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Galunisertib

Key Value
Synonyms: 700874-72-2
GALUNISERTIB
LY 2157299
LY-2157299
LY2157299
National Service Center# (NSC#):1,2 761216
CAS#: 700874-72-2
PubChem#: NA
Mechanism of Action: TGFB1|PK:GSK3B
Status: Clinical trial
Molecular Formula: C22H19N5O
Smiles: Cc1cccc(n1)c2nn3CCCc3c2c4ccnc5ccc(cc45)C(=O)N

Galunisertib is in CellMinerCDB, a searchable tool integrating cancer cell line pharmacogenomics data to link gene and drug activity signatures.

Click Here to Access CellMinerCDB

Galunisertib is in CellMiner (NCI-60),a database and query tool designed for the cancer research community to facilitate integration and study of molecular and pharmacological data for the NCI-60 cancerous cell lines.

Click Here to Access CellMiner (NCI-60)

If you use content from this page, CellMinerCDB or CellMiner (NCI-60), please cite: Luna A et al. 2021. PMID: 33196823, Rajapakse VN et al. 2018. PMID: 30553813, Luna et al. 2016., PMID: 26635141, and Reinhold et al. 2012., PMID: 22802077.

Available Data

Visit CellMinerCDB to interactively explore available pharmacogenomics data for Galunisertib.

Visit CellMiner (NCI-60) to explore NCI-60 related analysis for Galunisertib.

Galunisertib is available in the following datasets
NCI60 GDSC-MGH-Sanger GDSC1 drugs GDSC2 drugs CCLE-Broad-MIT CTRP-Broad-MIT NCI-DTP SCLC PRISM-Broad-MIT NCI60-DTP Almanac
NA NA NA NA NA NA 761216 NA NA
1 NSC#: Originally known as Cancer Chemotherapy National Service Center number, the NSC# is an identifying number assigned by NCI-DTP to an agent or product (e.g. small molecule or biological agent).
2 Most structures have a unique NSC number but over the years a small percentage of structures or agents may have been assigned more than one NSC number. In the case of salts, different salt forms (e.g. HCl, HOAc) are designated with separate NSC numbers.

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