| 740 |
Methotrexate |
Df|DHFR |
FDA approved |
FDA approved |
| 750 |
Busulfan |
A7|AlkAg |
FDA approved |
FDA approved |
| 752 |
6-Thioguanine |
Ds|IMPDH2|IMPDH |
FDA approved |
FDA approved |
| 755 |
6-Mercaptopurine |
Ds|PPAT |
FDA approved |
FDA approved |
| 757 |
Colchicine |
TUBB |
FDA approved |
FDA approved |
| 762 |
Nitrogen mustard |
A7|AlkAg |
FDA approved |
FDA approved |
| 1390 |
Allopurinol |
AM|XDH |
FDA approved |
FDA approved |
| 2821 |
Ferulic acid |
|
FDA approved |
FDA approved |
| 2833 |
phlorizin |
|
FDA approved |
FDA approved |
| 3053 |
Actinomycin D |
Db|RNA polymerase I |
FDA approved |
FDA approved |
| 3061 |
malacid |
DHFR |
FDA approved |
FDA approved |
| 3069 |
Chloramphenicol |
|
FDA approved |
FDA approved |
| 3088 |
Chlorambucil |
A7|AlkAg |
FDA approved |
FDA approved |
| 3090 |
badil |
|
FDA approved |
FDA approved |
| 3354 |
Estradiol Cypionate |
|
FDA approved |
FDA approved |
| 3590 |
Calcium leucovorin |
Df |
FDA approved |
FDA approved |
| 4291 |
Masoprocol |
|
FDA approved |
FDA approved |
| 4375 |
Hydroxychloroquine Sulfate |
Immunomodulatory |
FDA approved |
FDA approved |
| 4722 |
aloin |
|
FDA approved |
FDA approved |
| 5364 |
cinchonidine |
|
FDA approved |
FDA approved |
| 5366 |
Noscapine |
|
FDA approved |
FDA approved |
| 5751 |
salicin |
|
FDA approved |
FDA approved |
| 6396 |
Thiotepa |
A7|AlkAg |
FDA approved |
FDA approved |
| 8096 |
Beta-Sitosterol |
|
FDA approved |
FDA approved |
| 8797 |
degalol |
|
FDA approved |
FDA approved |
| 8806 |
Melphalan |
A7|AlkAg |
FDA approved |
FDA approved |
| 9706 |
Triethylenemelamine |
A7|AlkAg |
FDA approved |
FDA approved |
| 9896 |
diandron |
|
FDA approved |
FDA approved |
| 10023 |
Prednisone |
Ho |
FDA approved |
FDA approved |
| 10483 |
Desoximetasone |
|
FDA approved |
FDA approved |
| 10721 |
cortef fluid |
|
FDA approved |
FDA approved |
| 10973 |
Ethinyl Estradiol |
Ho |
FDA approved |
FDA approved |
| 12198 |
Dromostanolone Propionate |
Ho |
FDA approved |
FDA approved |
| 13397 |
Triamcinolone |
|
FDA approved |
FDA approved |
| 13875 |
Altretamine |
Db|AlkAg |
FDA approved |
FDA approved |
| 14229 |
Acrichine |
Db|AP |
FDA approved |
FDA approved |
| 15628 |
rozex |
|
FDA approved |
FDA approved |
| 17474 |
Eskazine |
|
FDA approved |
FDA approved |
| 18509 |
Aminolevulinic acid |
AM |
FDA approved |
FDA approved |
| 19893 |
Fluorouracil |
Ds|Rs|TYMS |
FDA approved |
FDA approved |
| 19987 |
Methylprednisolone |
NonCan:Anti-inflammatory |
FDA approved |
FDA approved |
| 20256 |
uridin |
|
FDA approved |
FDA approved |
| 23162 |
Nandrolone Phenpropionate |
Ho|NonCan:Ste |
FDA approved |
FDA approved |
| 23759 |
Testolactone |
Ho |
FDA approved |
FDA approved |
| 24559 |
Mithramycin |
Db|Rs |
FDA approved |
FDA approved |
| 25154 |
Pipobroman |
A7|AlkAg |
FDA approved |
FDA approved |
| 25953 |
Disulfiram |
|
FDA approved |
FDA approved |
| 26271 |
Cyclophosphamide |
A7|AlkAg |
FDA approved |
FDA approved |
| 26980 |
Mitomycin |
A2|AlkAg |
FDA approved |
FDA approved |
| 27640 |
Floxuridine |
Ds|TYMS |
FDA approved |
FDA approved |
| 32065 |
Hydroxyurea |
AM|Dr |
FDA approved |
FDA approved |
| 32982 |
Curcumin |
Apo |
FDA approved |
FDA approved |
| 33001 |
Fluorometholone |
|
FDA approved |
FDA approved |
| 33299 |
bena |
|
FDA approved |
FDA approved |
| 34462 |
Uracil Mustard |
A7|AlkAg |
FDA approved |
FDA approved |
| 34521 |
Dexamethasone Decadron |
Ho |
FDA approved |
FDA approved |
| 34936 |
naganol |
|
FDA approved |
FDA approved |
| 35347 |
biosone |
|
FDA approved |
FDA approved |
| 35443 |
Papaverine Hydrochloride |
|
FDA approved |
FDA approved |
| 38721 |
Mitotane |
A7|Ho|AlkAg|anti-Ho|CYP11A1 |
FDA approved |
FDA approved |
| 39661 |
Idoxuridine |
|
FDA approved |
FDA approved |
| 42199 |
Benztropine mesylate |
|
FDA approved |
FDA approved |
| 45388 |
Dacarbazine |
A7|AlkAg |
FDA approved |
FDA approved |
| 45923 |
Methoxsalen |
Db |
FDA approved |
FDA approved |
| 49842 |
Vinblastine |
TUBB|Tu-frag |
FDA approved |
FDA approved |
| 53477 |
hctz |
|
FDA approved |
FDA approved |
| 56423 |
Melatonin |
|
FDA approved |
FDA approved |
| 57197 |
Caffeic Acid |
|
FDA approved |
FDA approved |
| 59272 |
r-e-s |
|
FDA approved |
FDA approved |
| 59687 |
Acetalax |
NonCan:Cath |
FDA approved |
FDA approved |
| 61805 |
kantaridin |
|
FDA approved |
FDA approved |
| 62791 |
ergosterol |
|
FDA approved |
FDA approved |
| 63878 |
Cytarabine |
Ds |
FDA approved |
FDA approved |
| 66847 |
Thalidomide |
Ang|Immunomodulatory |
FDA approved |
FDA approved |
| 67574 |
Vincristine |
TUBB|Tu-frag |
FDA approved |
FDA approved |
| 71047 |
lactone |
|
FDA approved |
FDA approved |
| 71423 |
Megestrol Acetate |
Ho|PGR |
FDA approved |
FDA approved |
| 75520 |
tfdu |
TYMS |
FDA approved |
FDA approved |
| 77213 |
Procarbazine |
A7|AlkAg |
FDA approved |
FDA approved |
| 77541 |
amuno |
|
FDA approved |
FDA approved |
| 78206 |
Cyclobenzaprine Hydrochloride |
|
FDA approved |
FDA approved |
| 79037 |
Lomustine |
A6|AlkAg |
FDA approved |
FDA approved |
| 79269 |
Vistonuridine |
TUBB|FU-Antidote |
FDA approved |
FDA approved |
| 79389 |
Clofibrate |
|
FDA approved |
FDA approved |
| 80998 |
Cortivazol |
|
FDA approved |
FDA approved |
| 81549 |
Penicillamine |
|
FDA approved |
FDA approved |
| 82151 |
Daunorubicin |
TOP2 |
FDA approved |
FDA approved |
| 82174 |
Nalidixic Acid |
|
FDA approved |
FDA approved |
| 83142 |
Daunorubicin |
TOP2 |
FDA approved |
FDA approved |
| 85442 |
Amiodarone Hydrochloride |
|
FDA approved |
FDA approved |
| 85998 |
Streptozocin |
A7|AlkAg |
FDA approved |
FDA approved |
| 88536 |
Calusterone |
Ho |
FDA approved |
FDA approved |
| 88789 |
Cyclacillin |
|
FDA approved |
FDA approved |
| 89201 |
Estramustine |
A7|TUBB|AlkAg |
FDA approved |
FDA approved |
| 90636 |
Vinblastine |
TUBB|Tu-frag |
FDA approved |
FDA approved |
| 92339 |
Fluphenazine |
NonCan:Psy |
FDA approved |
FDA approved |
| 92859 |
Arsenic trioxide |
Apo |
FDA approved |
FDA approved |
| 93819 |
ergenyl |
PK:GSK3A,GSK3B |
FDA approved |
FDA approved |
| 94600 |
Camptothecin |
TOP1 |
FDA approved |
FDA approved |
| 95100 |
Digoxin |
NonCan:CardG |
FDA approved |
FDA approved |
| 100071 |
Haloprogin |
|
FDA approved |
FDA approved |
| 100880 |
Camptothecin |
TOP1 |
FDA approved |
FDA approved |
| 102816 |
Azacitidine |
DNMT |
FDA approved |
FDA approved |
| 103805 |
ancotil |
|
FDA approved |
FDA approved |
| 105014 |
Cladribine |
Ds|ADA |
FDA approved |
FDA approved |
| 105024 |
Mithramycin |
Db|Rs |
FDA approved |
FDA approved |
| 105823 |
Acadesine |
AM |
FDA approved |
FDA approved |
| 109229 |
Asparaginase |
AM|Pi |
FDA approved |
FDA approved |
| 109500 |
Cromolyn Sodium |
|
FDA approved |
FDA approved |
| 109724 |
Ifosfamide |
A7|AlkAg |
FDA approved |
FDA approved |
| 109929 |
Asparaginase |
AM|Pi |
FDA approved |
FDA approved |
| 111180 |
Acetylcysteine |
|
FDA approved |
FDA approved |
| 113891 |
Mesna |
|
FDA approved |
FDA approved |
| 113926 |
rifa |
|
FDA approved |
FDA approved |
| 117186 |
Acetalax |
NonCan:Cath |
FDA approved |
FDA approved |
| 118218 |
Fludarabine |
Ds|AM|Dr|STAT1 |
FDA approved |
FDA approved |
| 119875 |
Cisplatin |
A7|AlkAg |
FDA approved |
FDA approved |
| 122758 |
Isotretinoin |
Ho|RXR|Differentiator |
FDA approved |
FDA approved |
| 122819 |
Teniposide |
TOP2 |
FDA approved |
FDA approved |
| 123127 |
Doxorubicin |
TOP2 |
FDA approved |
FDA approved |
| 124463 |
Fludarabine |
Ds|AM|Dr|STAT1 |
FDA approved |
FDA approved |
| 125066 |
Bleomycin |
Db |
FDA approved |
FDA approved |
| 125973 |
Paclitaxel |
TUBB|Tu-stab |
FDA approved |
FDA approved |
| 127716 |
Decitabine |
AM|DNMT |
FDA approved |
FDA approved |
| 129185 |
melbex |
|
FDA approved |
FDA approved |
| 134727 |
Mitomycin |
A2|AlkAg |
FDA approved |
FDA approved |
| 138783 |
Bendamustine |
A2|A6|AlkAg |
FDA approved |
FDA approved |
| 141540 |
Etoposide |
TOP2 |
FDA approved |
FDA approved |
| 141549 |
M-AMSA |
TOP2 |
FDA approved |
FDA approved |
| 141633 |
Homoharringtonine |
Apo|Ang|Pi |
FDA approved |
FDA approved |
| 141993 |
Minocycline Hydrochloride |
|
FDA approved |
FDA approved |
| 143020 |
Mithramycin |
Db|Rs |
FDA approved |
FDA approved |
| 145668 |
Ancitabine hydrochloride |
Ds |
FDA approved |
FDA approved |
| 148958 |
Tegafur |
Df |
FDA approved |
FDA approved |
| 150817 |
nysert |
|
FDA approved |
FDA approved |
| 154948 |
M-AMSA |
TOP2 |
FDA approved |
FDA approved |
| 156303 |
M-AMSA |
TOP2 |
FDA approved |
FDA approved |
| 157035 |
Parthenolide |
Apo |
FDA approved |
FDA approved |
| 163039 |
ribavirin |
|
FDA approved |
FDA approved |
| 163661 |
3'-deoxy-2'-thymidinene |
|
FDA approved |
FDA approved |
| 165706 |
Cupric Chloride |
|
FDA approved |
FDA approved |
| 169434 |
florid |
|
FDA approved |
FDA approved |
| 169780 |
Dexrazoxane |
TOP2|NonCan:Cardioprotective |
FDA approved |
FDA approved |
| 170984 |
Pimozide |
NonCan:Psy |
FDA approved |
FDA approved |
| 170986 |
Miconazole |
|
FDA approved |
FDA approved |
| 177023 |
Levamisole Hydrochloride |
|
FDA approved |
FDA approved |
| 180973 |
Tamoxifen |
Ho|SERM |
FDA approved |
FDA approved |
| 184849 |
Mebendazole |
Tu-stab |
FDA approved |
FDA approved |
| 196515 |
Dinoprost Tromethamine |
|
FDA approved |
FDA approved |
| 208734 |
aclarubicin |
TOP2 |
FDA approved |
FDA approved |
| 218321 |
Pentostatin |
Ds|AM|ADA |
FDA approved |
FDA approved |
| 226080 |
Rapamycin |
PK:STK,MTOR |
FDA approved |
FDA approved |
| 227189 |
aloin |
|
FDA approved |
FDA approved |
| 241240 |
Carboplatin |
A7|AlkAg |
FDA approved |
FDA approved |
| 243115 |
Econazole Nitrate |
|
FDA approved |
FDA approved |
| 246131 |
Valrubicin |
TOP2 |
FDA approved |
FDA approved |
| 248616 |
Spectinomycin Hydrochloride |
|
FDA approved |
FDA approved |
| 249992 |
M-AMSA |
TOP2 |
FDA approved |
FDA approved |
| 256439 |
Idarubicin |
TOP2 |
FDA approved |
FDA approved |
| 256857 |
dolgit |
|
FDA approved |
FDA approved |
| 256942 |
Epirubicin |
TOP2 |
FDA approved |
FDA approved |
| 257473 |
Clotrimazole |
|
FDA approved |
FDA approved |
| 265489 |
bestatin |
|
FDA approved |
FDA approved |
| 266046 |
Oxaliplatin |
A7|AlkAg |
FDA approved |
FDA approved |
| 279836 |
Mitoxantrone |
TOP2 |
FDA approved |
FDA approved |
| 287459 |
Cytarabine |
Ds |
FDA approved |
FDA approved |
| 290193 |
ciclosporin |
|
FDA approved |
FDA approved |
| 292810 |
Prazosin Hydrochloride |
|
FDA approved |
FDA approved |
| 296961 |
Amifostine |
RP |
FDA approved |
FDA approved |
| 299589 |
Domperidone |
|
FDA approved |
FDA approved |
| 301739 |
Mitoxantrone |
TOP2 |
FDA approved |
FDA approved |
| 312887 |
Fludarabine |
Ds|AM|Dr|STAT1 |
FDA approved |
FDA approved |
| 315851 |
Bupropion Hydrochloride |
|
FDA approved |
FDA approved |
| 317629 |
ketoconazole |
CYP19A1 |
FDA approved |
FDA approved |
| 321521 |
auranofin |
|
FDA approved |
FDA approved |
| 337250 |
dfmo hcl |
|
FDA approved |
FDA approved |
| 352122 |
Trimetrexate glucuronate |
Df|DHFR |
FDA approved |
FDA approved |
| 356717 |
renoquid |
|
FDA approved |
FDA approved |
| 362856 |
Temozolomide |
A7|AlkAg |
FDA approved |
FDA approved |
| 367746 |
pentagastrin |
|
FDA approved |
FDA approved |
| 369100 |
Imiquimod |
AM|TLR7|ImmuneResMod |
FDA approved |
FDA approved |
| 407305 |
aloin |
|
FDA approved |
FDA approved |
| 409962 |
Carmustine |
A7|AlkAg |
FDA approved |
FDA approved |
| 526598 |
Mithramycin |
Db|Rs |
FDA approved |
FDA approved |
| 527017 |
Amphotericin B |
|
FDA approved |
FDA approved |
| 602670 |
timazid |
|
FDA approved |
FDA approved |
| 606170 |
Zalcitabine |
Ds |
FDA approved |
FDA approved |
| 606698 |
Rapamycin |
PK:STK,MTOR |
FDA approved |
FDA approved |
| 606869 |
Clofarabine |
Ds |
FDA approved |
FDA approved |
| 608000 |
Tamibarotene |
RXR |
FDA approved |
FDA approved |
| 608210 |
Vinorelbine |
TUBB|Tu-frag |
FDA approved |
FDA approved |
| 609699 |
Topotecan |
TOP1 |
FDA approved |
FDA approved |
| 612049 |
Didanosine |
|
FDA approved |
FDA approved |
| 613327 |
Gemcitabine |
Ds |
FDA approved |
FDA approved |
| 613680 |
Toremifene |
Ho |
FDA approved |
FDA approved |
| 614826 |
bisacodyl, active ingredient of viraplex |
NonCan:Cath |
FDA approved |
FDA approved |
| 615296 |
Haloperidol |
|
FDA approved |
FDA approved |
| 616348 |
Irinotecan |
TOP1 |
FDA approved |
FDA approved |
| 620107 |
pentamidine isethionate |
|
FDA approved |
FDA approved |
| 628503 |
Docetaxel |
TUBB|Tu-stab |
FDA approved |
FDA approved |
| 630176 |
Depsipeptide |
HDAC |
FDA approved |
FDA approved |
| 632307 |
Cetuximab |
Ab |
FDA approved |
FDA approved |
| 633770 |
Brivudine |
|
FDA approved |
FDA approved |
| 633781 |
Lovastatin |
|
FDA approved |
FDA approved |
| 633782 |
Simvastatin |
AM|NonCan:Chol |
FDA approved |
FDA approved |
| 639186 |
Raltitrexed |
Ds|DHFR|TYMS |
FDA approved |
FDA approved |
| 641530 |
Nevirapine |
|
FDA approved |
FDA approved |
| 648766 |
Trabectedin |
A2 |
FDA approved |
FDA approved |
| 652104 |
mifepristone |
|
FDA approved |
FDA approved |
| 656576 |
Midostaurin |
PK:PRKCA,STK,FLT3 |
FDA approved |
FDA approved |
| 661749 |
bergenin |
|
FDA approved |
FDA approved |
| 664312 |
Rilmenidine |
|
FDA approved |
FDA approved |
| 665970 |
artemether |
NonCan:Mal |
FDA approved |
FDA approved |
| 666076 |
Piroxicam |
PTGS2 |
FDA approved |
FDA approved |
| 673596 |
7-Ethyl-10-hydroxycamptothecin |
TOP1 |
FDA approved |
FDA approved |
| 676879 |
Phenothiazine, 2-azido-10-[4-(4-methyl-1-piperazinyl)butyl]-, difumarate |
NonCan:Psy |
FDA approved |
FDA approved |
| 677411 |
Leflunomide |
PK:JAK1,JAK2 |
FDA approved |
FDA approved |
| 681239 |
Bortezomib |
PSM |
FDA approved |
FDA approved |
| 683863 |
Irofulven |
Apo|AlkAg|RDI |
FDA approved |
FDA approved |
| 683864 |
Temsirolimus |
PK:STK,MTOR |
FDA approved |
FDA approved |
| 685524 |
CYTISINE |
|
FDA approved |
FDA approved |
| 685701 |
Flurbiprofen |
|
FDA approved |
FDA approved |
| 686673 |
Nelarabine |
Ds |
FDA approved |
FDA approved |
| 688097 |
Trastuzumab |
Ab |
FDA approved |
FDA approved |
| 693184 |
norvir |
|
FDA approved |
FDA approved |
| 697855 |
Nitazoxanide |
|
FDA approved |
FDA approved |
| 697979 |
Denileukin Diftitox Ontak |
IL |
FDA approved |
FDA approved |
| 698037 |
Pemetrexed |
Df|AM|GARTF|DHFR|TYMS |
FDA approved |
FDA approved |
| 701852 |
Vorinostat |
HDAC |
FDA approved |
FDA approved |
| 702294 |
Estramustine |
A7|TUBB|AlkAg |
FDA approved |
FDA approved |
| 706363 |
Arsenic trioxide |
Apo |
FDA approved |
FDA approved |
| 707389 |
Eribulin mesilate |
TUBB |
FDA approved |
FDA approved |
| 712571 |
artesunate |
|
FDA approved |
FDA approved |
| 712807 |
Capecitabine |
Ds|TYMS |
FDA approved |
FDA approved |
| 713563 |
Exemestane |
Ho|CYP19A1 |
FDA approved |
FDA approved |
| 715055 |
Gefitinib |
PK:YK,EGFR |
FDA approved |
FDA approved |
| 718781 |
Erlotinib |
PK:YK,EGFR |
FDA approved |
FDA approved |
| 719276 |
Fulvestrant |
AM|Ho|ESR|SERM |
FDA approved |
FDA approved |
| 719344 |
Anastrozole |
Ho|CYP19A1 |
FDA approved |
FDA approved |
| 719345 |
Letrozole |
Ho|CYP19A1 |
FDA approved |
FDA approved |
| 719627 |
Celecoxib |
AM|PTGS2|COX2|NonCan:NSAID |
FDA approved |
FDA approved |
| 721075 |
claritin |
|
FDA approved |
FDA approved |
| 721517 |
Zoledronate |
AM|NonCan:Anti-bone resorp |
FDA approved |
FDA approved |
| 722664 |
Nelfinavir |
PSM |
FDA approved |
FDA approved |
| 724772 |
Sorafenib |
PK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase |
FDA approved |
FDA approved |
| 726630 |
Belinostat |
HDAC |
FDA approved |
FDA approved |
| 727071 |
Ofloxacin |
|
FDA approved |
FDA approved |
| 727989 |
Lapatinib |
PK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR |
FDA approved |
FDA approved |
| 728073 |
Irinotecan |
TOP1 |
FDA approved |
FDA approved |
| 732517 |
Dasatinib |
BCR-ABL|PK:YK,PDGFR,KIT |
FDA approved |
FDA approved |
| 733504 |
Everolimus |
PK:STK,MTOR |
FDA approved |
FDA approved |
| 737754 |
Pazopanib |
PK:YK,PDGFR,FGFR,KIT,VEGFR |
FDA approved |
FDA approved |
| 741078 |
Selumetinib |
PK:STK,YK,MAP2K,MAP2K1,MAP2K2 |
FDA approved |
FDA approved |
| 741485 |
Finasteride |
AR |
FDA approved |
FDA approved |
| 743414 |
Imatinib |
BCR-ABL|PK:YK |
FDA approved |
FDA approved |
| 744009 |
Sildenafil |
|
FDA approved |
FDA approved |
| 745750 |
Lapatinib |
PK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR |
FDA approved |
FDA approved |
| 746847 |
Leuprolide |
Ho |
FDA approved |
FDA approved |
| 747167 |
Nelfinavir |
PSM |
FDA approved |
FDA approved |
| 747599 |
Nilotinib |
BCR-ABL|PK:YK |
FDA approved |
FDA approved |
| 747856 |
Olaparib |
PARP|PARP1 |
FDA approved |
FDA approved |
| 747971 |
Sorafenib |
PK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase |
FDA approved |
FDA approved |
| 747972 |
Lenalidomide |
FT|Immunomodulatory |
FDA approved |
FDA approved |
| 747973 |
Ixabepilone |
TUBB|Tu-stab |
FDA approved |
FDA approved |
| 747974 |
Raloxifene |
Ho|SERM |
FDA approved |
FDA approved |
| 749226 |
Abiraterone |
Ho|CYP17A1 |
FDA approved |
FDA approved |
| 749227 |
Abiraterone |
Ho|CYP17A1 |
FDA approved |
FDA approved |
| 750690 |
Sunitinib |
PK:YK,PDGFR,KIT,VEGFR,Multikinase |
FDA approved |
FDA approved |
| 750691 |
Afatinib |
PK:YK,EGFR |
FDA approved |
FDA approved |
| 751548 |
Salinomycin |
Apo|Ab|CD133 |
FDA approved |
FDA approved |
| 752782 |
Pazopanib |
PK:YK,PDGFR,FGFR,KIT,VEGFR |
FDA approved |
FDA approved |
| 753686 |
Olaparib |
PARP|PARP1 |
FDA approved |
FDA approved |
| 754143 |
Depsipeptide |
HDAC |
FDA approved |
FDA approved |
| 754230 |
Pralatrexate |
Df|CTNNB1|DHFR |
FDA approved |
FDA approved |
| 754355 |
Niraparib |
PARP|PARP1|PARP2 |
FDA approved |
FDA approved |
| 754363 |
Plerixafor |
CXCR4 |
FDA approved |
FDA approved |
| 754771 |
Itraconazole |
AM|NonCan:Ant |
FDA approved |
FDA approved |
| 755384 |
Pemetrexed |
Df|AM|GARTF|DHFR|TYMS |
FDA approved |
FDA approved |
| 755389 |
Bosutinib |
STAT|BCR-ABL|STAT5A/B|PK:YK,LYN,SRC,HCK |
FDA approved |
FDA approved |
| 755400 |
Masitinib |
PK:YK,PDGFR,FGFR,KIT,FGFR3 |
FDA approved |
FDA approved |
| 755401 |
Golotimod |
STAT|STAT3 |
FDA approved |
FDA approved |
| 755404 |
Flurbiprofen |
|
FDA approved |
FDA approved |
| 755605 |
Enzalutamide |
Ho|AR |
FDA approved |
FDA approved |
| 755606 |
Cediranib |
PK:YK,VEGF,VEGFR,KDR |
FDA approved |
FDA approved |
| 755764 |
Fluphenazine |
NonCan:Psy |
FDA approved |
FDA approved |
| 755767 |
Tacrolimus |
PK:MTOR |
FDA approved |
FDA approved |
| 755768 |
Fluphenazine |
NonCan:Psy |
FDA approved |
FDA approved |
| 755809 |
Vismodegib |
SMO|PK:YK |
FDA approved |
FDA approved |
| 755841 |
Actinomycin D |
Db|RNA polymerase I |
FDA approved |
FDA approved |
| 755843 |
ivermectin (usan) |
|
FDA approved |
FDA approved |
| 755871 |
Amphotericin B |
|
FDA approved |
FDA approved |
| 755880 |
Mitomycin |
A2|AlkAg |
FDA approved |
FDA approved |
| 755980 |
Lenvatinib |
PK:YK,PDGFR,FGFR,VEGFR,KDR,RET |
FDA approved |
FDA approved |
| 755984 |
Pralatrexate |
Df|CTNNB1|DHFR |
FDA approved |
FDA approved |
| 755985 |
Nelarabine |
Ds |
FDA approved |
FDA approved |
| 755986 |
Vismodegib |
SMO|PK:YK |
FDA approved |
FDA approved |
| 756643 |
KX-01 |
PK:YK,SRC |
FDA approved |
FDA approved |
| 756644 |
Rucaparib |
PARP|PARP1 |
FDA approved |
FDA approved |
| 756645 |
Crizotinib |
PK:YK,MET,ALK |
FDA approved |
FDA approved |
| 756647 |
Quizartinib |
PK:YK,PDGFR,FLT,KIT,FLT3 |
FDA approved |
FDA approved |
| 756655 |
Bortezomib |
PSM |
FDA approved |
FDA approved |
| 756656 |
MK-2206 |
PK:STK,AKT,AKT1,AKT2,AKT3 |
FDA approved |
FDA approved |
| 756659 |
Intedanib |
PK:YK,PDGFR,FGFR,VEGFR,FLT3 |
FDA approved |
FDA approved |
| 756661 |
Chlorpromazine |
NonCan:Psy |
FDA approved |
FDA approved |
| 756685 |
clemastine (usan) |
|
FDA approved |
FDA approved |
| 756689 |
Chlorpromazine |
NonCan:Psy |
FDA approved |
FDA approved |
| 756700 |
Clotrimazole |
|
FDA approved |
FDA approved |
| 756702 |
Colchicine |
TUBB |
FDA approved |
FDA approved |
| 756714 |
Cytarabine |
Ds |
FDA approved |
FDA approved |
| 756717 |
Daunorubicin |
TOP2 |
FDA approved |
FDA approved |
| 756734 |
dienestrol (usan) |
|
FDA approved |
FDA approved |
| 756738 |
Digoxin |
NonCan:CardG |
FDA approved |
FDA approved |
| 757027 |
Ethinyl estradiol |
Ho |
FDA approved |
FDA approved |
| 757036 |
Fluorouracil |
Ds|Rs|TYMS |
FDA approved |
FDA approved |
| 757050 |
badil |
|
FDA approved |
FDA approved |
| 757087 |
Nitrogen mustard |
A7|AlkAg |
FDA approved |
FDA approved |
| 757098 |
Melphalan |
A7|AlkAg |
FDA approved |
FDA approved |
| 757119 |
florid |
|
FDA approved |
FDA approved |
| 757120 |
Minocycline Hydrochloride |
|
FDA approved |
FDA approved |
| 757306 |
malacid |
DHFR |
FDA approved |
FDA approved |
| 757307 |
Acrichine |
Db|AP |
FDA approved |
FDA approved |
| 757345 |
Tamoxifen |
Ho|SERM |
FDA approved |
FDA approved |
| 757348 |
6-Thioguanine |
Ds|IMPDH2|IMPDH |
FDA approved |
FDA approved |
| 757349 |
metlaril |
|
FDA approved |
FDA approved |
| 757350 |
navan |
|
FDA approved |
FDA approved |
| 757363 |
Tyrothricin |
NonCan:Ant |
FDA approved |
FDA approved |
| 757369 |
Eskazine |
|
FDA approved |
FDA approved |
| 757384 |
Vinblastine |
TUBB|Tu-frag |
FDA approved |
FDA approved |
| 757400 |
pentamidine isethionate |
|
FDA approved |
FDA approved |
| 757424 |
melbex |
|
FDA approved |
FDA approved |
| 757425 |
ouabain |
|
FDA approved |
FDA approved |
| 757436 |
Cabozantinib |
PK:YK,MET,AXL,KIT,VEGFR,FLT3,RET |
FDA approved |
FDA approved |
| 757437 |
Salinomycin |
Apo|Ab|CD133 |
FDA approved |
FDA approved |
| 757439 |
Neratinib |
PK:YK,EGFR,ERBB2 |
FDA approved |
FDA approved |
| 757441 |
Axitinib |
PK:YK,PDGFR,VEGFR |
FDA approved |
FDA approved |
| 757442 |
Intedanib |
PK:YK,PDGFR,FGFR,VEGFR,FLT3 |
FDA approved |
FDA approved |
| 757443 |
Finasteride |
AR |
FDA approved |
FDA approved |
| 757804 |
Etoposide |
TOP2 |
FDA approved |
FDA approved |
| 757816 |
Fluphenazine |
NonCan:Psy |
FDA approved |
FDA approved |
| 757838 |
Mebendazole |
Tu-stab |
FDA approved |
FDA approved |
| 757849 |
sulconazole nitrate (usan) |
|
FDA approved |
FDA approved |
| 757854 |
Pimozide |
NonCan:Psy |
FDA approved |
FDA approved |
| 757882 |
Econazole Nitrate |
|
FDA approved |
FDA approved |
| 758007 |
Tivozanib |
PK:YK,MET,PDGFR,FGFR,KIT,VEGFR,FLT3,KDR |
FDA approved |
FDA approved |
| 758183 |
monensin sodium |
|
FDA approved |
FDA approved |
| 758186 |
Azacitidine |
DNMT |
FDA approved |
FDA approved |
| 758194 |
ciclosporin |
|
FDA approved |
FDA approved |
| 758230 |
Floxuridine |
Ds|TYMS |
FDA approved |
FDA approved |
| 758233 |
mefloquine (usan) |
|
FDA approved |
FDA approved |
| 758244 |
tepotinib |
PK:YK,MET |
FDA approved |
FDA approved |
| 758246 |
Trametinib |
PK:STK,MAP2K,MAP2K1,MAP2K2 |
FDA approved |
FDA approved |
| 758247 |
Palbociclib |
PK:STK,CDK,CDK4,CDK6 |
FDA approved |
FDA approved |
| 758252 |
Carfilzomib |
PSM |
FDA approved |
FDA approved |
| 758253 |
Homoharringtonine |
Apo|Ang|Pi |
FDA approved |
FDA approved |
| 758254 |
Ixazomib citrate |
PSM |
FDA approved |
FDA approved |
| 758255 |
Teniposide |
TOP2 |
FDA approved |
FDA approved |
| 758387 |
Triflupromazine Hydrochloride |
|
FDA approved |
FDA approved |
| 758390 |
bepridil hydrochloride (usan) |
|
FDA approved |
FDA approved |
| 758423 |
M-AMSA |
TOP2 |
FDA approved |
FDA approved |
| 758487 |
Ponatinib |
BCR-ABL|PK:YK |
FDA approved |
FDA approved |
| 758612 |
Bleomycin |
Db |
FDA approved |
FDA approved |
| 758645 |
Paclitaxel |
TUBB|Tu-stab |
FDA approved |
FDA approved |
| 758654 |
paroxetine hydrochloride (usan) |
|
FDA approved |
FDA approved |
| 758662 |
Lovastatin |
|
FDA approved |
FDA approved |
| 758664 |
Rapamycin |
PK:STK,MTOR |
FDA approved |
FDA approved |
| 758667 |
Teniposide |
TOP2 |
FDA approved |
FDA approved |
| 758671 |
Ancitabine hydrochloride |
Ds |
FDA approved |
FDA approved |
| 758682 |
artenimol |
|
FDA approved |
FDA approved |
| 758691 |
acrisorcin (usan) |
|
FDA approved |
FDA approved |
| 758706 |
Simvastatin |
AM|NonCan:Chol |
FDA approved |
FDA approved |
| 758774 |
Belinostat |
HDAC |
FDA approved |
FDA approved |
| 758896 |
fluvastatin |
|
FDA approved |
FDA approved |
| 758958 |
oxiconazole nitrate (usan) |
|
FDA approved |
FDA approved |
| 759106 |
nisoldipine (usan) |
|
FDA approved |
FDA approved |
| 759135 |
Methylene Blue |
|
FDA approved |
FDA approved |
| 759151 |
triclosan (usan) |
|
FDA approved |
FDA approved |
| 759155 |
Doxorubicin |
TOP2 |
FDA approved |
FDA approved |
| 759169 |
Tioconazole |
|
FDA approved |
FDA approved |
| 759174 |
Vincristine |
TUBB|Tu-frag |
FDA approved |
FDA approved |
| 759178 |
Pipamperone |
NonCan:Psy |
FDA approved |
FDA approved |
| 759195 |
Epirubicin |
TOP2 |
FDA approved |
FDA approved |
| 759224 |
Idelalisib |
PK:PIK3 |
FDA approved |
FDA approved |
| 759228 |
Idebenone |
|
FDA approved |
FDA approved |
| 759263 |
Topotecan |
TOP1 |
FDA approved |
FDA approved |
| 759274 |
Arsenic trioxide |
Apo |
FDA approved |
FDA approved |
| 759323 |
anafranil |
|
FDA approved |
FDA approved |
| 759559 |
amoxapine (usan) |
|
FDA approved |
FDA approved |
| 759560 |
Amiodarone Hydrochloride |
|
FDA approved |
FDA approved |
| 759614 |
6-Mercaptopurine |
Ds|PPAT |
FDA approved |
FDA approved |
| 759811 |
telmisartan (usan) |
|
FDA approved |
FDA approved |
| 759817 |
artesunate |
|
FDA approved |
FDA approved |
| 759850 |
Docetaxel |
TUBB|Tu-stab |
FDA approved |
FDA approved |
| 759852 |
Vorinostat |
HDAC |
FDA approved |
FDA approved |
| 759856 |
Gefitinib |
PK:YK,EGFR |
FDA approved |
FDA approved |
| 759857 |
Clofarabine |
Ds |
FDA approved |
FDA approved |
| 759877 |
Dasatinib |
BCR-ABL|PK:YK,PDGFR,KIT |
FDA approved |
FDA approved |
| 759878 |
Irinotecan |
TOP1 |
FDA approved |
FDA approved |
| 760057 |
Nitazoxanide |
|
FDA approved |
FDA approved |
| 760087 |
Vinorelbine |
TUBB|Tu-frag |
FDA approved |
FDA approved |
| 760424 |
moxidectin (usan) |
|
FDA approved |
FDA approved |
| 760443 |
Copanlisib |
PK:PIK3 |
FDA approved |
FDA approved |
| 760764 |
Voreloxin |
TOP2 |
FDA approved |
FDA approved |
| 760766 |
Vandetanib |
PK:STK,YK,PDGFR,EGFR,VEGFR,RET |
FDA approved |
FDA approved |
| 761068 |
Cabozantinib |
PK:YK,MET,AXL,KIT,VEGFR,FLT3,RET |
FDA approved |
FDA approved |
| 761190 |
Panobinostat |
HDAC |
FDA approved |
FDA approved |
| 761191 |
brigatinib |
PK:YK,IGF1R,ALK,EGFR |
FDA approved |
FDA approved |
| 761385 |
Sonidegib |
SMO|Hg-Smo |
FDA approved |
FDA approved |
| 761386 |
Sonidegib |
SMO|Hg-Smo |
FDA approved |
FDA approved |
| 761388 |
Plerixafor |
CXCR4 |
FDA approved |
FDA approved |
| 761389 |
Raloxifene |
Ho|SERM |
FDA approved |
FDA approved |
| 761431 |
Vemurafenib |
PK:YK,BRAF |
FDA approved |
FDA approved |
| 761432 |
Cabazitaxel |
TUBB|Tu-stab |
FDA approved |
FDA approved |
| 761910 |
Ibrutinib |
PK:YK,BTK |
FDA approved |
FDA approved |
| 762523 |
elvitegravir |
|
FDA approved |
FDA approved |
| 763371 |
Ruxolitinib |
PK:YK,JAK,JAK1,JAK2 |
FDA approved |
FDA approved |
| 763932 |
Regorafenib |
GTPase|PK:STK,YK,PDGFR,FGFR,KIT,MAP2K,RAF,VEGFR,KDR,RET,Multikinase |
FDA approved |
FDA approved |
| 764040 |
Alectinib |
PK:YK,ALK |
FDA approved |
FDA approved |
| 764042 |
ARRY-162 |
PK:STK,MAP2K,MAP2K1,MAP2K2 |
FDA approved |
FDA approved |
| 764134 |
Dabrafenib |
PK:BRAF |
FDA approved |
FDA approved |
| 764487 |
NVP-BGJ398 |
PK:FGFR,FGFR1,FGFR2,FGFR3,FGFR4 |
FDA approved |
FDA approved |
| 764581 |
ARRY-380 |
PK:ERBB2 |
FDA approved |
FDA approved |
| 764778 |
Ivacaftor |
|
FDA approved |
FDA approved |
| 764821 |
Alectinib |
PK:YK,ALK |
FDA approved |
FDA approved |
| 765396 |
BMN-673 |
PARP1|PARP2 |
FDA approved |
FDA approved |
| 765694 |
Bosutinib |
STAT|BCR-ABL|STAT5A/B|PK:YK,LYN,SRC,HCK |
FDA approved |
FDA approved |
| 765888 |
Dacomitinib |
PK:EGFR,ERBB2 |
FDA approved |
FDA approved |
| 765974 |
BYL-719 |
PK:PIK3 |
FDA approved |
FDA approved |
| 766118 |
Teriflunomide |
|
FDA approved |
FDA approved |
| 766270 |
ABT-199 |
BCL2 |
FDA approved |
FDA approved |
| 766907 |
Ixazomib |
PSM |
FDA approved |
FDA approved |
| 767125 |
BMN-673 |
PARP1|PARP2 |
FDA approved |
FDA approved |
| 767600 |
Fedratinib |
PK:FLT,JAK,FLT3,JAK2,RET |
FDA approved |
FDA approved |
| 768068 |
Cobimetinib (isomer 1) |
PK:MAP2K,MAP2K1 |
FDA approved |
FDA approved |
| 768069 |
Cobimetinib (isomer 1) |
PK:MAP2K,MAP2K1 |
FDA approved |
FDA approved |
| 768073 |
LY-2835219 |
PK:PIM1,CDK,CDK4,CDK6 |
FDA approved |
FDA approved |
| 771649 |
ARN-509 |
AR |
FDA approved |
FDA approved |
| 772469 |
IPI-145 |
PK:PIK3 |
FDA approved |
FDA approved |
| 773149 |
nitisinone |
|
FDA approved |
FDA approved |
| 774769 |
NMS-E628 |
PK:ROS1,ALK |
FDA approved |
FDA approved |
| 775351 |
Pomalidomide |
Immunomodulatory |
FDA approved |
FDA approved |
| 775772 |
PF-04449913 |
SMO |
FDA approved |
FDA approved |
| 776422 |
LDK-378 |
PK:ALK |
FDA approved |
FDA approved |
| 777109 |
E-7438 |
EZH2 |
FDA approved |
FDA approved |
| 777193 |
LDK-378 |
PK:ALK |
FDA approved |
FDA approved |
| 777878 |
TABRECTA |
PK:MET |
FDA approved |
FDA approved |
| 778304 |
Encorafenib |
PK:BRAF |
FDA approved |
FDA approved |
| 778590 |
Cobimetinib (isomer 1) |
PK:MAP2K,MAP2K1 |
FDA approved |
FDA approved |
| 778909 |
LEE-011 |
PK:CDK,CDK4,CDK6 |
FDA approved |
FDA approved |
| 779217 |
osimertinib |
PK:EGFR |
FDA approved |
FDA approved |
| 779405 |
CO-1686 |
PK:EGFR |
FDA approved |
FDA approved |
| 780108 |
PF-06463922 |
PK:ROS1,ALK |
FDA approved |
FDA approved |
| 780203 |
selinexor |
XPO1 |
FDA approved |
FDA approved |
| 781556 |
JNJ-42756493 |
PK:FGFR,FGFR1,FGFR2,FGFR3,FGFR4 |
FDA approved |
FDA approved |
| 782351 |
tofacitinib |
PK:JAK,JAK1,JAK3 |
FDA approved |
FDA approved |
| 785497 |
INCB-024360 |
IDO1 |
FDA approved |
FDA approved |
| 785570 |
LOXO-101 |
PK:NTRK |
FDA approved |
FDA approved |
| 787457 |
brigatinib |
PK:YK,IGF1R,ALK,EGFR |
FDA approved |
FDA approved |
| 787846 |
gilteritinib |
PK:AXL,FLT3 |
FDA approved |
FDA approved |
| 788120 |
enasidenib |
IDH1|IDH2 |
FDA approved |
FDA approved |
| 788948 |
Vistonuridine |
TUBB|FU-Antidote |
FDA approved |
FDA approved |
| 789102 |
ivosidenib |
IDH1 |
FDA approved |
FDA approved |
| 789300 |
PLX-3397 |
PK:CSF1R,KIT,FLT3 |
FDA approved |
FDA approved |
| 789925 |
ABL-001 |
BCR-ABL |
FDA approved |
FDA approved |
| 791164 |
acalabrutinib |
PK:BTK |
FDA approved |
FDA approved |
| 792848 |
olmutinib |
PK:EGFR,BTK,JAK3 |
FDA approved |
FDA approved |
| 797937 |
Sulfatinib |
PK:YK,FGFR,KDR |
FDA approved |
FDA approved |
| 799318 |
zanubrutinib |
PK:BTK |
FDA approved |
FDA approved |
| 800405 |
umbralisib |
|
FDA approved |
FDA approved |
| 801082 |
BLU-285 |
|
FDA approved |
FDA approved |
| 809693 |
Copanlisib |
PK:PIK3 |
FDA approved |
FDA approved |
| 811429 |
BLU-667 |
PK:RET |
FDA approved |
FDA approved |
| 813783 |
Trabectedin |
A2 |
FDA approved |
FDA approved |