740 |
METHOTREXATE |
Df|DHFR |
FDA approved |
FDA approved |
750 |
Busulfan |
A7|AlkAg |
FDA approved |
FDA approved |
752 |
6-THIOGUANINE |
Ds|IMPDH2|IMPDH |
FDA approved |
FDA approved |
755 |
6-MERCAPTOPURINE |
Ds|PPAT |
FDA approved |
FDA approved |
762 |
Nitrogen mustard |
A7|AlkAg |
FDA approved |
FDA approved |
1390 |
Allopurinol |
AM|XDH |
FDA approved |
FDA approved |
3053 |
Actinomycin D |
Db |
FDA approved |
FDA approved |
3088 |
Chlorambucil |
A7|AlkAg |
FDA approved |
FDA approved |
3590 |
CALCIUM LEUCOVORIN |
Df |
FDA approved |
FDA approved |
6396 |
Thiotepa |
A7|AlkAg |
FDA approved |
FDA approved |
8806 |
Melphalan |
A7|AlkAg |
FDA approved |
FDA approved |
9706 |
Triethylenemelamine |
A7|AlkAg |
FDA approved |
FDA approved |
10023 |
Prednisone |
Ho |
FDA approved |
FDA approved |
10973 |
Ethinyl estradiol |
Ho |
FDA approved |
FDA approved |
12198 |
Dromostanolone Propionate |
Ho |
FDA approved |
FDA approved |
13875 |
Altretamine |
Db|AlkAg |
FDA approved |
FDA approved |
14229 |
Acrichine |
Db|AP |
FDA approved |
FDA approved |
18509 |
Aminolevulinic acid |
AM |
FDA approved |
FDA approved |
19893 |
Fluorouracil |
Ds|Rs|TYMS |
FDA approved |
FDA approved |
23162 |
Nandrolone phenpropionate |
Ho|NonCan:Ste |
FDA approved |
FDA approved |
23759 |
TESTOLACTONE |
Ho |
FDA approved |
FDA approved |
24559 |
Mithramycin |
Db|Rs |
FDA approved |
FDA approved |
25154 |
Pipobroman |
A7|AlkAg |
FDA approved |
FDA approved |
26271 |
Cyclophosphamide |
A7|AlkAg |
FDA approved |
FDA approved |
26980 |
Mitomycin |
A2 |
FDA approved |
FDA approved |
27640 |
Floxuridine |
Ds|TYMS |
FDA approved |
FDA approved |
32065 |
Hydroxyurea |
AM|Dr |
FDA approved |
FDA approved |
34462 |
Uracil mustard |
A7|AlkAg |
FDA approved |
FDA approved |
34521 |
Dexamethasone Decadron |
Ho |
FDA approved |
FDA approved |
38721 |
Mitotane |
A7|Ho|AlkAg|anti-Ho|CYP11A1 |
FDA approved |
FDA approved |
45388 |
DACARBAZINE |
A7|AlkAg |
FDA approved |
FDA approved |
45923 |
Methoxsalen |
Db |
FDA approved |
FDA approved |
49842 |
Vinblastine |
TUBB|Tu-frag |
FDA approved |
FDA approved |
59687 |
Acetalax |
NonCan:Cath |
FDA approved |
FDA approved |
63878 |
Cytarabine |
Ds |
FDA approved |
FDA approved |
66847 |
Thalidomide |
Ang|Immunomodulatory |
FDA approved |
FDA approved |
67574 |
Vincristine |
TUBB|Tu-frag |
FDA approved |
FDA approved |
71423 |
Megestrol acetate |
Ho|PGR |
FDA approved |
FDA approved |
75520 |
tfdu |
TYMS |
FDA approved |
FDA approved |
77213 |
Procarbazine |
A7|AlkAg |
FDA approved |
FDA approved |
79037 |
Lomustine |
A6|AlkAg |
FDA approved |
FDA approved |
79269 |
Vistonuridine |
TUBB|FU-Antidote |
FDA approved |
FDA approved |
82151 |
Daunorubicin |
TOP2 |
FDA approved |
FDA approved |
83142 |
Daunorubicin |
TOP2 |
FDA approved |
FDA approved |
85998 |
STREPTOZOCIN |
A7|AlkAg |
FDA approved |
FDA approved |
88536 |
Calusterone |
Ho |
FDA approved |
FDA approved |
89201 |
Estramustine |
A7|TUBB|AlkAg |
FDA approved |
FDA approved |
90636 |
Vinblastine |
TUBB|Tu-frag |
FDA approved |
FDA approved |
92339 |
Fluphenazine |
NonCan:Psy |
FDA approved |
FDA approved |
92859 |
Arsenic trioxide |
Apo |
FDA approved |
FDA approved |
95100 |
Digoxin |
NonCan:CardG |
FDA approved |
FDA approved |
102816 |
AZACITIDINE |
DNMT |
FDA approved |
FDA approved |
105014 |
Cladribine |
Ds|ADA |
FDA approved |
FDA approved |
105024 |
Mithramycin |
Db|Rs |
FDA approved |
FDA approved |
109229 |
Asparaginase |
AM|Pi |
FDA approved |
FDA approved |
109724 |
Ifosfamide |
A7|AlkAg |
FDA approved |
FDA approved |
109929 |
Asparaginase |
AM|Pi |
FDA approved |
FDA approved |
113891 |
Mesna |
|
FDA approved |
FDA approved |
117186 |
Acetalax |
NonCan:Cath |
FDA approved |
FDA approved |
118218 |
Fludarabine |
Ds|AM|Dr|STAT1 |
FDA approved |
FDA approved |
119875 |
Cisplatin |
A7|AlkAg |
FDA approved |
FDA approved |
122758 |
Isotretinoin |
Ho|RXR|Differentiator |
FDA approved |
FDA approved |
122819 |
Teniposide |
TOP2 |
FDA approved |
FDA approved |
123127 |
Doxorubicin |
TOP2 |
FDA approved |
FDA approved |
124463 |
Fludarabine |
Ds|AM|Dr|STAT1 |
FDA approved |
FDA approved |
125066 |
Bleomycin |
Db |
FDA approved |
FDA approved |
125973 |
Paclitaxel |
TUBB|Tu-stab |
FDA approved |
FDA approved |
127716 |
DECITABINE |
AM|DNMT |
FDA approved |
FDA approved |
134727 |
Mitomycin |
A2 |
FDA approved |
FDA approved |
138783 |
Bendamustine |
A2|A6|AlkAg |
FDA approved |
FDA approved |
141540 |
Etoposide |
TOP2 |
FDA approved |
FDA approved |
141633 |
Homoharringtonine |
Apo|Ang|Pi |
FDA approved |
FDA approved |
143020 |
Mithramycin |
Db|Rs |
FDA approved |
FDA approved |
148958 |
Tegafur |
Df |
FDA approved |
FDA approved |
157035 |
Parthenolide |
Apo |
FDA approved |
FDA approved |
169780 |
Dexrazoxane |
TOP2|NonCan:Cardioprotective |
FDA approved |
FDA approved |
177023 |
Levamisole hydrochloride |
|
FDA approved |
FDA approved |
180973 |
Tamoxifen |
Ho|SERM |
FDA approved |
FDA approved |
218321 |
PENTOSTATIN |
Ds|AM|ADA |
FDA approved |
FDA approved |
226080 |
RAPAMYCIN |
PK:STK,MTOR |
FDA approved |
FDA approved |
241240 |
Carboplatin |
A7|AlkAg |
FDA approved |
FDA approved |
246131 |
Valrubicin |
TOP2 |
FDA approved |
FDA approved |
256439 |
Idarubicin |
TOP2 |
FDA approved |
FDA approved |
256942 |
Epirubicin |
TOP2 |
FDA approved |
FDA approved |
266046 |
Oxaliplatin |
A7|AlkAg |
FDA approved |
FDA approved |
279836 |
MITOXANTRONE |
TOP2 |
FDA approved |
FDA approved |
287459 |
Cytarabine |
Ds |
FDA approved |
FDA approved |
296961 |
Amifostine |
RP |
FDA approved |
FDA approved |
301739 |
Mitoxantrone |
TOP2 |
FDA approved |
FDA approved |
312887 |
Fludarabine |
Ds|AM|Dr|STAT1 |
FDA approved |
FDA approved |
362856 |
Temozolomide |
A7|AlkAg |
FDA approved |
FDA approved |
369100 |
Imiquimod |
AM|TLR7|ImmuneResMod |
FDA approved |
FDA approved |
409962 |
Carmustine |
A7|AlkAg |
FDA approved |
FDA approved |
526598 |
Mithramycin |
Db|Rs |
FDA approved |
FDA approved |
606698 |
Rapamycin |
PK:STK,MTOR |
FDA approved |
FDA approved |
606869 |
Clofarabine |
Ds |
FDA approved |
FDA approved |
608000 |
Tamibarotene |
RXR |
FDA approved |
FDA approved |
608210 |
Vinorelbine |
TUBB|Tu-frag |
FDA approved |
FDA approved |
609699 |
Topotecan |
TOP1 |
FDA approved |
FDA approved |
613327 |
Gemcitabine |
Ds |
FDA approved |
FDA approved |
613680 |
Toremifene |
Ho |
FDA approved |
FDA approved |
614826 |
Bisacodyl, active ingredient of Viraplex |
NonCan:Cath |
FDA approved |
FDA approved |
616348 |
Irinotecan |
TOP1 |
FDA approved |
FDA approved |
628503 |
Docetaxel |
TUBB|Tu-stab |
FDA approved |
FDA approved |
630176 |
Depsipeptide |
HDAC |
FDA approved |
FDA approved |
632307 |
Cetuximab |
Ab |
FDA approved |
FDA approved |
633782 |
Simvastatin |
AM|NonCan:Chol |
FDA approved |
FDA approved |
639186 |
Raltitrexed |
Ds|DHFR|TYMS |
FDA approved |
FDA approved |
648766 |
Trabectedin |
A2 |
FDA approved |
FDA approved |
656576 |
Midostaurin |
PK:PRKCA,STK |
FDA approved |
FDA approved |
673596 |
7-Ethyl-10-hydroxycamptothecin |
TOP1 |
FDA approved |
FDA approved |
676879 |
Phenothiazine, 2-azido-10-[4-(4-methyl-1-piperazinyl)butyl]-, difumarate |
NonCan:Psy |
FDA approved |
FDA approved |
681239 |
Bortezomib |
PSM |
FDA approved |
FDA approved |
683863 |
Irofulven |
Apo|AlkAg|RDI |
FDA approved |
FDA approved |
683864 |
Temsirolimus |
PK:STK,MTOR |
FDA approved |
FDA approved |
685701 |
Flurbiprofen |
|
FDA approved |
FDA approved |
686673 |
Nelarabine |
Ds |
FDA approved |
FDA approved |
688097 |
Trastuzumab |
Ab |
FDA approved |
FDA approved |
697979 |
Denileukin Diftitox Ontak |
IL |
FDA approved |
FDA approved |
698037 |
Pemetrexed |
Df|AM|GARTF|DHFR |
FDA approved |
FDA approved |
701852 |
Vorinostat |
HDAC |
FDA approved |
FDA approved |
702294 |
Estramustine |
A7|TUBB|AlkAg |
FDA approved |
FDA approved |
706363 |
Arsenic trioxide |
Apo |
FDA approved |
FDA approved |
707389 |
Eribulin mesilate |
TUBB |
FDA approved |
FDA approved |
712807 |
Capecitabine |
Ds|TYMS |
FDA approved |
FDA approved |
713563 |
Exemestane |
Ho|CYP19A1 |
FDA approved |
FDA approved |
715055 |
Gefitinib |
PK:YK,EGFR |
FDA approved |
FDA approved |
718781 |
Erlotinib |
PK:YK,EGFR |
FDA approved |
FDA approved |
719276 |
Fulvestrant |
AM|Ho|ESR|SERM |
FDA approved |
FDA approved |
719344 |
Anastrozole |
Ho|CYP19A1 |
FDA approved |
FDA approved |
719345 |
Letrozole |
Ho|CYP19A1 |
FDA approved |
FDA approved |
719627 |
Celecoxib |
AM|PTGS2|COX2|NonCan:NSAID |
FDA approved |
FDA approved |
721517 |
Zoledronate |
AM|NonCan:Anti-bone resorp |
FDA approved |
FDA approved |
722664 |
Nelfinavir |
PSM |
FDA approved |
FDA approved |
724772 |
Sorafenib |
PK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase |
FDA approved |
FDA approved |
726630 |
Belinostat |
HDAC |
FDA approved |
FDA approved |
727989 |
Lapatinib |
PK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR |
FDA approved |
FDA approved |
728073 |
Irinotecan |
TOP1 |
FDA approved |
FDA approved |
732517 |
Dasatinib |
BCR-ABL|PK:YK,PDGFR,KIT |
FDA approved |
FDA approved |
733504 |
Everolimus |
PK:STK,MTOR |
FDA approved |
FDA approved |
737754 |
Pazopanib |
PK:YK,PDGFR,FGFR,KIT,VEGFR |
FDA approved |
FDA approved |
741078 |
Selumetinib |
PK:STK,YK,MAP2K,MAP2K1,MAP2K2 |
FDA approved |
FDA approved |
741485 |
Finasteride |
|
FDA approved |
FDA approved |
743414 |
Imatinib |
BCR-ABL|PK:YK |
FDA approved |
FDA approved |
744009 |
Sildenafil |
|
FDA approved |
FDA approved |
745750 |
Lapatinib |
PK:STK,YK,MET,EGFR,ERBB2,KIT,RAF,VEGFR |
FDA approved |
FDA approved |
746847 |
Leuprolide |
Ho |
FDA approved |
FDA approved |
747167 |
Nelfinavir |
PSM |
FDA approved |
FDA approved |
747599 |
Nilotinib |
BCR-ABL|PK:YK |
FDA approved |
FDA approved |
747856 |
Olaparib |
PARP|PARP1 |
FDA approved |
FDA approved |
747971 |
Sorafenib |
PK:YK,PDGFR,BRAF,KIT,VEGFR,Multikinase |
FDA approved |
FDA approved |
747972 |
Lenalidomide |
FT|Immunomodulatory |
FDA approved |
FDA approved |
747973 |
Ixabepilone |
TUBB|Tu-stab |
FDA approved |
FDA approved |
747974 |
Raloxifene |
Ho|SERM |
FDA approved |
FDA approved |
749226 |
Abiraterone |
Ho|CYP17A1 |
FDA approved |
FDA approved |
749227 |
Abiraterone |
Ho|CYP17A1 |
FDA approved |
FDA approved |
750690 |
Sunitinib |
PK:YK,PDGFR,KIT,VEGFR,Multikinase |
FDA approved |
FDA approved |
750691 |
Afatinib |
PK:YK,EGFR |
FDA approved |
FDA approved |
752782 |
Pazopanib |
PK:YK,PDGFR,FGFR,KIT,VEGFR |
FDA approved |
FDA approved |
753686 |
Olaparib |
PARP|PARP1 |
FDA approved |
FDA approved |
754143 |
Depsipeptide |
HDAC |
FDA approved |
FDA approved |
754230 |
pralatrexate |
Df|CTNNB1|DHFR |
FDA approved |
FDA approved |
754355 |
Niraparib |
PARP|PARP1 |
FDA approved |
FDA approved |
754363 |
Plerixafor |
CXCR4 |
FDA approved |
FDA approved |
755384 |
Pemetrexed |
Df|AM|GARTF|DHFR |
FDA approved |
FDA approved |
755389 |
Bosutinib |
STAT|BCR-ABL|STAT5A/B|PK:YK,LYN,SRC,HCK |
FDA approved |
FDA approved |
755401 |
Golotimod |
STAT|STAT3 |
FDA approved |
FDA approved |
755404 |
Flurbiprofen |
|
FDA approved |
FDA approved |
755605 |
Enzalutamide |
Ho|AR |
FDA approved |
FDA approved |
755764 |
Fluphenazine |
NonCan:Psy |
FDA approved |
FDA approved |
755767 |
Tacrolimus |
|
FDA approved |
FDA approved |
755768 |
Fluphenazine |
NonCan:Psy |
FDA approved |
FDA approved |
755809 |
Vismodegib |
SMO|PK:YK |
FDA approved |
FDA approved |
755841 |
Actinomycin D |
Db |
FDA approved |
FDA approved |
755880 |
Mitomycin |
A2 |
FDA approved |
FDA approved |
755980 |
Lenvatinib |
PK:YK,PDGFR,FGFR,VEGFR,RET |
FDA approved |
FDA approved |
755984 |
Pralatrexate |
Df|CTNNB1|DHFR |
FDA approved |
FDA approved |
755985 |
Nelarabine |
Ds |
FDA approved |
FDA approved |
755986 |
Vismodegib |
SMO|PK:YK |
FDA approved |
FDA approved |
756644 |
Rucaparib |
PARP|PARP1 |
FDA approved |
FDA approved |
756645 |
Crizotinib |
PK:YK,MET,ALK |
FDA approved |
FDA approved |
756655 |
Bortezomib |
PSM |
FDA approved |
FDA approved |
756661 |
Chlorpromazine |
NonCan:Psy |
FDA approved |
FDA approved |
756689 |
Chlorpromazine |
NonCan:Psy |
FDA approved |
FDA approved |
756714 |
Cytarabine |
Ds |
FDA approved |
FDA approved |
756717 |
DAUNORUBICIN |
TOP2 |
FDA approved |
FDA approved |
756738 |
DIGOXIN |
NonCan:CardG |
FDA approved |
FDA approved |
757027 |
ETHINYL ESTRADIOL |
Ho |
FDA approved |
FDA approved |
757036 |
Fluorouracil |
Ds|Rs|TYMS |
FDA approved |
FDA approved |
757087 |
Nitrogen mustard |
A7|AlkAg |
FDA approved |
FDA approved |
757098 |
Melphalan |
A7|AlkAg |
FDA approved |
FDA approved |
757307 |
Acrichine |
Db|AP |
FDA approved |
FDA approved |
757345 |
Tamoxifen |
Ho|SERM |
FDA approved |
FDA approved |
757348 |
6-Thioguanine |
Ds|IMPDH2|IMPDH |
FDA approved |
FDA approved |
757363 |
TYROTHRICIN |
NonCan:Ant |
FDA approved |
FDA approved |
757384 |
Vinblastine |
TUBB|Tu-frag |
FDA approved |
FDA approved |
757436 |
Cabozantinib |
PK:YK,MET,AXL,KIT,VEGFR,FLT3,RET |
FDA approved |
FDA approved |
757439 |
Neratinib |
PK:YK,EGFR,ERBB2 |
FDA approved |
FDA approved |
757441 |
Axitinib |
PK:YK,PDGFR,VEGFR |
FDA approved |
FDA approved |
757443 |
Finasteride |
|
FDA approved |
FDA approved |
757804 |
Etoposide |
TOP2 |
FDA approved |
FDA approved |
757816 |
Fluphenazine |
NonCan:Psy |
FDA approved |
FDA approved |
758186 |
Azacitidine |
DNMT |
FDA approved |
FDA approved |
758230 |
Floxuridine |
Ds|TYMS |
FDA approved |
FDA approved |
758244 |
tepotinib |
PK:YK,MET |
FDA approved |
FDA approved |
758246 |
Trametinib |
PK:STK,MAP2K,MAP2K1,MAP2K2 |
FDA approved |
FDA approved |
758247 |
Palbociclib |
PK:STK,CDK,CDK4,CDK6 |
FDA approved |
FDA approved |
758252 |
Carfilzomib |
PSM |
FDA approved |
FDA approved |
758253 |
Homoharringtonine |
Apo|Ang|Pi |
FDA approved |
FDA approved |
758254 |
Ixazomib citrate |
PSM |
FDA approved |
FDA approved |
758255 |
Teniposide |
TOP2 |
FDA approved |
FDA approved |
758487 |
Ponatinib |
BCR-ABL|PK:YK |
FDA approved |
FDA approved |
758612 |
Bleomycin |
Db |
FDA approved |
FDA approved |
758645 |
Paclitaxel |
TUBB|Tu-stab |
FDA approved |
FDA approved |
758664 |
Rapamycin |
PK:STK,MTOR |
FDA approved |
FDA approved |
758667 |
Teniposide |
TOP2 |
FDA approved |
FDA approved |
758706 |
Simvastatin |
AM|NonCan:Chol |
FDA approved |
FDA approved |
758774 |
Belinostat |
HDAC |
FDA approved |
FDA approved |
759155 |
Doxorubicin |
TOP2 |
FDA approved |
FDA approved |
759174 |
Vincristine |
TUBB|Tu-frag |
FDA approved |
FDA approved |
759178 |
Pipamperone |
NonCan:Psy |
FDA approved |
FDA approved |
759195 |
Epirubicin |
TOP2 |
FDA approved |
FDA approved |
759224 |
Idelalisib |
PK:PIK3 |
FDA approved |
FDA approved |
759263 |
Topotecan |
TOP1 |
FDA approved |
FDA approved |
759274 |
ARSENIC TRIOXIDE |
Apo |
FDA approved |
FDA approved |
759614 |
6-Mercaptopurine |
Ds|PPAT |
FDA approved |
FDA approved |
759850 |
Docetaxel |
TUBB|Tu-stab |
FDA approved |
FDA approved |
759852 |
Vorinostat |
HDAC |
FDA approved |
FDA approved |
759856 |
Gefitinib |
PK:YK,EGFR |
FDA approved |
FDA approved |
759857 |
Clofarabine |
Ds |
FDA approved |
FDA approved |
759877 |
Dasatinib |
BCR-ABL|PK:YK,PDGFR,KIT |
FDA approved |
FDA approved |
759878 |
Irinotecan |
TOP1 |
FDA approved |
FDA approved |
760087 |
VINORELBINE |
TUBB|Tu-frag |
FDA approved |
FDA approved |
760443 |
Copanlisib |
PK:PIK3 |
FDA approved |
FDA approved |
760766 |
Vandetanib |
PK:STK,YK,PDGFR,EGFR,VEGFR,RET |
FDA approved |
FDA approved |
761068 |
Cabozantinib |
PK:YK,MET,AXL,KIT,VEGFR,FLT3,RET |
FDA approved |
FDA approved |
761190 |
Panobinostat |
HDAC |
FDA approved |
FDA approved |
761191 |
brigatinib |
PK:YK,ALK,EGFR |
FDA approved |
FDA approved |
761385 |
Sonidegib |
SMO|Hg-Smo |
FDA approved |
FDA approved |
761386 |
Sonidegib |
SMO|Hg-Smo |
FDA approved |
FDA approved |
761388 |
Plerixafor |
CXCR4 |
FDA approved |
FDA approved |
761389 |
Raloxifene |
Ho|SERM |
FDA approved |
FDA approved |
761431 |
Vemurafenib |
PK:YK,BRAF |
FDA approved |
FDA approved |
761432 |
Cabazitaxel |
TUBB|Tu-stab |
FDA approved |
FDA approved |
761910 |
Ibrutinib |
PK:YK,BTK |
FDA approved |
FDA approved |
763371 |
Ruxolitinib |
PK:YK,JAK,JAK1,JAK2 |
FDA approved |
FDA approved |
763932 |
Regorafenib |
GTPase|PK:STK,YK,PDGFR,FGFR,KIT,MAP2K,RAF,VEGFR,RET,Multikinase |
FDA approved |
FDA approved |
764040 |
Alectinib |
PK:YK,ALK |
FDA approved |
FDA approved |
764042 |
ARRY-162 |
PK:STK,MAP2K,MAP2K1,MAP2K2 |
FDA approved |
FDA approved |
764134 |
Dabrafenib |
PK:BRAF |
FDA approved |
FDA approved |
764778 |
Ivacaftor |
|
FDA approved |
FDA approved |
764821 |
Alectinib |
PK:YK,ALK |
FDA approved |
FDA approved |
765396 |
BMN-673 |
PARP1 |
FDA approved |
FDA approved |
765694 |
Bosutinib |
STAT|BCR-ABL|STAT5A/B|PK:YK,LYN,SRC,HCK |
FDA approved |
FDA approved |
765888 |
Dacomitinib |
PK:EGFR,ERBB2 |
FDA approved |
FDA approved |
766270 |
ABT-199 |
BCL2 |
FDA approved |
FDA approved |
767125 |
BMN-673 |
PARP1 |
FDA approved |
FDA approved |
768068 |
Cobimetinib (isomer 1) |
PK:MAP2K,MAP2K1 |
FDA approved |
FDA approved |
768069 |
Cobimetinib (isomer 1) |
PK:MAP2K,MAP2K1 |
FDA approved |
FDA approved |
768073 |
LY-2835219 |
PK:CDK,CDK4,CDK6 |
FDA approved |
FDA approved |
771649 |
ARN-509 |
AR |
FDA approved |
FDA approved |
772469 |
IPI-145 |
PK:PIK3 |
FDA approved |
FDA approved |
774769 |
NMS-E628 |
PK:ALK |
FDA approved |
FDA approved |
775351 |
Pomalidomide |
Immunomodulatory |
FDA approved |
FDA approved |
775772 |
PF-04449913 |
SMO |
FDA approved |
FDA approved |
776422 |
LDK-378 |
PK:ALK |
FDA approved |
FDA approved |
777193 |
LDK-378 |
PK:ALK |
FDA approved |
FDA approved |
777878 |
TABRECTA |
PK:MET |
FDA approved |
FDA approved |
778304 |
Encorafenib |
PK:BRAF |
FDA approved |
FDA approved |
778590 |
Cobimetinib (isomer 1) |
PK:MAP2K,MAP2K1 |
FDA approved |
FDA approved |
778909 |
LEE-011 |
PK:CDK,CDK4,CDK6 |
FDA approved |
FDA approved |
779217 |
Osimertinib |
PK:EGFR |
FDA approved |
FDA approved |
780108 |
PF-06463922 |
PK:ROS1,ALK |
FDA approved |
FDA approved |
781556 |
JNJ-42756493 |
PK:FGFR,FGFR1,FGFR2,FGFR3,FGFR4 |
FDA approved |
FDA approved |
785497 |
INCB-024360 |
IDO1 |
FDA approved |
FDA approved |
785570 |
LOXO-101 |
PK:NTRK |
FDA approved |
FDA approved |
787457 |
brigatinib |
PK:YK,ALK,EGFR |
FDA approved |
FDA approved |
787846 |
gilteritinib |
PK:AXL,FLT3 |
FDA approved |
FDA approved |
788120 |
Enasidenib |
IDH2 |
FDA approved |
FDA approved |
788948 |
Vistonuridine |
TUBB|FU-Antidote |
FDA approved |
FDA approved |
789102 |
ivosidenib |
IDH1 |
FDA approved |
FDA approved |
791164 |
Acalabrutinib |
PK:BTK |
FDA approved |
FDA approved |
797937 |
Sulfatinib |
PK:YK,FGFR |
FDA approved |
FDA approved |
800405 |
umbralisib |
|
FDA approved |
FDA approved |
809693 |
Copanlisib |
PK:PIK3 |
FDA approved |
FDA approved |
813783 |
Trabectedin |
A2 |
FDA approved |
FDA approved |