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MLN-7243

Key Value
Synonyms: MLN-7243
CT-M7243
TAK-243
MLN7243
A-1384
785004
National Service Center# (NSC#):1,2 785004
CAS#: NA
PubChem#: NA
Mechanism of Action: UB-activating
Status: Clinical trial
Molecular Formula: C19H20F3N5O5S2
Smiles: NS(=O)(=O)OC[C@H]1C[C@@H](Nc2ccnc3cc(nn23)c4cccc(SC(F)(F)F)c4)[C@H](O)[C@@H]1O

MLN-7243 is in CellMinerCDB, a searchable tool integrating cancer cell line pharmacogenomics data to link gene and drug activity signatures.

Click Here to Access CellMinerCDB

MLN-7243 is in CellMiner (NCI-60),a database and query tool designed for the cancer research community to facilitate integration and study of molecular and pharmacological data for the NCI-60 cancerous cell lines.

Click Here to Access CellMiner (NCI-60)

If you use content from this page, CellMinerCDB or CellMiner (NCI-60), please cite: Luna A et al. 2021. PMID: 33196823, Rajapakse VN et al. 2018. PMID: 30553813, Luna et al. 2016., PMID: 26635141, and Reinhold et al. 2012., PMID: 22802077.

Available Data

Visit CellMinerCDB to interactively explore available pharmacogenomics data for MLN-7243.

Visit CellMiner (NCI-60) to explore NCI-60 related analysis for MLN-7243.

MLN-7243 is available in the following datasets
NCI60 GDSC-MGH-Sanger GDSC1 drugs GDSC2 drugs CCLE-Broad-MIT CTRP-Broad-MIT NCI-DTP SCLC PRISM-Broad-MIT NCI60-DTP Almanac
785004 NA NA NA NA NA NA NA NA
1 NSC#: Originally known as Cancer Chemotherapy National Service Center number, the NSC# is an identifying number assigned by NCI-DTP to an agent or product (e.g. small molecule or biological agent).
2 Most structures have a unique NSC number but over the years a small percentage of structures or agents may have been assigned more than one NSC number. In the case of salts, different salt forms (e.g. HCl, HOAc) are designated with separate NSC numbers.

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