Clinical Trial NSCs

NSC Name Mechanism Current Status Previous Status
9219 Quercetin TOP2|AO|NonCan:COMT Clinical trial Clinical trial
36405 Chelerythrine BCL2|PK:PRKCA,STK Clinical trial Clinical trial
36586 GENISTEIN TOP2|PK:YK Clinical trial Clinical trial
62343 3-Bromopyruvate (acid) Mito|HK2 Clinical trial Clinical trial
63984 Cordycepin Ds Clinical trial Clinical trial
93766 Hydrastinine HCl NonCan:Antihemorrhagic Clinical trial Clinical trial
109874 Benzimate TUBB Clinical trial Clinical trial
112907 TETRAHYDROURIDINE Clinical trial Clinical trial
116069 Cerulenin FAS|FASN|HMGCS1/2 Clinical trial Clinical trial
130181 Tirapazamine DDI Clinical trial Clinical trial
142784 TEMPOL RP|FRS Clinical trial Clinical trial
174939 Elesclomol PK:ROS1 Clinical trial Clinical trial
217990 Pluripotin GTPase|RAS|RASA1|PK:STK,MAP3K Clinical trial Clinical trial
221019 WORTMANNIN PK:PIK3 Clinical trial Clinical trial
255109 geldanamycin analog HSP90 Clinical trial Clinical trial
264137 Elliptinium Acetate TOP2 Clinical trial Clinical trial
280594 TRICIRIBINE PHOSPHATE PK:STK,AKT1 Clinical trial Clinical trial
281612 benzaldehyde (BEN) A7 Clinical trial Clinical trial
308847 AMONAFIDE TOP2 Clinical trial Clinical trial
313425 Imexon Apo Clinical trial Clinical trial
320846 Batracylin TOP2|TOP1 Clinical trial Clinical trial
324360 Didox Clinical trial Clinical trial
326231 Buthionine sulphoximine AM Clinical trial Clinical trial
330507 Tanespimycin HSP90 Clinical trial Clinical trial
350625 tic10 Clinical trial Clinical trial
354258 8-Chloro-adenosine AM Clinical trial Clinical trial
354462 HYPOTHEMYCIN PK:YK,MAP2K1,MAP2K2 Clinical trial Clinical trial
365798 Fostamatinib Ds|Rs|PK:YK,SYK Clinical trial Clinical trial
366140 PYRAZOLOACRIDINE Db Clinical trial Clinical trial
374551 FENRETINIDE Ds Clinical trial Clinical trial
376128 DOLASTATIN 10 TUBB Clinical trial Clinical trial
377381 Antineoplaston A10 Clinical trial Clinical trial
600011 Tesmilifene hydrochloride Ho Clinical trial Clinical trial
609974 Carboxyamidotriazole AM Clinical trial Clinical trial
618487 Staurosporine PK:PRKCA,SRC,Multikinase Clinical trial Clinical trial
619130 Antineoplaston A10 Clinical trial Clinical trial
627168 Pyrazoloacridine Db Clinical trial Clinical trial
629749 Lapachone TOP2|TOP1 Clinical trial Clinical trial
637037 O-6-Benzylguanine DDR|MGMT Clinical trial Clinical trial
638646 7-Hydroxystaurosporine PK:STK,CDK1,CDK2,CDK4,CDK6 Clinical trial Clinical trial
638850 7-Hydroxystaurosporine PK:STK,CDK1,CDK2,CDK4,CDK6 Clinical trial Clinical trial
639966 Perifosine PK:STK,AKT,AKT1,AKT2,AKT3 Clinical trial Clinical trial
648539 Antineoplaston A10 Clinical trial Clinical trial
649890 Alvocidib CCNT1|PK:STK,CDK,CDK1,CDK2,CDK4,CDK6,CDK7,CDK8,CDK9 Clinical trial Clinical trial
656889 XK-469 TOP2 Clinical trial Clinical trial
663249 Triapine Dr|CC Clinical trial Clinical trial
668814 Kahalide F Clinical trial Clinical trial
677083 Okadaic acid Pase Clinical trial Clinical trial
678515 FAU Db Clinical trial Clinical trial
679828 PD-98059 PK:STK,MAP2K,MAP2K1,MAP2K2 Clinical trial Clinical trial
684363 Epothilone B TUBB|Tu-stab Clinical trial Clinical trial
684681 EF-5 Clinical trial Clinical trial
686288 AMINOFLAVONE Db|DDI Clinical trial Clinical trial
694501 BN-2629 Db Clinical trial Clinical trial
697286 LY-294002 PK:PIK3 Clinical trial Clinical trial
697726 RH1 PK:ROS1 Clinical trial Clinical trial
697887 XK-469 TOP2 Clinical trial Clinical trial
697912 5-Fluoro deoxy uridine 10mer Ds|AM Clinical trial Clinical trial
698215 XK-469 TOP2 Clinical trial Clinical trial
701554 Seliciclib PK:STK,CDK,CDK2,CDK7,CDK9 Clinical trial Clinical trial
702827 Orantinib PK:YK,PDGFR,FGFR,VEGFR,KDR Clinical trial Clinical trial
703081 SL-0101 RPS6 Clinical trial Clinical trial
706995 Entinostat HDAC Clinical trial Clinical trial
707545 Alvespimycin HSP90 Clinical trial Clinical trial
708298 AR-67 TOP1 Clinical trial Clinical trial
710270 Karenitecin TOP1 Clinical trial Clinical trial
710297 PX-316 PK:STK Clinical trial Clinical trial
710464 AFP464 Db|DDI Clinical trial Clinical trial
713763 Rebimastat PSM Clinical trial Clinical trial
714597 Imexon Apo Clinical trial Clinical trial
719239 E-7820 Ang|ITG Clinical trial Clinical trial
721782 D-1MT AM|INDO|IDO1|PK:ROS1 Clinical trial Clinical trial
722134 Sonolisib PK:PIK3 Clinical trial Clinical trial
724998 LMP-400 TOP1 Clinical trial Clinical trial
725776 LMP776 TOP1 Clinical trial Clinical trial
726188 IPdR Clinical trial Clinical trial
727859 (R)-(-)-Gossypol acetic acid Apo|BCL2 Clinical trial Clinical trial
728165 Lificguat HYP|HIF1|EPAS1 Clinical trial Clinical trial
732011 SR16157 Ho Clinical trial Clinical trial
734325 DMAPT NFkB Clinical trial Clinical trial
737664 Veliparib PARP|PARP1|PARP2 Clinical trial Clinical trial
741899 BML-277 PK:CHEK,CHEK2 Clinical trial Clinical trial
744912 Obatoclax Apo|BCL2 Clinical trial Clinical trial
749712 AT-13387 HSP90 Clinical trial Clinical trial
751249 Dactolisib PK:STK,PIK3,MTOR Clinical trial Clinical trial
751297 Y-27632 RHO Clinical trial Clinical trial
752493 Iniparib PARP|PARP1|PARP2 Clinical trial Clinical trial
752840 Veliparib PARP|PARP1|PARP2 Clinical trial Clinical trial
754344 Rigosertib RAS|Tu-stab|PK:STK,PLK1 Clinical trial Clinical trial
754345 JNJ-28312141 PK:YK,CSF1R Clinical trial Clinical trial
754346 AMG-458 PK:YK,MET Clinical trial Clinical trial
754347 Peptide [CRGDKGPDC - cys & cys bridge Clinical trial Clinical trial
754348 PF-03084014 diastereomer 1 PSM|APH1|Gamma secretase Clinical trial Clinical trial
754349 Amuvatinib RAD51|PK:YK,PDGFR,KIT,FLT3,Multikinase Clinical trial Clinical trial
754350 CB-64D Sig2Rec Clinical trial Clinical trial
754351 XL-147 PK:PIK3 Clinical trial Clinical trial
754352 Adavosertib PK:STK,YK,WEE1 Clinical trial Clinical trial
754353 Buparlisib PK:PIK3 Clinical trial Clinical trial
754354 GSK-461364 PK:STK,PLK1 Clinical trial Clinical trial
754356 PF-562271 PK:YK,FAK Clinical trial Clinical trial
754357 RAF-265 GTPase|PK:BRAF Clinical trial Clinical trial
754358 TDP-665759 Apo|MDM2 Clinical trial Clinical trial
754359 AEG-40730 Apo|IAP Clinical trial Clinical trial
754360 MI-219 Apo|MDM2 Clinical trial Clinical trial
754361 Astex FGF inhibitor PK:YK,FGFR Clinical trial Clinical trial
754362 SB-590885 GTPase|PK:YK,BRAF Clinical trial Clinical trial
754364 Targegen B-Raf/PDGFR inhibitor Cpd 6 GTPase|PK:YK,PDGFR,BRAF Clinical trial Clinical trial
754365 XR-11576 TOP2|TOP1 Clinical trial Clinical trial
754366 XR-5944 TOP2|TOP1 Clinical trial Clinical trial
754367 XR-5000 TOP2|TOP1 Clinical trial Clinical trial
755385 Pictilisib PK:PIK3 Clinical trial Clinical trial
755386 Ispinesib TUBB|CC|CDH16|KIF11|Kinesin|PK:YK Clinical trial Clinical trial
755387 Sepantronium bromide Apo|BIRC5 Clinical trial Clinical trial
755388 Fenoprofen Clinical trial Clinical trial
755402 Meclofenamate Clinical trial Clinical trial
755761 XAV-939 Wnt|PK:YK,TNKS Clinical trial Clinical trial
755762 Luminespib HSP90 Clinical trial Clinical trial
755763 Pimasertib PK:STK,YK,MAP2K,MAP2K1,MAP2K2 Clinical trial Clinical trial
755765 GW-5074 GTPase|PK:RAF,RAF1 Clinical trial Clinical trial
755766 H-89 Protein kinase A|PK:STK,AKT1 Clinical trial Clinical trial
755769 LY-294002 PK:PIK3 Clinical trial Clinical trial
755770 PD-0325901 PK:STK,MAP2K,MAP2K1 Clinical trial Clinical trial
755771 Salirasib GTPase|RAS|PK:YK,MTOR Clinical trial Clinical trial
755772 SB-203580 PK:STK,MAPK14,PDK1 Clinical trial Clinical trial
755773 1,9-Pyrazoleanthrone PK:STK,MAPK14,MAPK8 Clinical trial Clinical trial
755774 Staurosporine PK:PRKCA,SRC,Multikinase Clinical trial Clinical trial
755775 Foretinib PK:YK,MET,AXL,VEGFR,KDR,RON,Multikinase Clinical trial Clinical trial
755806 XL-147 PK:PIK3 Clinical trial Clinical trial
755807 Dactolisib PK:STK,PIK3,MTOR Clinical trial Clinical trial
755892 Hydrastinine HCl NonCan:Antihemorrhagic Clinical trial Clinical trial
755926 PF-03084014 diastereomer 1 PSM|APH1|Gamma secretase Clinical trial Clinical trial
755927 WZ-4002 PK:YK,EGFR Clinical trial Clinical trial
755981 WP-1034 STAT|PK:YK,JAK Clinical trial Clinical trial
755982 Semagacestat PSM|APH1|Gamma secretase Clinical trial Clinical trial
755983 BI-2536 PK:STK,PLK1 Clinical trial Clinical trial
756641 ICG-001 Apo|Wnt|CTNNB1 Clinical trial Clinical trial
756642 Entinostat HDAC Clinical trial Clinical trial
756646 IWR-1 Wnt|CTNNB1 Clinical trial Clinical trial
756648 AZD-1480 PK:YK,JAK,JAK1,JAK2 Clinical trial Clinical trial
756649 SB-431542 TGFB1|PK:STK,GSK3B Clinical trial Clinical trial
756650 RO-4929097 PSM|APH1|Gamma secretase Clinical trial Clinical trial
756651 Custom Peptide 835899 FGF|Protein kinase A|BAD|YWHA|PK:YK,PDGFR,RAF,VEGFR,MAP3K5 Clinical trial Clinical trial
756652 Linsitinib PK:YK,IGF1R Clinical trial Clinical trial
756653 SB-239063 PK:STK,MAPK14 Clinical trial Clinical trial
756654 ZM-336372 GTPase|PK:BRAF,RAF,RAF1 Clinical trial Clinical trial
756657 OSU-03012 PK:STK,PDK1 Clinical trial Clinical trial
756658 OSU-03013 PK:STK,PDK1 Clinical trial Clinical trial
756660 Quercetin TOP2|AO|NonCan:COMT Clinical trial Clinical trial
756662 sr 13654 BIRC5|PK:YK Clinical trial Clinical trial
756663 Obatoclax Apo|BCL2 Clinical trial Clinical trial
756874 NU-6027 PK:STK,ATR Clinical trial Clinical trial
756875 (+/-)-Nutlin-3 Apo|MDM2 Clinical trial Clinical trial
756876 (-)-Nutlin-3 Apo|MDM2 Clinical trial Clinical trial
756877 1st Precursor Intermediate to TDP 665759 Apo|MDM2 Clinical trial Clinical trial
756878 2nd Precursor Intermediate to TDP 665759 Apo|MDM2 Clinical trial Clinical trial
756879 Lificguat HYP|HIF1|EPAS1 Clinical trial Clinical trial
757148 AZD-7762 PK:STK,CHEK,CHEK1,CHEK2 Clinical trial Clinical trial
757149 Volasertib PK:STK,PLK1 Clinical trial Clinical trial
757333 SGI-1776 PK:STK,PIM1 Clinical trial Clinical trial
757334 Cpd-401 STAT|STAT3 Clinical trial Clinical trial
757438 PLX-4720 GTPase|PK:BRAF Clinical trial Clinical trial
757440 Deforolimius PK:STK,MTOR Clinical trial Clinical trial
757444 Barasertib PK:STK,AURK Clinical trial Clinical trial
758005 Sapitinib PK:YK,EGFR,ERBB2 Clinical trial Clinical trial
758006 BLZ-945 PK:CSF1R Clinical trial Clinical trial
758242 Tivantinib PK:YK,MET Clinical trial Clinical trial
758243 BMS-754807 PK:YK,IGF1R Clinical trial Clinical trial
758245 ENMD-2076 PK:STK,AURK,KDR Clinical trial Clinical trial
758248 RO-5126766 GTPase|PK:STK,YK,BRAF,MAP2K,RAF,MAP2K1,MAP2K2 Clinical trial Clinical trial
758249 Pracinostat HDAC Clinical trial Clinical trial
758250 SNS-314 PK:STK,AURK Clinical trial Clinical trial
758251 Amonafide TOP2 Clinical trial Clinical trial
758256 PKI-587 PK:STK,PIK3,MTOR Clinical trial Clinical trial
758257 LY-2606368 PK:STK,CHEK,CHEK1 Clinical trial Clinical trial
758484 Ezatiostat GSTP1|PK:STK,ROS1 Clinical trial Clinical trial
758485 BX-912 PK:STK,PDK1 Clinical trial Clinical trial
758486 HPI-1 SMO|Hg-Smo Clinical trial Clinical trial
758488 Lexibulin TUBB|Tu-frag|Tu-stab Clinical trial Clinical trial
758489 Indibulin TUBB|Tu-frag|PK:PTK Clinical trial Clinical trial
758490 Picoplatin A7|CC|AlkAg|IDNARep Clinical trial Clinical trial
758591 SGX-523 PK:YK,MET Clinical trial Clinical trial
758773 Varbulin TUBB|Tu-frag Clinical trial Clinical trial
758871 AZD-8055 PK:STK,MTOR Clinical trial Clinical trial
758872 Saracatinib PK:YK,FYN,LYN,FGFR,SRC,BLK,LCK,YES1 Clinical trial Clinical trial
758873 ABT-737 Apo|BCL2 Clinical trial Clinical trial
759094 ENMD-2076 Precursor PK:STK,AURK Clinical trial Clinical trial
759095 JNJ-38877605 PK:YK,MET Clinical trial Clinical trial
759096 Triapine Dr|CC Clinical trial Clinical trial
759498 CYC-116 PK:STK,AURK Clinical trial Clinical trial
759657 Quisinostat HDAC Clinical trial Clinical trial
759658 6-(4-pyrimidinyl)-1H-indazole derivative PK:STK,PDK1 Clinical trial Clinical trial
759659 Navitoclax Apo|BCL2 Clinical trial Clinical trial
759660 OSI-027 PK:STK,MTOR Clinical trial Clinical trial
759661 Dovitinib PK:YK,MET,PDGFR,EGFR,FGFR,KIT,VEGFR,FGFR1,FGFR3,FLT3 Clinical trial Clinical trial
759674 Pacritinib PK:YK,JAK,JAK2 Clinical trial Clinical trial
759675 KW-2449 BCR-ABL|PK:STK,AURK,FLT,FLT3 Clinical trial Clinical trial
759676 PI-103 PK:PIK3,MTOR Clinical trial Clinical trial
759677 Alisertib PK:STK,AURK Clinical trial Clinical trial
759905 4SC-202 HDAC Clinical trial Clinical trial
760143 Mocetinostat HDAC Clinical trial Clinical trial
760144 AT-9283 PK:STK,AURK Clinical trial Clinical trial
760183 (+)-JQ1 BRD Clinical trial Clinical trial
760419 Fenretinide Ds Clinical trial Clinical trial
760442 Daporinad NAMPT|PK:YK Clinical trial Clinical trial
760444 Tipifarnib FT|PK:YK Clinical trial Clinical trial
760536 PF-04691502 PK:PIK3 Clinical trial Clinical trial
760765 BMS-690514 PK:YK,EGFR,ERBB2,VEGFR Clinical trial Clinical trial
760841 Tandutinib PK:YK,PDGFR,FLT,KIT,FLT3 Clinical trial Clinical trial
760842 BIM-46187 Apo|GTPase|CASP Clinical trial Clinical trial
760843 Motesanib PK:YK,PDGFR,KIT,VEGFR,KDR,RET Clinical trial Clinical trial
761069 AMG-900 PK:STK,AURK Clinical trial Clinical trial
761070 VE-821 PK:STK,ATR Clinical trial Clinical trial
761188 Rabusertib PK:STK,CHEK,CHEK1 Clinical trial Clinical trial
761189 Teglarinad Apo|NAMPT Clinical trial Clinical trial
761192 Pevonedistat NFkB|NEDD8 Clinical trial Clinical trial
761193 Silmitasertib CK2|PK:STK Clinical trial Clinical trial
761194 CUDC-305 HSP90 Clinical trial Clinical trial
761215 TAK-733 PK:STK,MAP2K,MAP2K1,MAP2K2 Clinical trial Clinical trial
761216 Galunisertib TGFB1|PK:GSK3B Clinical trial Clinical trial
761217 Avagacestat PSM|APH1|Gamma secretase Clinical trial Clinical trial
761266 Motexafin Dr|TXNRD|PK:ROS1 Clinical trial Clinical trial
761387 CCT-128930 PK:STK,AKT,AKT1,AKT2,AKT3 Clinical trial Clinical trial
761390 By-Product of CUDC-305 HSP90 Clinical trial Clinical trial
761690 CP-91149 PYGL Clinical trial Clinical trial
761691 SCH-1473759 PK:STK,AURK Clinical trial Clinical trial
761692 MK-8033 PK:YK,MET Clinical trial Clinical trial
761693 Vertex ATR inhibitor Cpd 45 PK:STK,ATR Clinical trial Clinical trial
761759 TAK-960 analog PK:STK,PLK1 Clinical trial Clinical trial
761760 BMS-536924 PK:YK,IGF1R Clinical trial Clinical trial
761879 ITRI-260 PK:YK,FLT,FLT3 Clinical trial Clinical trial
761931 KHK-Indazole PK:YK,IGF1R Clinical trial Clinical trial
762151 TAK-901 PK:STK,AURK Clinical trial Clinical trial
762152 ONX-0914 PSM Clinical trial Clinical trial
762153 ST-3595 HDAC Clinical trial Clinical trial
762154 Des-fluoro-TAK-960 PK:STK,PLK1 Clinical trial Clinical trial
762381 CGI Diphenylurea PK inhibitor PK:YK,EPHA4,PDGFR,VEGFR Clinical trial Clinical trial
762382 CH-5132799 PK:PIK3 Clinical trial Clinical trial
762418 TAK Plk inhibitor PK:STK,PLK1 Clinical trial Clinical trial
762419 CT-32228 AGPAT2|PK:YK,VEGFR Clinical trial Clinical trial
762521 RO-4987655 PK:STK,MAP2K Clinical trial Clinical trial
762598 BAL-27862 TUBB|Tu-frag Clinical trial Clinical trial
762672 BMS-299897 PSM|APH1|Gamma secretase Clinical trial Clinical trial
762673 SB-1317 PK:STK,CDK,ERK,FLT,JAK,FLT3 Clinical trial Clinical trial
762829 MK-0752 PSM|APH1|Gamma secretase Clinical trial Clinical trial
762831 MK-0752 PSM|APH1|Gamma secretase Clinical trial Clinical trial
763094 JZL-184 MGLL Clinical trial Clinical trial
763443 (+)-Nutlin-3 Apo|MDM2 Clinical trial Clinical trial
763444 PF-477736 PK:STK,CHEK,CHEK1 Clinical trial Clinical trial
763525 Pluripotin GTPase|RAS|RASA1|PK:STK,MAP3K Clinical trial Clinical trial
763526 Crenolanib PK:YK,PDGFR,KIT,VEGFR,TEK,FLT3 Clinical trial Clinical trial
763527 JZL-195 MGLL Clinical trial Clinical trial
763564 EMD-534085 CDH16|KIF11|Kinesin|PK:YK Clinical trial Clinical trial
763579 AT-13387 HSP90 Clinical trial Clinical trial
763758 SEN-450 SMO Clinical trial Clinical trial
763832 LOR-253 KLF4|MYC|MTF1 Clinical trial Clinical trial
763929 Orantinib PK:YK,PDGFR,FGFR,VEGFR,KDR Clinical trial Clinical trial
763930 AS-703569 PK:AURK Clinical trial Clinical trial
763931 PF-04217903 PK:MET Clinical trial Clinical trial
764036 Dinaciclib PK:STK,CDK,CDK1,CDK2,CDK5,CDK9 Clinical trial Clinical trial
764037 BP-1-102 STAT|IL6|STAT3 Clinical trial Clinical trial
764039 AZD-5363 PK:STK,AKT,AKT1,AKT2,AKT3 Clinical trial Clinical trial
764041 TAE-684 PK:YK,ALK Clinical trial Clinical trial
764043 (+)-JQ1 BRD Clinical trial Clinical trial
764090 BMS-777607 PK:MET,RON Clinical trial Clinical trial
764091 Apitolisib PK:PIK3,MTOR Clinical trial Clinical trial
764092 GSK-2126458 PK:PIK3 Clinical trial Clinical trial
764135 BMS-599626 PK:YK,EGFR,ERBB2 Clinical trial Clinical trial
764136 Abexinostat HDAC Clinical trial Clinical trial
764237 Linifanib PK:YK,CSF1R,PDGFR,VEGFR,FLT3,KDR Clinical trial Clinical trial
764238 6-Bromoindirubin-3'-Acetoxime PK:GSK3A Clinical trial Clinical trial
764239 AZD-4547 PK:YK,FGFR,FGFR1,FGFR2,FGFR3 Clinical trial Clinical trial
764276 t-dcyd Clinical trial Clinical trial
764334 delanzomib PSM Clinical trial Clinical trial
764481 Brivanib PK:YK,FGFR,VEGFR,FGFR1,FGFR2,FGFR3,KDR Clinical trial Clinical trial
764488 Orteronel CYP17A1 Clinical trial Clinical trial
764515 Pp-242 PK:MTOR Clinical trial Clinical trial
764516 ZSTK-474 PK:PIK3 Clinical trial Clinical trial
764517 UNC-0638 EHMT2|EHMT1/2 Clinical trial Clinical trial
764579 Inolitazone hydrochloride PPARG Clinical trial Clinical trial
764580 MK-2461 PK:MET,FGFR Clinical trial Clinical trial
764582 10058-F4 MYC Clinical trial Clinical trial
764608 BAL-101553 Tu-frag Clinical trial Clinical trial
764609 10074-G5 MYC Clinical trial Clinical trial
764658 INK-128 PK:MTOR Clinical trial Clinical trial
764659 SCH-900776 PK:STK,CHEK,CHEK1 Clinical trial Clinical trial
764755 Cerulenin FAS|FASN|HMGCS1/2 Clinical trial Clinical trial
764756 C-75 FAS|FASN Clinical trial Clinical trial
764757 SM-406 IAP Clinical trial Clinical trial
764764 ONX-0801 TYMS Clinical trial Clinical trial
764765 ARQ-680 PK:BRAF Clinical trial Clinical trial
764820 Gandotinib PK:JAK,JAK2,JAK3 Clinical trial Clinical trial
764823 Varlitinib PK:YK,EGFR,ERBB2 Clinical trial Clinical trial
765262 R-428 PK:AXL Clinical trial Clinical trial
765395 MPC-3100 HSP90 Clinical trial Clinical trial
765435 Ganetespib HSP90 Clinical trial Clinical trial
765436 YK-4-279 ERG|ETV Clinical trial Clinical trial
765632 LY-2109761 TGFB1|PK:GSK3B Clinical trial Clinical trial
765672 S-49076 PK:MET,AXL,FGFR,MERTK Clinical trial Clinical trial
765673 Litronesib TUBB|CDH16|KIF11 Clinical trial Clinical trial
765695 PD 184352 PK:MAP2K Clinical trial Clinical trial
765775 Gemcitabine elaidate Ds Clinical trial Clinical trial
765776 AZD-3514 AR Clinical trial Clinical trial
765865 ASP-3026 PK:ALK Clinical trial Clinical trial
765866 Refametinib PK:MAP2K,MAP2K1,MAP2K2 Clinical trial Clinical trial
765889 ABT-348 PK:AURK,VEGFR Clinical trial Clinical trial
765898 GDC-0152 IAP Clinical trial Clinical trial
765949 AEE-788 PK:EGFR,ERBB2,VEGF,VEGFR Clinical trial Clinical trial
766254 Oprozomib PSM Clinical trial Clinical trial
766255 CT-GSK183 PK:IGF1R,ALK Clinical trial Clinical trial
766271 PHA-665752 PK:MET Clinical trial Clinical trial
766288 AMG-208 PK:MET Clinical trial Clinical trial
766811 Odanacatib CTSB Clinical trial Clinical trial
766819 Sotrastaurin PK:PRKCA Clinical trial Clinical trial
766820 LY-2228820 PK:MAPK14 Clinical trial Clinical trial
766821 BMS-911543 PK:JAK,JAK1,JAK2,JAK3 Clinical trial Clinical trial
766824 CEP-14083 PK:ALK Clinical trial Clinical trial
766887 OSI-930 PK:PDGFR,KIT,VEGFR,Multikinase Clinical trial Clinical trial
766888 BBOA AEMD Clinical trial Clinical trial
766906 MLN-2480 PK:BRAF,RAF,RAF1 Clinical trial Clinical trial
766908 PD 173074 PK:PDGFR,FGFR,SRC,VEGFR,FGFR1,FGFR3 Clinical trial Clinical trial
766991 GSK-690693 PK:AKT,AKT1,AKT2,AKT3 Clinical trial Clinical trial
766992 BAY 61-3606 PK:SYK Clinical trial Clinical trial
767006 AEW-541 PK:YK,IGF1R Clinical trial Clinical trial
767048 BMS-387032 PK:CDK,CDK2,CDK7,CDK9 Clinical trial Clinical trial
767123 Saridegib SMO Clinical trial Clinical trial
767124 Enzastaurin PK:PRKCA,STK,PIK3,AKT Clinical trial Clinical trial
767126 LEQ-506 SMO Clinical trial Clinical trial
767128 Birinapant IAP Clinical trial Clinical trial
767189 AZD-2014 PK:MTOR Clinical trial Clinical trial
767470 MLN-0905 PK:PLK1 Clinical trial Clinical trial
767533 BMN-673 enantiomer PARP1 Clinical trial Clinical trial
767598 Momelotinib PK:JAK,JAK1,JAK2,JAK3 Clinical trial Clinical trial
767599 I-BET-151 BRD Clinical trial Clinical trial
767601 VX-944 IMPDH2|IMPDH1|IMPDH Clinical trial Clinical trial
767745 Pelitrexol GARTF Clinical trial Clinical trial
767746 ADW-742 PK:IGF1R,KIT Clinical trial Clinical trial
767896 LY-2940680 SMO Clinical trial Clinical trial
767897 BPR1J-097 PK:FLT,FLT3 Clinical trial Clinical trial
767898 Ipatasertib PK:AKT,AKT1,AKT2,AKT3 Clinical trial Clinical trial
767951 GSK-1904529A PK:IGF1R Clinical trial Clinical trial
767952 Rocilinostat HDAC Clinical trial Clinical trial
767953 R-1530 PK:PDGFR,CDK,FGFR,VEGFR,KDR,Multikinase Clinical trial Clinical trial
767954 EMD-1204831 PK:MET Clinical trial Clinical trial
768011 XL-541 GEMIN2 Clinical trial Clinical trial
768070 enantiomer of PF-4176340 PK:AKT Clinical trial Clinical trial
768071 Enantiomer of PF-4176340 PK:AKT Clinical trial Clinical trial
768072 TAK-960 PK:PLK1 Clinical trial Clinical trial
768100 SAR-245409 PK:PIK3 Clinical trial Clinical trial
768112 SAR-402674 TOP1 Clinical trial Clinical trial
768508 GSK-2636771 PK:PIK3,MTOR Clinical trial Clinical trial
768509 SNX-5422 HSP90 Clinical trial Clinical trial
768536 BAM7 BCL2 Clinical trial Clinical trial
768539 IDH1-Comp 301 IDH1 Clinical trial Clinical trial
768593 CEP-9722 PARP1 Clinical trial Clinical trial
771531 RG-7112 MDM2 Clinical trial Clinical trial
771532 GDC-0349 PK:MTOR,PIM3 Clinical trial Clinical trial
771644 ARQ-621 CDH16|KIF11 Clinical trial Clinical trial
771650 AT-13148 PK:AKT,AKT1,AKT2,AKT3 Clinical trial Clinical trial
771651 VX-322 PK:FLT,KIT,FLT3 Clinical trial Clinical trial
771652 SAR-125844 PK:MET Clinical trial Clinical trial
771750 LY-2874455 PK:FGFR,VEGFR,FGFR1,FGFR2,FGFR3,FGFR4 Clinical trial Clinical trial
771751 CUDC-907 HDAC|PK:PIK3 Clinical trial Clinical trial
771858 TAK-441 SMO Clinical trial Clinical trial
772196 Lestaurtinib PK:YK,FLT,NTRK,FLT3,JAK2 Clinical trial Clinical trial
772197 LY-2801653 PK:MET,AXL,FLT3,MERTK,MST1R,Multikinase Clinical trial Clinical trial
772198 LY-2090314 PK:GSK3A,GSK3B Clinical trial Clinical trial
772254 ARRY-520 Isomer A CDH16 Clinical trial Clinical trial
772255 ARRY-520 Isomer A CDH16 Clinical trial Clinical trial
772290 Pelitrexol isomer A GARTF Clinical trial Clinical trial
772291 Pelitrexol isomer B GARTF Clinical trial Clinical trial
772351 XL-888 HSP90 Clinical trial Clinical trial
772498 r406 PK:SYK Clinical trial Clinical trial
772499 Vatalanib CYP19A1|PK:YK,PDGFR,KIT,VEGFR,KDR Clinical trial Clinical trial
772563 ARRY-704 PK:MAP2K,MAP2K1,MAP2K2 Clinical trial Clinical trial
772564 IDH-C227 IDH1 Clinical trial Clinical trial
772595 KPT-185 XPO1 Clinical trial Clinical trial
772868 LCL-161 IAP Clinical trial Clinical trial
772885 PF-4942847 HSP90 Clinical trial Clinical trial
772886 Apatinib PK:VEGFR Clinical trial Clinical trial
772887 XL-019 PK:JAK,JAK2 Clinical trial Clinical trial
772920 ONX-0805 PK:JAK,JAK2 Clinical trial Clinical trial
772991 PKM2 (9) PKM Clinical trial Clinical trial
772992 Fostamatinib Ds|Rs|PK:YK,SYK Clinical trial Clinical trial
773094 R-547 PK:CDK,CDK1,CDK2,CDK4 Clinical trial Clinical trial
773095 BGT-226 PK:PIK3 Clinical trial Clinical trial
773096 IDH-C35 IDH1 Clinical trial Clinical trial
773174 LDHA Inhibitor-33 LDHA Clinical trial Clinical trial
773230 AZD-2461 PARP1|PARP2 Clinical trial Clinical trial
773260 KPT-251 XPO1 Clinical trial Clinical trial
773261 GSK-921 CDH16|KIF11 Clinical trial Clinical trial
773262 VX-689 PK:AURK Clinical trial Clinical trial
773263 Bafetinib BCR-ABL|PK:YK,FYN,LYN Clinical trial Clinical trial
773264 R-306465 HDAC Clinical trial Clinical trial
773265 B-7100 HSP90 Clinical trial Clinical trial
773394 AT-7519 RNA polymerase I|PK:CDK,CDK1,CDK2,CDK4,CDK6 Clinical trial Clinical trial
774651 Cilengitide Ang|ITG Clinical trial Clinical trial
774829 I-BET-762 BRD Clinical trial Clinical trial
774830 Milciclib PK:CDK,CDK1,CDK2,CDK4,CDK5,Multikinase Clinical trial Clinical trial
774831 Rebastinib BCR-ABL|PK:LYN,FGFR,SRC,VEGFR,TEK Clinical trial Clinical trial
774901 AZD-2858 Wnt|PK:GSK3A Clinical trial Clinical trial
774911 BAY-1000394 PK:CDK Clinical trial Clinical trial
775018 LDHA Cmp 35 LDHA Clinical trial Clinical trial
775306 P-529 PK:PIK3,AKT,FGFR,MTOR,VEGFR Clinical trial Clinical trial
775636 SCH-772984 PK:ERK,MAP3K,MAPK1 Clinical trial Clinical trial
775637 AMD-070 CXCR4 Clinical trial Clinical trial
775665 VX-702 PK:MAPK14 Clinical trial Clinical trial
775727 Torin2 PK:MTOR Clinical trial Clinical trial
775771 BMS-863233 PK:CDC7,CDK7,CDK9 Clinical trial Clinical trial
775790 Maritoclax MCL1 Clinical trial Clinical trial
776017 Telatinib PK:PDGFR,KIT,VEGFR,KDR Clinical trial Clinical trial
776043 CEP-32496 PK:BRAF Clinical trial Clinical trial
776066 AZD-1208 PK:PIM1,PIM2,PIM3 Clinical trial Clinical trial
776762 EXEL-7647 PK:EGFR,ERBB2,SRC,VEGFR Clinical trial Clinical trial
776786 P505-15 PK:SYK Clinical trial Clinical trial
776787 AZD-3463 PK:IGF1R,ALK Clinical trial Clinical trial
776790 MK-0429 ITG Clinical trial Clinical trial
776821 CCT-241533 PK:CHEK,CHEK2 Clinical trial Clinical trial
776996 PI-103 PK:PIK3,MTOR Clinical trial Clinical trial
777194 Daporinad NAMPT|PK:YK Clinical trial Clinical trial
777425 GDC-0032 PK:PIK3 Clinical trial Clinical trial
777445 GSK-1070916 PK:AURK Clinical trial Clinical trial
777446 Talmapimod PK:MAPK14 Clinical trial Clinical trial
777447 VTX-2337 TLR8 Clinical trial Clinical trial
777448 PFI-1 BRD Clinical trial Clinical trial
777571 BIX-01294 EHMT2|EHMT1/2 Clinical trial Clinical trial
777572 AZD-8186 PI3KB|PK:PIK3 Clinical trial Clinical trial
777573 E-7820 Ang|ITG Clinical trial Clinical trial
777586 5-aza-T-dCyd Clinical trial Clinical trial
777638 AZD-6738 PK:ATR Clinical trial Clinical trial
777639 LGK-974 Wnt|PORCN Clinical trial Clinical trial
777671 BRD-4770 EHMT2|EHMT1/2 Clinical trial Clinical trial
777718 VE-822 PK:ATR Clinical trial Clinical trial
777877 PF-4989216 PK:PIK3 Clinical trial Clinical trial
777879 AM-5992 PK:CDK,FLT,FLT3 Clinical trial Clinical trial
778305 Afuresertib PK:AKT,AKT1,AKT2,AKT3 Clinical trial Clinical trial
778364 Defactinib PK:FAK Clinical trial Clinical trial
778365 EPZ-5676 DOT1L Clinical trial Clinical trial
778366 EXEL-2280 PK:IGF1R,AURK,FGFR,SRC Clinical trial Clinical trial
778367 ARRY-614 PK:MAPK14 Clinical trial Clinical trial
778368 GSK-2141795 PK:AKT Clinical trial Clinical trial
778448 Ombrabulin TUBB|Tu-frag Clinical trial Clinical trial
778746 FH-535 PPARG Clinical trial Clinical trial
778747 OTX-015 BRD Clinical trial Clinical trial
778809 TAK-632 PK:BRAF Clinical trial Clinical trial
778810 VS-5584 PK:PIK3,MTOR Clinical trial Clinical trial
779218 CEP-28122 PK:ALK Clinical trial Clinical trial
779404 RG-7388 MDM2 Clinical trial Clinical trial
779407 GNE-617 NAMPT Clinical trial Clinical trial
779408 Deltarasin PDE6D Clinical trial Clinical trial
780019 PD183805 PK:EGFR,ERBB2 Clinical trial Clinical trial
780020 spebrutinib PK:BTK Clinical trial Clinical trial
780041 GSK-126 EZH2 Clinical trial Clinical trial
780042 CP-724714 PK:ERBB2 Clinical trial Clinical trial
780043 EPZ-004777 DOT1L Clinical trial Clinical trial
780163 SOMCL-12-81 PK:ALK Clinical trial Clinical trial
780204 TAS-116 HSP90 Clinical trial Clinical trial
780205 dimethylfasudil RHO Clinical trial Clinical trial
780249 AZD-6738 PK:ATR Clinical trial Clinical trial
780250 AZD-6738 ( R,S-isomer) PK:ATR Clinical trial Clinical trial
780290 SAR-260301 (enantiomer 1) PI3KB Clinical trial Clinical trial
780291 SAR-260301 (enantiomer 1) PI3KB Clinical trial Clinical trial
780404 AZ-505 SETD8|SMYD2 Clinical trial Clinical trial
780812 BMS-906024 APH1|Gamma secretase Clinical trial Clinical trial
780965 MK-0731 CDH16|KIF11 Clinical trial Clinical trial
781008 maritoclax MCL1 Clinical trial Clinical trial
781009 MI-773 MDM2 Clinical trial Clinical trial
781016 BAY-87-2243 HIF1 Clinical trial Clinical trial
781148 CEP-37440 PK:ALK,FAK Clinical trial Clinical trial
781343 GDC-0994 PK:ERK,MAP3K,MAPK1 Clinical trial Clinical trial
781344 NMS-1286937 PK:PLK1 Clinical trial Clinical trial
781409 AGI-6780 IDH2 Clinical trial Clinical trial
781417 RN-486 PK:BTK Clinical trial Clinical trial
781468 CUDC-427 IAP Clinical trial Clinical trial
781469 BMS-833923 SMO Clinical trial Clinical trial
781470 PF-03758309 PK:PAK4 Clinical trial Clinical trial
781514 AMG-925 PK:CDK,CDK4,CDK6,FLT3 Clinical trial Clinical trial
781515 AMG-232 MDM2 Clinical trial Clinical trial
781516 entosplenitib PK:SYK Clinical trial Clinical trial
781626 Pacritinib PK:YK,JAK,JAK2 Clinical trial Clinical trial
781627 GSK-2606414 PK:EIF2AK3 Clinical trial Clinical trial
781652 ningetinib PK:MET Clinical trial Clinical trial
781761 LY-3009120 PK:BRAF,RAF1 Clinical trial Clinical trial
782006 PTC-691 PK:RET Clinical trial Clinical trial
782007 AZ-628 PK:BRAF Clinical trial Clinical trial
782017 H-89 Protein kinase A|PK:STK,AKT1 Clinical trial Clinical trial
782121 Volitinib PK:MET Clinical trial Clinical trial
782122 AMG-511 PK:PIK3 Clinical trial Clinical trial
782125 JNJ-54302833 FASN Clinical trial Clinical trial
782153 MG-132 PSM Clinical trial Clinical trial
782164 CX-5461 RNA polymerase I Clinical trial Clinical trial
782310 CPI-169 EZH2 Clinical trial Clinical trial
782362 PWT-33597 PK:PIK3,MTOR Clinical trial Clinical trial
782363 CH-5183284 PK:PDGFR,FGFR,VEGFR,FGFR1,FGFR2,FGFR3 Clinical trial Clinical trial
782457 VBY-825 CTSB Clinical trial Clinical trial
782549 Defactinib PK:FAK Clinical trial Clinical trial
782579 PCI-27483 F7 Clinical trial Clinical trial
782762 E-3810 PK:PDGFR,FGFR,VEGFR Clinical trial Clinical trial
782763 cs-1730 BRD Clinical trial Clinical trial
783015 CGM-097 MDM2 Clinical trial Clinical trial
783102 VS-4718 PK:FAK Clinical trial Clinical trial
783107 E-7449 PARP1|PARP2 Clinical trial Clinical trial
783249 JNJ-26483327 PK:EGFR,ERBB2,SRC,VEGFR,RET,Multikinase Clinical trial Clinical trial
783272 JNJ-47117096 PK:MELK Clinical trial Clinical trial
783294 VT-464 CYP17A1 Clinical trial Clinical trial
783296 Poziotinib PK:EGFR,ERBB2,Multikinase Clinical trial Clinical trial
783332 EPZ-5687 EZH2 Clinical trial Clinical trial
783333 SGI-1027 DNMT Clinical trial Clinical trial
783334 RG-108 DNMT Clinical trial Clinical trial
783360 IM-25 DNMT Clinical trial Clinical trial
783415 CB-839 GLS Clinical trial Clinical trial
783916 pyridoclax MCL1 Clinical trial Clinical trial
783917 GSK-2879552 KDM1A Clinical trial Clinical trial
784284 P-1446 PK:CDK,CDK1,CDK2,CDK4,CDK7,CDK9 Clinical trial Clinical trial
784415 Danusertib BCR-ABL|PK:YK,AURK,FGFR,RET Clinical trial Clinical trial
784590 Altiratinib PK:MET,NTRK,VEGFR,TEK,KDR Clinical trial Clinical trial
784591 CCT-251545 Wnt|PK:CDK19 Clinical trial Clinical trial
784722 aldoxorubicin TOP2 Clinical trial Clinical trial
784815 AZD-3147 PK:MTOR Clinical trial Clinical trial
784817 A-1210477 MCL1 Clinical trial Clinical trial
784856 CPI-0610 BRD Clinical trial Clinical trial
785004 MLN-7243 UB-activating Clinical trial Clinical trial
785117 PQR-309 PK:PIK3,MTOR Clinical trial Clinical trial
785222 BMS-983970 APH1|Gamma secretase Clinical trial Clinical trial
785299 EPZ-015666 PRMT5 Clinical trial Clinical trial
785300 BLU-9931 PK:FGFR,FGFR1,FGFR2,FGFR3,FGFR4 Clinical trial Clinical trial
785306 TAS-115 PK:MET,VEGFR Clinical trial Clinical trial
785345 Bet-BAY-002 BRD Clinical trial Clinical trial
785657 RX-3117 DNMT Clinical trial Clinical trial
786098 BAY-1143572 PK:CDK,CDK9 Clinical trial Clinical trial
786099 AZD-8835 PK:PIK3 Clinical trial Clinical trial
786100 CB-5083 VCP Clinical trial Clinical trial
786959 AZD-9496 SERD Clinical trial Clinical trial
787025 BAY-1161909 IDUA Clinical trial Clinical trial
787026 BAY-1217389 IDUA Clinical trial Clinical trial
787027 EGF-816 PK:EGFR Clinical trial Clinical trial
787038 AC-710 PK:CSF1R,PDGFR,FLT3 Clinical trial Clinical trial
787039 MI-503 KMT2A Clinical trial Clinical trial
787047 AZD-3965 SLC16A1|SLC16A7 Clinical trial Clinical trial
787048 azd5582 IAP Clinical trial Clinical trial
787081 SR 9243 NR1H1/2 Clinical trial Clinical trial
787137 AMG-319 PK:PIK3 Clinical trial Clinical trial
787251 Lomeguatrib MGMT Clinical trial Clinical trial
787252 TAE-226 PK:IGF1R,FAK Clinical trial Clinical trial
787253 LY-3039478 NOTCH Clinical trial Clinical trial
787269 SW-033291 HPGD Clinical trial Clinical trial
787312 PT-2385 EPAS1 Clinical trial Clinical trial
787326 GDC-0810 SERD Clinical trial Clinical trial
787780 Sabutoclax MCL1 Clinical trial Clinical trial
787827 CFG-920 CYP17A1 Clinical trial Clinical trial
787880 OTS-964 PK:PBK Clinical trial Clinical trial
787960 UMI-77 MCL1 Clinical trial Clinical trial
787962 KU-55933 PK:ATM Clinical trial Clinical trial
788121 AZD-3759 PK:EGFR Clinical trial Clinical trial
788186 Bafetinib BCR-ABL|PK:YK,FYN,LYN Clinical trial Clinical trial
788203 sitravatinib PK:PDGFR,AXL,NTRK,KDR,RET Clinical trial Clinical trial
788365 PF-06747775 PK:EGFR Clinical trial Clinical trial
788794 A-911 PK:CDK,CDK9 Clinical trial Clinical trial
788900 napabucasin CTNNB1|STAT3 Clinical trial Clinical trial
788992 OICR-9429 WDR5 Clinical trial Clinical trial
789040 CBL-0137 Clinical trial Clinical trial
789041 GSK-295 CENP Clinical trial Clinical trial
789042 LOR-253 KLF4|MYC|MTF1 Clinical trial Clinical trial
789043 ARV-825 BRD Clinical trial Clinical trial
789044 CCT-271850 IDUA Clinical trial Clinical trial
789099 LY-3154567 NAMPT Clinical trial Clinical trial
789223 AMG-337 PK:MET Clinical trial Clinical trial
789722 Litronesib TUBB|CDH16|KIF11 Clinical trial Clinical trial
789797 SW-044248 TOP1 Clinical trial Clinical trial
789968 LY-3023414 PK:PIK3,MTOR Clinical trial Clinical trial
789969 SB-202190 PK:MAPK14 Clinical trial Clinical trial
790182 Alofanib PK:FGFR Clinical trial Clinical trial
790865 EPZ-020411 PRMT6 Clinical trial Clinical trial
791059 MGCD-265 PK:MET,VEGFR Clinical trial Clinical trial
791163 RG-7602 PK:CHEK1 Clinical trial Clinical trial
791226 SAR-245409 PK:PIK3 Clinical trial Clinical trial
791227 XL-147 PK:PIK3 Clinical trial Clinical trial
791328 ARQ-092 PK:AKT Clinical trial Clinical trial
791495 GDC-0339 PK:PIM1,PIM2,PIM3 Clinical trial Clinical trial
791496 APR-246 Apo Clinical trial Clinical trial
791648 PF-2771 CENP Clinical trial Clinical trial
791783 eFT-508 MKNK1/2 Clinical trial Clinical trial
791785 Sapacitabine Ds Clinical trial Clinical trial
791966 CFI-400945 PK:PLK1 Clinical trial Clinical trial
791967 TAK-659 (isomer 1) PK:SYK Clinical trial Clinical trial
791968 TAK-659 (isomer 1) PK:SYK Clinical trial Clinical trial
792847 INCB-047775 PK:AKT Clinical trial Clinical trial
792849 Itacitinib PK:JAK1 Clinical trial Clinical trial
792955 GSK-2194069 FAS|FASN Clinical trial Clinical trial
792956 AZD-0156 PK:ATM Clinical trial Clinical trial
792969 VX-984 PK:PRKDC Clinical trial Clinical trial
792970 KPT-9274 PK:PAK4 Clinical trial Clinical trial
792971 CC-223 PK:MTOR Clinical trial Clinical trial
792987 GDC-0084 PK:PIK3,MTOR Clinical trial Clinical trial
792996 ARQ-087 PK:FGFR Clinical trial Clinical trial
792997 ARQ-087_Peak 2 Clinical trial Clinical trial
793103 ABBV-075 BRD Clinical trial Clinical trial
793148 RX-5902 Clinical trial Clinical trial
793149 BAY-876 SLC2A1 Clinical trial Clinical trial
793150 ensartinib PK:ALK Clinical trial Clinical trial
793151 CC-115 PK:MTOR Clinical trial Clinical trial
793322 naquotinib PK:EGFR Clinical trial Clinical trial
793323 BGB-283 PK:BRAF Clinical trial Clinical trial
793324 BAY-1125976 PK:AKT,AKT2 Clinical trial Clinical trial
793430 CPI-1205 EZH2 Clinical trial Clinical trial
793585 LY-3177833 PK:CDC7,CDK7 Clinical trial Clinical trial
793677 ASP-5878 PK:FGFR Clinical trial Clinical trial
793679 CNDAC Clinical trial Clinical trial
793726 CCT-245737 PK:CHEK1 Clinical trial Clinical trial
793727 CCT-251921 PK:CDK,CDK19 Clinical trial Clinical trial
794109 LGH-447 PK:PIM1 Clinical trial Clinical trial
794442 PQR-620 PK:MTOR Clinical trial Clinical trial
794443 KPT-8602 XPO1 Clinical trial Clinical trial
794487 BAY-1436032 IDH1 Clinical trial Clinical trial
794589 NTRC-0066-0 PK:TTK Clinical trial Clinical trial
794590 BAY-1082439 PK:PIK3 Clinical trial Clinical trial
794646 AMG-51 PK:MET Clinical trial Clinical trial
795067 IPI-549 Clinical trial Clinical trial
795142 M2698 PK:AKT,AKT1,AKT2,AKT3 Clinical trial Clinical trial
795384 serabelisib Clinical trial Clinical trial
795718 BLU-554 PK:FGFR,FGFR4 Clinical trial Clinical trial
795781 GSK-2795039 Clinical trial Clinical trial
796100 PF-06840003 IDO1 Clinical trial Clinical trial
796101 ABC-294640 SPHK2 Clinical trial Clinical trial
796433 PF-04136309 Clinical trial Clinical trial
797172 A-1331852 Clinical trial Clinical trial
797393 AT-265 HSP90 Clinical trial Clinical trial
797653 WT-161 HDAC Clinical trial Clinical trial
797769 ABC-1183 Clinical trial Clinical trial
797770 CEP-40783 Clinical trial Clinical trial
797771 ulixertinib PK:ERK Clinical trial Clinical trial
797772 Selonsertib PK:MAP3K5 Clinical trial Clinical trial
797932 PLX-8394 PK:BRAF Clinical trial Clinical trial
797933 tirabrutinib PK:BTK Clinical trial Clinical trial
797934 Plinabulin Clinical trial Clinical trial
797938 AZD-5153 Clinical trial Clinical trial
798200 TP-0903 PK:AXL Clinical trial Clinical trial
798201 VH-298 VHL Clinical trial Clinical trial
798202 fenebrutinib PK:BTK Clinical trial Clinical trial
798303 BPTES GLS Clinical trial Clinical trial
798304 EC-330 MDM2 Clinical trial Clinical trial
798517 SAR-20347 PK:TYK2 Clinical trial Clinical trial
798799 GS-9901 Clinical trial Clinical trial
798846 S-63845 Clinical trial Clinical trial
799644 DDP-38003 Clinical trial Clinical trial
799645 Aurigene Cmp 4 Clinical trial Clinical trial
799771 BMS-988205 IDO1 Clinical trial Clinical trial
799908 GNE-140 LDHA Clinical trial Clinical trial
800019 PF-06821497 EZH2 Clinical trial Clinical trial
800030 LXS-196 PK:PRKCA Clinical trial Clinical trial
800283 H3B-6527 PK:FGFR Clinical trial Clinical trial
800404 GSK-3326595 PRMT5 Clinical trial Clinical trial
800522 TPX-0005 PK:ROS1,ALK Clinical trial Clinical trial
800525 BAY-1895344 PK:ATR Clinical trial Clinical trial
800729 GDC-0077 Clinical trial Clinical trial
800888 CFI-402257 IDUA|PK:TTK Clinical trial Clinical trial
800890 MSC-2530818 PK:CDK Clinical trial Clinical trial
800892 Evobrutinib PK:BTK Clinical trial Clinical trial
800893 milademetan MDM2 Clinical trial Clinical trial
801089 PRN-1371 PK:FGFR Clinical trial Clinical trial
801230 BMS-986158 Clinical trial Clinical trial
801661 TAK-931 PK:CDC7 Clinical trial Clinical trial
801812 CPI-444 Clinical trial Clinical trial
801813 AZD-4205 PK:JAK Clinical trial Clinical trial
802100 ON-123300 PK:CDK,RET Clinical trial Clinical trial
802101 AZD-4635 Clinical trial Clinical trial
802450 BAY-1251152 Clinical trial Clinical trial
802451 LY-3200882 Clinical trial Clinical trial
802548 AZD-5069 CXCR2 Clinical trial Clinical trial
802820 FT-1518 PK:MTOR Clinical trial Clinical trial
802821 PQR-530 PK:MTOR Clinical trial Clinical trial
802822 nedisertib Clinical trial Clinical trial
803014 Tenalisib Clinical trial Clinical trial
803247 CB-1158 Clinical trial Clinical trial
803248 MTX-211 PK:EGFR Clinical trial Clinical trial
803408 EED-226 EED Clinical trial Clinical trial
803409 BAY-1816032 PK:BUB1 Clinical trial Clinical trial
803410 LY-3214996 PK:ERK Clinical trial Clinical trial
803552 SGN-2FF Clinical trial Clinical trial
803600 AG-881 IDH1|IDH2 Clinical trial Clinical trial
803601 LYC-55716 Clinical trial Clinical trial
803789 AZD-1390 PK:ATM Clinical trial Clinical trial
803790 Aurigene Cpm 16 Clinical trial Clinical trial
804040 E-7046 Clinical trial Clinical trial
804041 AMG-176 Clinical trial Clinical trial
804253 Pamiparib PARP1|PARP2 Clinical trial Clinical trial
804254 SHP-099 PTPN11 Clinical trial Clinical trial
804518 BAY-1163877 PK:FGFR Clinical trial Clinical trial
804520 HDM-201 MDM2 Clinical trial Clinical trial
804521 S-222611 PK:EGFR,ERBB2 Clinical trial Clinical trial
804861 ASTX-660 IAP Clinical trial Clinical trial
804862 EPZ-031686 SMYD3 Clinical trial Clinical trial
804962 FGF-401 PK:FGFR Clinical trial Clinical trial
805149 TP-3654 PK:PIM1,PIM3 Clinical trial Clinical trial
805500 SEL-120 PK:CDK Clinical trial Clinical trial
805596 IDF-11774 Clinical trial Clinical trial
805746 CC-671 PK:TTK Clinical trial Clinical trial
806387 CYC-065 PK:CDK Clinical trial Clinical trial
806388 E-7090 PK:FGFR Clinical trial Clinical trial
806595 PLX-51107 Clinical trial Clinical trial
806812 RG-6016 Clinical trial Clinical trial
807047 LXH-254 PK:RAF Clinical trial Clinical trial
807055 AZD-5991 Clinical trial Clinical trial
807398 INCB-057643 Clinical trial Clinical trial
807626 JNJ-3887618 Clinical trial Clinical trial
807627 BMS-986195 PK:BTK Clinical trial Clinical trial
808292 SGI-110 DNMT Clinical trial Clinical trial
808507 PF-6459988 PRMT5|PK:EGFR Clinical trial Clinical trial
808789 RG-7741 Clinical trial Clinical trial
808790 AZD-0364 PK:ERK Clinical trial Clinical trial
808792 CC-90003 PK:ERK Clinical trial Clinical trial
808793 Real Thiol Clinical trial Clinical trial
809099 EPZ-011989 EZH2 Clinical trial Clinical trial
809100 RG-7112 MDM2 Clinical trial Clinical trial
809251 ETC-159 Clinical trial Clinical trial
809252 PF-06855800 PRMT5 Clinical trial Clinical trial
809694 BOS-172722 Clinical trial Clinical trial
809970 LOXO-195 Clinical trial Clinical trial
809971 S-64315 Clinical trial Clinical trial
809972 IACS-10759 Clinical trial Clinical trial
809973 BAY-2402234 DHODH Clinical trial Clinical trial
810114 Vecabrutinib PK:BTK Clinical trial Clinical trial
810341 PF-6459988 PRMT5|PK:EGFR Clinical trial Clinical trial
810717 CG-806 PK:BTK Clinical trial Clinical trial
811953 IACS-8968 IDO1 Clinical trial Clinical trial
812052 CH-7057288 Clinical trial Clinical trial
812172 ARS-1620 KRAS Clinical trial Clinical trial
812415 ABBV-744 Clinical trial Clinical trial
812727 relacorilant Clinical trial Clinical trial
812728 AZD-4320 Clinical trial Clinical trial
812901 PRN-1008 PK:BTK Clinical trial Clinical trial
812926 TAS-6417 PK:EGFR Clinical trial Clinical trial
812927 PF-06873600 PK:CDK Clinical trial Clinical trial
812928 IDH-305 IDH1 Clinical trial Clinical trial
813380 AZD-3229 Clinical trial Clinical trial
813381 valemetostat EZH2 Clinical trial Clinical trial
813488 futibutinib PK:FGFR Clinical trial Clinical trial
813859 RGX-104 Clinical trial Clinical trial
813862 Lapachone TOP2|TOP1 Clinical trial Clinical trial
814025 LSZ-102 SERD Clinical trial Clinical trial