK,BRAF
681239Proscript boronic acidFDA approvedPSM754143RomidepsinFDA approvedHDAC
681239Proscript boronic acidFDA approvedPSM754230PralatrexateFDA approvedDf|CTNNB1|DHFR
681239Proscript boronic acidFDA approvedPSM755986VismodegibFDA approvedSMO|PK:YK
681239Proscript boronic acidFDA approvedPSM756645CrizotinibFDA approvedPK:YK,MET,ALK
681239Proscript boronic acidFDA approvedPSM757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
681239Proscript boronic acidFDA approvedPSM760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
681239Proscript boronic acidFDA approvedPSM761432CabazitaxelFDA approvedTUBB|Tu-stab
681239Proscript boronic acidFDA approvedPSM763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
686673NelarabineFDA approvedDs740MethotrexateFDA approvedDf|DHFR
686673NelarabineFDA approvedDs752ThioguanineFDA approvedDs|IMPDH2|IMPDH
686673NelarabineFDA approvedDs7556-MercaptopurineFDA approvedDs|PPAT
686673NelarabineFDA approvedDs3053DactinomycinFDA approvedDb|RNA polymerase I
686673NelarabineFDA approvedDs3088ChlorambucilFDA approvedA7|AlkAg
686673NelarabineFDA approvedDs6396ThiotepaFDA approvedA7|AlkAg
686673NelarabineFDA approvedDs8806MelphalanFDA approvedA7|AlkAg
686673NelarabineFDA approvedDs13875HexamethylmelamineFDA approvedDb|AlkAg
686673NelarabineFDA approvedDs19893FluorouracilFDA approvedDs|Rs|TYMS
686673NelarabineFDA approvedDs24559MithramycinFDA approvedDb|Rs
686673NelarabineFDA approvedDs27640FloxuridineFDA approvedDs|TYMS
686673NelarabineFDA approvedDs32065HydroxyureaFDA approvedAM|Dr
686673NelarabineFDA approvedDs34462Uracil mustardFDA approvedA7|AlkAg
686673NelarabineFDA approvedDs38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
686673NelarabineFDA approvedDs45388DacarbazineFDA approvedA7|AlkAg
686673NelarabineFDA approvedDs49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
686673NelarabineFDA approvedDs63878Cytarabine hydrochlorideFDA approvedDs
686673NelarabineFDA approvedDs67574Vincristine sulfateFDA approvedTUBB|Tu-frag
686673NelarabineFDA approvedDs71423Megestrol acetateFDA approvedHo|PGR
686673NelarabineFDA approvedDs79037LomustineFDA approvedA6|AlkAg
686673NelarabineFDA approvedDs82151Daunorubicin hydrochlorideFDA approvedTOP2
686673NelarabineFDA approvedDs105014CladribineFDA approvedDs|ADA
686673NelarabineFDA approvedDs118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
686673NelarabineFDA approvedDs122758TretinoinFDA approvedHo|RXR|Differentiator
686673NelarabineFDA approvedDs122819TeniposideFDA approvedTOP2
686673NelarabineFDA approvedDs138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
686673NelarabineFDA approvedDs141540EtoposideFDA approvedTOP2
686673NelarabineFDA approvedDs169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
686673NelarabineFDA approvedDs180973Tamoxifen citrateFDA approvedHo|SERM
686673NelarabineFDA approvedDs241240CarboplatinFDA approvedA7|AlkAg
686673NelarabineFDA approvedDs279836MitoxantroneFDA approvedTOP2
686673NelarabineFDA approvedDs362856TemozolomideFDA approvedA7|AlkAg
686673NelarabineFDA approvedDs608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
686673NelarabineFDA approvedDs698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
686673NelarabineFDA approvedDs713563ExemestaneFDA approvedHo|CYP19A1
686673NelarabineFDA approvedDs715055GefitinibFDA approvedPK:YK,EGFR
686673NelarabineFDA approvedDs719276FulvestrantFDA approvedAM|Ho|ESR|SERM
686673NelarabineFDA approvedDs719344AnastrozoleFDA approvedHo|CYP19A1
686673NelarabineFDA approvedDs719345LetrozoleFDA approvedHo|CYP19A1
686673NelarabineFDA approvedDs719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
686673NelarabineFDA approvedDs737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
686673NelarabineFDA approvedDs743414ImatinibFDA approvedBCR-ABL|PK:YK
686673NelarabineFDA approvedDs747599NilotinibFDA approvedBCR-ABL|PK:YK
686673NelarabineFDA approvedDs747972LenalidomideFDA approvedFT|Immunomodulatory
686673NelarabineFDA approvedDs747974RaloxifeneFDA approvedHo|SERM
686673NelarabineFDA approvedDs749226AbirateroneFDA approvedHo|CYP17A1
686673NelarabineFDA approvedDs753082VemurafenibFDA approvedPK:YK,BRAF
686673NelarabineFDA approvedDs755986VismodegibFDA approvedSMO|PK:YK
686673NelarabineFDA approvedDs756645CrizotinibFDA approvedPK:YK,MET,ALK
686673NelarabineFDA approvedDs757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
686673NelarabineFDA approvedDs760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
686673NelarabineFDA approvedDs761432CabazitaxelFDA approvedTUBB|Tu-stab
686673NelarabineFDA approvedDs763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS9706Triethylenemelamine-A7|AlkAg
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS123127Doxorubicin hydrochlorideFDA approvedTOP2
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS713563ExemestaneFDA approvedHo|CYP19A1
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS715055GefitinibFDA approvedPK:YK,EGFR
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS747972LenalidomideFDA approvedFT|Immunomodulatory
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS747974RaloxifeneFDA approvedHo|SERM
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS749226AbirateroneFDA approvedHo|CYP17A1
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS753082VemurafenibFDA approvedPK:YK,BRAF
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS755986VismodegibFDA approvedSMO|PK:YK
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS756645CrizotinibFDA approvedPK:YK,MET,ALK
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS761432CabazitaxelFDA approvedTUBB|Tu-stab
698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
701852VorinostatFDA approvedHDAC752ThioguanineFDA approvedDs|IMPDH2|IMPDH
701852VorinostatFDA approvedHDAC3053DactinomycinFDA approvedDb|RNA polymerase I
701852VorinostatFDA approvedHDAC3088ChlorambucilFDA approvedA7|AlkAg
701852VorinostatFDA approvedHDAC6396ThiotepaFDA approvedA7|AlkAg
701852VorinostatFDA approvedHDAC8806MelphalanFDA approvedA7|AlkAg
701852VorinostatFDA approvedHDAC13875HexamethylmelamineFDA approvedDb|AlkAg
701852VorinostatFDA approvedHDAC19893FluorouracilFDA approvedDs|Rs|TYMS
701852VorinostatFDA approvedHDAC27640FloxuridineFDA approvedDs|TYMS
701852VorinostatFDA approvedHDAC34462Uracil mustardFDA approvedA7|AlkAg
701852VorinostatFDA approvedHDAC45388DacarbazineFDA approvedA7|AlkAg
701852VorinostatFDA approvedHDAC49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
701852VorinostatFDA approvedHDAC63878Cytarabine hydrochlorideFDA approvedDs
701852VorinostatFDA approvedHDAC67574Vincristine sulfateFDA approvedTUBB|Tu-frag
701852VorinostatFDA approvedHDAC71423Megestrol acetateFDA approvedHo|PGR
701852VorinostatFDA approvedHDAC79037LomustineFDA approvedA6|AlkAg
701852VorinostatFDA approvedHDAC82151Daunorubicin hydrochlorideFDA approvedTOP2
701852VorinostatFDA approvedHDAC102816AzacitidineFDA approvedDNMT
701852VorinostatFDA approvedHDAC105014CladribineFDA approvedDs|ADA
701852VorinostatFDA approvedHDAC118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
701852VorinostatFDA approvedHDAC122758TretinoinFDA approvedHo|RXR|Differentiator
701852VorinostatFDA approvedHDAC122819TeniposideFDA approvedTOP2
701852VorinostatFDA approvedHDAC125973PaclitaxelFDA approvedTUBB|Tu-stab
701852VorinostatFDA approvedHDAC141540EtoposideFDA approvedTOP2
701852VorinostatFDA approvedHDAC169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
701852VorinostatFDA approvedHDAC180973Tamoxifen citrateFDA approvedHo|SERM
701852VorinostatFDA approvedHDAC226080RapamycinFDA approvedPK:STK,MTOR
701852VorinostatFDA approvedHDAC241240CarboplatinFDA approvedA7|AlkAg
701852VorinostatFDA approvedHDAC246131ValrubicinFDA approvedTOP2
701852VorinostatFDA approvedHDAC279836MitoxantroneFDA approvedTOP2
701852VorinostatFDA approvedHDAC362856TemozolomideFDA approvedA7|AlkAg
701852VorinostatFDA approvedHDAC606869ClofarabineFDA approvedDs
701852VorinostatFDA approvedHDAC608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
701852VorinostatFDA approvedHDAC613327Gemcitabine HCLFDA approvedDs
701852VorinostatFDA approvedHDAC628503DocetaxelFDA approvedTUBB|Tu-stab
701852VorinostatFDA approvedHDAC673596SN 38Clinical trialTOP1
701852VorinostatFDA approvedHDAC686673NelarabineFDA approvedDs
701852VorinostatFDA approvedHDAC698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
701852VorinostatFDA approvedHDAC712807CapecitabineFDA approvedDs|TYMS
701852VorinostatFDA approvedHDAC713563ExemestaneFDA approvedHo|CYP19A1
701852VorinostatFDA approvedHDAC715055GefitinibFDA approvedPK:YK,EGFR
701852VorinostatFDA approvedHDAC719344AnastrozoleFDA approvedHo|CYP19A1
701852VorinostatFDA approvedHDAC719345LetrozoleFDA approvedHo|CYP19A1
701852VorinostatFDA approvedHDAC719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
701852VorinostatFDA approvedHDAC737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
701852VorinostatFDA approvedHDAC743414ImatinibFDA approvedBCR-ABL|PK:YK
701852VorinostatFDA approvedHDAC747599NilotinibFDA approvedBCR-ABL|PK:YK
701852VorinostatFDA approvedHDAC747972LenalidomideFDA approvedFT|Immunomodulatory
701852VorinostatFDA approvedHDAC747974RaloxifeneFDA approvedHo|SERM
701852VorinostatFDA approvedHDAC749226AbirateroneFDA approvedHo|CYP17A1
701852VorinostatFDA approvedHDAC753082VemurafenibFDA approvedPK:YK,BRAF
701852VorinostatFDA approvedHDAC754143RomidepsinFDA approvedHDAC
701852VorinostatFDA approvedHDAC755986VismodegibFDA approvedSMO|PK:YK
701852VorinostatFDA approvedHDAC756645CrizotinibFDA approvedPK:YK,MET,ALK
701852VorinostatFDA approvedHDAC757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
701852VorinostatFDA approvedHDAC760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
701852VorinostatFDA approvedHDAC761432CabazitaxelFDA approvedTUBB|Tu-stab
701852VorinostatFDA approvedHDAC763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg740MethotrexateFDA approvedDf|DHFR
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg750BusulfanFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg752ThioguanineFDA approvedDs|IMPDH2|IMPDH
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg7556-MercaptopurineFDA approvedDs|PPAT
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg1390AllopurinolFDA approvedAM|XDH
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg3053DactinomycinFDA approvedDb|RNA polymerase I
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg3088ChlorambucilFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg6396ThiotepaFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg8806MelphalanFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg9706Triethylenemelamine-A7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg13875HexamethylmelamineFDA approvedDb|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg14229QuinacrineClinical trialDb|AP
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg18509Aminolevulinic Acid HydrochlorideFDA approvedAM
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg19893FluorouracilFDA approvedDs|Rs|TYMS
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg24559MithramycinFDA approvedDb|Rs
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg25154PipobromanFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg26271CyclophosphamideFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg26980MitomycinFDA approvedA2|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg27640FloxuridineFDA approvedDs|TYMS
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg32065HydroxyureaFDA approvedAM|Dr
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg34462Uracil mustardFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg45388DacarbazineFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg459238-MethoxypsoralenFDA approvedDb
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg63878Cytarabine hydrochlorideFDA approvedDs
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg66847ThalidomideFDA approvedAng|Immunomodulatory
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg67574Vincristine sulfateFDA approvedTUBB|Tu-frag
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg71423Megestrol acetateFDA approvedHo|PGR
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg79037LomustineFDA approvedA6|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg82151Daunorubicin hydrochlorideFDA approvedTOP2
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg85998StreptozocinFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg102816AzacitidineFDA approvedDNMT
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg105014CladribineFDA approvedDs|ADA
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg109724IfosfamideFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg122758TretinoinFDA approvedHo|RXR|Differentiator
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg122819TeniposideFDA approvedTOP2
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg123127Doxorubicin hydrochlorideFDA approvedTOP2
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg125066BleomycinFDA approvedDb
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg125973PaclitaxelFDA approvedTUBB|Tu-stab
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg127716DecitabineFDA approvedAM|DNMT
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg141540EtoposideFDA approvedTOP2
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg180973Tamoxifen citrateFDA approvedHo|SERM
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg218321PentostatinFDA approvedDs|AM|ADA
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg226080RapamycinFDA approvedPK:STK,MTOR
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg241240CarboplatinFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg246131ValrubicinFDA approvedTOP2
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg266046OxaliplatinFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg279836MitoxantroneFDA approvedTOP2
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg296961EthiofosFDA approvedRP
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg362856TemozolomideFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg409962CarmustineFDA approvedA7|AlkAg
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg606869ClofarabineFDA approvedDs
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg609699Topotecan hydrochlorideFDA approvedTOP1
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg613327Gemcitabine HCLFDA approvedDs
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg628503DocetaxelFDA approvedTUBB|Tu-stab
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg673596SN 38Clinical trialTOP1
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg686673NelarabineFDA approvedDs
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg701852VorinostatFDA approvedHDAC
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg712807CapecitabineFDA approvedDs|TYMS
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg713563ExemestaneFDA approvedHo|CYP19A1
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg715055GefitinibFDA approvedPK:YK,EGFR
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg719276FulvestrantFDA approvedAM|Ho|ESR|SERM
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg719344AnastrozoleFDA approvedHo|CYP19A1
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg719345LetrozoleFDA approvedHo|CYP19A1
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg733504EverolimusFDA approvedPK:STK,MTOR
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg743414ImatinibFDA approvedBCR-ABL|PK:YK
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg747599NilotinibFDA approvedBCR-ABL|PK:YK
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg747972LenalidomideFDA approvedFT|Immunomodulatory
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg747973IxabepiloneFDA approvedTUBB|Tu-stab
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg747974RaloxifeneFDA approvedHo|SERM
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg749226AbirateroneFDA approvedHo|CYP17A1
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg753082VemurafenibFDA approvedPK:YK,BRAF
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg754143RomidepsinFDA approvedHDAC
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg754230PralatrexateFDA approvedDf|CTNNB1|DHFR
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg755986VismodegibFDA approvedSMO|PK:YK
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg756645CrizotinibFDA approvedPK:YK,MET,ALK
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg761432CabazitaxelFDA approvedTUBB|Tu-stab
702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
712807CapecitabineFDA approvedDs|TYMS740MethotrexateFDA approvedDf|DHFR
712807CapecitabineFDA approvedDs|TYMS752ThioguanineFDA approvedDs|IMPDH2|IMPDH
712807CapecitabineFDA approvedDs|TYMS7556-MercaptopurineFDA approvedDs|PPAT
712807CapecitabineFDA approvedDs|TYMS3053DactinomycinFDA approvedDb|RNA polymerase I
712807CapecitabineFDA approvedDs|TYMS3088ChlorambucilFDA approvedA7|AlkAg
712807CapecitabineFDA approvedDs|TYMS6396ThiotepaFDA approvedA7|AlkAg
712807CapecitabineFDA approvedDs|TYMS8806MelphalanFDA approvedA7|AlkAg
712807CapecitabineFDA approvedDs|TYMS13875HexamethylmelamineFDA approvedDb|AlkAg
712807CapecitabineFDA approvedDs|TYMS19893FluorouracilFDA approvedDs|Rs|TYMS
712807CapecitabineFDA approvedDs|TYMS24559MithramycinFDA approvedDb|Rs
712807CapecitabineFDA approvedDs|TYMS27640FloxuridineFDA approvedDs|TYMS
712807CapecitabineFDA approvedDs|TYMS32065HydroxyureaFDA approvedAM|Dr
712807CapecitabineFDA approvedDs|TYMS34462Uracil mustardFDA approvedA7|AlkAg
712807CapecitabineFDA approvedDs|TYMS38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
712807CapecitabineFDA approvedDs|TYMS45388DacarbazineFDA approvedA7|AlkAg
712807CapecitabineFDA approvedDs|TYMS49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
712807CapecitabineFDA approvedDs|TYMS63878Cytarabine hydrochlorideFDA approvedDs
712807CapecitabineFDA approvedDs|TYMS67574Vincristine sulfateFDA approvedTUBB|Tu-frag
712807CapecitabineFDA approvedDs|TYMS71423Megestrol acetateFDA approvedHo|PGR
712807CapecitabineFDA approvedDs|TYMS79037LomustineFDA approvedA6|AlkAg
712807CapecitabineFDA approvedDs|TYMS82151Daunorubicin hydrochlorideFDA approvedTOP2
712807CapecitabineFDA approvedDs|TYMS105014CladribineFDA approvedDs|ADA
712807CapecitabineFDA approvedDs|TYMS118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
712807CapecitabineFDA approvedDs|TYMS122758TretinoinFDA approvedHo|RXR|Differentiator
712807CapecitabineFDA approvedDs|TYMS122819TeniposideFDA approvedTOP2
712807CapecitabineFDA approvedDs|TYMS138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
712807CapecitabineFDA approvedDs|TYMS141540EtoposideFDA approvedTOP2
712807CapecitabineFDA approvedDs|TYMS169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
712807CapecitabineFDA approvedDs|TYMS180973Tamoxifen citrateFDA approvedHo|SERM
712807CapecitabineFDA approvedDs|TYMS241240CarboplatinFDA approvedA7|AlkAg
712807CapecitabineFDA approvedDs|TYMS246131ValrubicinFDA approvedTOP2
712807CapecitabineFDA approvedDs|TYMS279836MitoxantroneFDA approvedTOP2
712807CapecitabineFDA approvedDs|TYMS362856TemozolomideFDA approvedA7|AlkAg
712807CapecitabineFDA approvedDs|TYMS608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
712807CapecitabineFDA approvedDs|TYMS686673NelarabineFDA approvedDs
712807CapecitabineFDA approvedDs|TYMS698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
712807CapecitabineFDA approvedDs|TYMS713563ExemestaneFDA approvedHo|CYP19A1
712807CapecitabineFDA approvedDs|TYMS715055GefitinibFDA approvedPK:YK,EGFR
712807CapecitabineFDA approvedDs|TYMS719276FulvestrantFDA approvedAM|Ho|ESR|SERM
712807CapecitabineFDA approvedDs|TYMS719344AnastrozoleFDA approvedHo|CYP19A1
712807CapecitabineFDA approvedDs|TYMS719345LetrozoleFDA approvedHo|CYP19A1
712807CapecitabineFDA approvedDs|TYMS719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
712807CapecitabineFDA approvedDs|TYMS737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
712807CapecitabineFDA approvedDs|TYMS743414ImatinibFDA approvedBCR-ABL|PK:YK
712807CapecitabineFDA approvedDs|TYMS747599NilotinibFDA approvedBCR-ABL|PK:YK
712807CapecitabineFDA approvedDs|TYMS747972LenalidomideFDA approvedFT|Immunomodulatory
712807CapecitabineFDA approvedDs|TYMS747974RaloxifeneFDA approvedHo|SERM
712807CapecitabineFDA approvedDs|TYMS749226AbirateroneFDA approvedHo|CYP17A1
712807CapecitabineFDA approvedDs|TYMS753082VemurafenibFDA approvedPK:YK,BRAF
712807CapecitabineFDA approvedDs|TYMS755986VismodegibFDA approvedSMO|PK:YK
712807CapecitabineFDA approvedDs|TYMS756645CrizotinibFDA approvedPK:YK,MET,ALK
712807CapecitabineFDA approvedDs|TYMS757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
712807CapecitabineFDA approvedDs|TYMS760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
712807CapecitabineFDA approvedDs|TYMS761432CabazitaxelFDA approvedTUBB|Tu-stab
712807CapecitabineFDA approvedDs|TYMS763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
713563ExemestaneFDA approvedHo|CYP19A19706Triethylenemelamine-A7|AlkAg
713563ExemestaneFDA approvedHo|CYP19A1123127Doxorubicin hydrochlorideFDA approvedTOP2
713563ExemestaneFDA approvedHo|CYP19A1715055GefitinibFDA approvedPK:YK,EGFR
713563ExemestaneFDA approvedHo|CYP19A1737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
713563ExemestaneFDA approvedHo|CYP19A1747972LenalidomideFDA approvedFT|Immunomodulatory
713563ExemestaneFDA approvedHo|CYP19A1747974RaloxifeneFDA approvedHo|SERM
713563ExemestaneFDA approvedHo|CYP19A1749226AbirateroneFDA approvedHo|CYP17A1
713563ExemestaneFDA approvedHo|CYP19A1753082VemurafenibFDA approvedPK:YK,BRAF
713563ExemestaneFDA approvedHo|CYP19A1755986VismodegibFDA approvedSMO|PK:YK
713563ExemestaneFDA approvedHo|CYP19A1756645CrizotinibFDA approvedPK:YK,MET,ALK
713563ExemestaneFDA approvedHo|CYP19A1757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
713563ExemestaneFDA approvedHo|CYP19A1760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
713563ExemestaneFDA approvedHo|CYP19A1761432CabazitaxelFDA approvedTUBB|Tu-stab
713563ExemestaneFDA approvedHo|CYP19A1763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
715055GefitinibFDA approvedPK:YK,EGFR9706Triethylenemelamine-A7|AlkAg
715055GefitinibFDA approvedPK:YK,EGFR123127Doxorubicin hydrochlorideFDA approvedTOP2
715055GefitinibFDA approvedPK:YK,EGFR737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
715055GefitinibFDA approvedPK:YK,EGFR747972LenalidomideFDA approvedFT|Immunomodulatory
715055GefitinibFDA approvedPK:YK,EGFR747974RaloxifeneFDA approvedHo|SERM
715055GefitinibFDA approvedPK:YK,EGFR749226AbirateroneFDA approvedHo|CYP17A1
715055GefitinibFDA approvedPK:YK,EGFR753082VemurafenibFDA approvedPK:YK,BRAF
715055GefitinibFDA approvedPK:YK,EGFR755986VismodegibFDA approvedSMO|PK:YK
715055GefitinibFDA approvedPK:YK,EGFR756645CrizotinibFDA approvedPK:YK,MET,ALK
715055GefitinibFDA approvedPK:YK,EGFR757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
715055GefitinibFDA approvedPK:YK,EGFR760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
715055GefitinibFDA approvedPK:YK,EGFR761432CabazitaxelFDA approvedTUBB|Tu-stab
715055GefitinibFDA approvedPK:YK,EGFR763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
718781Erlotinib HCLFDA approvedPK:YK,EGFR740MethotrexateFDA approvedDf|DHFR
718781Erlotinib HCLFDA approvedPK:YK,EGFR750BusulfanFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR752ThioguanineFDA approvedDs|IMPDH2|IMPDH
718781Erlotinib HCLFDA approvedPK:YK,EGFR7556-MercaptopurineFDA approvedDs|PPAT
718781Erlotinib HCLFDA approvedPK:YK,EGFR762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR1390AllopurinolFDA approvedAM|XDH
718781Erlotinib HCLFDA approvedPK:YK,EGFR3053DactinomycinFDA approvedDb|RNA polymerase I
718781Erlotinib HCLFDA approvedPK:YK,EGFR3088ChlorambucilFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR6396ThiotepaFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR8806MelphalanFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR9706Triethylenemelamine-A7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR13875HexamethylmelamineFDA approvedDb|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR14229QuinacrineClinical trialDb|AP
718781Erlotinib HCLFDA approvedPK:YK,EGFR18509Aminolevulinic Acid HydrochlorideFDA approvedAM
718781Erlotinib HCLFDA approvedPK:YK,EGFR19893FluorouracilFDA approvedDs|Rs|TYMS
718781Erlotinib HCLFDA approvedPK:YK,EGFR24559MithramycinFDA approvedDb|Rs
718781Erlotinib HCLFDA approvedPK:YK,EGFR25154PipobromanFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR26271CyclophosphamideFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR26980MitomycinFDA approvedA2|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR27640FloxuridineFDA approvedDs|TYMS
718781Erlotinib HCLFDA approvedPK:YK,EGFR32065HydroxyureaFDA approvedAM|Dr
718781Erlotinib HCLFDA approvedPK:YK,EGFR34462Uracil mustardFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
718781Erlotinib HCLFDA approvedPK:YK,EGFR45388DacarbazineFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR459238-MethoxypsoralenFDA approvedDb
718781Erlotinib HCLFDA approvedPK:YK,EGFR49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
718781Erlotinib HCLFDA approvedPK:YK,EGFR63878Cytarabine hydrochlorideFDA approvedDs
718781Erlotinib HCLFDA approvedPK:YK,EGFR66847ThalidomideFDA approvedAng|Immunomodulatory
718781Erlotinib HCLFDA approvedPK:YK,EGFR67574Vincristine sulfateFDA approvedTUBB|Tu-frag
718781Erlotinib HCLFDA approvedPK:YK,EGFR71423Megestrol acetateFDA approvedHo|PGR
718781Erlotinib HCLFDA approvedPK:YK,EGFR77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR79037LomustineFDA approvedA6|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR82151Daunorubicin hydrochlorideFDA approvedTOP2
718781Erlotinib HCLFDA approvedPK:YK,EGFR85998StreptozocinFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR102816AzacitidineFDA approvedDNMT
718781Erlotinib HCLFDA approvedPK:YK,EGFR105014CladribineFDA approvedDs|ADA
718781Erlotinib HCLFDA approvedPK:YK,EGFR109724IfosfamideFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
718781Erlotinib HCLFDA approvedPK:YK,EGFR122758TretinoinFDA approvedHo|RXR|Differentiator
718781Erlotinib HCLFDA approvedPK:YK,EGFR122819TeniposideFDA approvedTOP2
718781Erlotinib HCLFDA approvedPK:YK,EGFR123127Doxorubicin hydrochlorideFDA approvedTOP2
718781Erlotinib HCLFDA approvedPK:YK,EGFR125066BleomycinFDA approvedDb
718781Erlotinib HCLFDA approvedPK:YK,EGFR125973PaclitaxelFDA approvedTUBB|Tu-stab
718781Erlotinib HCLFDA approvedPK:YK,EGFR127716DecitabineFDA approvedAM|DNMT
718781Erlotinib HCLFDA approvedPK:YK,EGFR138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR141540EtoposideFDA approvedTOP2
718781Erlotinib HCLFDA approvedPK:YK,EGFR169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
718781Erlotinib HCLFDA approvedPK:YK,EGFR180973Tamoxifen citrateFDA approvedHo|SERM
718781Erlotinib HCLFDA approvedPK:YK,EGFR218321PentostatinFDA approvedDs|AM|ADA
718781Erlotinib HCLFDA approvedPK:YK,EGFR226080RapamycinFDA approvedPK:STK,MTOR
718781Erlotinib HCLFDA approvedPK:YK,EGFR241240CarboplatinFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR246131ValrubicinFDA approvedTOP2
718781Erlotinib HCLFDA approvedPK:YK,EGFR266046OxaliplatinFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR279836MitoxantroneFDA approvedTOP2
718781Erlotinib HCLFDA approvedPK:YK,EGFR296961EthiofosFDA approvedRP
718781Erlotinib HCLFDA approvedPK:YK,EGFR362856TemozolomideFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod
718781Erlotinib HCLFDA approvedPK:YK,EGFR409962CarmustineFDA approvedA7|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR606869ClofarabineFDA approvedDs
718781Erlotinib HCLFDA approvedPK:YK,EGFR608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
718781Erlotinib HCLFDA approvedPK:YK,EGFR609699Topotecan hydrochlorideFDA approvedTOP1
718781Erlotinib HCLFDA approvedPK:YK,EGFR613327Gemcitabine HCLFDA approvedDs
718781Erlotinib HCLFDA approvedPK:YK,EGFR628503DocetaxelFDA approvedTUBB|Tu-stab
718781Erlotinib HCLFDA approvedPK:YK,EGFR673596SN 38Clinical trialTOP1
718781Erlotinib HCLFDA approvedPK:YK,EGFR686673NelarabineFDA approvedDs
718781Erlotinib HCLFDA approvedPK:YK,EGFR698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
718781Erlotinib HCLFDA approvedPK:YK,EGFR701852VorinostatFDA approvedHDAC
718781Erlotinib HCLFDA approvedPK:YK,EGFR702294Estramustine disodium phosphateFDA approvedA7|TUBB|AlkAg
718781Erlotinib HCLFDA approvedPK:YK,EGFR712807CapecitabineFDA approvedDs|TYMS
718781Erlotinib HCLFDA approvedPK:YK,EGFR713563ExemestaneFDA approvedHo|CYP19A1
718781Erlotinib HCLFDA approvedPK:YK,EGFR715055GefitinibFDA approvedPK:YK,EGFR
718781Erlotinib HCLFDA approvedPK:YK,EGFR719276FulvestrantFDA approvedAM|Ho|ESR|SERM
718781Erlotinib HCLFDA approvedPK:YK,EGFR719344AnastrozoleFDA approvedHo|CYP19A1
718781Erlotinib HCLFDA approvedPK:YK,EGFR719345LetrozoleFDA approvedHo|CYP19A1
718781Erlotinib HCLFDA approvedPK:YK,EGFR719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
718781Erlotinib HCLFDA approvedPK:YK,EGFR721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
718781Erlotinib HCLFDA approvedPK:YK,EGFR732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
718781Erlotinib HCLFDA approvedPK:YK,EGFR733504EverolimusFDA approvedPK:STK,MTOR
718781Erlotinib HCLFDA approvedPK:YK,EGFR737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
718781Erlotinib HCLFDA approvedPK:YK,EGFR743414ImatinibFDA approvedBCR-ABL|PK:YK
718781Erlotinib HCLFDA approvedPK:YK,EGFR745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
718781Erlotinib HCLFDA approvedPK:YK,EGFR747599NilotinibFDA approvedBCR-ABL|PK:YK
718781Erlotinib HCLFDA approvedPK:YK,EGFR747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
718781Erlotinib HCLFDA approvedPK:YK,EGFR747972LenalidomideFDA approvedFT|Immunomodulatory
718781Erlotinib HCLFDA approvedPK:YK,EGFR747973IxabepiloneFDA approvedTUBB|Tu-stab
718781Erlotinib HCLFDA approvedPK:YK,EGFR747974RaloxifeneFDA approvedHo|SERM
718781Erlotinib HCLFDA approvedPK:YK,EGFR749226AbirateroneFDA approvedHo|CYP17A1
718781Erlotinib HCLFDA approvedPK:YK,EGFR750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
718781Erlotinib HCLFDA approvedPK:YK,EGFR753082VemurafenibFDA approvedPK:YK,BRAF
718781Erlotinib HCLFDA approvedPK:YK,EGFR754143RomidepsinFDA approvedHDAC
718781Erlotinib HCLFDA approvedPK:YK,EGFR754230PralatrexateFDA approvedDf|CTNNB1|DHFR
718781Erlotinib HCLFDA approvedPK:YK,EGFR755986VismodegibFDA approvedSMO|PK:YK
718781Erlotinib HCLFDA approvedPK:YK,EGFR756645CrizotinibFDA approvedPK:YK,MET,ALK
718781Erlotinib HCLFDA approvedPK:YK,EGFR757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
718781Erlotinib HCLFDA approvedPK:YK,EGFR760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
718781Erlotinib HCLFDA approvedPK:YK,EGFR761432CabazitaxelFDA approvedTUBB|Tu-stab
718781Erlotinib HCLFDA approvedPK:YK,EGFR763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
719276FulvestrantFDA approvedAM|Ho|ESR|SERM752ThioguanineFDA approvedDs|IMPDH2|IMPDH
719276FulvestrantFDA approvedAM|Ho|ESR|SERM3053DactinomycinFDA approvedDb|RNA polymerase I
719276FulvestrantFDA approvedAM|Ho|ESR|SERM3088ChlorambucilFDA approvedA7|AlkAg
719276FulvestrantFDA approvedAM|Ho|ESR|SERM6396ThiotepaFDA approvedA7|AlkAg
719276FulvestrantFDA approvedAM|Ho|ESR|SERM8806MelphalanFDA approvedA7|AlkAg
719276FulvestrantFDA approvedAM|Ho|ESR|SERM9706Triethylenemelamine-A7|AlkAg
719276FulvestrantFDA approvedAM|Ho|ESR|SERM13875HexamethylmelamineFDA approvedDb|AlkAg
719276FulvestrantFDA approvedAM|Ho|ESR|SERM19893FluorouracilFDA approvedDs|Rs|TYMS
719276FulvestrantFDA approvedAM|Ho|ESR|SERM24559MithramycinFDA approvedDb|Rs
719276FulvestrantFDA approvedAM|Ho|ESR|SERM27640FloxuridineFDA approvedDs|TYMS
719276FulvestrantFDA approvedAM|Ho|ESR|SERM32065HydroxyureaFDA approvedAM|Dr
719276FulvestrantFDA approvedAM|Ho|ESR|SERM34462Uracil mustardFDA approvedA7|AlkAg
719276FulvestrantFDA approvedAM|Ho|ESR|SERM38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
719276FulvestrantFDA approvedAM|Ho|ESR|SERM45388DacarbazineFDA approvedA7|AlkAg
719276FulvestrantFDA approvedAM|Ho|ESR|SERM49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
719276FulvestrantFDA approvedAM|Ho|ESR|SERM63878Cytarabine hydrochlorideFDA approvedDs
719276FulvestrantFDA approvedAM|Ho|ESR|SERM67574Vincristine sulfateFDA approvedTUBB|Tu-frag
719276FulvestrantFDA approvedAM|Ho|ESR|SERM71423Megestrol acetateFDA approvedHo|PGR
719276FulvestrantFDA approvedAM|Ho|ESR|SERM79037LomustineFDA approvedA6|AlkAg
719276FulvestrantFDA approvedAM|Ho|ESR|SERM82151Daunorubicin hydrochlorideFDA approvedTOP2
719276FulvestrantFDA approvedAM|Ho|ESR|SERM102816AzacitidineFDA approvedDNMT
719276FulvestrantFDA approvedAM|Ho|ESR|SERM105014CladribineFDA approvedDs|ADA
719276FulvestrantFDA approvedAM|Ho|ESR|SERM118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
719276FulvestrantFDA approvedAM|Ho|ESR|SERM122758TretinoinFDA approvedHo|RXR|Differentiator
719276FulvestrantFDA approvedAM|Ho|ESR|SERM122819TeniposideFDA approvedTOP2
719276FulvestrantFDA approvedAM|Ho|ESR|SERM123127Doxorubicin hydrochlorideFDA approvedTOP2
719276FulvestrantFDA approvedAM|Ho|ESR|SERM125066BleomycinFDA approvedDb
719276FulvestrantFDA approvedAM|Ho|ESR|SERM125973PaclitaxelFDA approvedTUBB|Tu-stab
719276FulvestrantFDA approvedAM|Ho|ESR|SERM138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
719276FulvestrantFDA approvedAM|Ho|ESR|SERM141540EtoposideFDA approvedTOP2
719276FulvestrantFDA approvedAM|Ho|ESR|SERM169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
719276FulvestrantFDA approvedAM|Ho|ESR|SERM180973Tamoxifen citrateFDA approvedHo|SERM
719276FulvestrantFDA approvedAM|Ho|ESR|SERM226080RapamycinFDA approvedPK:STK,MTOR
719276FulvestrantFDA approvedAM|Ho|ESR|SERM241240CarboplatinFDA approvedA7|AlkAg
719276FulvestrantFDA approvedAM|Ho|ESR|SERM246131ValrubicinFDA approvedTOP2
719276FulvestrantFDA approvedAM|Ho|ESR|SERM279836MitoxantroneFDA approvedTOP2
719276FulvestrantFDA approvedAM|Ho|ESR|SERM362856TemozolomideFDA approvedA7|AlkAg
719276FulvestrantFDA approvedAM|Ho|ESR|SERM606869ClofarabineFDA approvedDs
719276FulvestrantFDA approvedAM|Ho|ESR|SERM608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
719276FulvestrantFDA approvedAM|Ho|ESR|SERM613327Gemcitabine HCLFDA approvedDs
719276FulvestrantFDA approvedAM|Ho|ESR|SERM673596SN 38Clinical trialTOP1
719276FulvestrantFDA approvedAM|Ho|ESR|SERM686673NelarabineFDA approvedDs
719276FulvestrantFDA approvedAM|Ho|ESR|SERM698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
719276FulvestrantFDA approvedAM|Ho|ESR|SERM701852VorinostatFDA approvedHDAC
719276FulvestrantFDA approvedAM|Ho|ESR|SERM712807CapecitabineFDA approvedDs|TYMS
719276FulvestrantFDA approvedAM|Ho|ESR|SERM713563ExemestaneFDA approvedHo|CYP19A1
719276FulvestrantFDA approvedAM|Ho|ESR|SERM715055GefitinibFDA approvedPK:YK,EGFR
719276FulvestrantFDA approvedAM|Ho|ESR|SERM719345LetrozoleFDA approvedHo|CYP19A1
719276FulvestrantFDA approvedAM|Ho|ESR|SERM719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
719276FulvestrantFDA approvedAM|Ho|ESR|SERM732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
719276FulvestrantFDA approvedAM|Ho|ESR|SERM733504EverolimusFDA approvedPK:STK,MTOR
719276FulvestrantFDA approvedAM|Ho|ESR|SERM737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
719276FulvestrantFDA approvedAM|Ho|ESR|SERM743414ImatinibFDA approvedBCR-ABL|PK:YK
719276FulvestrantFDA approvedAM|Ho|ESR|SERM745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
719276FulvestrantFDA approvedAM|Ho|ESR|SERM747599NilotinibFDA approvedBCR-ABL|PK:YK
719276FulvestrantFDA approvedAM|Ho|ESR|SERM747972LenalidomideFDA approvedFT|Immunomodulatory
719276FulvestrantFDA approvedAM|Ho|ESR|SERM747974RaloxifeneFDA approvedHo|SERM
719276FulvestrantFDA approvedAM|Ho|ESR|SERM749226AbirateroneFDA approvedHo|CYP17A1
719276FulvestrantFDA approvedAM|Ho|ESR|SERM750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
719276FulvestrantFDA approvedAM|Ho|ESR|SERM753082VemurafenibFDA approvedPK:YK,BRAF
719276FulvestrantFDA approvedAM|Ho|ESR|SERM754143RomidepsinFDA approvedHDAC
719276FulvestrantFDA approvedAM|Ho|ESR|SERM755986VismodegibFDA approvedSMO|PK:YK
719276FulvestrantFDA approvedAM|Ho|ESR|SERM756645CrizotinibFDA approvedPK:YK,MET,ALK
719276FulvestrantFDA approvedAM|Ho|ESR|SERM757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
719276FulvestrantFDA approvedAM|Ho|ESR|SERM760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
719276FulvestrantFDA approvedAM|Ho|ESR|SERM761432CabazitaxelFDA approvedTUBB|Tu-stab
719276FulvestrantFDA approvedAM|Ho|ESR|SERM763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
719344AnastrozoleFDA approvedHo|CYP19A1750BusulfanFDA approvedA7|AlkAg
719344AnastrozoleFDA approvedHo|CYP19A1752ThioguanineFDA approvedDs|IMPDH2|IMPDH
719344AnastrozoleFDA approvedHo|CYP19A13053DactinomycinFDA approvedDb|RNA polymerase I
719344AnastrozoleFDA approvedHo|CYP19A13088ChlorambucilFDA approvedA7|AlkAg
719344AnastrozoleFDA approvedHo|CYP19A16396ThiotepaFDA approvedA7|AlkAg
719344AnastrozoleFDA approvedHo|CYP19A18806MelphalanFDA approvedA7|AlkAg
719344AnastrozoleFDA approvedHo|CYP19A19706Triethylenemelamine-A7|AlkAg
719344AnastrozoleFDA approvedHo|CYP19A113875HexamethylmelamineFDA approvedDb|AlkAg
719344AnastrozoleFDA approvedHo|CYP19A119893FluorouracilFDA approvedDs|Rs|TYMS
719344AnastrozoleFDA approvedHo|CYP19A124559MithramycinFDA approvedDb|Rs
719344AnastrozoleFDA approvedHo|CYP19A127640FloxuridineFDA approvedDs|TYMS
719344AnastrozoleFDA approvedHo|CYP19A132065HydroxyureaFDA approvedAM|Dr
719344AnastrozoleFDA approvedHo|CYP19A134462Uracil mustardFDA approvedA7|AlkAg
719344AnastrozoleFDA approvedHo|CYP19A138721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
719344AnastrozoleFDA approvedHo|CYP19A145388DacarbazineFDA approvedA7|AlkAg
719344AnastrozoleFDA approvedHo|CYP19A149842Vinblastine sulfateFDA approvedTUBB|Tu-frag
719344AnastrozoleFDA approvedHo|CYP19A163878Cytarabine hydrochlorideFDA approvedDs
719344AnastrozoleFDA approvedHo|CYP19A167574Vincristine sulfateFDA approvedTUBB|Tu-frag
719344AnastrozoleFDA approvedHo|CYP19A171423Megestrol acetateFDA approvedHo|PGR
719344AnastrozoleFDA approvedHo|CYP19A179037LomustineFDA approvedA6|AlkAg
719344AnastrozoleFDA approvedHo|CYP19A182151Daunorubicin hydrochlorideFDA approvedTOP2
719344AnastrozoleFDA approvedHo|CYP19A1102816AzacitidineFDA approvedDNMT
719344AnastrozoleFDA approvedHo|CYP19A1105014CladribineFDA approvedDs|ADA
719344AnastrozoleFDA approvedHo|CYP19A1118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
719344AnastrozoleFDA approvedHo|CYP19A1122758TretinoinFDA approvedHo|RXR|Differentiator
719344AnastrozoleFDA approvedHo|CYP19A1122819TeniposideFDA approvedTOP2
719344AnastrozoleFDA approvedHo|CYP19A1123127Doxorubicin hydrochlorideFDA approvedTOP2
719344AnastrozoleFDA approvedHo|CYP19A1125066BleomycinFDA approvedDb
719344AnastrozoleFDA approvedHo|CYP19A1125973PaclitaxelFDA approvedTUBB|Tu-stab
719344AnastrozoleFDA approvedHo|CYP19A1138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
719344AnastrozoleFDA approvedHo|CYP19A1141540EtoposideFDA approvedTOP2
719344AnastrozoleFDA approvedHo|CYP19A1169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
719344AnastrozoleFDA approvedHo|CYP19A1180973Tamoxifen citrateFDA approvedHo|SERM
719344AnastrozoleFDA approvedHo|CYP19A1226080RapamycinFDA approvedPK:STK,MTOR
719344AnastrozoleFDA approvedHo|CYP19A1241240CarboplatinFDA approvedA7|AlkAg
719344AnastrozoleFDA approvedHo|CYP19A1246131ValrubicinFDA approvedTOP2
719344AnastrozoleFDA approvedHo|CYP19A1279836MitoxantroneFDA approvedTOP2
719344AnastrozoleFDA approvedHo|CYP19A1362856TemozolomideFDA approvedA7|AlkAg
719344AnastrozoleFDA approvedHo|CYP19A1606869ClofarabineFDA approvedDs
719344AnastrozoleFDA approvedHo|CYP19A1608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
719344AnastrozoleFDA approvedHo|CYP19A1613327Gemcitabine HCLFDA approvedDs
719344AnastrozoleFDA approvedHo|CYP19A1673596SN 38Clinical trialTOP1
719344AnastrozoleFDA approvedHo|CYP19A1686673NelarabineFDA approvedDs
719344AnastrozoleFDA approvedHo|CYP19A1698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
719344AnastrozoleFDA approvedHo|CYP19A1701852VorinostatFDA approvedHDAC
719344AnastrozoleFDA approvedHo|CYP19A1712807CapecitabineFDA approvedDs|TYMS
719344AnastrozoleFDA approvedHo|CYP19A1713563ExemestaneFDA approvedHo|CYP19A1
719344AnastrozoleFDA approvedHo|CYP19A1715055GefitinibFDA approvedPK:YK,EGFR
719344AnastrozoleFDA approvedHo|CYP19A1719276FulvestrantFDA approvedAM|Ho|ESR|SERM
719344AnastrozoleFDA approvedHo|CYP19A1719345LetrozoleFDA approvedHo|CYP19A1
719344AnastrozoleFDA approvedHo|CYP19A1719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
719344AnastrozoleFDA approvedHo|CYP19A1721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
719344AnastrozoleFDA approvedHo|CYP19A1732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
719344AnastrozoleFDA approvedHo|CYP19A1733504EverolimusFDA approvedPK:STK,MTOR
719344AnastrozoleFDA approvedHo|CYP19A1737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
719344AnastrozoleFDA approvedHo|CYP19A1743414ImatinibFDA approvedBCR-ABL|PK:YK
719344AnastrozoleFDA approvedHo|CYP19A1745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
719344AnastrozoleFDA approvedHo|CYP19A1747599NilotinibFDA approvedBCR-ABL|PK:YK
719344AnastrozoleFDA approvedHo|CYP19A1747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
719344AnastrozoleFDA approvedHo|CYP19A1747972LenalidomideFDA approvedFT|Immunomodulatory
719344AnastrozoleFDA approvedHo|CYP19A1747974RaloxifeneFDA approvedHo|SERM
719344AnastrozoleFDA approvedHo|CYP19A1749226AbirateroneFDA approvedHo|CYP17A1
719344AnastrozoleFDA approvedHo|CYP19A1750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
719344AnastrozoleFDA approvedHo|CYP19A1753082VemurafenibFDA approvedPK:YK,BRAF
719344AnastrozoleFDA approvedHo|CYP19A1754143RomidepsinFDA approvedHDAC
719344AnastrozoleFDA approvedHo|CYP19A1755986VismodegibFDA approvedSMO|PK:YK
719344AnastrozoleFDA approvedHo|CYP19A1756645CrizotinibFDA approvedPK:YK,MET,ALK
719344AnastrozoleFDA approvedHo|CYP19A1757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
719344AnastrozoleFDA approvedHo|CYP19A1760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
719344AnastrozoleFDA approvedHo|CYP19A1761432CabazitaxelFDA approvedTUBB|Tu-stab
719344AnastrozoleFDA approvedHo|CYP19A1763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
719345LetrozoleFDA approvedHo|CYP19A1752ThioguanineFDA approvedDs|IMPDH2|IMPDH
719345LetrozoleFDA approvedHo|CYP19A13088ChlorambucilFDA approvedA7|AlkAg
719345LetrozoleFDA approvedHo|CYP19A18806MelphalanFDA approvedA7|AlkAg
719345LetrozoleFDA approvedHo|CYP19A113875HexamethylmelamineFDA approvedDb|AlkAg
719345LetrozoleFDA approvedHo|CYP19A119893FluorouracilFDA approvedDs|Rs|TYMS
719345LetrozoleFDA approvedHo|CYP19A134462Uracil mustardFDA approvedA7|AlkAg
719345LetrozoleFDA approvedHo|CYP19A145388DacarbazineFDA approvedA7|AlkAg
719345LetrozoleFDA approvedHo|CYP19A171423Megestrol acetateFDA approvedHo|PGR
719345LetrozoleFDA approvedHo|CYP19A179037LomustineFDA approvedA6|AlkAg
719345LetrozoleFDA approvedHo|CYP19A182151Daunorubicin hydrochlorideFDA approvedTOP2
719345LetrozoleFDA approvedHo|CYP19A1122819TeniposideFDA approvedTOP2
719345LetrozoleFDA approvedHo|CYP19A1141540EtoposideFDA approvedTOP2
719345LetrozoleFDA approvedHo|CYP19A1169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
719345LetrozoleFDA approvedHo|CYP19A1279836MitoxantroneFDA approvedTOP2
719345LetrozoleFDA approvedHo|CYP19A1608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
719345LetrozoleFDA approvedHo|CYP19A1698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
719345LetrozoleFDA approvedHo|CYP19A1713563ExemestaneFDA approvedHo|CYP19A1
719345LetrozoleFDA approvedHo|CYP19A1715055GefitinibFDA approvedPK:YK,EGFR
719345LetrozoleFDA approvedHo|CYP19A1737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
719345LetrozoleFDA approvedHo|CYP19A1747972LenalidomideFDA approvedFT|Immunomodulatory
719345LetrozoleFDA approvedHo|CYP19A1747974RaloxifeneFDA approvedHo|SERM
719345LetrozoleFDA approvedHo|CYP19A1749226AbirateroneFDA approvedHo|CYP17A1
719345LetrozoleFDA approvedHo|CYP19A1753082VemurafenibFDA approvedPK:YK,BRAF
719345LetrozoleFDA approvedHo|CYP19A1755986VismodegibFDA approvedSMO|PK:YK
719345LetrozoleFDA approvedHo|CYP19A1756645CrizotinibFDA approvedPK:YK,MET,ALK
719345LetrozoleFDA approvedHo|CYP19A1757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
719345LetrozoleFDA approvedHo|CYP19A1760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
719345LetrozoleFDA approvedHo|CYP19A1761432CabazitaxelFDA approvedTUBB|Tu-stab
719345LetrozoleFDA approvedHo|CYP19A1763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID740MethotrexateFDA approvedDf|DHFR
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID752ThioguanineFDA approvedDs|IMPDH2|IMPDH
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID3053DactinomycinFDA approvedDb|RNA polymerase I
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID3088ChlorambucilFDA approvedA7|AlkAg
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID8806MelphalanFDA approvedA7|AlkAg
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID13875HexamethylmelamineFDA approvedDb|AlkAg
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID19893FluorouracilFDA approvedDs|Rs|TYMS
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID34462Uracil mustardFDA approvedA7|AlkAg
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID45388DacarbazineFDA approvedA7|AlkAg
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID71423Megestrol acetateFDA approvedHo|PGR
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID79037LomustineFDA approvedA6|AlkAg
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID82151Daunorubicin hydrochlorideFDA approvedTOP2
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID122819TeniposideFDA approvedTOP2
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID141540EtoposideFDA approvedTOP2
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID279836MitoxantroneFDA approvedTOP2
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID713563ExemestaneFDA approvedHo|CYP19A1
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID715055GefitinibFDA approvedPK:YK,EGFR
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID719345LetrozoleFDA approvedHo|CYP19A1
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID747972LenalidomideFDA approvedFT|Immunomodulatory
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID747974RaloxifeneFDA approvedHo|SERM
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID749226AbirateroneFDA approvedHo|CYP17A1
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID753082VemurafenibFDA approvedPK:YK,BRAF
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID755986VismodegibFDA approvedSMO|PK:YK
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID756645CrizotinibFDA approvedPK:YK,MET,ALK
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID761432CabazitaxelFDA approvedTUBB|Tu-stab
719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp752ThioguanineFDA approvedDs|IMPDH2|IMPDH
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp3053DactinomycinFDA approvedDb|RNA polymerase I
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp3088ChlorambucilFDA approvedA7|AlkAg
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp6396ThiotepaFDA approvedA7|AlkAg
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp8806MelphalanFDA approvedA7|AlkAg
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp13875HexamethylmelamineFDA approvedDb|AlkAg
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp18509Aminolevulinic Acid HydrochlorideFDA approvedAM
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp19893FluorouracilFDA approvedDs|Rs|TYMS
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp27640FloxuridineFDA approvedDs|TYMS
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp34462Uracil mustardFDA approvedA7|AlkAg
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp45388DacarbazineFDA approvedA7|AlkAg
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp63878Cytarabine hydrochlorideFDA approvedDs
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp67574Vincristine sulfateFDA approvedTUBB|Tu-frag
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp71423Megestrol acetateFDA approvedHo|PGR
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp79037LomustineFDA approvedA6|AlkAg
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp82151Daunorubicin hydrochlorideFDA approvedTOP2
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp102816AzacitidineFDA approvedDNMT
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp105014CladribineFDA approvedDs|ADA
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp122758TretinoinFDA approvedHo|RXR|Differentiator
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp122819TeniposideFDA approvedTOP2
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp125973PaclitaxelFDA approvedTUBB|Tu-stab
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp141540EtoposideFDA approvedTOP2
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp180973Tamoxifen citrateFDA approvedHo|SERM
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp226080RapamycinFDA approvedPK:STK,MTOR
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp241240CarboplatinFDA approvedA7|AlkAg
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp246131ValrubicinFDA approvedTOP2
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp279836MitoxantroneFDA approvedTOP2
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp362856TemozolomideFDA approvedA7|AlkAg
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp606869ClofarabineFDA approvedDs
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp613327Gemcitabine HCLFDA approvedDs
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp628503DocetaxelFDA approvedTUBB|Tu-stab
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp673596SN 38Clinical trialTOP1
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp686673NelarabineFDA approvedDs
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp701852VorinostatFDA approvedHDAC
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp712807CapecitabineFDA approvedDs|TYMS
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp713563ExemestaneFDA approvedHo|CYP19A1
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp715055GefitinibFDA approvedPK:YK,EGFR
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp719276FulvestrantFDA approvedAM|Ho|ESR|SERM
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp719345LetrozoleFDA approvedHo|CYP19A1
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp733504EverolimusFDA approvedPK:STK,MTOR
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp743414ImatinibFDA approvedBCR-ABL|PK:YK
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp747599NilotinibFDA approvedBCR-ABL|PK:YK
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp747972LenalidomideFDA approvedFT|Immunomodulatory
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp747974RaloxifeneFDA approvedHo|SERM
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp749226AbirateroneFDA approvedHo|CYP17A1
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp753082VemurafenibFDA approvedPK:YK,BRAF
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp754143RomidepsinFDA approvedHDAC
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp755986VismodegibFDA approvedSMO|PK:YK
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp756645CrizotinibFDA approvedPK:YK,MET,ALK
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp761432CabazitaxelFDA approvedTUBB|Tu-stab
721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT752ThioguanineFDA approvedDs|IMPDH2|IMPDH
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT3053DactinomycinFDA approvedDb|RNA polymerase I
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT3088ChlorambucilFDA approvedA7|AlkAg
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT6396ThiotepaFDA approvedA7|AlkAg
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT8806MelphalanFDA approvedA7|AlkAg
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT13875HexamethylmelamineFDA approvedDb|AlkAg
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT19893FluorouracilFDA approvedDs|Rs|TYMS
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT27640FloxuridineFDA approvedDs|TYMS
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT34462Uracil mustardFDA approvedA7|AlkAg
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT45388DacarbazineFDA approvedA7|AlkAg
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT63878Cytarabine hydrochlorideFDA approvedDs
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT67574Vincristine sulfateFDA approvedTUBB|Tu-frag
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT71423Megestrol acetateFDA approvedHo|PGR
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT79037LomustineFDA approvedA6|AlkAg
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT82151Daunorubicin hydrochlorideFDA approvedTOP2
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT102816AzacitidineFDA approvedDNMT
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT105014CladribineFDA approvedDs|ADA
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT122758TretinoinFDA approvedHo|RXR|Differentiator
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT122819TeniposideFDA approvedTOP2
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT125973PaclitaxelFDA approvedTUBB|Tu-stab
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT141540EtoposideFDA approvedTOP2
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT180973Tamoxifen citrateFDA approvedHo|SERM
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT226080RapamycinFDA approvedPK:STK,MTOR
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT241240CarboplatinFDA approvedA7|AlkAg
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT279836MitoxantroneFDA approvedTOP2
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT362856TemozolomideFDA approvedA7|AlkAg
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT606869ClofarabineFDA approvedDs
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT613327Gemcitabine HCLFDA approvedDs
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT628503DocetaxelFDA approvedTUBB|Tu-stab
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT673596SN 38Clinical trialTOP1
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT686673NelarabineFDA approvedDs
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT701852VorinostatFDA approvedHDAC
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT712807CapecitabineFDA approvedDs|TYMS
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT713563ExemestaneFDA approvedHo|CYP19A1
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT715055GefitinibFDA approvedPK:YK,EGFR
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT719345LetrozoleFDA approvedHo|CYP19A1
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT743414ImatinibFDA approvedBCR-ABL|PK:YK
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT747599NilotinibFDA approvedBCR-ABL|PK:YK
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT747972LenalidomideFDA approvedFT|Immunomodulatory
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT747974RaloxifeneFDA approvedHo|SERM
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT749226AbirateroneFDA approvedHo|CYP17A1
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT753082VemurafenibFDA approvedPK:YK,BRAF
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT754143RomidepsinFDA approvedHDAC
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT755986VismodegibFDA approvedSMO|PK:YK
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT756645CrizotinibFDA approvedPK:YK,MET,ALK
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT761432CabazitaxelFDA approvedTUBB|Tu-stab
732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
733504EverolimusFDA approvedPK:STK,MTOR752ThioguanineFDA approvedDs|IMPDH2|IMPDH
733504EverolimusFDA approvedPK:STK,MTOR3053DactinomycinFDA approvedDb|RNA polymerase I
733504EverolimusFDA approvedPK:STK,MTOR3088ChlorambucilFDA approvedA7|AlkAg
733504EverolimusFDA approvedPK:STK,MTOR6396ThiotepaFDA approvedA7|AlkAg
733504EverolimusFDA approvedPK:STK,MTOR8806MelphalanFDA approvedA7|AlkAg
733504EverolimusFDA approvedPK:STK,MTOR13875HexamethylmelamineFDA approvedDb|AlkAg
733504EverolimusFDA approvedPK:STK,MTOR19893FluorouracilFDA approvedDs|Rs|TYMS
733504EverolimusFDA approvedPK:STK,MTOR27640FloxuridineFDA approvedDs|TYMS
733504EverolimusFDA approvedPK:STK,MTOR34462Uracil mustardFDA approvedA7|AlkAg
733504EverolimusFDA approvedPK:STK,MTOR45388DacarbazineFDA approvedA7|AlkAg
733504EverolimusFDA approvedPK:STK,MTOR63878Cytarabine hydrochlorideFDA approvedDs
733504EverolimusFDA approvedPK:STK,MTOR67574Vincristine sulfateFDA approvedTUBB|Tu-frag
733504EverolimusFDA approvedPK:STK,MTOR71423Megestrol acetateFDA approvedHo|PGR
733504EverolimusFDA approvedPK:STK,MTOR79037LomustineFDA approvedA6|AlkAg
733504EverolimusFDA approvedPK:STK,MTOR82151Daunorubicin hydrochlorideFDA approvedTOP2
733504EverolimusFDA approvedPK:STK,MTOR102816AzacitidineFDA approvedDNMT
733504EverolimusFDA approvedPK:STK,MTOR105014CladribineFDA approvedDs|ADA
733504EverolimusFDA approvedPK:STK,MTOR118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
733504EverolimusFDA approvedPK:STK,MTOR122758TretinoinFDA approvedHo|RXR|Differentiator
733504EverolimusFDA approvedPK:STK,MTOR122819TeniposideFDA approvedTOP2
733504EverolimusFDA approvedPK:STK,MTOR125973PaclitaxelFDA approvedTUBB|Tu-stab
733504EverolimusFDA approvedPK:STK,MTOR141540EtoposideFDA approvedTOP2
733504EverolimusFDA approvedPK:STK,MTOR169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
733504EverolimusFDA approvedPK:STK,MTOR180973Tamoxifen citrateFDA approvedHo|SERM
733504EverolimusFDA approvedPK:STK,MTOR226080RapamycinFDA approvedPK:STK,MTOR
733504EverolimusFDA approvedPK:STK,MTOR241240CarboplatinFDA approvedA7|AlkAg
733504EverolimusFDA approvedPK:STK,MTOR279836MitoxantroneFDA approvedTOP2
733504EverolimusFDA approvedPK:STK,MTOR362856TemozolomideFDA approvedA7|AlkAg
733504EverolimusFDA approvedPK:STK,MTOR606869ClofarabineFDA approvedDs
733504EverolimusFDA approvedPK:STK,MTOR608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
733504EverolimusFDA approvedPK:STK,MTOR613327Gemcitabine HCLFDA approvedDs
733504EverolimusFDA approvedPK:STK,MTOR628503DocetaxelFDA approvedTUBB|Tu-stab
733504EverolimusFDA approvedPK:STK,MTOR673596SN 38Clinical trialTOP1
733504EverolimusFDA approvedPK:STK,MTOR686673NelarabineFDA approvedDs
733504EverolimusFDA approvedPK:STK,MTOR698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
733504EverolimusFDA approvedPK:STK,MTOR701852VorinostatFDA approvedHDAC
733504EverolimusFDA approvedPK:STK,MTOR712807CapecitabineFDA approvedDs|TYMS
733504EverolimusFDA approvedPK:STK,MTOR713563ExemestaneFDA approvedHo|CYP19A1
733504EverolimusFDA approvedPK:STK,MTOR715055GefitinibFDA approvedPK:YK,EGFR
733504EverolimusFDA approvedPK:STK,MTOR719345LetrozoleFDA approvedHo|CYP19A1
733504EverolimusFDA approvedPK:STK,MTOR719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
733504EverolimusFDA approvedPK:STK,MTOR732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
733504EverolimusFDA approvedPK:STK,MTOR737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
733504EverolimusFDA approvedPK:STK,MTOR743414ImatinibFDA approvedBCR-ABL|PK:YK
733504EverolimusFDA approvedPK:STK,MTOR747599NilotinibFDA approvedBCR-ABL|PK:YK
733504EverolimusFDA approvedPK:STK,MTOR747972LenalidomideFDA approvedFT|Immunomodulatory
733504EverolimusFDA approvedPK:STK,MTOR747974RaloxifeneFDA approvedHo|SERM
733504EverolimusFDA approvedPK:STK,MTOR749226AbirateroneFDA approvedHo|CYP17A1
733504EverolimusFDA approvedPK:STK,MTOR753082VemurafenibFDA approvedPK:YK,BRAF
733504EverolimusFDA approvedPK:STK,MTOR754143RomidepsinFDA approvedHDAC
733504EverolimusFDA approvedPK:STK,MTOR755986VismodegibFDA approvedSMO|PK:YK
733504EverolimusFDA approvedPK:STK,MTOR756645CrizotinibFDA approvedPK:YK,MET,ALK
733504EverolimusFDA approvedPK:STK,MTOR757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
733504EverolimusFDA approvedPK:STK,MTOR760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
733504EverolimusFDA approvedPK:STK,MTOR761432CabazitaxelFDA approvedTUBB|Tu-stab
733504EverolimusFDA approvedPK:STK,MTOR763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR747974RaloxifeneFDA approvedHo|SERM
737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR749226AbirateroneFDA approvedHo|CYP17A1
737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR753082VemurafenibFDA approvedPK:YK,BRAF
737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR755986VismodegibFDA approvedSMO|PK:YK
737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR756645CrizotinibFDA approvedPK:YK,MET,ALK
737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
743414ImatinibFDA approvedBCR-ABL|PK:YK740MethotrexateFDA approvedDf|DHFR
743414ImatinibFDA approvedBCR-ABL|PK:YK752ThioguanineFDA approvedDs|IMPDH2|IMPDH
743414ImatinibFDA approvedBCR-ABL|PK:YK3053DactinomycinFDA approvedDb|RNA polymerase I
743414ImatinibFDA approvedBCR-ABL|PK:YK3088ChlorambucilFDA approvedA7|AlkAg
743414ImatinibFDA approvedBCR-ABL|PK:YK6396ThiotepaFDA approvedA7|AlkAg
743414ImatinibFDA approvedBCR-ABL|PK:YK8806MelphalanFDA approvedA7|AlkAg
743414ImatinibFDA approvedBCR-ABL|PK:YK13875HexamethylmelamineFDA approvedDb|AlkAg
743414ImatinibFDA approvedBCR-ABL|PK:YK19893FluorouracilFDA approvedDs|Rs|TYMS
743414ImatinibFDA approvedBCR-ABL|PK:YK27640FloxuridineFDA approvedDs|TYMS
743414ImatinibFDA approvedBCR-ABL|PK:YK34462Uracil mustardFDA approvedA7|AlkAg
743414ImatinibFDA approvedBCR-ABL|PK:YK45388DacarbazineFDA approvedA7|AlkAg
743414ImatinibFDA approvedBCR-ABL|PK:YK63878Cytarabine hydrochlorideFDA approvedDs
743414ImatinibFDA approvedBCR-ABL|PK:YK67574Vincristine sulfateFDA approvedTUBB|Tu-frag
743414ImatinibFDA approvedBCR-ABL|PK:YK71423Megestrol acetateFDA approvedHo|PGR
743414ImatinibFDA approvedBCR-ABL|PK:YK79037LomustineFDA approvedA6|AlkAg
743414ImatinibFDA approvedBCR-ABL|PK:YK82151Daunorubicin hydrochlorideFDA approvedTOP2
743414ImatinibFDA approvedBCR-ABL|PK:YK105014CladribineFDA approvedDs|ADA
743414ImatinibFDA approvedBCR-ABL|PK:YK118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
743414ImatinibFDA approvedBCR-ABL|PK:YK122758TretinoinFDA approvedHo|RXR|Differentiator
743414ImatinibFDA approvedBCR-ABL|PK:YK122819TeniposideFDA approvedTOP2
743414ImatinibFDA approvedBCR-ABL|PK:YK141540EtoposideFDA approvedTOP2
743414ImatinibFDA approvedBCR-ABL|PK:YK169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
743414ImatinibFDA approvedBCR-ABL|PK:YK180973Tamoxifen citrateFDA approvedHo|SERM
743414ImatinibFDA approvedBCR-ABL|PK:YK241240CarboplatinFDA approvedA7|AlkAg
743414ImatinibFDA approvedBCR-ABL|PK:YK279836MitoxantroneFDA approvedTOP2
743414ImatinibFDA approvedBCR-ABL|PK:YK362856TemozolomideFDA approvedA7|AlkAg
743414ImatinibFDA approvedBCR-ABL|PK:YK608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
743414ImatinibFDA approvedBCR-ABL|PK:YK698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
743414ImatinibFDA approvedBCR-ABL|PK:YK713563ExemestaneFDA approvedHo|CYP19A1
743414ImatinibFDA approvedBCR-ABL|PK:YK715055GefitinibFDA approvedPK:YK,EGFR
743414ImatinibFDA approvedBCR-ABL|PK:YK719345LetrozoleFDA approvedHo|CYP19A1
743414ImatinibFDA approvedBCR-ABL|PK:YK719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
743414ImatinibFDA approvedBCR-ABL|PK:YK737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
743414ImatinibFDA approvedBCR-ABL|PK:YK747972LenalidomideFDA approvedFT|Immunomodulatory
743414ImatinibFDA approvedBCR-ABL|PK:YK747974RaloxifeneFDA approvedHo|SERM
743414ImatinibFDA approvedBCR-ABL|PK:YK749226AbirateroneFDA approvedHo|CYP17A1
743414ImatinibFDA approvedBCR-ABL|PK:YK753082VemurafenibFDA approvedPK:YK,BRAF
743414ImatinibFDA approvedBCR-ABL|PK:YK755986VismodegibFDA approvedSMO|PK:YK
743414ImatinibFDA approvedBCR-ABL|PK:YK756645CrizotinibFDA approvedPK:YK,MET,ALK
743414ImatinibFDA approvedBCR-ABL|PK:YK757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
743414ImatinibFDA approvedBCR-ABL|PK:YK760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
743414ImatinibFDA approvedBCR-ABL|PK:YK761432CabazitaxelFDA approvedTUBB|Tu-stab
743414ImatinibFDA approvedBCR-ABL|PK:YK763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR752ThioguanineFDA approvedDs|IMPDH2|IMPDH
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR3053DactinomycinFDA approvedDb|RNA polymerase I
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR3088ChlorambucilFDA approvedA7|AlkAg
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR6396ThiotepaFDA approvedA7|AlkAg
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR8806MelphalanFDA approvedA7|AlkAg
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR13875HexamethylmelamineFDA approvedDb|AlkAg
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR19893FluorouracilFDA approvedDs|Rs|TYMS
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR27640FloxuridineFDA approvedDs|TYMS
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR34462Uracil mustardFDA approvedA7|AlkAg
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR45388DacarbazineFDA approvedA7|AlkAg
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR63878Cytarabine hydrochlorideFDA approvedDs
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR67574Vincristine sulfateFDA approvedTUBB|Tu-frag
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR71423Megestrol acetateFDA approvedHo|PGR
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR79037LomustineFDA approvedA6|AlkAg
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR82151Daunorubicin hydrochlorideFDA approvedTOP2
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR102816AzacitidineFDA approvedDNMT
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR105014CladribineFDA approvedDs|ADA
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR122758TretinoinFDA approvedHo|RXR|Differentiator
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR122819TeniposideFDA approvedTOP2
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR125973PaclitaxelFDA approvedTUBB|Tu-stab
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR141540EtoposideFDA approvedTOP2
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR180973Tamoxifen citrateFDA approvedHo|SERM
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR226080RapamycinFDA approvedPK:STK,MTOR
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR241240CarboplatinFDA approvedA7|AlkAg
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR279836MitoxantroneFDA approvedTOP2
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR362856TemozolomideFDA approvedA7|AlkAg
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR606869ClofarabineFDA approvedDs
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR613327Gemcitabine HCLFDA approvedDs
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR628503DocetaxelFDA approvedTUBB|Tu-stab
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR673596SN 38Clinical trialTOP1
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR686673NelarabineFDA approvedDs
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR701852VorinostatFDA approvedHDAC
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR712807CapecitabineFDA approvedDs|TYMS
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR713563ExemestaneFDA approvedHo|CYP19A1
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR715055GefitinibFDA approvedPK:YK,EGFR
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR719345LetrozoleFDA approvedHo|CYP19A1
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR733504EverolimusFDA approvedPK:STK,MTOR
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR743414ImatinibFDA approvedBCR-ABL|PK:YK
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR747599NilotinibFDA approvedBCR-ABL|PK:YK
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR747972LenalidomideFDA approvedFT|Immunomodulatory
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR747974RaloxifeneFDA approvedHo|SERM
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR749226AbirateroneFDA approvedHo|CYP17A1
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR753082VemurafenibFDA approvedPK:YK,BRAF
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR754143RomidepsinFDA approvedHDAC
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR755986VismodegibFDA approvedSMO|PK:YK
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR756645CrizotinibFDA approvedPK:YK,MET,ALK
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR761432CabazitaxelFDA approvedTUBB|Tu-stab
745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
747599NilotinibFDA approvedBCR-ABL|PK:YK740MethotrexateFDA approvedDf|DHFR
747599NilotinibFDA approvedBCR-ABL|PK:YK752ThioguanineFDA approvedDs|IMPDH2|IMPDH
747599NilotinibFDA approvedBCR-ABL|PK:YK7556-MercaptopurineFDA approvedDs|PPAT
747599NilotinibFDA approvedBCR-ABL|PK:YK3053DactinomycinFDA approvedDb|RNA polymerase I
747599NilotinibFDA approvedBCR-ABL|PK:YK3088ChlorambucilFDA approvedA7|AlkAg
747599NilotinibFDA approvedBCR-ABL|PK:YK6396ThiotepaFDA approvedA7|AlkAg
747599NilotinibFDA approvedBCR-ABL|PK:YK8806MelphalanFDA approvedA7|AlkAg
747599NilotinibFDA approvedBCR-ABL|PK:YK13875HexamethylmelamineFDA approvedDb|AlkAg
747599NilotinibFDA approvedBCR-ABL|PK:YK19893FluorouracilFDA approvedDs|Rs|TYMS
747599NilotinibFDA approvedBCR-ABL|PK:YK24559MithramycinFDA approvedDb|Rs
747599NilotinibFDA approvedBCR-ABL|PK:YK27640FloxuridineFDA approvedDs|TYMS
747599NilotinibFDA approvedBCR-ABL|PK:YK32065HydroxyureaFDA approvedAM|Dr
747599NilotinibFDA approvedBCR-ABL|PK:YK34462Uracil mustardFDA approvedA7|AlkAg
747599NilotinibFDA approvedBCR-ABL|PK:YK38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
747599NilotinibFDA approvedBCR-ABL|PK:YK45388DacarbazineFDA approvedA7|AlkAg
747599NilotinibFDA approvedBCR-ABL|PK:YK49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
747599NilotinibFDA approvedBCR-ABL|PK:YK63878Cytarabine hydrochlorideFDA approvedDs
747599NilotinibFDA approvedBCR-ABL|PK:YK67574Vincristine sulfateFDA approvedTUBB|Tu-frag
747599NilotinibFDA approvedBCR-ABL|PK:YK71423Megestrol acetateFDA approvedHo|PGR
747599NilotinibFDA approvedBCR-ABL|PK:YK79037LomustineFDA approvedA6|AlkAg
747599NilotinibFDA approvedBCR-ABL|PK:YK82151Daunorubicin hydrochlorideFDA approvedTOP2
747599NilotinibFDA approvedBCR-ABL|PK:YK105014CladribineFDA approvedDs|ADA
747599NilotinibFDA approvedBCR-ABL|PK:YK118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
747599NilotinibFDA approvedBCR-ABL|PK:YK122758TretinoinFDA approvedHo|RXR|Differentiator
747599NilotinibFDA approvedBCR-ABL|PK:YK122819TeniposideFDA approvedTOP2
747599NilotinibFDA approvedBCR-ABL|PK:YK138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
747599NilotinibFDA approvedBCR-ABL|PK:YK141540EtoposideFDA approvedTOP2
747599NilotinibFDA approvedBCR-ABL|PK:YK169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
747599NilotinibFDA approvedBCR-ABL|PK:YK180973Tamoxifen citrateFDA approvedHo|SERM
747599NilotinibFDA approvedBCR-ABL|PK:YK241240CarboplatinFDA approvedA7|AlkAg
747599NilotinibFDA approvedBCR-ABL|PK:YK279836MitoxantroneFDA approvedTOP2
747599NilotinibFDA approvedBCR-ABL|PK:YK362856TemozolomideFDA approvedA7|AlkAg
747599NilotinibFDA approvedBCR-ABL|PK:YK608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
747599NilotinibFDA approvedBCR-ABL|PK:YK698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
747599NilotinibFDA approvedBCR-ABL|PK:YK713563ExemestaneFDA approvedHo|CYP19A1
747599NilotinibFDA approvedBCR-ABL|PK:YK715055GefitinibFDA approvedPK:YK,EGFR
747599NilotinibFDA approvedBCR-ABL|PK:YK719344AnastrozoleFDA approvedHo|CYP19A1
747599NilotinibFDA approvedBCR-ABL|PK:YK719345LetrozoleFDA approvedHo|CYP19A1
747599NilotinibFDA approvedBCR-ABL|PK:YK719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
747599NilotinibFDA approvedBCR-ABL|PK:YK737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
747599NilotinibFDA approvedBCR-ABL|PK:YK743414ImatinibFDA approvedBCR-ABL|PK:YK
747599NilotinibFDA approvedBCR-ABL|PK:YK747972LenalidomideFDA approvedFT|Immunomodulatory
747599NilotinibFDA approvedBCR-ABL|PK:YK747974RaloxifeneFDA approvedHo|SERM
747599NilotinibFDA approvedBCR-ABL|PK:YK749226AbirateroneFDA approvedHo|CYP17A1
747599NilotinibFDA approvedBCR-ABL|PK:YK753082VemurafenibFDA approvedPK:YK,BRAF
747599NilotinibFDA approvedBCR-ABL|PK:YK755986VismodegibFDA approvedSMO|PK:YK
747599NilotinibFDA approvedBCR-ABL|PK:YK756645CrizotinibFDA approvedPK:YK,MET,ALK
747599NilotinibFDA approvedBCR-ABL|PK:YK757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
747599NilotinibFDA approvedBCR-ABL|PK:YK760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
747599NilotinibFDA approvedBCR-ABL|PK:YK761432CabazitaxelFDA approvedTUBB|Tu-stab
747599NilotinibFDA approvedBCR-ABL|PK:YK763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase752ThioguanineFDA approvedDs|IMPDH2|IMPDH
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase3053DactinomycinFDA approvedDb|RNA polymerase I
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase3088ChlorambucilFDA approvedA7|AlkAg
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase6396ThiotepaFDA approvedA7|AlkAg
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase8806MelphalanFDA approvedA7|AlkAg
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase9706Triethylenemelamine-A7|AlkAg
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase13875HexamethylmelamineFDA approvedDb|AlkAg
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase19893FluorouracilFDA approvedDs|Rs|TYMS
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase24559MithramycinFDA approvedDb|Rs
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase27640FloxuridineFDA approvedDs|TYMS
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase32065HydroxyureaFDA approvedAM|Dr
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase34462Uracil mustardFDA approvedA7|AlkAg
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase45388DacarbazineFDA approvedA7|AlkAg
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase63878Cytarabine hydrochlorideFDA approvedDs
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase67574Vincristine sulfateFDA approvedTUBB|Tu-frag
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase71423Megestrol acetateFDA approvedHo|PGR
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase79037LomustineFDA approvedA6|AlkAg
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase82151Daunorubicin hydrochlorideFDA approvedTOP2
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase102816AzacitidineFDA approvedDNMT
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase105014CladribineFDA approvedDs|ADA
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase122758TretinoinFDA approvedHo|RXR|Differentiator
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase122819TeniposideFDA approvedTOP2
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase125066BleomycinFDA approvedDb
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase125973PaclitaxelFDA approvedTUBB|Tu-stab
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase141540EtoposideFDA approvedTOP2
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase180973Tamoxifen citrateFDA approvedHo|SERM
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase226080RapamycinFDA approvedPK:STK,MTOR
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase241240CarboplatinFDA approvedA7|AlkAg
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase279836MitoxantroneFDA approvedTOP2
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase362856TemozolomideFDA approvedA7|AlkAg
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase606869ClofarabineFDA approvedDs
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase613327Gemcitabine HCLFDA approvedDs
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase628503DocetaxelFDA approvedTUBB|Tu-stab
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase673596SN 38Clinical trialTOP1
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase686673NelarabineFDA approvedDs
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase701852VorinostatFDA approvedHDAC
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase712807CapecitabineFDA approvedDs|TYMS
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase713563ExemestaneFDA approvedHo|CYP19A1
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase715055GefitinibFDA approvedPK:YK,EGFR
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase719276FulvestrantFDA approvedAM|Ho|ESR|SERM
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase719345LetrozoleFDA approvedHo|CYP19A1
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase733504EverolimusFDA approvedPK:STK,MTOR
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase743414ImatinibFDA approvedBCR-ABL|PK:YK
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase747599NilotinibFDA approvedBCR-ABL|PK:YK
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase747972LenalidomideFDA approvedFT|Immunomodulatory
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase747974RaloxifeneFDA approvedHo|SERM
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase749226AbirateroneFDA approvedHo|CYP17A1
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase753082VemurafenibFDA approvedPK:YK,BRAF
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase754143RomidepsinFDA approvedHDAC
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase755986VismodegibFDA approvedSMO|PK:YK
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase756645CrizotinibFDA approvedPK:YK,MET,ALK
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase761432CabazitaxelFDA approvedTUBB|Tu-stab
747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
747972LenalidomideFDA approvedFT|Immunomodulatory9706Triethylenemelamine-A7|AlkAg
747972LenalidomideFDA approvedFT|Immunomodulatory123127Doxorubicin hydrochlorideFDA approvedTOP2
747972LenalidomideFDA approvedFT|Immunomodulatory737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
747972LenalidomideFDA approvedFT|Immunomodulatory747974RaloxifeneFDA approvedHo|SERM
747972LenalidomideFDA approvedFT|Immunomodulatory749226AbirateroneFDA approvedHo|CYP17A1
747972LenalidomideFDA approvedFT|Immunomodulatory753082VemurafenibFDA approvedPK:YK,BRAF
747972LenalidomideFDA approvedFT|Immunomodulatory755986VismodegibFDA approvedSMO|PK:YK
747972LenalidomideFDA approvedFT|Immunomodulatory756645CrizotinibFDA approvedPK:YK,MET,ALK
747972LenalidomideFDA approvedFT|Immunomodulatory757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
747972LenalidomideFDA approvedFT|Immunomodulatory760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
747972LenalidomideFDA approvedFT|Immunomodulatory761432CabazitaxelFDA approvedTUBB|Tu-stab
747972LenalidomideFDA approvedFT|Immunomodulatory763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
747973IxabepiloneFDA approvedTUBB|Tu-stab740MethotrexateFDA approvedDf|DHFR
747973IxabepiloneFDA approvedTUBB|Tu-stab750BusulfanFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab752ThioguanineFDA approvedDs|IMPDH2|IMPDH
747973IxabepiloneFDA approvedTUBB|Tu-stab7556-MercaptopurineFDA approvedDs|PPAT
747973IxabepiloneFDA approvedTUBB|Tu-stab762Nitrogen mustard hydrochlorideFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab1390AllopurinolFDA approvedAM|XDH
747973IxabepiloneFDA approvedTUBB|Tu-stab3053DactinomycinFDA approvedDb|RNA polymerase I
747973IxabepiloneFDA approvedTUBB|Tu-stab3088ChlorambucilFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab6396ThiotepaFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab8806MelphalanFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab9706Triethylenemelamine-A7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab13875HexamethylmelamineFDA approvedDb|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab14229QuinacrineClinical trialDb|AP
747973IxabepiloneFDA approvedTUBB|Tu-stab18509Aminolevulinic Acid HydrochlorideFDA approvedAM
747973IxabepiloneFDA approvedTUBB|Tu-stab19893FluorouracilFDA approvedDs|Rs|TYMS
747973IxabepiloneFDA approvedTUBB|Tu-stab24559MithramycinFDA approvedDb|Rs
747973IxabepiloneFDA approvedTUBB|Tu-stab25154PipobromanFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab26271CyclophosphamideFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab26980MitomycinFDA approvedA2|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab27640FloxuridineFDA approvedDs|TYMS
747973IxabepiloneFDA approvedTUBB|Tu-stab32065HydroxyureaFDA approvedAM|Dr
747973IxabepiloneFDA approvedTUBB|Tu-stab34462Uracil mustardFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
747973IxabepiloneFDA approvedTUBB|Tu-stab45388DacarbazineFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab459238-MethoxypsoralenFDA approvedDb
747973IxabepiloneFDA approvedTUBB|Tu-stab49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
747973IxabepiloneFDA approvedTUBB|Tu-stab63878Cytarabine hydrochlorideFDA approvedDs
747973IxabepiloneFDA approvedTUBB|Tu-stab66847ThalidomideFDA approvedAng|Immunomodulatory
747973IxabepiloneFDA approvedTUBB|Tu-stab67574Vincristine sulfateFDA approvedTUBB|Tu-frag
747973IxabepiloneFDA approvedTUBB|Tu-stab71423Megestrol acetateFDA approvedHo|PGR
747973IxabepiloneFDA approvedTUBB|Tu-stab77213Procarbazine hydrochlorideFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab79037LomustineFDA approvedA6|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab82151Daunorubicin hydrochlorideFDA approvedTOP2
747973IxabepiloneFDA approvedTUBB|Tu-stab85998StreptozocinFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab102816AzacitidineFDA approvedDNMT
747973IxabepiloneFDA approvedTUBB|Tu-stab105014CladribineFDA approvedDs|ADA
747973IxabepiloneFDA approvedTUBB|Tu-stab109724IfosfamideFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
747973IxabepiloneFDA approvedTUBB|Tu-stab122758TretinoinFDA approvedHo|RXR|Differentiator
747973IxabepiloneFDA approvedTUBB|Tu-stab122819TeniposideFDA approvedTOP2
747973IxabepiloneFDA approvedTUBB|Tu-stab123127Doxorubicin hydrochlorideFDA approvedTOP2
747973IxabepiloneFDA approvedTUBB|Tu-stab125066BleomycinFDA approvedDb
747973IxabepiloneFDA approvedTUBB|Tu-stab125973PaclitaxelFDA approvedTUBB|Tu-stab
747973IxabepiloneFDA approvedTUBB|Tu-stab127716DecitabineFDA approvedAM|DNMT
747973IxabepiloneFDA approvedTUBB|Tu-stab138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab141540EtoposideFDA approvedTOP2
747973IxabepiloneFDA approvedTUBB|Tu-stab169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
747973IxabepiloneFDA approvedTUBB|Tu-stab180973Tamoxifen citrateFDA approvedHo|SERM
747973IxabepiloneFDA approvedTUBB|Tu-stab218321PentostatinFDA approvedDs|AM|ADA
747973IxabepiloneFDA approvedTUBB|Tu-stab226080RapamycinFDA approvedPK:STK,MTOR
747973IxabepiloneFDA approvedTUBB|Tu-stab241240CarboplatinFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab246131ValrubicinFDA approvedTOP2
747973IxabepiloneFDA approvedTUBB|Tu-stab266046OxaliplatinFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab279836MitoxantroneFDA approvedTOP2
747973IxabepiloneFDA approvedTUBB|Tu-stab296961EthiofosFDA approvedRP
747973IxabepiloneFDA approvedTUBB|Tu-stab362856TemozolomideFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab369100ImiquimodFDA approvedAM|TLR7|ImmuneResMod
747973IxabepiloneFDA approvedTUBB|Tu-stab409962CarmustineFDA approvedA7|AlkAg
747973IxabepiloneFDA approvedTUBB|Tu-stab606869ClofarabineFDA approvedDs
747973IxabepiloneFDA approvedTUBB|Tu-stab608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
747973IxabepiloneFDA approvedTUBB|Tu-stab609699Topotecan hydrochlorideFDA approvedTOP1
747973IxabepiloneFDA approvedTUBB|Tu-stab613327Gemcitabine HCLFDA approvedDs
747973IxabepiloneFDA approvedTUBB|Tu-stab628503DocetaxelFDA approvedTUBB|Tu-stab
747973IxabepiloneFDA approvedTUBB|Tu-stab673596SN 38Clinical trialTOP1
747973IxabepiloneFDA approvedTUBB|Tu-stab686673NelarabineFDA approvedDs
747973IxabepiloneFDA approvedTUBB|Tu-stab698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
747973IxabepiloneFDA approvedTUBB|Tu-stab701852VorinostatFDA approvedHDAC
747973IxabepiloneFDA approvedTUBB|Tu-stab712807CapecitabineFDA approvedDs|TYMS
747973IxabepiloneFDA approvedTUBB|Tu-stab713563ExemestaneFDA approvedHo|CYP19A1
747973IxabepiloneFDA approvedTUBB|Tu-stab715055GefitinibFDA approvedPK:YK,EGFR
747973IxabepiloneFDA approvedTUBB|Tu-stab719276FulvestrantFDA approvedAM|Ho|ESR|SERM
747973IxabepiloneFDA approvedTUBB|Tu-stab719344AnastrozoleFDA approvedHo|CYP19A1
747973IxabepiloneFDA approvedTUBB|Tu-stab719345LetrozoleFDA approvedHo|CYP19A1
747973IxabepiloneFDA approvedTUBB|Tu-stab719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
747973IxabepiloneFDA approvedTUBB|Tu-stab721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
747973IxabepiloneFDA approvedTUBB|Tu-stab732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
747973IxabepiloneFDA approvedTUBB|Tu-stab733504EverolimusFDA approvedPK:STK,MTOR
747973IxabepiloneFDA approvedTUBB|Tu-stab737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
747973IxabepiloneFDA approvedTUBB|Tu-stab743414ImatinibFDA approvedBCR-ABL|PK:YK
747973IxabepiloneFDA approvedTUBB|Tu-stab745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
747973IxabepiloneFDA approvedTUBB|Tu-stab747599NilotinibFDA approvedBCR-ABL|PK:YK
747973IxabepiloneFDA approvedTUBB|Tu-stab747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
747973IxabepiloneFDA approvedTUBB|Tu-stab747972LenalidomideFDA approvedFT|Immunomodulatory
747973IxabepiloneFDA approvedTUBB|Tu-stab747974RaloxifeneFDA approvedHo|SERM
747973IxabepiloneFDA approvedTUBB|Tu-stab749226AbirateroneFDA approvedHo|CYP17A1
747973IxabepiloneFDA approvedTUBB|Tu-stab750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
747973IxabepiloneFDA approvedTUBB|Tu-stab753082VemurafenibFDA approvedPK:YK,BRAF
747973IxabepiloneFDA approvedTUBB|Tu-stab754143RomidepsinFDA approvedHDAC
747973IxabepiloneFDA approvedTUBB|Tu-stab754230PralatrexateFDA approvedDf|CTNNB1|DHFR
747973IxabepiloneFDA approvedTUBB|Tu-stab755986VismodegibFDA approvedSMO|PK:YK
747973IxabepiloneFDA approvedTUBB|Tu-stab756645CrizotinibFDA approvedPK:YK,MET,ALK
747973IxabepiloneFDA approvedTUBB|Tu-stab757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
747973IxabepiloneFDA approvedTUBB|Tu-stab760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
747973IxabepiloneFDA approvedTUBB|Tu-stab761432CabazitaxelFDA approvedTUBB|Tu-stab
747973IxabepiloneFDA approvedTUBB|Tu-stab763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
747974RaloxifeneFDA approvedHo|SERM9706Triethylenemelamine-A7|AlkAg
747974RaloxifeneFDA approvedHo|SERM123127Doxorubicin hydrochlorideFDA approvedTOP2
747974RaloxifeneFDA approvedHo|SERM737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
747974RaloxifeneFDA approvedHo|SERM749226AbirateroneFDA approvedHo|CYP17A1
747974RaloxifeneFDA approvedHo|SERM753082VemurafenibFDA approvedPK:YK,BRAF
747974RaloxifeneFDA approvedHo|SERM755986VismodegibFDA approvedSMO|PK:YK
747974RaloxifeneFDA approvedHo|SERM756645CrizotinibFDA approvedPK:YK,MET,ALK
747974RaloxifeneFDA approvedHo|SERM757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
747974RaloxifeneFDA approvedHo|SERM760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
747974RaloxifeneFDA approvedHo|SERM761432CabazitaxelFDA approvedTUBB|Tu-stab
747974RaloxifeneFDA approvedHo|SERM763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
749226AbirateroneFDA approvedHo|CYP17A1737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
749226AbirateroneFDA approvedHo|CYP17A1747974RaloxifeneFDA approvedHo|SERM
749226AbirateroneFDA approvedHo|CYP17A1753082VemurafenibFDA approvedPK:YK,BRAF
749226AbirateroneFDA approvedHo|CYP17A1755986VismodegibFDA approvedSMO|PK:YK
749226AbirateroneFDA approvedHo|CYP17A1756645CrizotinibFDA approvedPK:YK,MET,ALK
749226AbirateroneFDA approvedHo|CYP17A1757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
749226AbirateroneFDA approvedHo|CYP17A1760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
749226AbirateroneFDA approvedHo|CYP17A1761432CabazitaxelFDA approvedTUBB|Tu-stab
749226AbirateroneFDA approvedHo|CYP17A1763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase752ThioguanineFDA approvedDs|IMPDH2|IMPDH
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase3053DactinomycinFDA approvedDb|RNA polymerase I
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase3088ChlorambucilFDA approvedA7|AlkAg
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase6396ThiotepaFDA approvedA7|AlkAg
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase8806MelphalanFDA approvedA7|AlkAg
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase13875HexamethylmelamineFDA approvedDb|AlkAg
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase19893FluorouracilFDA approvedDs|Rs|TYMS
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase27640FloxuridineFDA approvedDs|TYMS
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase34462Uracil mustardFDA approvedA7|AlkAg
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase45388DacarbazineFDA approvedA7|AlkAg
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase63878Cytarabine hydrochlorideFDA approvedDs
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase67574Vincristine sulfateFDA approvedTUBB|Tu-frag
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase71423Megestrol acetateFDA approvedHo|PGR
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase79037LomustineFDA approvedA6|AlkAg
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase82151Daunorubicin hydrochlorideFDA approvedTOP2
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase102816AzacitidineFDA approvedDNMT
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase105014CladribineFDA approvedDs|ADA
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase122758TretinoinFDA approvedHo|RXR|Differentiator
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase122819TeniposideFDA approvedTOP2
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase125973PaclitaxelFDA approvedTUBB|Tu-stab
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase141540EtoposideFDA approvedTOP2
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase180973Tamoxifen citrateFDA approvedHo|SERM
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase226080RapamycinFDA approvedPK:STK,MTOR
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase241240CarboplatinFDA approvedA7|AlkAg
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase279836MitoxantroneFDA approvedTOP2
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase362856TemozolomideFDA approvedA7|AlkAg
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase606869ClofarabineFDA approvedDs
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase613327Gemcitabine HCLFDA approvedDs
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase628503DocetaxelFDA approvedTUBB|Tu-stab
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase673596SN 38Clinical trialTOP1
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase686673NelarabineFDA approvedDs
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase701852VorinostatFDA approvedHDAC
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase712807CapecitabineFDA approvedDs|TYMS
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase713563ExemestaneFDA approvedHo|CYP19A1
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase715055GefitinibFDA approvedPK:YK,EGFR
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase719345LetrozoleFDA approvedHo|CYP19A1
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase733504EverolimusFDA approvedPK:STK,MTOR
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase743414ImatinibFDA approvedBCR-ABL|PK:YK
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase747599NilotinibFDA approvedBCR-ABL|PK:YK
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase747972LenalidomideFDA approvedFT|Immunomodulatory
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase747974RaloxifeneFDA approvedHo|SERM
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase749226AbirateroneFDA approvedHo|CYP17A1
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase753082VemurafenibFDA approvedPK:YK,BRAF
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase754143RomidepsinFDA approvedHDAC
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase755986VismodegibFDA approvedSMO|PK:YK
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase756645CrizotinibFDA approvedPK:YK,MET,ALK
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase761432CabazitaxelFDA approvedTUBB|Tu-stab
750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
753082VemurafenibFDA approvedPK:YK,BRAF752ThioguanineFDA approvedDs|IMPDH2|IMPDH
753082VemurafenibFDA approvedPK:YK,BRAF3088ChlorambucilFDA approvedA7|AlkAg
753082VemurafenibFDA approvedPK:YK,BRAF8806MelphalanFDA approvedA7|AlkAg
753082VemurafenibFDA approvedPK:YK,BRAF13875HexamethylmelamineFDA approvedDb|AlkAg
753082VemurafenibFDA approvedPK:YK,BRAF19893FluorouracilFDA approvedDs|Rs|TYMS
753082VemurafenibFDA approvedPK:YK,BRAF34462Uracil mustardFDA approvedA7|AlkAg
753082VemurafenibFDA approvedPK:YK,BRAF45388DacarbazineFDA approvedA7|AlkAg
753082VemurafenibFDA approvedPK:YK,BRAF71423Megestrol acetateFDA approvedHo|PGR
753082VemurafenibFDA approvedPK:YK,BRAF79037LomustineFDA approvedA6|AlkAg
753082VemurafenibFDA approvedPK:YK,BRAF82151Daunorubicin hydrochlorideFDA approvedTOP2
753082VemurafenibFDA approvedPK:YK,BRAF122819TeniposideFDA approvedTOP2
753082VemurafenibFDA approvedPK:YK,BRAF141540EtoposideFDA approvedTOP2
753082VemurafenibFDA approvedPK:YK,BRAF169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
753082VemurafenibFDA approvedPK:YK,BRAF279836MitoxantroneFDA approvedTOP2
753082VemurafenibFDA approvedPK:YK,BRAF608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
753082VemurafenibFDA approvedPK:YK,BRAF698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
753082VemurafenibFDA approvedPK:YK,BRAF713563ExemestaneFDA approvedHo|CYP19A1
753082VemurafenibFDA approvedPK:YK,BRAF715055GefitinibFDA approvedPK:YK,EGFR
753082VemurafenibFDA approvedPK:YK,BRAF747972LenalidomideFDA approvedFT|Immunomodulatory
753082VemurafenibFDA approvedPK:YK,BRAF747974RaloxifeneFDA approvedHo|SERM
754143RomidepsinFDA approvedHDAC752ThioguanineFDA approvedDs|IMPDH2|IMPDH
754143RomidepsinFDA approvedHDAC3053DactinomycinFDA approvedDb|RNA polymerase I
754143RomidepsinFDA approvedHDAC3088ChlorambucilFDA approvedA7|AlkAg
754143RomidepsinFDA approvedHDAC6396ThiotepaFDA approvedA7|AlkAg
754143RomidepsinFDA approvedHDAC8806MelphalanFDA approvedA7|AlkAg
754143RomidepsinFDA approvedHDAC13875HexamethylmelamineFDA approvedDb|AlkAg
754143RomidepsinFDA approvedHDAC19893FluorouracilFDA approvedDs|Rs|TYMS
754143RomidepsinFDA approvedHDAC27640FloxuridineFDA approvedDs|TYMS
754143RomidepsinFDA approvedHDAC34462Uracil mustardFDA approvedA7|AlkAg
754143RomidepsinFDA approvedHDAC45388DacarbazineFDA approvedA7|AlkAg
754143RomidepsinFDA approvedHDAC49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
754143RomidepsinFDA approvedHDAC63878Cytarabine hydrochlorideFDA approvedDs
754143RomidepsinFDA approvedHDAC67574Vincristine sulfateFDA approvedTUBB|Tu-frag
754143RomidepsinFDA approvedHDAC71423Megestrol acetateFDA approvedHo|PGR
754143RomidepsinFDA approvedHDAC79037LomustineFDA approvedA6|AlkAg
754143RomidepsinFDA approvedHDAC82151Daunorubicin hydrochlorideFDA approvedTOP2
754143RomidepsinFDA approvedHDAC105014CladribineFDA approvedDs|ADA
754143RomidepsinFDA approvedHDAC118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
754143RomidepsinFDA approvedHDAC122758TretinoinFDA approvedHo|RXR|Differentiator
754143RomidepsinFDA approvedHDAC122819TeniposideFDA approvedTOP2
754143RomidepsinFDA approvedHDAC125973PaclitaxelFDA approvedTUBB|Tu-stab
754143RomidepsinFDA approvedHDAC141540EtoposideFDA approvedTOP2
754143RomidepsinFDA approvedHDAC169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
754143RomidepsinFDA approvedHDAC180973Tamoxifen citrateFDA approvedHo|SERM
754143RomidepsinFDA approvedHDAC226080RapamycinFDA approvedPK:STK,MTOR
754143RomidepsinFDA approvedHDAC241240CarboplatinFDA approvedA7|AlkAg
754143RomidepsinFDA approvedHDAC246131ValrubicinFDA approvedTOP2
754143RomidepsinFDA approvedHDAC279836MitoxantroneFDA approvedTOP2
754143RomidepsinFDA approvedHDAC362856TemozolomideFDA approvedA7|AlkAg
754143RomidepsinFDA approvedHDAC606869ClofarabineFDA approvedDs
754143RomidepsinFDA approvedHDAC608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
754143RomidepsinFDA approvedHDAC613327Gemcitabine HCLFDA approvedDs
754143RomidepsinFDA approvedHDAC628503DocetaxelFDA approvedTUBB|Tu-stab
754143RomidepsinFDA approvedHDAC686673NelarabineFDA approvedDs
754143RomidepsinFDA approvedHDAC698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
754143RomidepsinFDA approvedHDAC712807CapecitabineFDA approvedDs|TYMS
754143RomidepsinFDA approvedHDAC713563ExemestaneFDA approvedHo|CYP19A1
754143RomidepsinFDA approvedHDAC715055GefitinibFDA approvedPK:YK,EGFR
754143RomidepsinFDA approvedHDAC719344AnastrozoleFDA approvedHo|CYP19A1
754143RomidepsinFDA approvedHDAC719345LetrozoleFDA approvedHo|CYP19A1
754143RomidepsinFDA approvedHDAC719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
754143RomidepsinFDA approvedHDAC737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
754143RomidepsinFDA approvedHDAC743414ImatinibFDA approvedBCR-ABL|PK:YK
754143RomidepsinFDA approvedHDAC747599NilotinibFDA approvedBCR-ABL|PK:YK
754143RomidepsinFDA approvedHDAC747972LenalidomideFDA approvedFT|Immunomodulatory
754143RomidepsinFDA approvedHDAC747974RaloxifeneFDA approvedHo|SERM
754143RomidepsinFDA approvedHDAC749226AbirateroneFDA approvedHo|CYP17A1
754143RomidepsinFDA approvedHDAC753082VemurafenibFDA approvedPK:YK,BRAF
754143RomidepsinFDA approvedHDAC755986VismodegibFDA approvedSMO|PK:YK
754143RomidepsinFDA approvedHDAC756645CrizotinibFDA approvedPK:YK,MET,ALK
754143RomidepsinFDA approvedHDAC757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
754143RomidepsinFDA approvedHDAC760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
754143RomidepsinFDA approvedHDAC761432CabazitaxelFDA approvedTUBB|Tu-stab
754143RomidepsinFDA approvedHDAC763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
754230PralatrexateFDA approvedDf|CTNNB1|DHFR752ThioguanineFDA approvedDs|IMPDH2|IMPDH
754230PralatrexateFDA approvedDf|CTNNB1|DHFR3053DactinomycinFDA approvedDb|RNA polymerase I
754230PralatrexateFDA approvedDf|CTNNB1|DHFR3088ChlorambucilFDA approvedA7|AlkAg
754230PralatrexateFDA approvedDf|CTNNB1|DHFR6396ThiotepaFDA approvedA7|AlkAg
754230PralatrexateFDA approvedDf|CTNNB1|DHFR8806MelphalanFDA approvedA7|AlkAg
754230PralatrexateFDA approvedDf|CTNNB1|DHFR9706Triethylenemelamine-A7|AlkAg
754230PralatrexateFDA approvedDf|CTNNB1|DHFR13875HexamethylmelamineFDA approvedDb|AlkAg
754230PralatrexateFDA approvedDf|CTNNB1|DHFR19893FluorouracilFDA approvedDs|Rs|TYMS
754230PralatrexateFDA approvedDf|CTNNB1|DHFR24559MithramycinFDA approvedDb|Rs
754230PralatrexateFDA approvedDf|CTNNB1|DHFR27640FloxuridineFDA approvedDs|TYMS
754230PralatrexateFDA approvedDf|CTNNB1|DHFR32065HydroxyureaFDA approvedAM|Dr
754230PralatrexateFDA approvedDf|CTNNB1|DHFR34462Uracil mustardFDA approvedA7|AlkAg
754230PralatrexateFDA approvedDf|CTNNB1|DHFR38721MitotaneFDA approvedA7|Ho|AlkAg|anti-Ho|CYP11A1
754230PralatrexateFDA approvedDf|CTNNB1|DHFR45388DacarbazineFDA approvedA7|AlkAg
754230PralatrexateFDA approvedDf|CTNNB1|DHFR49842Vinblastine sulfateFDA approvedTUBB|Tu-frag
754230PralatrexateFDA approvedDf|CTNNB1|DHFR63878Cytarabine hydrochlorideFDA approvedDs
754230PralatrexateFDA approvedDf|CTNNB1|DHFR67574Vincristine sulfateFDA approvedTUBB|Tu-frag
754230PralatrexateFDA approvedDf|CTNNB1|DHFR71423Megestrol acetateFDA approvedHo|PGR
754230PralatrexateFDA approvedDf|CTNNB1|DHFR79037LomustineFDA approvedA6|AlkAg
754230PralatrexateFDA approvedDf|CTNNB1|DHFR82151Daunorubicin hydrochlorideFDA approvedTOP2
754230PralatrexateFDA approvedDf|CTNNB1|DHFR102816AzacitidineFDA approvedDNMT
754230PralatrexateFDA approvedDf|CTNNB1|DHFR105014CladribineFDA approvedDs|ADA
754230PralatrexateFDA approvedDf|CTNNB1|DHFR118218Fludarabine BaseFDA approvedDs|AM|Dr|STAT1
754230PralatrexateFDA approvedDf|CTNNB1|DHFR122758TretinoinFDA approvedHo|RXR|Differentiator
754230PralatrexateFDA approvedDf|CTNNB1|DHFR122819TeniposideFDA approvedTOP2
754230PralatrexateFDA approvedDf|CTNNB1|DHFR125066BleomycinFDA approvedDb
754230PralatrexateFDA approvedDf|CTNNB1|DHFR125973PaclitaxelFDA approvedTUBB|Tu-stab
754230PralatrexateFDA approvedDf|CTNNB1|DHFR138783Bendamustine HydrochlorideFDA approvedA2|A6|AlkAg
754230PralatrexateFDA approvedDf|CTNNB1|DHFR141540EtoposideFDA approvedTOP2
754230PralatrexateFDA approvedDf|CTNNB1|DHFR169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
754230PralatrexateFDA approvedDf|CTNNB1|DHFR180973Tamoxifen citrateFDA approvedHo|SERM
754230PralatrexateFDA approvedDf|CTNNB1|DHFR226080RapamycinFDA approvedPK:STK,MTOR
754230PralatrexateFDA approvedDf|CTNNB1|DHFR241240CarboplatinFDA approvedA7|AlkAg
754230PralatrexateFDA approvedDf|CTNNB1|DHFR246131ValrubicinFDA approvedTOP2
754230PralatrexateFDA approvedDf|CTNNB1|DHFR279836MitoxantroneFDA approvedTOP2
754230PralatrexateFDA approvedDf|CTNNB1|DHFR362856TemozolomideFDA approvedA7|AlkAg
754230PralatrexateFDA approvedDf|CTNNB1|DHFR606869ClofarabineFDA approvedDs
754230PralatrexateFDA approvedDf|CTNNB1|DHFR608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
754230PralatrexateFDA approvedDf|CTNNB1|DHFR613327Gemcitabine HCLFDA approvedDs
754230PralatrexateFDA approvedDf|CTNNB1|DHFR628503DocetaxelFDA approvedTUBB|Tu-stab
754230PralatrexateFDA approvedDf|CTNNB1|DHFR673596SN 38Clinical trialTOP1
754230PralatrexateFDA approvedDf|CTNNB1|DHFR686673NelarabineFDA approvedDs
754230PralatrexateFDA approvedDf|CTNNB1|DHFR698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
754230PralatrexateFDA approvedDf|CTNNB1|DHFR701852VorinostatFDA approvedHDAC
754230PralatrexateFDA approvedDf|CTNNB1|DHFR712807CapecitabineFDA approvedDs|TYMS
754230PralatrexateFDA approvedDf|CTNNB1|DHFR713563ExemestaneFDA approvedHo|CYP19A1
754230PralatrexateFDA approvedDf|CTNNB1|DHFR715055GefitinibFDA approvedPK:YK,EGFR
754230PralatrexateFDA approvedDf|CTNNB1|DHFR719276FulvestrantFDA approvedAM|Ho|ESR|SERM
754230PralatrexateFDA approvedDf|CTNNB1|DHFR719344AnastrozoleFDA approvedHo|CYP19A1
754230PralatrexateFDA approvedDf|CTNNB1|DHFR719345LetrozoleFDA approvedHo|CYP19A1
754230PralatrexateFDA approvedDf|CTNNB1|DHFR719627CelecoxibFDA approvedAM|PTGS2|COX2|NonCan:NSAID
754230PralatrexateFDA approvedDf|CTNNB1|DHFR721517Zoledronic AcidFDA approvedAM|NonCan:Anti-bone resorp
754230PralatrexateFDA approvedDf|CTNNB1|DHFR732517DasatinibFDA approvedBCR-ABL|PK:YK,PDGFR,KIT
754230PralatrexateFDA approvedDf|CTNNB1|DHFR733504EverolimusFDA approvedPK:STK,MTOR
754230PralatrexateFDA approvedDf|CTNNB1|DHFR737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
754230PralatrexateFDA approvedDf|CTNNB1|DHFR743414ImatinibFDA approvedBCR-ABL|PK:YK
754230PralatrexateFDA approvedDf|CTNNB1|DHFR745750LapatinibFDA approvedPK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR
754230PralatrexateFDA approvedDf|CTNNB1|DHFR747599NilotinibFDA approvedBCR-ABL|PK:YK
754230PralatrexateFDA approvedDf|CTNNB1|DHFR747971SorafenibFDA approvedPK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase
754230PralatrexateFDA approvedDf|CTNNB1|DHFR747972LenalidomideFDA approvedFT|Immunomodulatory
754230PralatrexateFDA approvedDf|CTNNB1|DHFR747974RaloxifeneFDA approvedHo|SERM
754230PralatrexateFDA approvedDf|CTNNB1|DHFR749226AbirateroneFDA approvedHo|CYP17A1
754230PralatrexateFDA approvedDf|CTNNB1|DHFR750690Sunitinib (free base)FDA approvedPK:YK,PDGFR,KIT,VEGFR,Multikinase
754230PralatrexateFDA approvedDf|CTNNB1|DHFR753082VemurafenibFDA approvedPK:YK,BRAF
754230PralatrexateFDA approvedDf|CTNNB1|DHFR754143RomidepsinFDA approvedHDAC
754230PralatrexateFDA approvedDf|CTNNB1|DHFR755986VismodegibFDA approvedSMO|PK:YK
754230PralatrexateFDA approvedDf|CTNNB1|DHFR756645CrizotinibFDA approvedPK:YK,MET,ALK
754230PralatrexateFDA approvedDf|CTNNB1|DHFR757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
754230PralatrexateFDA approvedDf|CTNNB1|DHFR760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
754230PralatrexateFDA approvedDf|CTNNB1|DHFR761432CabazitaxelFDA approvedTUBB|Tu-stab
754230PralatrexateFDA approvedDf|CTNNB1|DHFR763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
755986VismodegibFDA approvedSMO|PK:YK737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
755986VismodegibFDA approvedSMO|PK:YK747974RaloxifeneFDA approvedHo|SERM
755986VismodegibFDA approvedSMO|PK:YK749226AbirateroneFDA approvedHo|CYP17A1
755986VismodegibFDA approvedSMO|PK:YK753082VemurafenibFDA approvedPK:YK,BRAF
755986VismodegibFDA approvedSMO|PK:YK756645CrizotinibFDA approvedPK:YK,MET,ALK
755986VismodegibFDA approvedSMO|PK:YK757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
755986VismodegibFDA approvedSMO|PK:YK760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
755986VismodegibFDA approvedSMO|PK:YK761432CabazitaxelFDA approvedTUBB|Tu-stab
755986VismodegibFDA approvedSMO|PK:YK763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
756645CrizotinibFDA approvedPK:YK,MET,ALK752ThioguanineFDA approvedDs|IMPDH2|IMPDH
756645CrizotinibFDA approvedPK:YK,MET,ALK3088ChlorambucilFDA approvedA7|AlkAg
756645CrizotinibFDA approvedPK:YK,MET,ALK8806MelphalanFDA approvedA7|AlkAg
756645CrizotinibFDA approvedPK:YK,MET,ALK13875HexamethylmelamineFDA approvedDb|AlkAg
756645CrizotinibFDA approvedPK:YK,MET,ALK19893FluorouracilFDA approvedDs|Rs|TYMS
756645CrizotinibFDA approvedPK:YK,MET,ALK34462Uracil mustardFDA approvedA7|AlkAg
756645CrizotinibFDA approvedPK:YK,MET,ALK45388DacarbazineFDA approvedA7|AlkAg
756645CrizotinibFDA approvedPK:YK,MET,ALK71423Megestrol acetateFDA approvedHo|PGR
756645CrizotinibFDA approvedPK:YK,MET,ALK79037LomustineFDA approvedA6|AlkAg
756645CrizotinibFDA approvedPK:YK,MET,ALK82151Daunorubicin hydrochlorideFDA approvedTOP2
756645CrizotinibFDA approvedPK:YK,MET,ALK122819TeniposideFDA approvedTOP2
756645CrizotinibFDA approvedPK:YK,MET,ALK141540EtoposideFDA approvedTOP2
756645CrizotinibFDA approvedPK:YK,MET,ALK169780ICRF-187FDA approvedTOP2|NonCan:Cardioprotective
756645CrizotinibFDA approvedPK:YK,MET,ALK279836MitoxantroneFDA approvedTOP2
756645CrizotinibFDA approvedPK:YK,MET,ALK608210Vinorelbine tartrateFDA approvedTUBB|Tu-frag
756645CrizotinibFDA approvedPK:YK,MET,ALK698037PemetrexedFDA approvedDf|AM|GARTF|DHFR|TYMS
756645CrizotinibFDA approvedPK:YK,MET,ALK713563ExemestaneFDA approvedHo|CYP19A1
756645CrizotinibFDA approvedPK:YK,MET,ALK715055GefitinibFDA approvedPK:YK,EGFR
756645CrizotinibFDA approvedPK:YK,MET,ALK737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
756645CrizotinibFDA approvedPK:YK,MET,ALK747972LenalidomideFDA approvedFT|Immunomodulatory
756645CrizotinibFDA approvedPK:YK,MET,ALK747974RaloxifeneFDA approvedHo|SERM
756645CrizotinibFDA approvedPK:YK,MET,ALK749226AbirateroneFDA approvedHo|CYP17A1
756645CrizotinibFDA approvedPK:YK,MET,ALK753082VemurafenibFDA approvedPK:YK,BRAF
756645CrizotinibFDA approvedPK:YK,MET,ALK755986VismodegibFDA approvedSMO|PK:YK
756645CrizotinibFDA approvedPK:YK,MET,ALK757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
756645CrizotinibFDA approvedPK:YK,MET,ALK760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
756645CrizotinibFDA approvedPK:YK,MET,ALK761432CabazitaxelFDA approvedTUBB|Tu-stab
756645CrizotinibFDA approvedPK:YK,MET,ALK763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR747974RaloxifeneFDA approvedHo|SERM
757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR749226AbirateroneFDA approvedHo|CYP17A1
757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR753082VemurafenibFDA approvedPK:YK,BRAF
757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR755986VismodegibFDA approvedSMO|PK:YK
757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR756645CrizotinibFDA approvedPK:YK,MET,ALK
757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR761432CabazitaxelFDA approvedTUBB|Tu-stab
757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET747974RaloxifeneFDA approvedHo|SERM
760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET749226AbirateroneFDA approvedHo|CYP17A1
760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET753082VemurafenibFDA approvedPK:YK,BRAF
760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET755986VismodegibFDA approvedSMO|PK:YK
760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET756645CrizotinibFDA approvedPK:YK,MET,ALK
760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET761432CabazitaxelFDA approvedTUBB|Tu-stab
760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
761431VemurafenibFDA approvedPK:YK,BRAF737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
761431VemurafenibFDA approvedPK:YK,BRAF747974RaloxifeneFDA approvedHo|SERM
761431VemurafenibFDA approvedPK:YK,BRAF749226AbirateroneFDA approvedHo|CYP17A1
761431VemurafenibFDA approvedPK:YK,BRAF753082VemurafenibFDA approvedPK:YK,BRAF
761431VemurafenibFDA approvedPK:YK,BRAF755986VismodegibFDA approvedSMO|PK:YK
761431VemurafenibFDA approvedPK:YK,BRAF756645CrizotinibFDA approvedPK:YK,MET,ALK
761431VemurafenibFDA approvedPK:YK,BRAF757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
761431VemurafenibFDA approvedPK:YK,BRAF760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
761431VemurafenibFDA approvedPK:YK,BRAF761432CabazitaxelFDA approvedTUBB|Tu-stab
761431VemurafenibFDA approvedPK:YK,BRAF763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
761432CabazitaxelFDA approvedTUBB|Tu-stab737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
761432CabazitaxelFDA approvedTUBB|Tu-stab747974RaloxifeneFDA approvedHo|SERM
761432CabazitaxelFDA approvedTUBB|Tu-stab749226AbirateroneFDA approvedHo|CYP17A1
761432CabazitaxelFDA approvedTUBB|Tu-stab753082VemurafenibFDA approvedPK:YK,BRAF
761432CabazitaxelFDA approvedTUBB|Tu-stab755986VismodegibFDA approvedSMO|PK:YK
761432CabazitaxelFDA approvedTUBB|Tu-stab756645CrizotinibFDA approvedPK:YK,MET,ALK
761432CabazitaxelFDA approvedTUBB|Tu-stab757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
761432CabazitaxelFDA approvedTUBB|Tu-stab760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
761432CabazitaxelFDA approvedTUBB|Tu-stab763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2
763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2737754Pazopanib hydrochlorideFDA approvedPK:YK,PDGFR,FGFR,KIT,VEGFR
763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2747974RaloxifeneFDA approvedHo|SERM
763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2749226AbirateroneFDA approvedHo|CYP17A1
763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2753082VemurafenibFDA approvedPK:YK,BRAF
763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2755986VismodegibFDA approvedSMO|PK:YK
763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2756645CrizotinibFDA approvedPK:YK,MET,ALK
763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2757441AxitinibFDA approvedPK:YK,PDGFR,VEGFR
763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2760766VandetanibFDA approvedPK:STK,YK,PDGFR,EGFR,VEGFR,RET
763371RuxolitinibFDA approvedPK:YK,JAK,JAK1,JAK2761432CabazitaxelFDA approvedTUBB|Tu-stab